Patents
Patents for C07D 413 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms (64,687)
03/2004
03/16/2004US6706710 Form of (R)-N-[5-methyl-8-(4-methylpiperazin-1-yl)-1,2,3,4-tetrahydro-2-naphthyl]-4-morpholinobenzamide
03/16/2004US6706708 Cytotoxic agents comprising taxanes and their therapeutic use
03/16/2004US6706707 Phenylethynyl and styryl derivatives of imidazole and fused ring heterocycles
03/11/2004WO2004020441A1 Hetereoaryl nitrile derivatives
03/11/2004WO2004020432A1 Arylamides
03/11/2004WO2004020430A2 Derivatives of dioxane-2-alkyl carbamates, preparation method thereof and application of same in therapeutics
03/11/2004WO2004020412A1 Dihydropyridine derivatives for use as human neutrophil elastase inhibitors
03/11/2004WO2004020409A1 Indoles having anti-diabetic activity
03/11/2004WO2004020408A1 Indoles having anti-diabetic activity
03/11/2004WO2004019943A1 Anabaseine derivatives useful in the treatment of neurodegenerative diseases
03/11/2004WO2004019941A1 Glycinamide derivatives as raf-kinase inhibitors
03/11/2004WO2004019938A1 Oxazolidin-2-one and thiazolidin-2-one derivatives for use as ep4 receptor agonists in the treatment of glaucoma
03/11/2004WO2004019935A1 -3 (sulfonamidoethyl) -indole derivaties for use as glucocorticoid mimetics in the treatment of inflammatory, allergic and proliferative diseases
03/11/2004WO2004019869A2 Indoles having anti-diabetic activity
03/11/2004WO2004019868A2 N-biarylmethyl aminocycloalkanecarboxamide derivatives
03/11/2004WO2004005279A3 Substituted anthranilic amide derivatives and methods of use
03/11/2004WO2003082861A3 Morpholinyl-urea derivatives for use of the treatment of inflammatory diseases
03/11/2004WO2003065789A3 N-biphenylmethyl aminocycloalkanecarboxamide derivatives
03/11/2004WO2003053945A3 Urea derivatives and their use as vanilloid receptor antagonists
03/11/2004US20040049051 Produced by fermenting DSM 6773
03/11/2004US20040049038 N-substituted with a methylene-bridged nonaromatic ring system, e.g., N-(2-(benzyloxy)-5,6,7,8,9,10-hexahydro-6,9-methanobenzo(a)(8)annulen-11-yl)-N'-(2,2,2-trifluoroethyl)-sulfamide; preventing or treating Alzheimer's Disease
03/11/2004US20040049035 Pyrrolecarboxamides and pyrrolethioamides as fungicides
03/11/2004US20040048908 E.g., 3-(5-(3,4-dichlorophenyl)- 4-isoxazolyl)propan-1-ol; prophylaxis or treatment of diabetes, impaired glucose tolerance or diabetic complications
03/11/2004US20040048903 Nicotinamide biaryl derivatives useful as inhibitors of PDE4 isozymes
03/11/2004US20040048901 Increased water solubility and bioabsorption; treatment of CNS disorders such as depression and emesis
03/11/2004US20040048895 Caspase-1 inhibitors and methods for their use
03/11/2004US20040048894 Compounds which mimic the chemical and biological properties of discodermolide
03/11/2004US20040048884 3-aminoalkyluracil derivatives, e.g., 1-(2,6-Difluorobenzyl)-5-(3-methoxyphenyl)-6-methyl-3-(N-methyl-N-(2 -pyridylethyl)-aminoethyl)uracil; contraceptives; treating lupus, sex hormone related cancer, benign prostatic hypertrophy, etc.
03/11/2004US20040048882 4-phenyl-6-alpha-(imidazolyl-, 1,2,4-triazolyl- or pyridyl)-benzyl substituted
03/11/2004US20040048880 Bicyclic heterocyclic compounds, pharmaceutical compositions containing these compounds, their use and process for preparing them
03/11/2004US20040048868 Benzimidazoles
03/11/2004US20040048864 Fungicidal heterocyclic aromatic amides and their compositions, methods of use and preparation
03/11/2004US20040048863 Treating osteoarthritis or rheumatoid arthritis
03/11/2004US20040048858 Chalcone derivatives and their use to treat diseases
03/11/2004US20040048852 Aromatic sulfone hydroxamic acid metalloprotease inhibitor
03/11/2004US20040048848 Novel gamma secretase inhibitors
03/11/2004US20040048843 And aza- and diaza-derivatives thereof; especially treating allergy or nasal congestion
03/11/2004US20040048774 Inhibitors of IMPDH enzyme
03/11/2004CA2496580A1 3-(sulfonamidoethyl)-indole derivaties for use as glucocorticoid mimetics in the treatment of inflammatory, allergic and proliferative diseases
03/11/2004CA2495917A1 Oxazolidin-2-one and thiazolidin-2-one derivatives for use as ep4 receptor agonists in the treatment of glaucoma
03/11/2004CA2495915A1 Indoles having anti-diabetic activity
03/11/2004CA2495914A1 N-biarylmethyl aminocycloalkanecarboxamide derivatives
03/11/2004CA2495248A1 Anabaseine derivatives useful in the treatment of neurodegenerative diseases
03/11/2004CA2494931A1 Hetereoaryl nitrile derivatives
03/10/2004EP1396490A1 3-quinoline-2-(1h)-ylideneindolin-2-one derivatives
03/10/2004EP1396487A1 Phenylpyridine carbonyl piperazine derivative
03/10/2004EP1395606A1 Pyrrolidin-2-one derivatives as inhibitors of factor xa
