Patents for C07D 409 - Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms (52,226) |
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10/21/1999 | WO1999052493A2 Compounds that inhibit the binding of integrins to their receptors |
10/21/1999 | WO1999040061A3 Novel dihydroxyhexanoic acid derivatives |
10/21/1999 | DE19817265A1 Treating hepatitis B using new or known dihydropyrimidine derivative antiviral agents |
10/21/1999 | CA2328878A1 Thienylazolylalcoxyethanamines, their preparation and their application as medicaments |
10/21/1999 | CA2328211A1 Substituted pyrrolidine hydroxamate metalloprotease inhibitors |
10/21/1999 | CA2327793A1 Thienylalkylamino-1,3,5-triazines |
10/21/1999 | CA2327695A1 Amine compounds, their production and their use as somatostatin receptor antagonists or agonists |
10/21/1999 | CA2327282A1 Treatment of parasitic diseases by inhibition of cysteine proteases of the papain superfamily |
10/21/1999 | CA2326665A1 Heterocyclic glycyl beta-alanine derivatives as vitronectin antagonists |
10/21/1999 | CA2325559A1 Non-endogenous, constitutively activated human serotonin receptors and small molecule modulators thereof |
10/20/1999 | EP0950657A2 Substituted carbazoles, process for their preparation and their use as sPLA2 inhibitors |
10/20/1999 | EP0950656A1 Sulfonated amino acid derivatives and metalloproteinase inhibitors containing the same |
10/20/1999 | EP0950405A1 Remedies for renal diseases and organ-preserving agents |
10/20/1999 | EP0950046A1 3,4-disubstituted azetidin-2-one derivatives useful as cysteine proteinase regulators |
10/20/1999 | CN1232462A Muscarinic antagonists |
10/20/1999 | CN1232457A 1,4-heterocyclic metalloprotease inhibitors |
10/20/1999 | CN1232453A Ether muscarinic antagonists |
10/20/1999 | CN1232451A Substd. cyclic amine metalloprotease inhibitors |
10/20/1999 | CN1232450A 2- and 2,5-substd. phenylketoenols |
10/20/1999 | CN1045774C Substd. arylthioalkylthiopyridines, their preparing method and pharmaceutical use |
10/20/1999 | CN1045772C Polyazacycloalkanes as dichelants |
10/20/1999 | CN1045770C Method for preparation of 1-biphenylmethyl imidazole derivs. |
10/20/1999 | CN1045768C Angiotension II antagonists compounds, preparing method and use thereof |
10/19/1999 | US5969151 Pyrazole compounds |
10/19/1999 | US5969141 Intermediates for 7-amino-1-cyclopropyl-6,8-dihalogeno-1,4-dihydro-4-oxo-3-quinolinecarbox ylic acid antibacterial agents |
10/19/1999 | US5969139 Inhibitors of herpes simplex virus thymidine kinase |
10/19/1999 | US5968977 Ketonitrile derivatives and antibacterial agent and drugs containing the same |
10/19/1999 | US5968971 Endothelin receptor antagonists |
10/19/1999 | US5968969 Stable, long acting salts of carboxamides for the treatment of joint disease |
10/19/1999 | US5968956 Substituted piperidine derivative and medicine comprising the same |
10/19/1999 | US5968954 Exhibit selective binding affinity for 5-hydroxytryptamine receptors |
10/19/1999 | US5968948 Annelated dihydropyridines and the use thereof for preparing pharmaceutical preparations |
10/19/1999 | US5968935 Agent for potentiating nerve growth factor activity containing 1,2-ethanediol derivative or salt thereof |
10/19/1999 | CA2197298C Novel pyrimidine derivatives and processes for the preparation thereof |
10/17/1999 | CA2269262A1 Substituted tricyclics |
10/14/1999 | WO1999051593A1 4-thionaphthyl-1h-imidazoles with alpha-2-adrenergic activity |
