Patents
Patents for C07D 409 - Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms (52,226)
10/1999
10/21/1999WO1999052493A2 Compounds that inhibit the binding of integrins to their receptors
10/21/1999WO1999040061A3 Novel dihydroxyhexanoic acid derivatives
10/21/1999DE19817265A1 Treating hepatitis B using new or known dihydropyrimidine derivative antiviral agents
10/21/1999CA2328878A1 Thienylazolylalcoxyethanamines, their preparation and their application as medicaments
10/21/1999CA2328211A1 Substituted pyrrolidine hydroxamate metalloprotease inhibitors
10/21/1999CA2327793A1 Thienylalkylamino-1,3,5-triazines
10/21/1999CA2327695A1 Amine compounds, their production and their use as somatostatin receptor antagonists or agonists
10/21/1999CA2327282A1 Treatment of parasitic diseases by inhibition of cysteine proteases of the papain superfamily
10/21/1999CA2326665A1 Heterocyclic glycyl beta-alanine derivatives as vitronectin antagonists
10/21/1999CA2325559A1 Non-endogenous, constitutively activated human serotonin receptors and small molecule modulators thereof
10/20/1999EP0950657A2 Substituted carbazoles, process for their preparation and their use as sPLA2 inhibitors
10/20/1999EP0950656A1 Sulfonated amino acid derivatives and metalloproteinase inhibitors containing the same
10/20/1999EP0950405A1 Remedies for renal diseases and organ-preserving agents
10/20/1999EP0950046A1 3,4-disubstituted azetidin-2-one derivatives useful as cysteine proteinase regulators
10/20/1999CN1232462A Muscarinic antagonists
10/20/1999CN1232457A 1,4-heterocyclic metalloprotease inhibitors
10/20/1999CN1232453A Ether muscarinic antagonists
10/20/1999CN1232451A Substd. cyclic amine metalloprotease inhibitors
10/20/1999CN1232450A 2- and 2,5-substd. phenylketoenols
10/20/1999CN1045774C Substd. arylthioalkylthiopyridines, their preparing method and pharmaceutical use
10/20/1999CN1045772C Polyazacycloalkanes as dichelants
10/20/1999CN1045770C Method for preparation of 1-biphenylmethyl imidazole derivs.
10/20/1999CN1045768C Angiotension II antagonists compounds, preparing method and use thereof
10/19/1999US5969151 Pyrazole compounds
10/19/1999US5969141 Intermediates for 7-amino-1-cyclopropyl-6,8-dihalogeno-1,4-dihydro-4-oxo-3-quinolinecarbox ylic acid antibacterial agents
10/19/1999US5969139 Inhibitors of herpes simplex virus thymidine kinase
10/19/1999US5968977 Ketonitrile derivatives and antibacterial agent and drugs containing the same
10/19/1999US5968971 Endothelin receptor antagonists
10/19/1999US5968969 Stable, long acting salts of carboxamides for the treatment of joint disease
10/19/1999US5968956 Substituted piperidine derivative and medicine comprising the same
10/19/1999US5968954 Exhibit selective binding affinity for 5-hydroxytryptamine receptors
10/19/1999US5968948 Annelated dihydropyridines and the use thereof for preparing pharmaceutical preparations
10/19/1999US5968935 Agent for potentiating nerve growth factor activity containing 1,2-ethanediol derivative or salt thereof
10/19/1999CA2197298C Novel pyrimidine derivatives and processes for the preparation thereof
10/17/1999CA2269262A1 Substituted tricyclics
10/14/1999WO1999051593A1 4-thionaphthyl-1h-imidazoles with alpha-2-adrenergic activity
10/14/1999WO1999051589A1 Substituted piperidines, method for their preparation and their use as pesticides and fungicides
10/14/1999WO1999051587A1 Fused thiophene derivatives and drugs containing the same as the active ingredient
10/14/1999WO1999051580A1 Pyrazole inhibitors of cytokine production
10/14/1999WO1999051578A1 Biocidal benzylbiphenyl derivatives
10/14/1999WO1999051574A1 Indole derivatives
10/14/1999WO1999051225A1 Antidiabetic agents
10/14/1999WO1999045011A8 Glycine transport inhibitors
10/14/1999WO1999032447A3 2,4,6-trisubstituted pyridines with estrogenic activity and methods for the solid phase synthesis thereof
10/14/1999DE19909541A1 New pyrimidine derivatives useful as herbicides, especially for selective weed control
10/14/1999DE19816055A1 Thienylalkylamino-1,3,5-triazine Thienylalkylamino-1,3,5-triazines
10/14/1999CA2328607A1 Antidiabetic agents
10/14/1999CA2327397A1 Indole derivatives
10/14/1999CA2327185A1 Pyrazole inhibitors of cytokine production
10/14/1999CA2326159A1 Biocidal benzylbiphenyl derivatives
10/13/1999EP0948498A1 Sulfonamide compounds having 5-ht receptor activity
10/13/1999EP0948497A2 Substituted pyrimidine compounds and their use
10/13/1999EP0948496A2 Substituted pyrimidinone and pyridone compounds and methods of use
10/13/1999EP0948495A1 Aryl and heteroaryl substituted fused pyrrole antiinflammatory agents
10/13/1999EP0948489A1 Piperazine compounds as inhibitors of mmp or tnf
10/13/1999EP0948483A1 Farnesyl transferase inhibitors
