Patents
Patents for C07D 417 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group (62,773)
09/2003
09/11/2003US20030171359 Suitable for treatment of illnesses characterised by excessive or abnormal cell proliferation; viral, bacterial, fungal and/or parasitic infections, skin diseases, bone diseases, cardiovascular diseases
09/11/2003US20030171354 Indole derivatives
09/11/2003US20030171309 Pharmaceutically active pyrrolidine derivatives as bax inhibitors
09/11/2003US20030171219 2,4,5-trisubstituted phenylketo-enols for use as pesticides and herbicides
09/11/2003US20030171218 Substituted 3-heteroaryl(amino- or oxy) pyrrolidin-2-ones of the formula (I), processes for preparing them, and their use as herbicides or as plant growth regulators.
09/11/2003US20030168970 Luminescent element material and luminescent element comprising the same
09/10/2003EP1342721A1 Sulfonamides and derivatives thereof that modulate the activity of endothelin
09/10/2003EP1341782A2 Inhibitors of p38 kinase
09/10/2003EP1341776A1 Benzazolonylcarbonyl cyclohexenones and use thereof as herbicides
09/10/2003EP1341771A2 Benzimidazole derivatives useful as tie-2 and/or vegfr-2 inhibitors
09/10/2003EP1341761A1 SUBSTITUTED INDOLES, PHARMACEUTICAL COMPOSITIONS CONTAINING SUCH INDOLES AND THEIR USE AS PPAR-$g(g) BINDING AGENTS
09/10/2003EP1341755A1 Carboxylic acid amide derivatives and their use in the treatment of thromboembolic diseases and tumours
09/10/2003EP1341540A2 Tyrosine kinase inhibitors
09/10/2003EP1131321B1 Indole derivatives and their use as serotonin receptor ligands
09/10/2003EP0873341B1 Epothilone derivatives, preparation and use
09/10/2003EP0851862B1 1(hetero)aryl-4-(condensed thiazol-2-ylalkyl)-piperazine derivatives, their preparation and their use in the treatment of 5-ht1a-receptor mediated disorders
09/10/2003CN1441800A Beta 3 adrenergic agonists
09/10/2003CN1441788A Novel arylethene-sulfonamides compounds
09/10/2003CN1441785A Tetrahydroixoquinoline analogs useful as growth hormone secretagogues
09/10/2003CN1441783A Medicine comprising dicyanopyridine derivative
09/10/2003CN1441782A N-oxides as NK1 receptor antagonist prodrugs of 4-phenyl-pyridine derivatives
09/10/2003CN1441781A Pharmaceutically active piperidine derivatives, in particular as modulators of chemokine receptor activity
09/10/2003CN1441780A Piperidine compounds for use as CCR-3 inhibitors
09/10/2003CN1441779A Proline derivatives and use thereof as drugs
09/09/2003US6617341 Insecticidal 2-iminothiazole derivatives
09/09/2003US6617339 Oxazolidinone derivatives, process for their preparation and pharmaceutical compositions containing them
09/09/2003US6617324 Substituted pyrazoles as p38 kinase inhibitors
09/09/2003CA2078814C Substituted pyridinylamino-1h-indoles, 1h-indazoles, 2h-indazoles, benzo[b]thiophenes and 1,2-benzisothiazoles, a process for their preparation and their use as medicaments
09/04/2003WO2003072577A1 Thiazole derivatives as npy receptor antagonists
09/04/2003WO2003072575A1 3-cyclyl-5-(nitrogen-containing 5-membered ring) methyl-oxazolidinone derivatives and their use as antibacterial agents
09/04/2003WO2003072574A1 Piperidine ouracil used as a medicament for treating bacterial infections
09/04/2003WO2003072566A1 Fused tricyclic heterocycles useful for treating hyper-proliferative disorders
