Patents
Patents for C07D 413 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms (64,687)
03/2004
03/04/2004US20040044221 Anticancer ganets; drug resistance
03/04/2004US20040044213 Process for making substituted 8-arylquinolinium benzenesulfonate
03/04/2004US20040044212 (Dihydro) Isoquinoline derivatives as phosphodiesterase inhibitors
03/04/2004US20040044203 Anticancer agents
03/04/2004US20040044057 5- substituted tetralones as inhibitors of ras farnesyl trransferase
03/04/2004US20040044053 Antitumor agents; kinase inhibitor
03/04/2004US20040044052 N-Aryl-2-oxazolidinone-5-carboxamides and their derivatives
03/04/2004US20040044049 Compounds for inhibiting insulin secretion and methods related thereto
03/04/2004US20040044041 2-(Biarylalkyl)amino-3-(cyanoalkanoylamino)pyridine derivatives
03/04/2004US20040044037 Sleep disorders; antidepressants; analgesics; central nervous system disorders
03/04/2004US20040044030 Cardiovascular disorders; antiarrhythmia agents
03/04/2004US20040044029 Azabicyclic compounds are central nervous system active agents
03/04/2004US20040044027 Induce immunology response; central nervous system disorders;sleep disorders; gastrointestinal disorders
03/04/2004US20040044000 Cardiovascular disorders; antiarthritic agents; inflammatory bowel disorders; vision defects; respiratory system disorders
03/04/2004US20040043989 Therapy for drug resistant bacteria; topoisomerase inhibitor
03/04/2004US20040043988 Cycloalkyl alkanoic acids as intergrin receptor antagonists
03/04/2004US20040043984 3,4-Dihydroquinolin-2-one, 5,6-fused oxazin-3-one, and 5,6-fused thiazin-3-one derivatives as matrix metalloproteinase inhibitors
03/04/2004US20040043983 Cardiovascular disorders; antiarthritic agents; inflammatory bowel disorders; vision defects; respiratory system disorders
03/04/2004US20040043979 Antiarthritic agents; cardiovascular disorders; imflammatory bowel disorders; skin disordfers; vision disorders
03/04/2004US20040043903 2-Aryl-5-trifluoromethylpyridines
03/04/2004DE10238742A1 New N-(maleimidyl- or thiohydantoinyl-alkyl)-piperazine derivatives, are androgen receptor destabilizers and/or inhibitors useful e.g. for treating prostate carcinoma or hyperplasia
03/04/2004DE10238045A1 2-Thio-substituierte Imidazolderivate und ihre Verwendung in der Pharmazie 2-thio-substituted imidazole derivatives and their use in the pharmaceutical
03/04/2004DE10238002A1 Benzimidazolderivate Benzimidazole derivatives
03/04/2004DE10237883A1 Substituierte Isoxazolderivate und ihre Verwendung in der Pharmazie Substituted isoxazole derivatives and their use in the pharmaceutical
03/04/2004CA2513416A1 Novel antibacterial agents
03/04/2004CA2501849A1 2-thio-substituted imidazole derivatives and their use in treating diseases associated with a disorder of the immune system
03/04/2004CA2497632A1 Novel thiophene derivatives, preparation method thereof and pharmaceutical compositions containing same
03/04/2004CA2496246A1 Pyrrole based inhibitors of glycogen synthase kinase 3
03/04/2004CA2496197A1 5-substituted-2-arylpyrazines as modulators of crf receptors
03/04/2004CA2496097A1 Keto cannabinoids with therapeutic indications
03/04/2004CA2495964A1 Substituted isoxazole derivatives and their use in pharmaceutics
03/04/2004CA2494634A1 Piperidine-pyridazones and phthalazones as pde4 inhibitors
03/04/2004CA2494263A1 Microbiocidal (e.g. fungicidal) 1,2,3-triazole derivatives
03/04/2004CA2494164A1 Pyridyl substituted heterocycles useful for treating or preventing hcv infection
03/03/2004EP1394162A1 Intermediates of azole antifungal agents and processes for the preparation thereof
03/03/2004EP1394159A1 New thiophene derivatives, process for their preparation and pharmaceutical compositions containing them
03/03/2004EP1394154A1 Five-membered heterocyclic alkanoic acid derivative
03/03/2004EP1394152A1 2-iminoimidazole derivatives (1)
03/03/2004EP1394150A1 4-Phenylpyridine derivatives and their use as NK-1 receptor antagonists
03/03/2004EP1394142A1 Carboxylic acid intermediates of antifungal agents and processes for the preparation thereof
03/03/2004EP1392681A1 Triazole compounds useful in treating diseases associated with unwanted cytokine activity
03/03/2004EP1392677A2 Chiral broad-spectrum antibacterial 7-substituted piperidino-quinolone carboxylic acid derivatives, their preparation and compositions
03/03/2004EP1392676A2 Heterocyclic urea derivatives and their use as dopamine d3 receptor ligands
03/03/2004EP1392662A1 Cdk inhibiting pyrimidines, production thereof and their use as medicaments
03/03/2004EP1392656A2 Process for preparing chiral diol sulfones and dihydroxy acid hmg coa reductase inhibitors
03/03/2004EP1392317A2 Substituted 1-benzazepines and derivatives thereof
03/03/2004EP1392309A1 Substituted pyrazinones, pyridines and pyrimidines as corticotropin releasing factor ligands
03/03/2004EP1392306A1 Substituted tetrahydroisoquinolines for use in the treatment of inflammatory diseases
03/03/2004EP1392302A1 5-substituted-2-arylpyridines as crf1 modulators
