Patents
Patents for C07D 409 - Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms (52,226)
01/2000
01/20/2000WO2000002870A1 Antiviral macrocyclic compounds
01/20/2000WO2000002865A1 Pharmaceutical agents
01/20/2000WO2000002851A1 Sulfur substituted sulfonylaminocarboxylic acid n-arylamides, their preparation, their use and pharmaceutical preparations comprising them
01/20/2000WO2000002850A2 Sulfonylamino carboxylic acid n-arylamides as guanylate cyclase activators
01/20/2000WO1999059526A3 Protease inhibitors
01/20/2000WO1999058518A3 Biphenyl oxo-acetic acids useful in the treatment of insulin resistance and hyperglycemia
01/20/2000CA2337795A1 Pharmaceutical agents
01/19/2000EP0972767A1 CYCLOALKA[b]PYRIDINE-3-CARBONYLGUANIDINE DERIVATIVES, PROCESS FOR PRODUCING THE SAME, AND DRUGS CONTAINING THE SAME
01/19/2000EP0971916A1 N-(arginyl)benzenesulphonamide derivatives and use thereof as antithrombotic agents
01/19/2000EP0971901A1 Phthalazinones
01/19/2000EP0971894A1 Nicotinamide derivatives
01/19/2000EP0971891A1 Thrombin inhibitors
01/19/2000EP0971744A2 COMBINATION THERAPY EMPLOYING ILEAL BILE ACID TRANSPORT INHIBITING BENZOTHIEPINES AND HMG Co-A REDUCTASE INHIBITORS
01/19/2000CN1242007A Cycloalkyl, lactam lactone and related compounds as 'beta'-amyloid peptide release inhibitors
01/19/2000CN1242000A Farnesyl transferase inhibitors
01/19/2000CN1048484C A process for preparing a composition containing benzoheterocycles
01/18/2000US6015826 Insecticides, aphidicides, and miticides
01/18/2000US6015818 Quinoline derivatives as bradykinin agonists
01/13/2000WO2000001687A1 Benzothiepines having activity as inhibitors of ileal bile acid transport and taurocholate uptake
01/13/2000WO2000001675A1 Novel benzimidazoles as corticotropin release factor antagonists
01/13/2000WO1999050252A3 Barbituric acid derivative and preventive and therapeutic agent for bone and cartilage containing the same
01/13/2000DE19830431A1 Sulfonylamino-carbonsäure-N-arylamide als Guanylatcyclase-Aktivatoren Sulfonylamino-carboxylic acid N-arylamides as guanylate cyclase activators
01/13/2000CA2336315A1 Benzothiepines having activity as inhibitors of ileal bile acid transport and taurocholate uptake
01/13/2000CA2335779A1 Novel benzimidazoles as corticotropin release factor antagonists
01/12/2000EP0970956A1 Pyrazole derivatives
01/12/2000EP0970954A1 3-piperidyl-4-oxoquinazoline derivatives and medicincal compositions containing the same
01/12/2000EP0970073A1 Process for preparing eprosartan
01/12/2000EP0970057A2 Substituted aminosalicyclic acid amides with fungicidal effect and intermediate products for production thereof
01/12/2000EP0970055A2 Hiv protease inhibitors
01/12/2000EP0970046A1 N-hydroxy-2-(alkyl, aryl, or heteroaryl sulfanyl, sulfinyl or sulfonyl)-3-substituted alkyl, aryl or heteroarylamides as matrix metalloproteinase inhibitors
01/12/2000EP0969841A1 Use of carboxylic acid derivatives for treating cancer
01/12/2000EP0862566B1 1-(1,2-disubstituted piperidinyl)-4-substituted piperazine derivatives
01/12/2000CN1241188A Heterocyclylmethyl-substed pyrazol derivs.
01/12/2000CN1241187A Piperazino derivs as neurokinin antagonists
01/12/2000CN1241116A Methyl substed fungicides and arthropodicides
01/12/2000CN1048159C Method for preparing pharmaceutical composition contg. imidazolyl-alkenoic acid
01/11/2000US6013809 Analgesics
01/11/2000US6013666 Oxirane carboxylic acid derivative and its manufacturing method
01/11/2000US6013663 Dithiolan derivatives, their preparation and their therapeutic effect
01/11/2000US6013662 Farnesyl transferase inhibitors, their preparation, the pharmaceutical compositions which contain them and their use in the preparation of medicaments
01/11/2000CA2195027C Hiv protease inhibitors useful for the treatment of aids
01/06/2000WO2000000488A1 Muscarinic antagonists
01/06/2000WO2000000487A1 5-ht1f agonists
01/06/2000WO2000000486A1 Thiophene and furan 2,5-dicarboxamides useful in the treatment of cancer
01/06/2000WO2000000477A1 Non-peptidyl inhibitors of vla-4 dependent cell binding useful in treating inflammatory, autoimmune, and respiratory diseases
01/06/2000WO2000000473A1 Carboxylic and hydroxamic acid compounds inhibiting metalloproteases, method for preparing same and pharmaceutical compositions containing them
01/06/2000WO2000000472A1 5-ht7 receptor antagonists
01/06/2000WO2000000470A1 Amino acid derivatives and drugs containing the same as the active ingredient
01/06/2000WO2000000465A1 Hydrazine derivatives
01/06/2000WO2000000203A1 Azepine derivatives having effects on serotonin related systems
01/06/2000WO2000000198A1 Piperidine derivatives having effects on serotonin related systems
01/06/2000WO2000000197A1 4-benzyl piperidine alkylsulfoxide heterocycles and their use as subtype-selective nmda receptor antagonists
