Patents
Patents for C07D 409 - Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms (52,226)
07/1999
07/08/1999CA2316382A1 N-phenylamide and n-pyridylamide derivatives, method of preparing them and pharmaceutical compositions containing them
07/08/1999CA2316352A1 Acyl guanidine sodium/proton exchange inhibitors and method
07/08/1999CA2316341A1 4-[aryl(piperidin-4-yl)] aminobenzamides which bind to the delta-opioid receptor
07/08/1999CA2315144A1 Novel farnesyl transferase inhibitors, preparation, pharmaceutical compositions containing them and use for preparing medicines
07/07/1999EP0927192A1 Modified aminoacids, pharmaceuticals containing these compounds and method for their production
07/07/1999EP0927179A1 Substituted benzocycloheptapyridine derivatives useful for inhibition of farnesyl protein transferase
07/07/1999EP0927170A1 Piperazino derivatives as neurokinin antagonists
07/07/1999EP0927168A1 1,3-diheterocyclic metalloprotease inhibitors
07/07/1999EP0927166A1 Amides as npy5 receptor antagonists
07/07/1999EP0927164A1 8-hydroxy-7-substituted quinolines as anti-viral agents
07/07/1999EP0927161A1 Substituted cyclic amine metalloprotease inhibitors
07/07/1999CN1221743A Substituted heterocyclic benzoeycloalkenes and the use thereof as substances having analgesic effect
07/06/1999US5919940 Tert-leucine-thiazol-2-ylamide
07/06/1999US5919809 3-substituted-2-oxindole derivatives
07/06/1999US5919801 N-substituted piperidines as PDE4 inhibitors
07/06/1999US5919795 Atherosclerosis therapy
07/06/1999US5919786 N,N-disubstituted amic acid derivatives
07/06/1999US5919778 Alzheimer*s disease
07/01/1999WO1999032483A1 New pharmaceutically active compounds
07/01/1999WO1999032482A1 Hypoglycemic imidazoline compounds
07/01/1999WO1999032477A1 Ortho-anthranilamide derivatives as anti-coagulants
07/01/1999WO1999032468A1 Anilide derivative, production and use thereof
07/01/1999WO1999032463A1 INHIBITION OF p38 KINASE USING SYMMETRICAL AND UNSYMMETRICAL DIPHENYL UREAS
07/01/1999WO1999032455A1 Inhibition of raf kinase using aryl and heteroaryl substituted heterocyclic ureas
07/01/1999WO1999032452A1 Carboxyl acid substituted heterocycles as metalloproteinase inhibitors
07/01/1999WO1999032451A1 Azepine or larger medium ring derivatives and their use as pharmaceuticals
07/01/1999WO1999032450A1 4-hydroxyquinoline-3-carboxamides and hydrazides as antiviral agents
07/01/1999WO1999032448A1 Substituted pyridine and pyridazine compounds and their pharmaceutical use
07/01/1999WO1999032447A2 2,4,6-trisubstituted pyridines with estrogenic activity and methods for the solid phase synthesis thereof
07/01/1999WO1999032436A1 Inhibition of raf kinase using symmetrical and unsymmetrical substituted diphenyl ureas
07/01/1999WO1999032112A1 Method for treating diabetes
07/01/1999WO1999032111A1 INHIBITION OF p38 KINASE ACTIVITY USING SUBSTITUTED HETEROCYCLIC UREAS
07/01/1999WO1999032106A1 Inhibition of raf kinase using substituted heterocyclic ureas
07/01/1999WO1999019324A3 Antipsychotic substituted piperidine derivatives
07/01/1999DE19756261A1 Neue arylsubstituierte Pyridylalkan-, alken- und alkincarbonsäureamide New pyridylalkane aryl, alkene and alkincarbonsäureamide
07/01/1999DE19756236A1 Neue piperazinylsubstituierte Pyridylalkan-, alken- und -alkincarbonsäureamide New piperazinyl substituted pyridylalkane, alkene and -alkincarbonsäureamide
07/01/1999DE19756235A1 Neue piperidinylsubstituierte Pyridylalkan- alken- und -alkincarbonsäureamide New piperidinylsubstituierte pyridylalkane alkene and -alkincarbonsäureamide
07/01/1999DE19756212A1 Neue, mit einem cyclischen Imid substituierte Pyridylalkan-, alken- und -alkincarbonsäureamide Novel substituted with a cyclic imide pyridylalkane, alkene and -alkincarbonsäureamide
07/01/1999CA2315720A1 Inhibition of p38 kinase activity using substituted heterocyclic ureas
07/01/1999CA2315226A1 Hypoglycemic imidazoline compounds
07/01/1999CA2315070A1 Ortho-anthranilamide derivatives as anti-coagulants
07/01/1999CA2311428A1 Anilide derivative, production and use thereof
07/01/1999CA2309882A1 4-hydroxyquinoline-3-carboxamides and hydrazides as antiviral agents
06/1999
06/30/1999EP0926146A1 Chromene compounds
06/30/1999EP0926145A1 Napthalene compounds, method for their preparation and pharmaceutical compositions containing them
06/30/1999EP0925297A1 Endothelin receptor antagonists
06/30/1999EP0925296A1 New pharmaceutically active compounds
06/30/1999EP0925287A1 Heterocyclic metalloprotease inhibitors
06/30/1999EP0925286A1 Substituted pyrimidine derivatives and their pharmaceutical use
06/30/1999CN1221414A Novel benzothiepines having activity as inhibitors of ileal bile acid transport and taurocholate uptake