03/10/2004EP1395583A1 New phenylpiperazines
03/10/2004EP1395582A1 Novel piperidinecarboxamide derivatives, method for preparing same and pharmaceutical compositions containing same
03/10/2004EP1395581A2 Novel benzothienyl or indole derivatives, preparation and use thereof as inhibitors of prenyl transferase proteins
03/10/2004EP1395578A1 Carbazole derivatives and their use for the preparation of pharmaceutical compositions for the treatment of npy related diseases
03/10/2004EP1395568A1 4-aminopyrimidine derivatives
03/10/2004EP1395565A1 Herbicidal substituted benzoylpyrazoles
03/10/2004EP1395561A1 Carbamate and oxamide compounds as inhibitors of cytokine production
03/10/2004EP1395553A1 Pyrrolidine derivatives as factor xa inhibitors
03/10/2004EP1395257A1 Macrocycles useful in the treatment of alzheimer's disease
03/10/2004EP1395251A2 Aminediols as agents for the treatment of alzheimer's disease
03/10/2004CN1481382A Isoindolin-1-one glucokinase activators
03/10/2004CN1481380A Novel benzazepines and related heterocyclic derivatives which are useful as orexin receptor antagonists
03/10/2004CN1481377A Cyclic Beta-amino acid derivatives as inhibitors of matrix metalloproteases and TNF alhpa
03/10/2004CN1481376A Oxybenzamides derivatives as factor xa inhibitors
03/10/2004CN1481369A Substituted phenyluracils compound
03/10/2004CN1481368A Gyrase imhibitors and uses thereof
03/10/2004CN1481361A Piperidine MCH antagonists and their use in treatment of obesity
03/10/2004CN1481245A 2-amino-benzoxazinones for treatment of herpes simplex virus
03/10/2004CN1480451A Photoactive compound used as intermediate for preparing photoactive 2-imidazoline-5-ketone or 2-imdazoline-5-thio-ketone derivative
03/10/2004CN1141306C Novel benzoylpyrazole compounds, prepn. of intermediates and herbicides
03/09/2004US6703503 Pyridazin-3-one derivatives, their use, and intermediates for their production
03/09/2004US6703397 Pyrimidinyl methyl indole derivatives with antibacterial activity
03/09/2004US6703387 Inhibitors of HPV E1 helicase enzyme
03/09/2004US6703368 Peptide-containing α-ketoamide cysteine and serine protease inhibitors
03/04/2004WO2004018463A2 Pyridyl substituted heterocycles useful for treating or preventing hcv infection
03/04/2004WO2004018462A1 Quinazolinone derivatives
03/04/2004WO2004018461A2 Antibacterial benzoic acid derivatives
03/04/2004WO2004018458A1 2-thio-substituted imidazole derivatives and their use in pharmaceutics
03/04/2004WO2004018457A1 Pyrrolidinedione substituted piperidine-phthalazones as pde4 inhibitors
03/04/2004WO2004018455A1 Pyrrole based inhibitors of glycogen synthase kinase 3
03/04/2004WO2004018449A1 Piperidine-derivatives as pde4 inhibitors
03/04/2004WO2004018448A1 Novel thiophene derivatives, preparation method thereof and pharmaceutical compositions containing same
03/04/2004WO2004018441A1 Aryl and heteroaryl morpholine derivatives
03/04/2004WO2004018439A1 Novel antibacterial agents
03/04/2004WO2004018438A2 Microbiocidal (e.g. fungicidal) 1,2,3-triazole derivatives
03/04/2004WO2004018437A1 5-substituted-2-arylpyrazines as modulators of crf receptors
03/04/2004WO2004018435A1 Pyrimidine derivatives as modulators of chemokine receptor activity
03/04/2004WO2004018428A1 Antibacterial benzoic acid derivatives
03/04/2004WO2004018419A2 Benzimidazole quinolinones and uses thereof
03/04/2004WO2004018414A2 Antibacterial agents
03/04/2004WO2004018044A2 N-(3-methoxy-5-methylpyrazin-2-yl)-2-(4-'1,3,4-oxadiazol-2-yl!phenyl)pyridine-3 sulphonamide as an anticancer agent
03/04/2004WO2004017974A1 Piperidine-pyridazones and phthalazones as pde4 inhibitors
03/04/2004WO2004017968A1 Substituted isoxazole derivatives and their use in pharmaceutics
03/04/2004WO2004017963A1 Benzimidazole derivatives
03/04/2004WO2004017961A2 Derivatives of 3-hydroxy-4-(cyclyl-alkylaminoalkyl)-5-phenyl-1h-pyrazole as antagonists of the gonadotropin releasing hormone (gnrh) for use in the treatment of sex hormone related conditions, such as prostatic of uterine cancer
03/04/2004WO2004017922A2 Keto cannabinoids with therapeutic indications
03/04/2004WO2004017911A2 Protease inhibitors
03/04/2004WO2003106448A3 Nicotinoyl derivatives as herbicidal compounds
03/04/2004WO2003082350A3 Radiolabelled quinoline and quinolinone derivatives and their use as metabotropic glutamate receptor ligands
03/04/2004WO2003022844A3 Synthesis of epothilones intermediates thereto and analogues thereof
03/04/2004WO2002098856A3 Piperazine oxyquinoline (naphthaline) platelet adenosine diphosphate receptor antagonists
03/04/2004WO2002070469A3 Selective pde3b inhibitors and use of the same in therapy
03/04/2004US20040044222 New substituted indolinones, preparation thereof and their use as pharmaceutical compositions