Patents
Patents for C07D 413 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms (64,687)
04/2002
04/30/2002US6380221 Ortho-anthranilamide derivatives as anti-coagulants
04/30/2002US6380220 Therapy of neurodegenerative diseases and neuronal injuries which are casued by ischemia, trauma or massive hemorrhages
04/30/2002US6380218 For therapy of respiratory, allergic, and inflammatory disorders comprising asthma, chronic obstructive pulmonary disease, acute respiratory disease syndrome, pulmonary hypersensitivity, and allergic rhinitis in a mammal
04/30/2002US6380215 For prevention and/or treatment of diseases caused by thrombus formation such as arterial thrombosis, arterial sclerosis, ischemic heart diseases
04/30/2002US6380213 Compounds useful as neuro-protective agents
04/30/2002US6380204 Alpha-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid receptor antagonist activity
04/30/2002US6380201 Methods of treating or ameliorating the symptoms of common cold or allergic rhinitis with serotonin 5-HT1F agonists
04/30/2002US6380191 Arylthiazolidinedione and aryloxazolidinedione derivatives
04/30/2002US6380189 2-amino benzoxazinones for the treatment of viral infections
04/30/2002US6380186 Psychotherapeutic agents
04/30/2002US6379823 Electroluminescence device, cyclic azine compound and production process of cyclic azine dye
04/25/2002WO2002032900A2 Aryl or heteroaryl fused imidazole compounds as anti-inflammatory and analgesic agents
04/25/2002WO2002032897A1 Alpha-aryl ethanolamines and their use as beta-3 adrenergic receptor agonists
04/25/2002WO2002032896A1 Furazanyl-triazole derivates for the treatment of diseases
04/25/2002WO2002032894A1 Substituted imidazoles useful in the treatment of inflammatory diseases
04/25/2002WO2002032893A2 Piperidine compounds as anti-allergic
04/25/2002WO2002032886A1 A process for the preparation of bis-benzazolyl compounds
04/25/2002WO2002032884A2 Methods for the preparation of biphenyl isoxazole sulfonamides
04/25/2002WO2002032872A1 Nitrogenous aromatic ring compounds
04/25/2002WO2002032857A1 Methods of producing oxazolidinone compounds
04/25/2002WO2002032422A2 Ep4 receptor inhibitors to treat rheumatoid arthritis
04/25/2002WO2002010137A3 Indazole derivatives as JNK inhibitors
04/25/2002WO2001081341A3 9-oxa-epothilon derivatives, method for the production and use thereof in pharmaceutical preparations
04/25/2002WO2001002369A3 Indazole compounds and pharmaceutical compositions for inhibiting protein kinases, and methods for their use
04/25/2002US20020049337 4-(2-amino-1-hydroxyethyl)oxazoline derivative and method for producing same
04/25/2002US20020049330 Such as 5-(N,N-dibenzyl)aminocarbonyl-2-pyridone; enzyme inhibitors; for treatment of Alzheimer's disease
04/25/2002US20020049329 Novel human NK3 receptor-selective antagonist compounds, method for obtaining them and pharmaceutical compositions containing them
04/25/2002US20020049243 Pyrrolidine derivatives
04/25/2002US20020049241 Conformationally rigid bicyclic and adamantane derivatives useful as alpha2-adrenergic blocking agents
04/25/2002US20020049236 Non-peptidyl inhibitors of VLA-4 dependent cell binding useful in treating inflammatory, autoimmune, and respiratory diseases
04/25/2002US20020049223 Quinoline and naphthyridine carboxylic acid antibacterials
04/25/2002US20020049222 Cyclopentyl modulators of chemokine receptor activity
04/25/2002US20020049220 Substituted azoles
04/25/2002US20020049217 Peptidomimetic macrocyclic compounds which inhibit prenyl-protein transferase and the prenylation of the oncogene protein Ras
04/25/2002US20020049213 Converting a benzaldehyde compound to an oxime in presence of hydroxylamine/hydrochloric acid and pyridine in methylene chloride, converting to intermediateand racting it with methoxyphenyl acetylene to form intermediate then final comp
04/25/2002US20020049211 Combination treatment for depression and anxiety
04/25/2002US20020049204 1,4-dihydro-benzo(d)oxazin-2-one derivatives useful for treating hormone-dependent neoplastic disease is selected from uterine myometrial fibroids, endometriosis, benign prostatic hypertrophy, carcinomas, and adenocarcinoma
04/25/2002US20020049202 Administering halogenated amidino or oxyamidino compound to treat diseases caused by nitric oxide synthase
04/25/2002US20020049201 Sulfonamide inhibitors of aspartyl protease
04/25/2002US20020049197 Aminoquinazolines and their use as medicaments
04/25/2002US20020049195 Urea compounds that are muscarinic receptor antagonists and agonists, administering to the mammal the urea compound to treat urinary incontinence, chronic pulmonary obstructive disease, asthma, hyper salivation, blurred vision etc.
