Patents
Patents for C07D 413 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms (64,687)
01/2002
01/03/2002WO2002000645A1 Indole derivatives useful for the treatment of cns disorders
01/03/2002WO2002000632A1 Benzodiazepines as inhibitors of hpv e1 helicase
01/03/2002WO2002000631A2 Benzhydryl derivatives
01/03/2002WO2002000626A1 Fused azepine derivatives and their use as antidiuretic agents
01/03/2002WO2002000590A1 Synthesis of functionalized and unfunctionalized olefins via cross and ring-closing metathesis
01/03/2002WO2001062233A3 Adenosine receptor modulators
01/03/2002US20020002199 Suitable for treating type I diabetes, type II diabetes, impaired glucose tolerance, insulin resistance or obesity
01/03/2002US20020002194 Synthesis of epothilones, intermediates thereto, analogues and uses thereof
01/03/2002US20020002169 Protein kinase inhibitors
01/03/2002US20020002164 Morpholine and thiomorpholine tachykinin receptor antagonists
01/03/2002DE10027514A1 Liganden von Integrinrezeptoren Ligands of integrin
01/03/2002CA2414115A1 Indole derivatives useful for the treatment of cns disorders
01/03/2002CA2412592A1 Substituted quinazoline derivatives and their use as inhibitors
01/03/2002CA2412555A1 Fused azepine derivatives and their use as antidiuretic agents
01/03/2002CA2411157A1 Benzodiazepines as inhibitors of hpv e1 helicase
01/03/2002CA2409762A1 Heteroaryl-phenyl substituted factor xa inhibitors
01/02/2002EP1167366A1 Amine derivatives
01/02/2002EP1165693A2 Squaraine dyes
01/02/2002EP1165554A1 New endothelin converting enzyme inhibitors, their production and their use
01/02/2002EP1165547A1 Substituted benzoylpyrazoles as herbicides
01/02/2002EP1165545A1 Novel compounds
01/02/2002EP1165542A1 4-substituted quinoline derivatives as nk-3 and/or gaba(a) receptor ligands
01/02/2002EP1165540A1 Tetrahydropyran derivatives and their use as therapeutic agents
01/02/2002EP1165530A2 Dihetero-substituted metalloprotease inhibitors
01/02/2002EP1165528A1 Novel morpholine derivatives, method for the production thereof and pharmaceutical preparations containing said derivatives
01/02/2002EP1165516A2 Heterocyclic urea and related compounds useful as anti-inflammatory agents
01/02/2002EP1165515A1 Pyridine-2,3-dicarboxylic acid diamides
01/02/2002EP1165501A1 Alkenyl- and alkynyl-containing metalloprotease inhibitors
01/02/2002EP1165496A1 Substituted aniline compounds
01/02/2002EP1165472A1 Methods for the preparation of biphenyl isoxazole sulfonamides
01/02/2002EP1135151A4 Peptoid and nonpeptoid containing alpha-keto oxadiazoles as serine protease inhibitors
01/02/2002EP0912553B1 BENZO[g]QUINOLINE DERIVATIVES
01/02/2002EP0835256B1 Microbicidal benzotriazoles
01/02/2002EP0825189B1 1,4-benzodioxin derivatives
01/02/2002CN1329609A Tetrahydrobenza epine derivatives useful as modulators of dopamine D3 receptors (antipsychotic agents)
01/02/2002CN1329607A Substituted benzopyran analogs for treatment of inflammation
01/02/2002CN1329596A Picolinamide derivatives and pest controllers containing same as active ingredient
01/02/2002CN1329594A Ureidopiperidine derivatives as selective human NK3 receptor antagonists
01/02/2002CN1329002A Intermediate product for preparing aralkyl and aryl alkylene heterocyclic lactam and imide
01/02/2002CN1077107C Heterocyclic compounds, their production and use
01/01/2002US6335336 Treating tumor necrosis factor and mitogen-activated protein kinase(map) mediated disorders; antiinflammatory and antiarthritic agents; inflammatory bowel disease
01/01/2002US6335334 Hypertensive agents, anticoagulants; cardiovascular and sexual disorders, angina pectoris, and atherosclerosis
01/01/2002US6335333 Matrix metalloproteinase inhibitors
01/01/2002US6335327 1-benzazepine derivatives; agonists or antagonists of vasopressin and/or oxytocin
01/01/2002US6335326 Dopamine agonist and antagonists; central nervous system and psychological disorders; anxiolytic, antidepressant and antiischemic agents; parkinson*s disease
01/01/2002US6335325 Crop protection
01/01/2002CA2056799C 1,4-dihydropyridine derivatives and methods of producing the same
01/01/2002CA2051830C Tricyclic heterocycles
12/2001
12/27/2001WO2001098296A2 2-(3,5-disubstituted-4-pyridyl)-4-(thienyl, thiazolyl or arylphenyl)-1,3-oxazoline compounds
12/27/2001WO2001098291A2 1,3-bis-(substituted-phenyl)-2-propen-1-ones and their use to treat vcam-1 mediated disorders
