Patents
Patents for C07D 413 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms (64,687)
01/2004
01/22/2004WO2004007458A1 Substituted 2-alkylamine nicotinic amide derivatives and use there of
01/22/2004WO2004007457A2 Substituted benzylamine derivatives and methods of use
01/22/2004WO2004007454A1 Piperidinetriol derivatives as inhibitors of glycosylceramidsynthase
01/22/2004WO2004007453A1 Piperidinetriol derivatives as inhibitors of glycosylceramide synthase
01/22/2004WO2004007427A1 N-methyl amino acids
01/22/2004WO2004006926A1 Sulphonylpiperidine derivatives containing an aryl or heteroaryl group for use as matrix metalloproteinase inhibitors
01/22/2004WO2004006924A1 Aryl piperidine derivatives and use thereof to reduce elevated levels of ldl-cholesterol
01/22/2004WO2004006923A1 Aryl piperidine derivatives as inducers of ldl-receptor expression for the treatment of hypercholesterolemia
01/22/2004WO2004006922A1 Aryl piperidine derivatives as inducers of ldl-receptor expression for the treatment of hypercholesterolemia
01/22/2004WO2004006886A2 Injectable depot formulation comprising crystals of iloperidone
01/22/2004WO2004006846A2 Receptor-type kinase modulators and methods of use
01/22/2004WO2003099206A3 Indole compounds useful as impdh inhibitors
01/22/2004WO2003080545A3 Substituted phenylacetic acids
01/22/2004WO2003055447A3 Heterocyclic acridone inhibitors of impdh enzyme
01/22/2004WO2003049690A3 Hiv integrase inhibitors
01/22/2004US20040014977 Benzoxazole compound, process for producing the same, and herbicide
01/22/2004US20040014967 Amide-containing compound having improved solubility and method of improving the solubility of an amide-containing compound
01/22/2004US20040014798 Skin disorders; hormone replacement therapy
01/22/2004US20040014793 Stability in blood
01/22/2004US20040014783 Antiinflammatory agents; autoimmune diseases; rheumatic diseases; anticholesterol agents; cardiovascular disorders
01/22/2004US20040014776 Anticancer agents; cyclin-dependent kinase inhibitor
01/22/2004US20040014767 Central nervous system diosrders; antidepressants, anxiolytic agents, anxiolytic agents
01/22/2004US20040014765 Chk-1 inhibitors
01/22/2004US20040014758 Benzylcycloalkyl amines as modulators of chemokine receptor activity
01/22/2004US20040014741 Dietetics; antidiabetic agents; antiinflammatory agents
01/22/2004US20040013619 Heteroaryl substituted hydroxyphenyltriazine uv-absorbers
01/22/2004DE10231711A1 Bicyclische Heterocyclen, diese Verbindungen enthaltende Arzneimittel, deren Verwendung und Verfahren zu ihrer Herstellung Bicyclic heterocycles, pharmaceutical compositions containing them, their use and process for their preparation
01/22/2004CA2492743A1 Antimicrobial oxazolidinones, process of their preparation, and pharmaceutical compositions containing them
01/22/2004CA2492194A1 Antibacterial cyano-(substituted)-methylenepiperidinophenyl oxazolidinones targeting multiple ribonucleoproteins sites
01/22/2004CA2492164A1 Substituted benzylamine derivatives and methods of use
01/22/2004CA2492100A1 Substituted 2-alkylamine nicotinic amide derivatives and use there of
01/22/2004CA2492086A1 Sulphonylpiperidine derivatives containing an aryl or heteroaryl group for use as matrix metalloproteinase inhibitors
01/22/2004CA2492045A1 Substituted amine derivatives and methods of use
01/22/2004CA2491191A1 Receptor-type kinase modulators and methods of use
01/21/2004EP1382604A1 Quinoline derivative having azolyl group and quinazoline derivative
01/21/2004EP1382603A1 NITROGENOUS FUSED−RING COMPOUND HAVING PYRAZOLYL GROUP AS SUBSTITUENT AND MEDICINAL COMPOSITION THEREOF
01/21/2004EP1382598A1 Novel heterocyclic derivatives
01/21/2004EP1382597A2 Steroid receptor modulator compounds and methods
01/21/2004EP1382336A1 Abc expression promoters
01/21/2004EP1381601A1 Clathrate of azithromycin hydrate with 1,2-propyleneglycol, method for the manufacture thereof and pharmaceutical composition comprising same
01/21/2004EP1381598A1 Novel tyrosine kinase inhibitors
01/21/2004EP1381594A1 Urea compounds useful as anti-inflammatory agents
01/21/2004EP1381592A1 1,4-disubstituted benzo-fused compounds
01/21/2004EP1381590A1 3,4-di-substituted cyclobutene-1,2-diones as cxc-chemokine receptor ligands
01/21/2004EP1381382A2 Methods and compositions for the treatment of diseases of the eye
01/21/2004EP1282601B1 Process and intermediates for the preparation of 1-(9h-carbazol-4-yloxy)-3-[2-(2-methoxy-phenoxy)-ethylamino]-propan-2-ol, carvedilol or acid addition salt thereof
01/21/2004EP0727998B1 Oxazoles for treating cytokine mediated diseases
01/21/2004CN1469876A Alpha-aryl ethanolamines and their use as beta-3 adrenergic receptor agonists
01/21/2004CN1469875A Pyrazole compounds useful as protein kinase inhibitors
01/21/2004CN1469874A Pyrazole compounds useful as protein kinase inhibitors
01/21/2004CN1469873A Piperidine compounds as anti-allergic