04/25/2002US20020049194 A benzoazepin or benzodiazepin derivatives, shows excellent anti-vasopressin activity, vasopressin agonistic activity and oxytocin antagonistic activity, and are useful as antagonist
04/25/2002US20020049193 Inhibitors of the enzyme activity associated with immunophilin proteins, particularly peptidyl-prolyl isomerase, or rotamase, enzyme activity.
04/25/2002US20020049187 2-(azetidin-2-on-1-yl) acetic acid derivatives; treatment of obsessive-compulsive disorder
04/25/2002DE10051321A1 New 2-(4-amino-piperidin-1-yl)-2-aryl-N-(phenylalkyl)-acetamides, are potent neurokinin antagonists, useful e.g. for treating allergic, inflammatory or central nervous system diseases
04/25/2002CA2426487A1 Ep4 receptor inhibitors to treat rheumatoid arthritis
04/25/2002CA2426337A1 Substituted imidazoles useful in the treatment of inflammatory diseases
04/25/2002CA2425911A1 Methods for the preparation of biphenyl isoxazole sulfonamides
04/25/2002CA2423792A1 Alpha-aryl ethanolamines and their use as beta-3 adrenergic receptor agonists
04/25/2002CA2423599A1 Methods of producing oxazolidinone compounds
04/24/2002EP0714299B1 Benzoxazinone and benzopyrimidinone piperidinyl tocolytic oxytocin receptor antagonists
04/24/2002CN1346354A Substituted benzoylpyrazoles as herbicides
04/24/2002CN1346350A Compound which inhibiti leukocyte adhesion mediated by VLA-4
04/24/2002CN1346282A Use of a cyclooxygenase-2 inhibitor and one or more antineoplastic agents as combination therapy method in treating neoplasia
04/24/2002CN1346271A Quinazoline derivatives as angiogenesis inhibitors
04/24/2002CN1083450C Processes for preparing intermediate product used in method of diastereoselective syntheses of nucleosides
04/24/2002CN1083445C Thiodepsipeptides for combating endoparasites and a method for producing the same
04/24/2002CN1083443C 吲哚衍生物 Indole derivatives
04/24/2002CN1083439C 2-amino-4-bicyclomino-1,3,5-triazines as herbicides and plant growth regulators
04/24/2002CN1083431C Novel heterocyclic compounds
04/23/2002US6376548 Enhanced propertied pesticides
04/23/2002US6376538 Antiinflammatory agents; autoimmune diseases
04/23/2002US6376520 Pesticides
04/23/2002US6376507 NK-1 receptor antagonists for the treatment of neuronal injury and stroke
04/23/2002US6376503 Alpha 1a adrenergic receptor antagonists
04/23/2002US6376499 Piperazine-amide compound with anticoagulant activity
04/23/2002US6376491 Benzofuran derivatives for treatment or prevention of mycosis in mammals
04/23/2002US6376490 Strong n-methyl-d-asparate receptor antagonists; useful in treating strokes, ischemia, and central nervous system injuries
04/23/2002US6376487 Oxadiazine derivatives
04/23/2002US6376485 Benzoxazoles with PDE-inhibiting activity
04/23/2002US6376484 For prevention and/or treatment of various kinds of inflammatory disease
04/23/2002US6376230 Stereoselective process for producing intermediates of cryptophycins
04/18/2002WO2002030929A1 Novel pleuromutilin derivatives
04/18/2002WO2002030927A1 Novel aminophenyl piperazine or aminophenyl piperidine derivatives inhibiting prenyl transferase proteins and methods for preparing same
