Patents
Patents for C07D 409 - Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms (52,226)
06/2000
06/29/2000WO2000037422A2 Ion channel modulating agents
06/29/2000CA2357760A1 Process for preparing n6-substituted deaza-adenosine derivatives
06/29/2000CA2355137A1 Non-peptide nk1 receptors antagonists
06/29/2000CA2353635A1 Anilide derivative, production and use thereof
06/28/2000EP1012166A1 1-amino-7-isoquinoline derivatives as serine protease inhibitors
06/28/2000EP1012147A2 O-substituted hydroxycumaranone derivatives as antitumor and antimetastatic agents
06/28/2000EP1012139A1 AZETIDINONE DERIVATIVES AS $g(b)-LACTAMASE INHIBITORS
06/28/2000EP1011663A1 BETA-LACTAM INHIBITORS OF CoA-IT
06/28/2000CN1258296A Pyridine derivatives and pharmaceutical compositions contg. them
06/28/2000CN1258291A Polymerisable, optically active dioxolane diesters
06/28/2000CN1258289A Substd. 2-benzoyl-cyclohexane-1,3-diones
06/28/2000CN1258286A Non-steroidal (hetero) cyclically substd. acylanilides with mixed gestagen and androgen activity
06/28/2000CN1258219A Benzocycloheptathiophene compounds
06/28/2000CN1053904C N-pyridyl carboxamides and derivs. processes for their preparation and pharmaceutical compositions contg. them
06/28/2000CN1053895C Substd. sulfonic acid amide, preparation process and pharmaceutical composition of same
06/27/2000US6080869 Chemical reduction process; forming dopamine da2 receptor agonists and beta2 adrenoreceptor agonists for treating obstructive airways diseases
06/27/2000US6080861 Herbicidal 6-thienyloxypyrid-2-carboxamides
06/27/2000US6080776 Used as a microbiocide for crop protection
06/27/2000US6080767 Substituted n-[(aminoiminomethyl or aminomethyl)phenyl]propyl amides
06/27/2000US6080764 Superoxide radical inhibitor
06/27/2000US6080763 Inhibit the release of inflammatory cytokines, e.g., tumor necrosis factor and interleukin-1; useful to treat chronic inflammatory disease; autoimmune diseases, e.g. rheumatoid arthritis, osteoporosis; pyrazolylureas
06/27/2000US6080757 Treatment of helicobacter (campylobacter) pylori infections; treatment and prevention of peptic ulcers, gastritis, dyspepsia, and gastric cancer
06/27/2000US6080743 2,3-dioxo-1,2,3,4-tetrahydro-quinoxalinyl derivatives
06/27/2000CA2017193C N-(aryloxyalkyl)heteroarylpiperidines and-heteroarylpiperazines, a pro cess for their preparation and their use as medicaments
06/22/2000WO2000035915A1 Piperazine derivatives
06/22/2000WO2000035911A1 Heteroaryl-cyclic acetals
06/22/2000WO2000035909A1 4-aryloxindoles as inhibitors of jnk protein kinases
06/22/2000WO2000035908A1 4-alkenyl (and alkynyl) oxindoles as inhibitors of cyclin-dependent kinases, in particular cdk2
06/22/2000WO2000035906A2 4- and 5-alkynyloxindoles and 4- and 5-alkenyloxindoles
06/22/2000WO2000035903A2 Thiochromanoyl cyclohexenone derivatives
06/22/2000WO2000035886A2 (hetero)aryl-bicyclic heteroaryl derivatives, their preparation and their use as protease inhibitors
06/22/2000WO2000035877A1 Heterocyclic piperidines as modulators of chemokine receptor activity
06/22/2000WO2000035865A2 Tubulin-binding agents
06/22/2000WO2000035864A1 New biphenyl and biphenyl-analogous compounds as integrin antagonists
06/22/2000CA2355249A1 Protease inhibitors
06/22/2000CA2355161A1 Biphenyl and biphenyl-analogous compounds as integrin antagonists
06/22/2000CA2355125A1 Thiochromanoylcyclohexenone derivatives
06/22/2000CA2354875A1 Piperazine derivatives
06/22/2000CA2354873A1 4-alkenyl (and alkynyl) oxindoles as inhibitors of cyclin-dependent kinases, in particular cdk2
06/22/2000CA2354591A1 4-aryloxindoles as inhibitors of jnk protein kinases
06/22/2000CA2354510A1 4- and 5-alkynyloxindoles and 4- and 5-alkenyloxindoles
06/22/2000CA2347912A1 Heterocyclic piperidines as modulators of chemokine receptor activity
06/21/2000EP1009758A1 Meta-benzamidine derivatives as serine protease inhibitors
06/21/2000EP1009747A1 Ureido and thioureido derivatives of 4-amino-2(5h)-furanones and 4-amino-2(5h)-thiophenones as antitumor agents
06/21/2000EP1009741A1 Novel carboxylic acid derivatives, their production and their use as mixed et a?/et b? endothelin-receptor antagonists
06/21/2000EP1009405A1 Pyrrolidine and piperidine modulators of chemokine receptor activity
06/21/2000CN1257491A 4-tetrahydropyridylpyrimidine derivatives
06/21/2000CN1257489A Substituted benzopyran derivatives for the treatment of inflammation
06/21/2000CN1053667C Inhibiting photodecomposition of 3-substituted-2-oxindoles
06/21/2000CN1053666C Benzoheterocylic compounds and process for preparing medicated salt thereof
06/21/2000CN1053665C 2,4-diaryl-1,3-dithiolanes, 2,4-diaryl-1,3-dioxolanes, 2,4-diaryl-1,3-oxathiolanes derivant
06/21/2000CN1053659C Pesticidal 1-aryl-5-(substituted alkylideneimino) pyrazoles
