Patents
Patents for C07D 471 - Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups (64,559)
12/1997
12/23/1997US5700808 5- or 6-substituted β-carboline-3-carboxylic acid esters
12/23/1997US5700796 Useful for treating congestive heart failure, disease conditions with excess renal water reabsorption and conditions with increased vasular resistance and coronary vasoconstriction
12/23/1997US5700757 Triazolopyridine dyes and intermediates therefor
12/23/1997US5700448 Contrast media
12/23/1997CA2027206C Sulphonylaminocarbonyltriazolinones
12/19/1997CA2208136A1 Inhibition of abnormal accumulation of extracellular matrices
12/18/1997WO1997047625A1 Tricyclic benzazepine vasopressin antagonists
12/18/1997WO1997047622A1 Cytokine production inhibitors, triazepine compounds, and intermediates thereof
12/18/1997WO1997047601A1 Fused heterocyclic compounds and medicinal uses thereof
12/18/1997CA2258053A1 Cytokine production inhibitors, triazepine compounds, and intermediates thereof
12/17/1997EP0812843A2 Process for the preparation of 2,3-pyridinedicarboximides
12/17/1997EP0812842A2 Process for the preparation of 5-(alkoxymethyl)-2,3-pyridine-dicarboximide compounds
12/17/1997EP0812841A1 Crystal of N-((quinolin-2-yl)-phenyl)sulfonamides and process for producing the same
12/17/1997EP0812838A1 Pyridonecarboxylic acid derivative substituted by bicyclic amino group, ester thereof, salt thereof, and bicyclic amine as intermediate therefor
12/17/1997EP0729456B1 Novel process for preparing (s)-1-[2(s)-(1,3-dihydro-1,3-dioxo-isoindol-2-yl)-1-oxo-3-phenylpropyl]-1,2,3,4-tetrahydro-2-pyridine-carboxylic acid methyl ester and intermediates thereof
12/17/1997EP0698025B1 Ampa antagonists and a method of treatment therewith
12/17/1997EP0644762B1 Pyrazolopyridine compounds for the treatment of anemia
12/17/1997CN1168151A Process for producing and purifying perylene-3,4-dicarboxylic acid imides
12/17/1997CN1168138A Aryl and heteroaryl purine compounds
12/17/1997CN1036711C Process for preparation of imidazoindolizine derivs.
12/16/1997US5698692 Inhibit binding between platelet membrane glycoprotein and fibrinogen
12/16/1997US5698675 Reagents for peptide couplings
12/16/1997US5698577 Compositions of bicyclic β-lactams and uses thereof
12/16/1997US5698570 Quinoline carboxylic acid derivatives having 7-(4-amino-methyl-3-oxime)pyrrolidine substituent and processes for preparing thereof
12/16/1997US5698568 Substance p antagonists
12/16/1997US5698567 Heterocyclic spiro compounds
12/16/1997US5698561 Medicament for treating or preventing cerebrovascular dementia
12/16/1997US5698559 Disubstituted polycyclic systems as cognition enhancers
12/16/1997US5698555 Hetaryloxy-β-carbolines, their production and use in pharmaceutical agents
12/16/1997US5698548 Spirocycloalkyl-substituted azetidinones useful as hypocholesterolemic agents
12/16/1997CA2120360C Fluoroalkylated amphiphilic ligands, their metallic complexes and their uses
12/13/1997CA2207464A1 Crystal of n-{(quinolin-2-yl)phenylsulfonamides and process for producing the same
12/11/1997WO1997046559A1 Process for preparing 9-hydroxyellipticine
12/11/1997WO1997046558A1 Pyrrolo[2,3-b]pyridine derivatives, useful as radiolabelled d4 receptor ligands
12/11/1997WO1997020841A3 New macrobicyclic compounds, methods of preparing them and pharmaceutical agents containing them
12/11/1997CA2256351A1 Pyrrolo[2,3-b]pyridine derivatives, useful as radiolabelled d4 receptor ligands
12/10/1997EP0811613A1 Antibiotic Quinolones and derivatives
12/10/1997EP0810995A1 Photochromic material for electro-optic storage memory
12/10/1997EP0810991A1 1-aryl-2-acylamino-ethane compounds and their use as neurokinin especially neurokinin 1 antagonists
12/10/1997EP0686158B1 Methods for purifying 20(s)-camptothecin
12/10/1997EP0570575B1 Bicycloazamacrocyclophosphonic acid, conjugates, contrast agents and preparation
12/10/1997CN1036653C Heterocyclic ring spiroring compounds and process for preparing same
12/10/1997CN1036652C Quaternary basic amides, method of preparing them and pharmaceutical compositions in which they are present
12/10/1997CA2207453A1 Process for the preparation of 5-(alkoxymethyl)-2,3-pyridinedicarboximide compounds
12/10/1997CA2207261A1 Process for the preparation of 2,3-pyridinedicarboximides
12/09/1997US5696254 Processes for the diastereoselective synthesis of nucleoside analogues
12/09/1997US5696145 Vasopressin and oxytocin receptor
