Patents
Patents for C07D 413 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms (64,687)
10/1999
10/21/1999WO1999052906A1 Substituted oxazolyle and thiazolyl uracil herbicides
10/21/1999WO1999052905A1 Process for producing indolmycins
10/21/1999WO1999052898A1 N,n-disubstituted amides that inhibit the binding of integrins to their receptors
10/21/1999WO1999052875A1 Amine compounds, their production and their use as somatostatin receptor antagonists or agonists
10/21/1999WO1999052869A1 Substituted indolinones having an inhibiting effect on kinases and cycline/cdk complexes
10/21/1999WO1999052868A1 Substituted pyrrolidine hydroxamate metalloprotease inhibitors
10/21/1999WO1999052851A1 Phosphate-mediated cyclization
10/21/1999WO1999052529A1 Antioxidant stabilizer system for pharmaceutical formulations
10/21/1999WO1999052493A2 Compounds that inhibit the binding of integrins to their receptors
10/21/1999DE19817459A1 New heterocyclic amide derivatives useful as cysteine protease inhibitors for treating neurodegenerative diseases, neuronal damage, stroke, cranial trauma, Alzheimer's disease, etc.
10/21/1999DE19817262A1 New dihydropyrimidine derivatives and their corresponding mesomers useful in treatment of hepatitis
10/21/1999DE19816624A1 Neue substituierte Indolinone, ihre Herstellung und ihre Verwendung als Arzneimittel New substituted indolinones, their preparation and their use as medicaments
10/21/1999CA2328211A1 Substituted pyrrolidine hydroxamate metalloprotease inhibitors
10/21/1999CA2327928A1 Phosphate-mediated cyclization
10/21/1999CA2327708A1 Antioxidant stabilizer system for pharmaceutical formulations
10/21/1999CA2327695A1 Amine compounds, their production and their use as somatostatin receptor antagonists or agonists
10/21/1999CA2327689A1 Process for producing indolmycins
10/21/1999CA2327282A1 Treatment of parasitic diseases by inhibition of cysteine proteases of the papain superfamily
10/20/1999EP0950656A1 Sulfonated amino acid derivatives and metalloproteinase inhibitors containing the same
10/20/1999EP0832078B1 N-hydroxyureas as antiinflammatory agents
10/20/1999EP0717738B1 Substituted oxazine and thiazine oxazolidinone antimicrobials
10/20/1999CN1232462A Muscarinic antagonists
10/20/1999CN1232457A 1,4-heterocyclic metalloprotease inhibitors
10/20/1999CN1232451A Substd. cyclic amine metalloprotease inhibitors
10/20/1999CN1232397A Use of H+, K+-ATPase inhibitor in treatment of nasal polyps
10/20/1999CN1045776C Thiazolidines and oxazolidines substd. by pyridine ring and their use as hypoglycemic agents
10/20/1999CN1045770C Method for preparation of 1-biphenylmethyl imidazole derivs.
10/20/1999CN1045768C Angiotension II antagonists compounds, preparing method and use thereof
10/19/1999US5969184 Amide compounds
10/19/1999US5969146 Monoamine oxidase inhibitors
10/19/1999US5969141 Intermediates for 7-amino-1-cyclopropyl-6,8-dihalogeno-1,4-dihydro-4-oxo-3-quinolinecarbox ylic acid antibacterial agents
10/19/1999US5969140 Aminopyridine derivatives of naphthalene for treatment of asthma and bronchoconstrictor inhibitors
10/19/1999US5968962 Phenyloxazolidinones having a C-C bond to 4-8 membered heterocyclic rings
10/19/1999US5968959 Administering phospholamban inhibitor
10/19/1999US5968955 Disubstituted piperidine derivatives as neuroprotective agents
10/19/1999US5968954 Exhibit selective binding affinity for 5-hydroxytryptamine receptors
10/19/1999US5968953 For side effect reduction
10/19/1999US5968947 Bicyclic amine derivatives
10/19/1999US5968934 Treatment of pain, inflammation, migraines, emesis and postherapeutic neuralgia
10/19/1999US5968923 (Azetidin-1-ylalkyl) lactams as tachykinin antagonists
10/14/1999WO1999051592A1 Indol-3-yl-cyclohexyl amine derivatives for the treatment of depression (5-ht1 receptor antagonists)
10/14/1999WO1999051587A1 Fused thiophene derivatives and drugs containing the same as the active ingredient
10/14/1999WO1999051580A1 Pyrazole inhibitors of cytokine production
10/14/1999WO1999045011A8 Glycine transport inhibitors
10/14/1999DE19854082A1 Substituierte Oxazolyl- und Thiazolyl-uracile Substituted oxazolyl and thiazolyl-uracils
10/14/1999CA2327360A1 Indol-3-yl-cyclohexyl amine derivatives for the treatment of depression (5-ht1 receptor antagonists)
10/14/1999CA2327185A1 Pyrazole inhibitors of cytokine production
10/13/1999EP0949261A1 Substituted piperidinedione derivatives and herbicides
10/13/1999EP0948498A1 Sulfonamide compounds having 5-ht receptor activity
10/13/1999EP0948494A1 Substituted benzo 1,4]dioxanes as antiobesity agents
10/13/1999EP0948489A1 Piperazine compounds as inhibitors of mmp or tnf
10/13/1999EP0948327A1 Antidiabetic agents
10/13/1999EP0948324A2 Methods and pharmaceutical compositions for inhibiting tumour cell growth
10/13/1999EP0692977B1 Novel heterocycle based nitrogen-sulfur ligands useful in radiographic imaging agents
