Patents
Patents for C07D 413 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms (64,687)
01/2004
01/06/2004US6673803 Quinazoline derivatives and pharmaceutical compositions containing them
01/06/2004US6673800 4,5,-dihydroisoxazolylakylpiperazine derivatives having selective biological activity at dopamine D3 or D4 receptor, and preparation thereof
01/06/2004US6673797 Cyclooxygenase-2 inhibitors; treating inflammatory disease induced by cyclooxygenase-2
01/02/2004EP1375499A1 Process for the production of 2-(5-methyl-4-oxazolyl)ethanol derivatives
01/02/2004EP1375486A1 Nitrogen-containing heteroaryl compounds having hiv integrase inhibitory activity
01/02/2004EP1375482A1 Benzamidine derivative
01/02/2004EP1375474A2 Intermediate for the preparation of carvedilol
01/02/2004EP1373562A2 Method for determining whether a test compound binds to a large rna target
01/02/2004EP1373264A1 3-heterocyclylpropanohydroxamic acid as procollagen c-proteinase inhibitors
01/02/2004EP1373263A1 Heterocyclic compounds for aging-related and diabetic vascular complications
01/02/2004EP1373262A2 Azacycloalkyl substituted acetic acid derivatives for use as mmp inhibitors
01/02/2004EP1373261A2 Cyclopropaheterocycles as non-nucleoside reverse transcriptase inhibitors
01/02/2004EP1373258A1 Ether derivatives useful as inhibitors of pde4 isozymes
01/02/2004EP1373257A1 Inhibitors of c-jun n-terminal kinases (jnk) and other protein kinases
01/02/2004EP1373251A2 Non-imidazole compounds as histamine h3 antagonists
01/02/2004EP1373248A1 Benzimidazol derivatives modulate chemokine receptors
01/02/2004EP1373244A2 Substituted benzopyranones as telomerase inhibitors
01/02/2004EP1373233A1 Derivatives of n-(arylsulfonyl)beta-aminoacids comprising a substituted aminomethyl group, the preparation method thereof and the pharmaceutical compositions containing same
01/02/2004EP1373231A1 3-heterocyclylpropanohydroxamic acid pcp inhibitors
01/02/2004EP1373224A1 New spirotricyclic derivatives and their use as phosphodiesterase-7 inhibitors
01/02/2004EP1373223A1 Cyano-substituted dihydropyrimidine compounds and their use to treat diseases
01/02/2004EP1373221A2 Novel cyano-substituted dihydropyrimidine compounds and their use to treat diseases
01/02/2004EP1373219A1 Thiohydantoins and use thereof for treating diabetes
01/02/2004EP1373210A1 Heterocyclic diamide invertebrate pest control agents
01/02/2004EP1372657A2 A method of treating proliferative diseases using eg5 inhibitors
01/02/2004EP1372653A2 Acylated piperidine derivatives as melanocortin-4 receptor agonists
01/02/2004EP0836595B1 Triazoline and isoxazoline bis-oxime derivatives and their use as pesticides
01/01/2004US20040002539 Enzyme inhibitors; anticoagulants; blood collecting device
01/01/2004US20040002527 Indolylalkylidenehydrazine-carboximidamide derivatives as 5-hydroxytryptamine-6 ligands
01/01/2004US20040002525 Obesity; osteoporosis
01/01/2004US20040002524 Cardiovascular disorders; osteoporosis; central nervous system disorders
01/01/2004US20040002522 Antiinflammatory agents; analgesics
01/01/2004US20040002515 Antihistamines; antiallergens; antiinflammatory agents; autoimmune diseases; rheumatic diseases
01/01/2004US20040002508 Antitumor agents; anticancer agents; sexual disorders; cardiovascular disorders
01/01/2004US20040002496 Compositions useful as inhibitors of protein kinases