03/03/2004EP1392299A1 Isoxazolone compounds useful in treating diseases associated with unwanted cytokine activity
03/03/2004EP1392295A1 Carboxylic acid substituted oxazole derivatives for use as ppar-alpha and -gamma activators in the treatment of diabetes
03/03/2004EP1392291A2 Tripeptidyl peptidase inhibitors
03/03/2004EP1307460B1 METHOD FOR THE PRODUCTION OF IMIDAZO-[1,2-c][2,3]-BENZODIAZEPINES AND INTERMEDIATES IN THE PRODUCTION THEREOF
03/03/2004EP1210345B1 Oxazole ppar antagonists
03/03/2004EP1124797B1 N-arylsulfonyl amino acid omega amides
03/03/2004EP1045839B1 Novel amines as pharmaceutical agents
03/03/2004EP1038874B1 Oxime derivatives and agricultural chemicals containing the same
03/03/2004EP0853617B1 Novel 2,3-dioxo-1,2,3,4-tetrahydro-quinoyxalinyl derivatives
03/03/2004EP0738268B1 Trisubstituted phenyl derivatives, processes for their preparation and their use as phosphodiesterase (type iv) inhibitors
03/03/2004CN1479728A Pexoxisome proliferator activated receptor alpha agonists
03/03/2004CN1479727A Piperazinylpyrazine compounds as agonist or antagonist of 5-hydroxytryptamine 5HT-2 receptor
03/03/2004CN1479618A Treatment of sexual dysfunction using boonbesin antagonist
03/03/2004CN1478778A 抗真菌剂及其制备方法和中间体 Antifungal agent and its preparation method and intermediates
03/02/2004US6699996 Production method of isoxazolidinedione compound
03/02/2004US6699995 Process for the preparation of oxazole derivatives
03/02/2004US6699896 Oxazole-aryl-carboxylic acids useful in the treatment of insulin resistance and hyperglycemia
03/02/2004US6699893 Glucocorticoid receptor modulators
03/02/2004US6699887 Administering a therapeutically effective amount of a pyrrazole sulfide or ether compound to treat the human immunodeficiency virus infection
03/02/2004US6699879 Phenyl urea and phenyl thiourea derivatives as orexin receptor antagonists
03/02/2004US6699867 4-(4-Methyl-piperazin-1-ylmethyl)-4,5-dihydrothiazol-2-ylamine
03/02/2004US6699866 For therapy of addiction, anxiety, depression, sexual dysfunction, hypertension, migraine, alzheimer's disease, obesity, emesis, psychosis, analgesia, schizophrenia, parkinson's disease, restless leg syndrome, sleeping disorders
03/02/2004US6699860 Di-substituted aminomethyl-chroman derivative beta-3 adrenoreceptor agonists
03/02/2004US6699856 Pyrazinones, compositions containing such compounds and methods of use
03/02/2004US6699853 Protecting useful plants against the undesirable action of harmful insects, acarids and nematodes,
03/02/2004US6699818 Trifluoromethylpyrrole carboxamides and trifluoromethylpyrrolethioamides as fungicides
03/02/2004US6699651 Base precursors for use in a photothermographic element
02/2004
02/26/2004WO2004016622A1 Derivatives of 4-4'-bipyridyl-2-2'-bisoxazoles and 4-4'-bipyridyl-2-2'-bistiazoles as antineoplasic agents
02/26/2004WO2004016604A2 Azabicyclic compounds are central nervous system active agents
02/26/2004WO2004016587A1 Nitrogen-containing compounds
02/26/2004WO2003101444A8 Diarylurea compounds and derivatives as chk-1 inhibitors for the treatment of cancer
02/26/2004WO2003099211A3 Mitotic kinesin inhibitors
02/26/2004WO2003050261A3 (1-phenyl-2-heteroaryl)ethyl-guanidine compounds as inhibitors of mitochondrial f1f0 atp hydrolase
02/26/2004WO2003047517A3 Novel-n-[4-(1h-imidazol-1-yl)-2-fluorophenyl]-3-(trifluoromethyl)-1-h-pyrazole-5-carboxamides as factor xa
02/26/2004WO2002098424B1 Novel anti-infectives
02/26/2004WO2002041910A8 Methods and compositions for the treatment of diseases of the eye
02/26/2004US20040039033 Administering (1-phenyl-2-heteroaryl)ethyl-guanidine compounds for treating ischemic conditions including myocardial infarction, congestive heart failure, and cardiac arrhythmias
02/26/2004US20040039016 HIV protease inhibitors
02/26/2004US20040038998 Aminopiperidine quinolines and their azaisosteric analogues with antibacterical activity
02/26/2004US20040038991 Imidazolyl-cyclic acetals
02/26/2004US20040038987 Novel cyclic diamine compounds and medicine containing the same
02/26/2004US20040038979 Novel 6-heteroarylphenanthridines
02/26/2004US20040038977 Treating arthritis, pain and cancer
02/26/2004US20040038976 S,N-diarylsulfonamide derivatives; treating inflammatory diseases such as Celiac's disease, Crohn's disease or colitis.
02/26/2004US20040038969 Substituted aminopyrimidines and aminopyridazines; analgesics particularly for migraines, neuropathic pain and associated hyperalgesia and allodynia; antiinflammatory agents; treating asthma, gastrointestinal disorders, etc.
02/26/2004US20040038962 Treatment of nocturnal enuresis, nocturia, polyuria resulting from central diabetes insipidus, urinary incontinence or bleeding disorders such a hemophilia
02/26/2004US20040038941 Compounds for the treatment of inflammatory disorders
02/26/2004CA2495589A1 Azabicyclic compounds are central nervous system active agents
02/25/2004EP1391456A1 2-iminoimidazole derivative (2)
02/25/2004EP1391454A1 Substituted benzamide compounds with antihypertensive activity
02/25/2004EP1391451A1 2-iminopyrrolidine derivates