09/04/2003WO2003072561A1 Benzofuran and benzothiophene derivatives useful in the treatment of hyper-proliferative disorders
09/04/2003WO2003072557A1 5-phenylthiazole derivatives and use as pi3 kinase inhibitors
09/04/2003WO2003072554A1 Azole compounds
09/04/2003WO2003072553A1 N-aryl-2-oxazolidinone-5-carboxamides and their derivates and their use as antibacterials
09/04/2003WO2003072551A1 Uracil-thioether
09/04/2003WO2003072528A2 (substituted)acyl dipeptidyl inhibitors of the ice/ced-3 family of cysteine proteases
09/04/2003WO2003072197A1 Acc inhibitors
09/04/2003WO2003072107A1 Substituted pyrimidinones and pyrimidinthiones
09/04/2003WO2003072102A1 Peroxisome proliferator activated receptor modulators
09/04/2003WO2003072100A1 Peroxisome proliferator activated receptor modulators
09/04/2003WO2003072033A2 Common ligand mimics: thiazolidinediones and rhodanines
09/04/2003WO2003062209A3 Substituted quinazolin-4-ylamine analogues as modulators of capsaicin
09/04/2003WO2003053367A3 Hydrogenation of precursors to thiazolidinedione antihyperglycemics
09/04/2003WO2003045313A3 2-aminoquinoline compounds
09/04/2003WO2003037891A8 Heteroaryl amines as glycogen synthase kinase 3beta inhibitors (gsk3 inhibitors)
09/04/2003WO2003037262A3 Novel anit-infectives
09/04/2003WO2003018002A3 Cyclopropyl and cyclobutyl epothilone analogs
09/04/2003US20030166927 1,5-Benzothiazepines and their use as hypolipidaemics
09/04/2003US20030166697 Divalent aromatic heterocyclic compounds useful in prevention or treatment of hyperlipidemia, arteriosclerosis, diabetes mellitus, hypertension, obesity, and the like
09/04/2003US20030166690 Use of compounds for decreasing activity of hormone-sensitive
09/04/2003US20030166689 Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1
09/04/2003US20030166685 Acid derivatives of benzene useful as anticoagulants in treating and preventing cardiovascular diseases, as anti-inflammatory agents, and as metastasis inhibitors in treating cancer
09/04/2003US20030166675 Substituted quinolin-2-one derivatives useful as antiproliferative agents
09/04/2003US20030166668 Substituted heteroarylalkanoic acids
09/04/2003US20030166664 E.g. 3-(1-(2-(5-(acetylamino)-2-methylphenyl)ethyl)piperidin--4-yl)-6-chloro-1H -indole; potent dopamine D4 ligands, dopamine antagonists; antiseratonin agents; psychoses; anxiolytic agents; antidepressants; side effects reduction
09/04/2003US20030166658 Condensing a heterocyclic ketone or aldehyde with a 2-(NH2-NH-)benzimidazole, -oxazole or -thiazole; ribonucleotide reductase inhibitors; anticarcinogenic and -tumor agents; also useful against multidrug resistant cells
09/04/2003US20030166652 Chemical compounds
09/04/2003US20030166649 E.g., 4-(2-(1-Benzhydryl-2-(2-((benzylsulfonyl)amino)ethyl)-5-chloro-1H-indol-3 -yl)ethoxy)benzoic acid; inhibitors of phospholipase enzymes, esp. phospholipase A2; antiarthritic and -inflammatory agents; analgesics; rheumatoid diseases
09/04/2003US20030166646 Nitric oxide synthase inhibitors such as 4-(morpholin-4-yl methyl)-4,5-dihydro-1,3-thiazol-2-ylamine, administered for prophylaxis of neurodegenerative diseases
09/04/2003US20030166644 Compounds and uses thereof for decreasing activity of hormone-sensitive lipase
09/04/2003US20030166635 Novel 2-nitromethylidene/2-cyanimino/2-nitro-imino-pyrrolidines and piperidines, intermediates, and their use as pesticides