10/14/1999 | WO1999051589A1 Substituted piperidines, method for their preparation and their use as pesticides and fungicides |
10/14/1999 | WO1999051587A1 Fused thiophene derivatives and drugs containing the same as the active ingredient |
10/14/1999 | WO1999051580A1 Pyrazole inhibitors of cytokine production |
10/14/1999 | WO1999051578A1 Biocidal benzylbiphenyl derivatives |
10/14/1999 | WO1999051574A1 Indole derivatives |
10/14/1999 | WO1999051225A1 Antidiabetic agents |
10/14/1999 | WO1999045011A8 Glycine transport inhibitors |
10/14/1999 | WO1999032447A3 2,4,6-trisubstituted pyridines with estrogenic activity and methods for the solid phase synthesis thereof |
10/14/1999 | DE19909541A1 New pyrimidine derivatives useful as herbicides, especially for selective weed control |
10/14/1999 | DE19816055A1 Thienylalkylamino-1,3,5-triazine Thienylalkylamino-1,3,5-triazines |
10/14/1999 | CA2328607A1 Antidiabetic agents |
10/14/1999 | CA2327397A1 Indole derivatives |
10/14/1999 | CA2327185A1 Pyrazole inhibitors of cytokine production |
10/14/1999 | CA2326159A1 Biocidal benzylbiphenyl derivatives |
10/13/1999 | EP0948498A1 Sulfonamide compounds having 5-ht receptor activity |
10/13/1999 | EP0948497A2 Substituted pyrimidine compounds and their use |
10/13/1999 | EP0948496A2 Substituted pyrimidinone and pyridone compounds and methods of use |
10/13/1999 | EP0948495A1 Aryl and heteroaryl substituted fused pyrrole antiinflammatory agents |
10/13/1999 | EP0948489A1 Piperazine compounds as inhibitors of mmp or tnf |
10/13/1999 | EP0948483A1 Farnesyl transferase inhibitors |
10/13/1999 | EP0948478A1 ARYL OR HETEROARYL SUBSTITUTED 3,4-DIHYDROANTHRACENE AND ARYL OR HETEROARYL SUBSTITUTED BENZO 1,2-g]-CHROM-3-ENE, BENZO 1,2-g]-THIOCHROM-3-ENE AND BENZO 1,2-g]-1,2-DIHYDROQUINOLINE DERIVATIVES HAVING RETINOID ANTAGONIST OR RETINOID INVERSE AGONIST TYPE BIOLOGICAL ACTIVITY |
10/13/1999 | EP0948327A1 Antidiabetic agents |
10/13/1999 | EP0948257A1 Triaryl substituted imidazoles, compositions containing such compounds and methods of use |
10/13/1999 | EP0579618B1 Pyridine- and imidazole-derived agents for cardiovascular diseases |
10/13/1999 | CN1231664A Sulfonamicles and derivatives thereof that moulate the activity of endothelin |
10/13/1999 | CN1231287A Benzosulfone derivatives |
10/13/1999 | CN1045597C Alkylenediamine derivatives having heterocyclic group and medicinal composition thereof |
10/13/1999 | CN1045595C Process for the preparation of the intermediates used in the synthesis of 3-aminopiperidine derivatives |
10/12/1999 | US5965739 Oxazolidine protected taxol analogs of given formula, and methods of synthesis from an oxazolidine free acid and a baccatin compound in the presence of a dehydrating agent; useful intermediates to make various taxol analogues |
10/12/1999 | US5965730 Selective phosphodiestearase iv inhibitor having bronchodialation and anti-inflammatory activity; prophylaxis and treatment of asthma |
10/12/1999 | US5965609 An antitumor agent, antimalaria agent, bactericide treating gram-negative bacteria and active drug treating stroke, traumatic brain injury, chronic neurodegenerative disease, alzheimer's disease or amyotropic lateral schlerosis |
10/12/1999 | US5965592 Acyl compounds |
10/12/1999 | US5965575 N-aryl piperidine compounds as 5HT1B antagonists |
10/12/1999 | US5965574 Heteroaryl amines as novel acetylcholinesterase inhibitors |