06/20/2000US6077858 Administering a substituted indole compound to the patients for the treatment of a variety of sex-hormone related and other conditions in both men and women
06/20/2000US6077850 Useful for treating cyclooxygenase-2 mediated disorders, such as inflammation and inflammation-related disorders
06/20/2000US6077849 Administering to a diabetic patient an antidiabetic fused bicyclic heteroaryl compound
06/20/2000US6077840 For treating or preventing progesterone-related diseases, for having an abortion, or for orally preventing conception, breast cancer, ovarian cancer, hysteromyoma, endometriosis, meningioma, myeloma, osteoporosis
06/20/2000US6077813 Substituted aromatic thiocarboxylic acid amides and their use as herbicides
06/15/2000WO2000034271A1 Method for producing pyrazolylbenzoyl derivatives and novel pyrazolylbenzoyl derivatives
06/15/2000WO2000034270A1 Thiochromanoylpyrazolone derivatives
06/15/2000WO2000034265A2 Quinoline-indole antimicrobial agents
06/15/2000WO2000034262A1 Benzofuran derivatives, process for the preparation of the same and uses thereof
06/15/2000WO2000009500A3 Nematicidal pyrazoles
06/15/2000WO2000006531A3 Nitric esters and nitrate salts of specific drugs
06/15/2000CA2353572A1 Method for producing pyrazolylbenzoyl derivatives and novel pyrazolylbenzoyl derivatives
06/15/2000CA2353542A1 Thiochromanoylpyrazolone derivatives
06/14/2000EP1008594A1 Compounds derived from thophene and benzothiophene, and related utilisation and composition
06/14/2000EP1008589A1 Fungicidal imidazolinones
06/14/2000EP1007524A1 Indole derivatives as 5-ht1b and 5-ht1d agonists
06/14/2000EP1007523A1 Indole and 2,3-dihydroindole derivatives, their preparation and use
06/14/2000EP1007515A1 Arylpyridazinones as prostaglandin endoperoxide h synthase biosynthesis inhibitors
06/14/2000EP1007042A1 Novel heteroaryl compounds for the modulation of protein tyrosine enzyme related cellular signal transduction
06/13/2000USRE36736 Substituted pyrroles
06/13/2000US6075151 Inhibiting bone loss or bone resorption, particularly osteoporosis, and cardiovascular-related hyperlipidemia, cardiovascular disorders
06/13/2000US6075146 Process for preparing benzoic acid derivative intermediates and benzothiophene pharmaceuticals
06/13/2000US6075144 9-hydroxyamino tetrahydroacridine and related compounds
06/13/2000US6075040 Obesity and diabetes
06/13/2000US6075026 Certain substituted 1-aryl-3-piperazin-1'-yl propanones
06/13/2000CA2085878C Bis-benzo or benzopyrido cyclo hepta piperidene, piperidylidene and piperazine compounds and compositions
06/13/2000CA1341023C Peptide derivatives
06/08/2000WO2000032590A1 SUBSTITUTED OXOAZAHETEROCYCLYL FACTOR Xa INHIBITORS
06/08/2000WO2000032588A2 Carboxylic acids and carboxylic acid isosteres of n-heterocyclic compounds
06/08/2000WO2000032577A2 Substituted benzo[de]isoquinoline-1,3-diones
06/08/2000CA2352045A1 Substituted benzo[de]isoquinoline-1,3-diones
06/07/2000EP1006113A1 Derivatives of 2-(2-oxo-ethylidene)-imidazolidin-4-one and their use to inhibit abnormal cell growth
06/07/2000EP1006110A1 Derivatives of acyl-piperazinil-pyrimidins, preparation thereof and application as medicaments
06/07/2000EP1005467A1 Benzothiophene derivatives as herbicides
06/07/2000EP1005460A1 Prostaglandin endoperoxide h synthase biosynthesis inhibitors
06/07/2000CN1255864A Combination of ileal bile acid transport inhibiting benzothiepines and HMG Co-A reductase inhibitors
06/07/2000CN1255495A Process for synthesizing beta-halobutenolide
06/06/2000US6071937 Oxymethoxy-3-aryl-pyrone derivatives
06/06/2000US6071931 AT1 -receptor antagonists for preventing and treating postischemic renal failure and for protecting ischemic kidneys
06/06/2000US6071921 4-phenyl-7-arylquinoazolines; angiogenisis inhibitors and/or vascular permeability reducing effects in warm-blooded animals; anticarcinogenic and -arthritic agents; rheumatic diseases; vascular endothelium growth factor inhibitors
06/06/2000US6071920 Bind to 5ht 1a receptors for treating disorders of the lower urinary tract; cns disorders; anxiolytic agents; antidepressants; hypotensive agents; sleep and eating disorders
06/06/2000US6071908 Radiation-activated cytotoxin therapy of neoplastic disease
06/06/2000US6071903 2,3,4,5-tetrahydro-1H-[1,4]-benzodiazepine-3-hydroxyamic acids
06/06/2000US6071860 For selective control of broad-leaved and grass weeds in crops of useful plants
06/02/2000WO2000031072A1 Process for making 5-substituted pyrazoles using dithietanes
06/02/2000WO2000031063A1 SUBSTITUTED PYRAZOLES AS p38 KINASE INHIBITORS
06/02/2000WO2000031039A1 Substituted benzo[de]isoquinoline-1,3-diones
06/02/2000WO2000031032A1 Pyrrolidine derivatives-ccr-3 receptor antagonists