04/18/2002WO2002030925A1 Benzopyranyl heterocycle derivatives, process for preparation thereof, and pharmaceutical compositions containing them
04/18/2002WO2002030923A1 Novel aminotriazolone compounds, method for preparing same and pharmaceutical compositions containing same
04/18/2002WO2002030907A1 Pyrazole derivatives for the treatment of viral diseases
04/18/2002WO2002030895A1 SUBSTITUTED INDOLES, PHARMACEUTICAL COMPOSITIONS CONTAINING SUCH INDOLES AND THEIR USE AS PPAR-η BINDING AGENTS
04/18/2002WO2002030890A1 Nitrogenous five-membered ring compounds
04/18/2002WO2002008177A8 N-substituted-1-amino-1,1-dialkylcarboxylic acid derivatives
04/18/2002WO2001087830A3 Substituted thioacetamides
04/18/2002WO2001026656A3 5-membered heterocycle derivatives and use thereof as monoamine oxidase inhibitors
04/18/2002WO2000066106A9 Use of benzodiazepines for treating autoimmune diseases induced by apoptosis
04/18/2002US20020045771 Reacting 7-OH-protected baccatin III with 3-tert-butyl-2,2-dimethyl4-phenyloxazolidine-5-carboxylic acid
04/18/2002US20020045654 Sulfonylbenzene compounds as anti-inflammatory/analgesic agents
04/18/2002US20020045652 Prophylactic or therapeutic drug for renal diseases
04/18/2002US20020045642 Antiinflammatory, -arthritic and -emetic agents; central nervous system disorders; Parkinson's disease; antidepressants; psychological disorders; anxiolytic agents; antagonists of substance P receptors
04/18/2002US20020045641 Multiple heteroatom containing heterocyclic ring compounds substituted with carboxylic acids and isosteres thereof
04/18/2002US20020045629 Sleep, eating and brain disorders, wakefulness promoters; Parkinson's disease, antiischemic agents, stroke, chronic fatigue syndrome; antidepressants; schizophrenia, nervous system disorders; multiple sclerosis, cognition activators
04/18/2002US20020045625 Oxazolidinone chemotherapeutic agents
04/18/2002US20020045620 Readily metabolized by the metabolic drug detoxification systems; metabolized by serum or intracellular hydrolases and esterases; shorthalf-life; noninsulin-dependent diabetes mellitus (NIDDM) (Type II); side effect reduction
04/18/2002US20020045619 4-oxo-1,4-dihydro-3-cinnolinecarboxamides as antiviral agents
04/18/2002US20020045616 Lactam inhibitors of FXa and method
04/18/2002US20020044899 Controlled, super-fine grinding so particles react completely during leaching; extraction of copper from copper sulfide ores and concentrates
04/18/2002CA2427499A1 Substituted indoles, pharmaceutical compositions containing such indoles and their use as ppar-.gamma. binding agents
04/18/2002CA2425416A1 Novel aminophenyl piperazine or aminophenyl piperidine derivatives inhibiting prenyl transferase proteins and methods for preparing same
04/18/2002CA2424802A1 Novel aminotriazolone compounds, method for preparing same and pharmaceutical compositions containing same
04/18/2002CA2423515A1 Pyrazole derivatives for the treatment of viral diseases
04/17/2002EP1197493A1 Benzimidazole compounds
04/17/2002EP1197226A1 Preventives for the recurrence of cerebrovascular failure and agents for ameliorating troubles following cerebrovascular failure and inhibiting progress thereof