10/12/1999 | US5965560 Substituted piperazines and piperidines as central nervous system agents |
10/12/1999 | US5965559 Aminoheterocyclic derivatives as antithrombotic or anticoagulant |
10/12/1999 | US5965556 Keto-acid amide derivatives, pharmaceutical compositions containing them and methods for inhibiting the activity of serine protease or thiol protease by administering the derivative to a mammal; alzheimer's disease |
10/12/1999 | US5965492 Triketone derivatives |
10/07/1999 | WO1999050266A1 Benzoheterocyclic distamycin derivatives, process for preparing them, and their use as antitumor agents |
10/07/1999 | WO1999050263A1 Quinolones as serine protease inhibitors |
10/07/1999 | WO1999050253A1 4,4-disubstituted-3,4-dihydro-2(1h)-quinazolinthione derivatives, their preparation and their use as hiv reverse transcriptase inhibitors |
10/07/1999 | WO1999050252A2 Barbituric acid derivative and preventive and therapeutic agent for bone and cartilage containing the same |
10/07/1999 | WO1999050250A1 Hiv inhibiting pyrimidine derivatives |
10/07/1999 | WO1999050243A1 The use of derivatives of 2-oxopyrrole as crop protection agents and novel 2-oxopyrroles |
10/07/1999 | WO1999049856A2 Antagonists for treatment of cd11/cd18 adhesion receptor mediated disorders |
10/07/1999 | DE19815026A1 Substituierte Piperidine, Verfahren zu ihrer Herstellung und ihre Verwendung als Schädlingsbekämpfungsmittel und Fungizide Substituted piperidines, process for their preparation and their use as pesticides and fungicides |
10/07/1999 | DE19812058C1 New 2-heterocyclyl-1,4-phenylenediamine derivatives |
10/07/1999 | CA2325986A1 Antagonists for treatment of cd11/cd18 adhesion receptor mediated disorders |
10/07/1999 | CA2325904A1 The use of derivatives of 2-oxopyrrole as crop protection agents and novel 2-oxopyrroles |
10/07/1999 | CA2324584A1 Barbituric acid derivative and preventive and therapeutic agent for bone and cartilage containing the same |
10/07/1999 | CA2322203A1 4,4-disubstituted-3,4-dihydro-2(1h)-quinazolinthione derivatives, their preparation and their use as hiv reverse transcriptase inhibitors |
10/07/1999 | CA2312953A1 Quinolones as serine protease inhibitors |
10/06/1999 | EP0947507A1 Novel tetrahydrobenzindolone derivatives |
10/06/1999 | EP0946587A2 New amide compounds |
10/06/1999 | EP0946552A1 Sulfonamides and derivatives thereof that modulate the activity of endothelin |
10/06/1999 | EP0946550A1 PREPARATION OF 1S- 1a,2b,3b,4a(S*)]]-4- 7- 1-(3-CHLORO-2-THIENYL) METHYL]PROPYL]AMINO]-3H-IMIDAZO 4,5-b]PYRIDIN-3-yl]-N-ETHYL-2,3-DIHYDROXYCYCLOPENTANECARBOXAMIDE |
10/06/1999 | EP0946546A1 Pyridin-2-yl-methylamine derivatives, method of preparing and application as medicine |
10/06/1999 | EP0946540A1 Substituted benzothiopyranes salts and their use as herbicides |
10/06/1999 | EP0946539A1 Sulphonamide derivatives, process for their preparation, and their use as medicaments |
10/06/1999 | EP0946538A1 Indane or dihydroindole derivatives |
10/06/1999 | EP0946528A2 OXYGEN OR SULFUR CONTAINING 5-MEMBERED HETEROAROMATICS AS FACTOR Xa INHIBITORS |
10/06/1999 | EP0946518A1 Modulators of proteins with phosphotyrosine recognition units |
10/06/1999 | EP0946517A1 N-(imidazolylbutyl) benzenesulphonamide derivatives, their preparation and therapeutic application |
10/06/1999 | EP0946511A1 Novel compounds with analgesic effect |