10/13/1999EP0948478A1 ARYL OR HETEROARYL SUBSTITUTED 3,4-DIHYDROANTHRACENE AND ARYL OR HETEROARYL SUBSTITUTED BENZO 1,2-g]-CHROM-3-ENE, BENZO 1,2-g]-THIOCHROM-3-ENE AND BENZO 1,2-g]-1,2-DIHYDROQUINOLINE DERIVATIVES HAVING RETINOID ANTAGONIST OR RETINOID INVERSE AGONIST TYPE BIOLOGICAL ACTIVITY
10/13/1999EP0948327A1 Antidiabetic agents
10/13/1999EP0948257A1 Triaryl substituted imidazoles, compositions containing such compounds and methods of use
10/13/1999EP0579618B1 Pyridine- and imidazole-derived agents for cardiovascular diseases
10/13/1999CN1231664A Sulfonamicles and derivatives thereof that moulate the activity of endothelin
10/13/1999CN1231287A Benzosulfone derivatives
10/13/1999CN1045597C Alkylenediamine derivatives having heterocyclic group and medicinal composition thereof
10/13/1999CN1045595C Process for the preparation of the intermediates used in the synthesis of 3-aminopiperidine derivatives
10/12/1999US5965739 Oxazolidine protected taxol analogs of given formula, and methods of synthesis from an oxazolidine free acid and a baccatin compound in the presence of a dehydrating agent; useful intermediates to make various taxol analogues
10/12/1999US5965730 Selective phosphodiestearase iv inhibitor having bronchodialation and anti-inflammatory activity; prophylaxis and treatment of asthma
10/12/1999US5965609 An antitumor agent, antimalaria agent, bactericide treating gram-negative bacteria and active drug treating stroke, traumatic brain injury, chronic neurodegenerative disease, alzheimer's disease or amyotropic lateral schlerosis
10/12/1999US5965592 Acyl compounds
10/12/1999US5965575 N-aryl piperidine compounds as 5HT1B antagonists
10/12/1999US5965574 Heteroaryl amines as novel acetylcholinesterase inhibitors
10/12/1999US5965560 Substituted piperazines and piperidines as central nervous system agents
10/12/1999US5965559 Aminoheterocyclic derivatives as antithrombotic or anticoagulant
10/12/1999US5965556 Keto-acid amide derivatives, pharmaceutical compositions containing them and methods for inhibiting the activity of serine protease or thiol protease by administering the derivative to a mammal; alzheimer's disease
10/12/1999US5965492 Triketone derivatives
10/07/1999WO1999050266A1 Benzoheterocyclic distamycin derivatives, process for preparing them, and their use as antitumor agents
10/07/1999WO1999050263A1 Quinolones as serine protease inhibitors
10/07/1999WO1999050253A1 4,4-disubstituted-3,4-dihydro-2(1h)-quinazolinthione derivatives, their preparation and their use as hiv reverse transcriptase inhibitors
10/07/1999WO1999050252A2 Barbituric acid derivative and preventive and therapeutic agent for bone and cartilage containing the same
10/07/1999WO1999050250A1 Hiv inhibiting pyrimidine derivatives
10/07/1999WO1999050243A1 The use of derivatives of 2-oxopyrrole as crop protection agents and novel 2-oxopyrroles
10/07/1999WO1999049856A2 Antagonists for treatment of cd11/cd18 adhesion receptor mediated disorders
10/07/1999DE19815026A1 Substituierte Piperidine, Verfahren zu ihrer Herstellung und ihre Verwendung als Schädlingsbekämpfungsmittel und Fungizide Substituted piperidines, process for their preparation and their use as pesticides and fungicides
10/07/1999DE19812058C1 New 2-heterocyclyl-1,4-phenylenediamine derivatives
10/07/1999CA2325986A1 Antagonists for treatment of cd11/cd18 adhesion receptor mediated disorders
10/07/1999CA2325904A1 The use of derivatives of 2-oxopyrrole as crop protection agents and novel 2-oxopyrroles
10/07/1999CA2324584A1 Barbituric acid derivative and preventive and therapeutic agent for bone and cartilage containing the same
10/07/1999CA2322203A1 4,4-disubstituted-3,4-dihydro-2(1h)-quinazolinthione derivatives, their preparation and their use as hiv reverse transcriptase inhibitors
10/07/1999CA2312953A1 Quinolones as serine protease inhibitors
10/06/1999EP0947507A1 Novel tetrahydrobenzindolone derivatives
10/06/1999EP0946587A2 New amide compounds
10/06/1999EP0946552A1 Sulfonamides and derivatives thereof that modulate the activity of endothelin
10/06/1999EP0946550A1 PREPARATION OF 1S- 1a,2b,3b,4a(S*)]]-4- 7- 1-(3-CHLORO-2-THIENYL) METHYL]PROPYL]AMINO]-3H-IMIDAZO 4,5-b]PYRIDIN-3-yl]-N-ETHYL-2,3-DIHYDROXYCYCLOPENTANECARBOXAMIDE
10/06/1999EP0946546A1 Pyridin-2-yl-methylamine derivatives, method of preparing and application as medicine
10/06/1999EP0946540A1 Substituted benzothiopyranes salts and their use as herbicides
10/06/1999EP0946539A1 Sulphonamide derivatives, process for their preparation, and their use as medicaments
10/06/1999EP0946538A1 Indane or dihydroindole derivatives
10/06/1999EP0946528A2 OXYGEN OR SULFUR CONTAINING 5-MEMBERED HETEROAROMATICS AS FACTOR Xa INHIBITORS
10/06/1999EP0946518A1 Modulators of proteins with phosphotyrosine recognition units
10/06/1999EP0946517A1 N-(imidazolylbutyl) benzenesulphonamide derivatives, their preparation and therapeutic application
10/06/1999EP0946511A1 Novel compounds with analgesic effect