01/01/2004US20040002495 Lactam glycogen phosphorylase inhibitors and method of use
01/01/2004US20040002487 Bone disorders; osteoporosis; oral diseases; antiarthritic agents
01/01/2004US20040002424 2-Amino-4-bicyclylamino-6H-1,3,5-triazines, processes for their preparation and their use as herbicides and plant growth regulators
12/2003
12/31/2003WO2004000838A1 Peptidic compounds as cysteine protease inhibitors
12/31/2003WO2004000837A1 Novel benzoxazolinone derivative
12/31/2003WO2004000819A1 New use of pyrimidine - or triazine- 2-carbonitiles for treating diseases associated with cysteine protease activity and novel pyrimidine-2-carbonitile derivatives
12/31/2003WO2004000817A2 Benzimidazole compounds and their use as estrogen agonists/antagonists
12/31/2003WO2004000814A1 8-(biaryl) quinoline pde4 inhibitors
12/31/2003WO2004000811A1 Arylsulfonylhydroxamic acid and amide derivatives and their use as protease inhibitors
12/31/2003WO2004000808A2 N-substituted piperidine derivatives as serotonin receptor agents
12/31/2003WO2004000230A2 Cyclothiocarbamative derivatives as pr modulators and use thereof for treatment of skin disorders
12/31/2003WO2004000214A2 Use of compounds having an amine nucleus in manufacture of a medicament useful for treating factor viia-associated conditions
12/31/2003WO2003072576A3 Oxazolidinone derivatives, processes for their preparation, and pharmaceutical compositions containing them
12/31/2003WO2003059269A3 Acridone inhibitors of impdh enzyme
12/31/2003WO2002060378A3 Substituted aryl compounds as cyclooxygenase-2 selective inhibitors, compositions and methods of use
12/31/2003CA2490646A1 Arylsulfonylhydroxamic acid and amide derivatives and their use as protease inhibitors
12/31/2003CA2490397A1 N-substituted piperidine derivatives as serotonin receptor agents
12/31/2003CA2490043A1 8-(biaryl) quinoline pde4 inhibitors
12/31/2003CA2489815A1 Cyclothiocarbamative derivatives as pr modulators and use thereof for treatment of skin disorders
12/31/2003CA2487266A1 Benzimidazole compounds and their use as estrogen agonists/antagonists
12/31/2003CA2445515A1 Transcription factor modulating compounds and methods of use thereof
12/30/2003US6670482 Process and novel intermediates for preparing isoxazolin-3-ylacyl benzenes
12/30/2003US6670473 Inhibitors of nitric oxide synthase (nos)
12/30/2003US6670447 Amino acid N-carboxyanhydrides with acyl substituents on nitrogen atoms thereof
12/30/2003US6670376 Aryl aniline β2 adrenergic receptor agonists
12/30/2003US6670358 Substituted thioacetamides
12/30/2003US6670307 1,3-oxazoline and 1,3-thiazoline derivatives, their preparation, and their use as pesticides
12/30/2003US6668527 Non-peptidyl inhibitors of VLA-4 dependent cell binding useful in treating inflammatory, autoimmune, and respiratory diseases
12/29/2003CA2433983A1 Aryl- and heteroarylcarbonylpiperazines and their use for the treatment of benign and malignant oncoses
12/25/2003US20030236402 A caspase-3 enzyme inhibitors, 3-(3-alkyl-amino-2-oxo-1,2-dihydro-1-pyrazinyl-alkanoylamino) -4-oxopentanoic acid; treating cardiac or cerebral ischemia or reperfusion injury, diabetes, AIDS
12/25/2003US20030236290 Inhibitors of animal cell motility and growth
12/25/2003US20030236287 Central nervous system disorders; analgesics; antiinflammatory agents; cognition activators; anticancer agents; antidiabetic agents