10/13/1999CN1231664A Sulfonamicles and derivatives thereof that moulate the activity of endothelin
10/13/1999CN1231663A Arthropodicidal and fungicidal cyclic amides
10/13/1999CN1231662A Quinazoline derivatives and pharmaceutical compositions containing them
10/13/1999CN1231661A Aralkyl and aralkylidene heterocyclic lactams and imides
10/13/1999CN1045602C Tetrahydropyrido-indole derivant and medicinal composition and pharmaceutical use thereof
10/13/1999CN1045597C Alkylenediamine derivatives having heterocyclic group and medicinal composition thereof
10/13/1999CN1045595C Process for the preparation of the intermediates used in the synthesis of 3-aminopiperidine derivatives
10/12/1999US5965745 Asthma; antiarthritic,-shock agents; bronchitis; respiratory system diseases, e.g. chronic obstructive airways diseases; psoriasis; allergic rhinitis; atopic dermatitis
10/12/1999US5965740 Alpha-substituted benzyl heterocyclic derivatives, intermediates for producing the same and pesticides containing the same as active ingredient
10/12/1999US5965739 Oxazolidine protected taxol analogs of given formula, and methods of synthesis from an oxazolidine free acid and a baccatin compound in the presence of a dehydrating agent; useful intermediates to make various taxol analogues
10/12/1999US5965580 Piperidine derivatives, process for obtaining them and pharmaceutical compositions containing them
10/12/1999US5965579 Antagonists of the neurotensin receptors; increasing affinity for human neurotensin receptors
10/12/1999US5965565 Piperidines, pyrrolidines, and hexahydro-1h-azepines of given formula; can be used to promote growth of livestock and in humans treat physiological or medical conditions characterized by grwoth hormone defiency
10/12/1999US5965558 2 or 2,3-di((2-carboxyethylenearyl)quinoxalines; purification of proteins and glycoproteins; units including protein tyrosine phosphatases and proteins with src-homology-2 domains; antidiabetics,-allergens,-coagulants
10/12/1999US5965554 Antipsychotic agents, compositions and method of use
10/12/1999US5965553 Anticholesterol agents, hypotriglyceridemic agents, antiatherosclerosis agents, antifungal agents, alzheimer's agents or anti-acne agents
10/12/1999US5965546 1-[(2-pyrimidinyloxy)alkyl]4-(heteroaryl)piperazines and related compounds and their therapeutic utility
10/12/1999CA1340785C Platelet activating factor antagonists
10/07/1999WO1999050267A1 Process for producing isooxazolidinedione compound
10/07/1999WO1999050263A1 Quinolones as serine protease inhibitors
10/07/1999WO1999050257A1 Benzoxazinones/benzothiazinones as serine protease inhibitors
10/07/1999WO1999050253A1 4,4-disubstituted-3,4-dihydro-2(1h)-quinazolinthione derivatives, their preparation and their use as hiv reverse transcriptase inhibitors
10/07/1999WO1999050249A2 Pyrimidines and triazines as integrin antagonists
10/07/1999WO1999050245A1 Indole derivatives with antiviral activity
10/07/1999WO1999050243A1 The use of derivatives of 2-oxopyrrole as crop protection agents and novel 2-oxopyrroles
10/07/1999CA2333927A1 Pyrimidines and triazines as integrin antagonists
10/07/1999CA2326166A1 Indole derivatives with antiviral activity
10/07/1999CA2325904A1 The use of derivatives of 2-oxopyrrole as crop protection agents and novel 2-oxopyrroles
10/07/1999CA2322203A1 4,4-disubstituted-3,4-dihydro-2(1h)-quinazolinthione derivatives, their preparation and their use as hiv reverse transcriptase inhibitors
10/07/1999CA2319551A1 Benzoxazinones/benzothiazinones as serine protease inhibitors
10/07/1999CA2312953A1 Quinolones as serine protease inhibitors
10/06/1999EP0946587A2 New amide compounds
10/06/1999EP0946552A1 Sulfonamides and derivatives thereof that modulate the activity of endothelin
10/06/1999EP0946546A1 Pyridin-2-yl-methylamine derivatives, method of preparing and application as medicine
10/06/1999EP0946545A1 Novel carboxy substituted cyclic carboxamide derivatives
10/06/1999EP0946541A1 Quinolines and their therapeutic use
10/06/1999EP0946528A2 OXYGEN OR SULFUR CONTAINING 5-MEMBERED HETEROAROMATICS AS FACTOR Xa INHIBITORS
10/06/1999EP0946519A1 Benzamide derivatives having a vasopressin antagonistic activity
10/06/1999EP0946512A1 6-phenylpyridyl-2-amine derivatives useful as nos inhibitors
10/06/1999EP0946508A1 NITROGEN CONTAINING HETEROAROMATICS AS FACTOR Xa INHIBITORS
10/06/1999EP0946175A1 USE OF AN H+, K+ -ATPase INHIBITOR IN THE TREATMENT OF NASAL POLYPS
10/06/1999CN1230958A Oxazolone derivatives and their use as anti-helicobacter pylori agents
10/06/1999CN1230950A Method of production and method of separation of 2,4'-dipyridyl derivatives and methods of production of benzoxazepine derivatives and salts thereof
10/06/1999CN1230542A Sidechain-bearing taxanes
10/06/1999CN1045441C Antifungal agents, processes for the preparation thereof, and intermediates
10/06/1999CN1045439C Heterarylation acyl iso-oxazole derivative its preparation and use and composition with the same