12/09/1997US5696133 Administering compound which modulates activity of progesterone receptor
12/09/1997US5696132 Microbiocides
12/09/1997US5696130 Tricyclic steroid receptor modulator compounds and methods
12/09/1997US5696129 5-HT4 antagonists
12/09/1997US5696127 Steroid receptor modulator compounds and methods
12/09/1997CA1339572C Macrocyclic amine complexes for ligand extraction and generation
12/06/1997CA2206914A1 Antibiotic quinolones and derivatives
12/04/1997WO1997045429A1 Beta-lactams
12/04/1997WO1997045428A1 Novel pyridazine compounds
12/04/1997WO1997045427A1 PYRIDOCARBAZOLE DERIVATIVES HAVING cGMP-PDE INHIBITORY EFFECT
12/04/1997WO1997045421A1 Oxocoumarin and barbituric acid derivates, their preparation and their use as ligand inhibitors of a corticotropin-releasing factor (crf) and/or a crf-binding protein complex
12/04/1997CA2256889A1 Pyridocarbazole derivatives having cgmp-pde inhibitory effect
12/04/1997CA2254943A1 Beta-lactams
12/04/1997CA2254744A1 Oxocoumarin and barbituric acid derivates, their preparation and their use as ligand inhibitors of a corticotropin-releasing factor (crf) and/or a crf-binding protein complex
12/04/1997CA2252747A1 Novel pyridazine compounds
12/03/1997EP0809642A1 Imidazo 1,2-a]pyridines for the treatment of cns and cardiac diseases
12/03/1997EP0809494A1 The use of heterocyclic compounds
12/03/1997CN1166831A Novel benzyl pyrimidines
12/03/1997CN1166490A Prep of novel mercaptoacetylamide derivatives
12/03/1997CN1166489A Prep. of novel alkyl-substituted alpha-ketone ester
12/03/1997CN1036590C Process for preparation of mercaptoacetylamide derivatives
12/02/1997US5693814 Crystals of antimicrobial compound
12/02/1997US5693812 Polymorphic forms of an angiotensin II antagonist
12/02/1997US5693811 Process for preparing tetrahdroimidazoquinolinamines
12/02/1997US5693808 Process for the preparation of peryleneimides, novel di-, tri- and tetrachromophoric perylene dyes and their use
12/02/1997US5693801 Anticonvulsants; anxiolytic agents; stimulants; treatment of overdoses of benzodiazepines
12/02/1997US5693787 Stereospecific
12/02/1997US5693663 Substituted bicyclic 3-aryl-pyrrolidine-2,4-dione derivatives
12/02/1997US5693657 Useful for treating hypercholesterolemia or atherosclerosis
12/02/1997US5693652 Benzimidazoles for ischemic heart conditions
12/02/1997US5693647 Steroid receptor modulator compounds and methods
12/02/1997US5693646 Steroid receptor modulator compounds and methods
12/02/1997US5693643 Hydantoin and succinimide-substituted derivatives of spiroindanylcamphorsulfonyl oxytocin antagonists
12/02/1997US5693636 Bicyclic fibrinogen antagonists
12/02/1997US5693635 Tricyclic benzazepine vasopressin antagonists
12/02/1997US5693633 Angiotensin II antagonists
11/1997
11/27/1997WO1997044342A1 PROCESS FOR PREPARING 1-ARYL-4-OXOPYRROLO[3,2-c]QUINOLINE DERIVATIVES
11/27/1997WO1997044337A1 Benzofuran carboxamides and their therapeutic use
11/27/1997WO1997044321A1 Antagonists of gonadotropin releasing hormone
11/27/1997WO1997044040A1 Hexahydro-pyrido(4,3-b)indole derivatives as antipsychotic drugs
11/27/1997WO1997044039A1 Aqueous suspensions of 9-hydroxyrisperidone fatty acid esters
11/27/1997WO1997044038A1 Tetrahydropteridines and pyridylpiperazines for treatment of neurological disorders
11/27/1997CA2255650A1 Tetrahydropteridines and pyridylpiperazines for treatment of neurological disorders
11/27/1997CA2254768A1 Antagonists of gonadotropin releasing hormone
11/27/1997CA2252537A1 Benzofuran carboxamides and their therapeutic use
11/26/1997EP0808835A1 Process for the preparation of optically active compounds
11/26/1997EP0808318A1 Tricyclic substituted hexahydrobenz e]isoindole alpha-1 adrenergic antagonists
11/26/1997EP0808313A1 Antipsychotic 4-(1h-indolyl-1-yl)-1-substituted piperidine derivatives
11/26/1997EP0808303A1 5-(4-subst.-piperidinyl-1)-3-aryl-pentanoic acid derivatives as tachykinin receptor antagonist
11/26/1997EP0808166A1 Medicament intended to the treatment of obsessive compulsive troubles, sleep apnoea, sexual dysfunctions, emesa and transport sickness
11/26/1997CN1166169A Heterocyclic compounds, useful as allosteric effectors at muscarinic receptors
11/26/1997CN1165817A New inhibitors of metalloprotease, process for preparing them and pharmaceutical compositions containing them
11/25/1997US5691366 Unsaturated nitro oxime formed by reaction of dinitrogen trioxide with diolefin ether, sulfide or amine to be used as vasodilators