06/30/1999CN1221408A Substituted pyrazolyl-pyrazole derivatives and their use as herbicides
06/30/1999CN1221407A Aminoisoquinolines and aminothienopyridine derivatives and their use as anti-inflammatory agents
06/30/1999CN1043888C Fungicidal and herbicidal triazoles
06/29/1999US5917034 Antithrombotic n-amidinopiperidine and benzamidine derivatives
06/29/1999US5916908 Pharmaceutical pyrazole compositions useful as inhibitors of protein kinases
06/29/1999US5916891 Cytokine mediated diseases
06/29/1999US5916889 1,4-disubstituted piperazines
06/24/1999WO1999031096A1 Piperazine derivatives useful as hypoglycemic agents
06/24/1999WO1999031088A1 Triazine angiogenesis inhibitors
06/24/1999WO1999031087A1 Cyclic imide-substituted pyridylalkane, alkene and alkine carboxamides useful as cytostatic and immunosuppressive agents
06/24/1999WO1999031085A1 3-piperidyl-4-oxoquinazoline derivatives and medicincal compositions containing the same
06/24/1999WO1999031075A1 1-substituted-1-aminomethyl-cycloalkane derivatives (=gabapentin analogues), their preparation and their use in the treatment of neurological disorders
06/24/1999WO1999031074A2 ((cyclo)alkyl substituted)-.gamma.-aminobutyric acid derivatives (=gaba analogues), their preparation and their use in the treatment of neurological disorders
06/24/1999WO1999031073A1 Novel pyrimidine-5-carboxamide derivatives
06/24/1999WO1999031070A1 Substituted phenylpyrazolones, method and intermediate products for the production thereof, and their utilization for combating parasitic fungi and animal parasites
06/24/1999WO1999031068A1 Substituted isoquinoline derivatives and their use as anticonvulsants
06/24/1999WO1999031066A1 Pyridones as src family sh2 domain inhibitors
06/24/1999WO1999031064A1 Aryl-substituted pyridylalkane, alkene, and alkine carboxamides useful as cytostatic and immunosuppressive agents
06/24/1999WO1999031063A1 New piperazinyl-substituted pyridylalkane, alkene and alkine carboxamides
06/24/1999WO1999031060A2 Piperidinyl-substituted pyridylalkane, alkene and alkine carboxamides as cytostatics and immunesuppressants
06/24/1999WO1999031057A1 4(3)substituted-4(3)-aminomethyl-(thio)pyran or -piperidine derivatives (=gabapentin analogues), their preparation and their use in the treatment of neurological disorders
06/24/1999DE19756115A1 Substituierte Phenylpyrazolone, Verfahren und Zwischenprodukte zu ihrer Herstellung und ihre Verwendung zur Bekämpfung von Schadpilzen und tierischen Schädlingen Substituted phenylpyrazolones, processes and intermediates for their preparation and their use for controlling harmful fungi and animal pests
06/24/1999CA2315079A1 Substituted isoquinoline derivatives and their use as anticonvulsants
06/24/1999CA2313776A1 Triazine angiogenesis inhibitors
06/24/1999CA2280705A1 3-piperidyl-4-oxoquinazoline derivatives and pharmaceutical compositionscomprising the same
06/23/1999EP0924209A1 Hypoglycemic imidazoline compounds
06/23/1999EP0924207A1 Chromene-3-carboxylate derivatives
06/23/1999EP0924201A1 Tricyclic-substituted pyrazolyl benzenesulfonamides and their use as cyclooxygenase II inhibitors
06/23/1999EP0923933A1 Substituted pyrazolyl benzenesulfonamides for use in the treatment of inflammation
06/23/1999EP0923576A1 4-aminoethoxy-indolone derivatives as dopamine d2 agonists
06/23/1999EP0923570A1 Pyridyl alkene- and pyridyl alkine- acid amides as cytostatics and immunosuppressives
06/23/1999EP0923569A1 Butyric acid matrix metalloproteinase inhibitors
06/23/1999EP0923563A1 1,4-heterocyclic metallprotease inhibitors
06/23/1999EP0923562A1 Substituted p-trifluoromethylphenyluracils
06/23/1999EP0923561A1 Heterocyclic metalloprotease inhibitors
06/23/1999EP0923558A1 Substituted 1-(3-pyrazolyl)-pyrazoles
06/23/1999EP0923542A1 Aryl substituted cyclic amines as selective dopamine d3 ligands
06/23/1999EP0923536A1 Arylcycloalkane carboxylic esters, their use, pharmaceutical compositions and preparation
06/23/1999CN1220602A Anti-viral compounds
06/23/1999CN1220265A New piperazine and piperidine compounds
06/23/1999CN1220264A Novel thiophenesulfonylurea derivatives
06/22/1999US5914334 Stable gel formulation for topical treatment of skin conditions
06/22/1999US5914333 Treatment of psychotic disorders
06/22/1999US5914332 Retroviral protease inhibiting compounds
06/22/1999CA2151674C Methods of administering crf antagonists
06/17/1999WO1999029677A1 Substituted 2,4-diamino-1,3,5-triazines
06/17/1999WO1999029674A1 Retinoic acid mimetic anilides
06/17/1999WO1999029673A1 SELECTIVE β3 ADRENERGIC AGONISTS
06/17/1999WO1999029670A2 Aminocarbonyltetralin and dihydronaphtalene derivates as thrombin inhibitors
06/17/1999DE19755016A1 Substituierte 2,4-Diamino-1,3,5-triazine Substituted 2,4-diamino-1,3,5-triazines