12/27/2001WO2001098290A2 Thiophene derivatives active as kinase inhibitors, process for their preparation and pharmaceutical compositions comprising them
12/27/2001WO2001098282A1 Benzoxazepinones and their use as squalene synthase inhibitors
12/27/2001WO2001098277A2 Substituted bicyclic derivatives for the treatment of abnormal cell growth
12/27/2001WO2001098272A1 Novel compounds
12/27/2001WO2001098270A2 N-ureidoalkyl-piperidines as modulators of chemokine receptor activity
12/27/2001WO2001098269A2 N-ureidoalkyl-piperidines as modulators of chemokine receptor activity
12/27/2001WO2001098268A2 Piperidine amides as modulators of chemokine receptor activity
12/27/2001WO2001098267A1 3-azabicyclo (3.1.0) hexane derivatives having opioid receptor affinity
12/27/2001US20010056183 Sulfonamides and derivatives thereof that modulate the activity of endothelin
12/27/2001CA2414085A1 Thiophene derivatives active as kinase inhibitors, process for their preparation and pharmaceutical compositions comprising them
12/27/2001CA2413878A1 1,3-bis-(substituted-phenyl)-2-propen-1-ones and their use to treat vcam-1 mediated disorders
12/27/2001CA2413429A1 Benzoxazepinones and their use as squalene synthase inhibitors
12/27/2001CA2413421A1 N-ureidoalkyl-piperidines as modulators of chemokine receptor activity
12/27/2001CA2413418A1 Piperidine amides as modulators of chemokine receptor activity
12/27/2001CA2413274A1 N-ureidoalkyl-piperidines as modulators of chemokine receptor activity
12/27/2001CA2412188A1 3-azabicyclo¬3.1.0|hexane derivatives useful in therapy
12/27/2001CA2411255A1 Novel compounds
12/26/2001CN1328550A Oxazole compounds as prostaglandin E2 agonists or antagonists
12/26/2001CN1328546A Pyrrolidines as inhibitors of neuraminidases
12/26/2001CN1327978A Oxime additives and its use as fungicide
12/25/2001US6333416 Chemical intermediate for protease inhibitor
12/25/2001US6333414 By reaction of thiourea with the corresponding diketone ester; carried out under reaction conditions, particularly with respect to ph, which are industrially more favorable.
12/25/2001US6333344 Prolines as antimicrobial agents
12/25/2001US6333341 Tumor necrosis factor, antiinflammatory agents and analgesics
12/25/2001US6333338 Anticoagulants, cardiovascular disorders
12/25/2001US6333328 Serotonin 5-HT3 receptor partial activator
12/25/2001US6333325 Method of treating cytokine mediated diseases or conditions
12/25/2001US6333324 For therapy and prophylaxis of matrix metalloproteinases (mmp) or tumor necrosis factor .alpha. (tnf.alpha.), mediated diseases
12/25/2001US6333323 Indole derivatives with antiviral activity
12/25/2001CA2032602C 4-carbonyl-substituted coumarin compound
12/20/2001WO2001096334A2 Heteroarylalkanoic acids as integrin receptor antagonists
12/20/2001WO2001096333A1 Hetaryl-substituted heterocycles
12/20/2001WO2001096331A1 Lactam inhibitors of factor xa and method
12/20/2001WO2001096330A2 Thrombin receptor antagonists
12/20/2001WO2001096328A1 Indole derivatives useful for the treatment of cns disorders
12/20/2001WO2001096327A1 BIOISOSTERIC BENZAMIDE DERIVATIVES AND THEIR USE AS APoB-100 SECRETION INHIBITORS
12/20/2001WO2001096315A1 Process for the preparation of 1,2,4-triazolin-5-one derivatives
12/20/2001WO2001096308A1 1,2-dihydropyridine compounds, process for preparation of the same and use thereof
12/20/2001WO2001096307A2 Cycloalkyl alkanoic acids as integrin receptor antagonists
12/20/2001WO2001096302A1 Piperidines for use as orexin receptor antagonists
12/20/2001WO2001095911A1 Protease inhibitors
12/20/2001WO2001077107B1 Oxazole derivatives and their uses as tyrosine kinase inhibitors
12/20/2001WO2001062245A3 Bilirubin or biliverdin degradation fragments
12/20/2001WO2001058896A8 Benzoxazole derivatives as tnf and pde iv inhibitors
12/20/2001WO2001016108A3 Bicyclic androgen and progesterone receptor modulator compounds and methods
12/20/2001WO1999019304A3 Alpha-alkylthio substituted pyrimidine ethers and thioethers as viral reverse transcriptase inhibitors
12/20/2001US20010053779 Antiinflammatory agents; respiratory system disorders
12/20/2001DE10029077A1 New heterocyclic-substituted thiazole derivatives, useful as total or selective herbicides, insecticides, acaricides, nematocides, ectoparasiticides or antifouling agents
12/20/2001CA2412353A1 Protease inhibitors
12/20/2001CA2412216A1 Lactam inhibitors of factor xa and method