09/04/2003US20030166633 Pyridinylimidazoles
09/04/2003US20030166590 Microsomal triglyceride transfer protein
09/04/2003US20030166574 1,3,4-Oxadiazoline derivatives and drugs containing these derivatives as active ingredient
09/04/2003US20030165640 Filters for electronic display device
09/04/2003CA2477344A1 3-cyclyl-5-(nitrogen-containing 5-membered ring) methyl-oxazolidinone derivatives and their use as antibacterial agents
09/04/2003CA2477287A1 Uracil-thioether
09/04/2003CA2477224A1 Piperidine ouracil used as a medicament for treating bacterial infections
09/04/2003CA2477008A1 Substituted pyrimidinones and pyrimidinthiones
09/04/2003CA2476038A1 N-aryl-2-oxazolidinone-5-carboxamides and their derivates and their use as antibacterials
09/04/2003CA2475653A1 (substituted)acyl dipeptidyl inhibitors of the ice/ced-3 family of cysteine proteases
09/04/2003CA2475299A1 Thiazole derivatives as npy receptor antagonists
09/03/2003EP1341403A1 Luminescent element material and luminescent element comprising the same
09/03/2003EP1340754A1 Substituted heterocyclic compounds, process for their preparation and pharmaceutical compositions containing them
09/03/2003EP1340750A1 Amide derivatives
09/03/2003EP1340749A1 Isoxazole derivatives
09/03/2003EP1340744A2 Hiv protease inhibitors
09/03/2003EP1340498A1 Use of epothilones in the treatment of brain diseases associated with proliferative processes
09/03/2003EP1339711A1 Aminothiazoles and their use as adenosine receptor antagonists
09/03/2003EP1339709A1 Farnesyl transferase inhibiting benzoheterocyclic derivatives
09/03/2003EP1339702A1 5-amide substituted diarylamines as mek inhibitors
09/03/2003EP1339701A1 Heteroaryl alkyl piperazine derivatives as fatty acid oxidation inhibitors
09/03/2003EP1339696A1 Benzyl(idene)-lactams and their use as 5ht1-receptor ligands
09/03/2003EP1339692A1 Novel compounds for use as hiv protease inhibitors
09/03/2003EP1339688A1 N-type calcium channel antagonists for the treatment of pain
09/03/2003EP1339680A1 Substituted oxindole derivatives as tyrosine kinase inhibitors
09/03/2003EP1339678A2 Ep4 receptor selective agonists in the treatment of osteoporosis
09/03/2003EP1339670A1 Substituted cyclohexane derivates and the use thereof in medicaments for treating cardiovascular diseases
09/03/2003EP1339403A2 Repinotan kit
09/03/2003EP1131319B1 3- benz(ox/thi)azol-7-yl -1h-pyrimidine-2,4-diones
09/03/2003EP1077947B1 Novel 1,5 and 3-o-substituted 1h-indazoles with anti-asthmatic, anti-allergic, anti-inflammatory, immuno-modulating and neuro-protective effect, method for the production and use thereof as medicaments
09/03/2003EP1060178B1 Heterocyclic compounds as inhibitors of rotamase enzymes
09/03/2003EP0929533B1 4,4-disubstituted-1,4-dihydro-2h-3,1-benzoxazin-2-ones useful as hiv reverse transcriptase inhibitors and intermediates and processes for making the same
09/03/2003EP0783496B9 Thiazolidinedione derivatives, their production and use
09/03/2003EP0612318B1 Heteroarylpiperidines, pyrrolidines and piperazines and their use as antipsychotics and analgetics
09/03/2003CN1440403A Quinazoline ditosylate salt compounds
09/03/2003CN1440402A N-ureidoheterocycloaklyl-piperidines as modulators of chemokine receptor activity
09/03/2003CN1440401A Amino substituted dibenzothiophene derivatives for treatmnt of disorders mediated by NP Y5 receptor