01/21/2004CN1469870A A process for the preparation of bis-benzazolyl compounds
01/21/2004CN1469865A Pyrazole derivatives for the treatment of viral diseases
01/21/2004CN1135229C Water soluble azoles as broad-spectrum antifungals
01/21/2004CN1135223C Aryl-substd propanolamine derivate medicine containing them and their use
01/20/2004US6680387 Materials and methods for the treatment of diabetes, hyperlipidemia, hypercholesterolemia, and atherosclerosis
01/20/2004US6680312 Sulfonamide derivatives, their production and use
01/20/2004US6680311 Cryptophycin compounds
01/20/2004CA2303498C Dioxocyclopentyl hydroxamic acids
01/20/2004CA2223936C Novel substituted aryl and cycloalkyl imidazolones; a new class of gaba brain receptor ligands
01/17/2004CA2435399A1 New anthracene derivatives and their use as pharmaceutical preparations
01/15/2004WO2004005283A1 Imidazoles, oxazoles and thiazoles with protein kinase inhibiting activities
01/15/2004WO2004005279A2 Substituted anthranilic amide derivatives and methods of use
01/15/2004WO2004005267A2 Heteroaryl compounds useful in treating inflammatory disorders
01/15/2004WO2004005252A1 Azabicyclo derivatives as muscarinic receptor antagonists
01/15/2004WO2004005229A1 Modulators of the glucocorticoid receptor
01/15/2004WO2004004732A1 Quinazoline derivatives for use in the treatment of cancer
01/15/2004WO2004004730A2 2-aminopyrazine derivatives as inhibitors of cyclin dependent kinases for the treatment of proliferative disorders
01/15/2004WO2004004727A1 3,4-dihydroisoquinolin-1-one derivatives as inducers of apoptosis
01/15/2004WO2004004722A1 1-amido-4-phenyl-4-benzyloxymethyl-piperidine derivatives and related compounds as neurokinin-1(nk-1) antagonists for the treatment of emesis, depression, anxiety and cough
01/15/2004WO2004004720A1 3-`(hetero) arylmethoxy ! pyridines and their analogues as p38 map kinase inhibitors
01/15/2004WO2004004716A1 Naphthalimide synthesis including amonafide synthesis and pharmaceutical preparations thereof
01/15/2004WO2004004665A2 Substituted heterocyclic derivatives useful as antidiabetic and antiobesity agents and method
01/15/2004WO2004004657A2 Hiv integrase inhibitors
01/15/2004WO2004004655A2 Substituted heterocyclic derivatives useful as antidiabetic and antiobesity agents and method
01/15/2004WO2004004629A2 3,6-disubstituted azabicyclo [3.1.0]hexane derivatives useful as muscarinic receptor antagonists
01/15/2004WO2003099798A8 Morpholinylmethylureas ccr-3 receptor antagonist
01/15/2004WO2003091247A3 Piperidinyl-and piperazinyl-sulfonylmethyl hydroxamic acids and their use as protease inhibitors
01/15/2004WO2003066060A3 Use of tyrosine kinase inhibitors for the treatment of inflammatory processes
01/15/2004WO2003047520A3 SUBSTITUTED AMINO METHYL FACTOR Xa INHIBITORS
01/15/2004WO2003045307A3 Pharmaceutical formulations comprising indolinone derivatives
01/15/2004US20040010145 Insecticides, miticides, nematocides
01/15/2004US20040010027 Tumor angiogenesis and metastasis inhibition.
01/15/2004US20040010022 2-aminooxazole derivatives
01/15/2004US20040010019 Aromatic sulfone hydroxamates and their use as protease inhibitors
01/15/2004US20040010014 Novel compounds as opioid receptor modulators
01/15/2004US20040010013 Cannabinoid receptor ligands
01/15/2004US20040010012 Selective inhibitor of the biological activity of human osteoclast cells
01/15/2004US20040010011 Aminoalkoxybenzoyl-benzofuran or benzothiophene derivatives, method for preparing same and compositions containing same
01/15/2004US20040009996 4-(1,2- or 2,1-benzoxazol-5-yl)-2-aminopyrimidines
01/15/2004US20040009995 Treating the symptoms of an acute or chronic disorder mediated by the classical pathway of the complement cascade
01/15/2004US20040009992 Azolylalkylazole derivatives, their preparation, and their use as pesticides
01/15/2004US20040009990 Especially piperidinylcarbonyl- and piperazinylcarbonyl-derivatives of indoles having oxalyl groups
01/15/2004US20040009988 Inhibiting hepatic production of apoprotein B-100 and microsomal triglyceride transfer protein to decrease VLDL and chylomicrons production
01/15/2004US20040009981 Oxazole, thiazole, 1,3,4-oxadiazole and 1,3,4-thiadiazole derivatives of pyrimidines, 1,2,4- and 1,3,5-triazines
01/15/2004US20040009974 Pyrimidylamino- or triazinylamino- substituted pyrazoles or 1,2,3-triazoles
01/15/2004US20040009972 Benzodiazepine inhibitors of mitochondial F1F0 ATP hydrolase and methods of inhibiting F1F0 ATP hydrolase
01/15/2004US20040009969 Diazacycloalkanes containing a 2,5-dioxo-1H-pyrrolyl- or 4-oxo-2-thioxoimidazolidinyl- groups; treating prostate cancer, benign prostate hyperplasia, androgenetic alopecia, hirsutism and androgen-dependent acne.
01/15/2004US20040009968 Indazole compounds useful as protein kinase inhibitors
01/15/2004US20040009967 May contain further anticancer or immunosuppressive agents