01/06/2000WO2000000196A1 Pyrrolidine and pyrroline derivatives having effects on serotonin related systems
01/06/2000WO1999043661A3 Substituted cycloalkyl-4-oxonicotinic carboxamides; gaba brain receptor ligands
01/06/2000CA2336625A1 Non-peptidyl inhibitors of vla-4 dependent cell binding useful in treating inflammatory, autoimmune, and respiratory diseases
01/06/2000CA2336254A1 5-ht1f agonists
01/06/2000CA2336162A1 Amino acid derivatives and pharmaceutical composition comprising, as active ingredients, them
01/06/2000CA2336117A1 Piperidine derivatives having effects on serotonin related systems
01/06/2000CA2335921A1 Carboxylic and hydroxamic acid compounds inhibiting metalloproteases, method for preparing same and pharmaceutical compositions containing them
01/06/2000CA2335310A1 Azepine derivatives having effects on serotonin related systems
01/06/2000CA2335245A1 Hydrazine derivatives
01/06/2000CA2334897A1 Pyrrolidine and pyrroline derivatives having effects on serotonin related systems
01/06/2000CA2330110A1 1,3-benzodiazepin-2-ones and 1,3-benzoxazepin-2-ones useful as hiv reverse transcriptase inhibitors
01/06/2000CA2327888A1 4-benzyl piperidine alkylsulfoxide heterocycles and their use as subtype-selective nmda receptor antagonists
01/05/2000EP0969071A1 Alkenyl compound having a negative delta epsilon value, liquid crystal composition and liquid crystal display device
01/05/2000EP0968250A1 Soluble chromophores having improved solubilising groups
01/05/2000EP0968208A1 Quinoline and quinazoline compounds useful in therapy, particularly in the treatment of benign prostatic hyperplasia
01/05/2000EP0968206A1 N-heterocyclic derivatives as nos inhibitors
01/05/2000EP0968198A1 HETEROCYCLIC COMPOUNDS AND THEIR USE FOR INHIBITING $g(b)-AMYLOID PEPTIDE
01/05/2000EP0968190A1 Substituted isoquinoline derivatives and their use as anticonvulsants
01/05/2000EP0664792B1 Fibrinogen receptor antagonists
01/05/2000CN1240445A Preparation of [1S-[1a,2b,3b,4a(S*)]]-4-[7-[[1-(3-chloro-2-thienyl)methyl] propyl] amino]-3H-imidazo [4,5-b] pyridin-3-y1]-n-ethyl-2
01/05/2000CN1240444A Piperidine derivatives
01/05/2000CN1240440A Substituted benzothiopyranes salts and their use as herbicides
01/05/2000CN1240437A Preparation and use of ortho-sulfonamido heteroaryl hydroxamic acids as matrix metalloproteinase and tace inhibitors
01/05/2000CN1240429A The preparation and use of ortho-sulfonamido aryl hydroxamic acids as matrix metalloproteinase and tace inhibitors
01/05/2000CN1240426A Novel tetrahydrobenzindolone derivatives
01/05/2000CN1240354A Use of condensated (hetaryl-substituted) 1-benzal-3-pyarzol derivates for treating special diseases of the cardiovascular and the central nerous systems
01/04/2000US6011059 Acyl guanidine sodium/proton exchange inhibitors and method
01/04/2000US6011056 C9 taxane derivatives and pharmaceutical compositions containing them
01/04/2000US6011055 Administering indomethacin, naproxen, ibuprofen, tenidap and imiquod in a pharmacologically acceptable carrier, excipient or diluent.
01/04/2000US6011039 Aminopyridine derivatives
01/04/2000US6011029 Benzodiazepine compounds
01/04/2000US6011028 Cyclic amidino agents useful as nitric oxide synthase inhibitors
12/1999
12/29/1999WO1999067252A2 Epothilone derivatives and their synthesis and use
12/29/1999WO1999067221A1 Compounds for inhibiting beta-amyloid peptide release and/or its synthesis
12/29/1999WO1999067220A1 Compounds for inhibiting beta-amyloid peptide release and/or its synthesis
12/29/1999WO1999067219A1 Compounds for inhibiting beta-amyloid peptide release and/or its synthesis
12/29/1999WO1999067215A1 Amidino and guanidino azetidinone tryptase inhibitors
12/29/1999WO1999066934A1 CYCLIC AMINO ACID COMPOUNDS, PHARMACEUTICAL COMPOSITIONS COMPRISING SAME, AND METHODS FOR INHIBITING β-AMYLOID PEPTIDE RELEASE AND/OR ITS SYNTHESIS BY USE OF SUCH COMPOUNDS
12/29/1999EP0967207A1 Nitrone derivatives, process for their preparation and pharmaceutical compositions containing them
12/29/1999EP0966454A1 Disubstituted bicyclic heterocycles, their production and use as medicaments
12/29/1999EP0966447A1 Small molecules useful in the treatment of inflammatory disease
12/29/1999EP0966446A1 Bicyclic inhibitors of protein farnesyl transferase
12/29/1999EP0966444A1 Process for preparing pyrazole derivatives
12/29/1999EP0966443A1 Heteroaryl-hexanoic acid amide derivatives, their preparation and their use as selective inhibitors of mip-1-alpha binding to its ccr1 receptor
12/29/1999EP0966430A1 Anti-inflammatory compounds
12/29/1999EP0966282A1 Use of angiotensin ii antagonists to treat symptomatic heart failure
12/29/1999EP0612314B1 2-pyrazinylethylamine derivatives and their use as pharmaceuticals
12/29/1999CN1239960A Thienylsulfonylamino (THIO) carbonyl compounds