12/25/2003US20030236262 Dietetics; antidiabetic agents; sexual disorders
12/25/2003US20030236256 N-phenyl-4-(4-pyridyl)-2-pyrimidineamine derivatives
12/25/2003US20030236252 Brain disorders, cardiovascular disorders, strokes, Parkinson's disease
12/25/2003US20030236240 Macrocycles useful in the treatment of alzheimer's disease
12/25/2003US20030236227 Materials and methods for the treatment of diabetes, hyperlipidemia, hypercholesterolemia, and atherosclerosis
12/25/2003US20030236199 Mycrocycles useful in the teatment of Alzheimer's disease
12/25/2003US20030236198 For treatment of infections by drug resistant bacteria
12/24/2003WO2003106628A2 Benzodiazepine inhibitors of mitochondial f>10< atp hydrolase and methods of inhibiting f>10< atp hydrolase
12/24/2003WO2003106610A1 Use of transition metal complexes with nitrogen-containing polydentate ligands as a bleaching catalyst and bleaching agent composition
12/24/2003WO2003106454A1 1h-isoquinoline-oxazolidinone derivaties and their use as antibacterial agents
12/24/2003WO2003106452A2 Antagonists of melanin concentrating hormone receptor
12/24/2003WO2003106451A1 Substituted diaminopyrimidines
12/24/2003WO2003106448A2 Novel herbicides
12/24/2003WO2003106437A1 2-oxazolidinones and their use as inhibitors of animal cell motility and growth
12/24/2003WO2003106431A2 Novel hexahydro-pyridazine-3-carbocylic acid hydrazide or hydrazone derivatives, combinatorial libraries containing same, use thereof as medicines, pharmaceutical compositions containing same and methods for preparing same
12/24/2003WO2003106430A1 Benzimidazole inhibitors of poly(adp-ribosyl) polymerase
12/24/2003WO2003106413A2 Process for the preparation of oxazolidinones and method of use thereof
12/24/2003WO2003105855A1 Mitotic kinesin inhibitors
12/24/2003WO2003105850A1 2-aminoquinolines as melanin concentrating hormone receptor antagonists
12/24/2003WO2003105849A1 Tetrahydroquinolines for modulating the expression of exogenous genes via an ecdysone receptor complex
12/24/2003WO2003105847A1 Ophthalmic compositions for treating ocular hypertension
12/24/2003WO2003105781A2 Ophthalmic compositions for treating ocular hypertension
12/24/2003WO2003105771A2 1-((5-aryl-1,2,4-oxadiazol-3-yl)benzyl)azetidine-3-carboxylates and 1-((5-aryl-1,2,4-oxadiazol-3-yl)benzyl)pyrrolidine-3-carboxylates as edg receptor agonists
12/24/2003WO2003093247A3 Antibacterial agents
12/24/2003WO2003091675A3 Ultrasonic doppler effect speed measurement
12/24/2003WO2003084916A3 Compounds that modulate ppar activity and methods for their preparation
12/24/2003WO2003068760A3 Compounds possessing affinity at 5ht1-type receptors and use thereof in therapy of cns disorders
12/24/2003WO2003061653A9 3-(imidazolyl)-2-aminopropanoic acids for use as tafi-a inhibitors for the treatment of thrombotic diseases
12/24/2003CN1463269A Phenylpiperazine
12/24/2003CN1131864C 吗啉衍生物的化学合成方法 Morpholine derivatives chemical synthesis
12/24/2003CN1131863C 噁二唑啉衍生物及其作为杀虫剂的用途 Oxadiazole derivatives and their use as pesticides
12/24/2003CN1131856C 作为黄体酮受体调节剂的环硫代氨基甲酸酯衍生物 As cyclic thiocarbamate derivative of progesterone receptor modulators
12/24/2003CN1131855C 1-取代-1-氨基甲基-环烷衍生物(=加巴喷丁类似物)、其制备及其在治疗神经病方面的用途 L-amino-1-substituted methyl - naphthenic derivative (= gabapentin analogs), their preparation and their use in the treatment of neuropathy