Patents for C07D 409 - Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms (52,226) |
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12/11/2003 | CA2482838A1 Pyrazole compounds and pharmaceutical compositions containing the compound |
12/10/2003 | EP1369414A1 Enantiomerically pure Arylcycloalkyl hydroxycarboxylic esters, processes for their preparation and their use as modulators of muscarinic receptors |
12/10/2003 | EP1369410A1 Process for the stereoselective reduction of derivatives of 4-aryl-4-oxobutyric acid |
12/10/2003 | EP1368346A1 Substituted benzofuran-2-carboxamides derivatives |
12/10/2003 | EP1368344A1 Piperazine derivatives, their preparation and uses in therapy (5ht1b receptor activity) |
12/10/2003 | EP1368342A2 Benzimidazole and pyridylimidazole derivatives as ligands for gaba receptors |
12/10/2003 | EP1368340A1 Piperazine derivatives as melanocortin receptor agonists |
12/10/2003 | EP1368336A2 Thiophene substituted amine derivatives as glyt-1 inhibitors |
12/10/2003 | EP1368325A1 New asymmetric process for the preparation of diarylmethylpiperazines derivatives and novel asymmetric diarylmetylamines as intermediates |
12/10/2003 | EP1368324A1 Quinazolines as mmp-13 inhibitors |
12/10/2003 | EP1368323A1 Pyrimidine matrix metalloproteinase inhibitors |
12/10/2003 | EP1368320A1 Substituted 2-oxy-3,5-dicyano-4-aryl-6-aminopyridines and use thereof |
12/10/2003 | EP1368318A2 Calcilytic compounds |
12/10/2003 | EP1368032A1 Excitatory amino acid receptor antagonists |
12/10/2003 | EP1367893A1 Pyridyl pyrimidines for use as pesticides |
12/10/2003 | EP1115721B1 Pyrimidone derivatives |
12/10/2003 | EP1091953B1 Novel benzothiepines having activity as inhibitors of ileal bile acid transport and taurocholate uptake |
12/10/2003 | EP0970046B1 N-hydroxy-2-(alkyl, aryl, or heteroaryl sulfanyl, sulfinyl or sulfonyl)-3-substituted alkyl, aryl or heteroarylamides as matrix metalloproteinase inhibitors |
12/10/2003 | EP0714396B1 Vasocontrictive dihydrobenzopyran derivatives |
12/10/2003 | EP0628064B2 Photochromic naphthopyrans |
12/10/2003 | CN1130360C Substituted thienocycloalk (en)ylamino-1,3,5-triazine |
12/10/2003 | CN1130358C Imidzzole compounds and preparing method and application thereof |
12/10/2003 | CN1130351C 1,5-benzodiazepine derivatives |
12/09/2003 | US6660866 C10 carbonate substituted taxanes |
12/09/2003 | US6660760 Heterocyclic aromatic compounds useful as growth hormone secretagogues |
12/09/2003 | US6660752 2,6-Substituted chroman derivatives useful as beta-3 adrenoreceptor agonists |
12/09/2003 | US6660751 Sulfonamide derivatives as 5-HT7 receptor antagonists |
12/09/2003 | US6660740 Sorbitol dehydrogenase inhibitors |
12/09/2003 | US6660739 Heterocyclic amides as inhibitors of factor Xa |
12/09/2003 | US6660738 Such as (3R,5S)-1-pyrimidin-2-yl-5-(2,4,5-trifluoro-benzyloxymethyl)-pyrrolidine-3 -thiol trifluoro-acetate useful as inhibitors of metalloproteases for treating diseases associated with vasoconstriction |
12/09/2003 | US6660736 MAO-B inhibitors |
12/09/2003 | US6660732 Ureas and thioureas inhibit production of cytokines |
12/09/2003 | US6660731 Pyrazole compounds useful as protein kinase inhibitors |
12/09/2003 | US6660728 Thienyl substituted acylguanidines as inhibitors of bone resorption and vitronectin receptor antagonists |
12/09/2003 | CA2189593C Sulphonylaminocarbonyltriazolinones having substituents bonded via oxygen |
12/04/2003 | WO2003099812A1 Phenyl-furan or phenyl-thiophene derivatives, their preparation and their use as medicine |
12/04/2003 | WO2003099805A1 Novel thiophene amidines, compositions thereof, and methods of treating complement-mediated diseases and conditions |
12/04/2003 | WO2003099795A1 4-substituted imidazole-2-thiones and imidazol-2-ones as agonists of the alpha-2b and alpha-2c adrenergic receptors |
12/04/2003 | WO2003099787A1 Novel piperidine compound |
12/04/2003 | WO2003099786A2 Aromatic sulfones and their medical use |
12/04/2003 | WO2003099773A1 Ccr9 inhibitors and methods of use thereof |
12/04/2003 | WO2003099765A1 β-ALANINE DERIVATIVE AND USE THEREOF |
12/04/2003 | WO2003099284A1 Amino-pyridine, -pyridine and pyridazine derivatives for use as vanilloid receptor ligands for the treatment of pain |
12/04/2003 | WO2003099276A1 1,1-disubstituted cycloalkyl derivatives as factor xa inhibitors |
12/04/2003 | WO2003099266A2 Acetamides and benzamides that are useful in treating sexual dysfunction |
12/04/2003 | WO2003063794A3 2,4-pyrimidinediamine compounds and their uses |
12/04/2003 | WO2003027085A3 3-pyridyl or 4-isoquinolinyl thiazoles as c17,20 lyase inhibitors |
12/04/2003 | WO2002094796A3 Benzo[g]quinoxaline derivatives as effective compounds against infectious diseases |
12/04/2003 | WO2002068397A8 Diaminoquinazoline esters for use as dihydrofolate reductade inhibitors |
12/04/2003 | US20030225288 Small organic compounds to modulate chemokine receptor activity; treating psoriasis, autoimmune diseases, multiple sclerosis, graft rejection, infectious diseases; anti-allergen, -arthritic, -inflammatory, carcinogenic agents |
12/04/2003 | US20030225283 2-Substituted phenyl,3-polar ring,N-heroaromatic propion-amides, e.g., 1-(2-(3,4-Dichlorophenyl)-3-(tetrahydro-furan-2-yl)-propionyl)-3- methylurea; antidiabetic agents; increase the flux of glucose metabolism in beta-cells and hepatocytes |
12/04/2003 | US20030225281 Piperidines derivatives and their use as serotonin receptor antagonists |
12/04/2003 | US20030225276 Prostaglandin endoperoxide H synthase biosynthesis inhibitors |
12/04/2003 | US20030225269 Inhibitors of interleukin-1beta converting enzyme |
12/04/2003 | US20030225228 A catalyst for the polymerization of olefins, contains a titanium zirconium or hafnium complex of a dianionic bidentate ligand, (at least one of donor atoms of the ligand is a nitrogen atom substituted by a pyrrolyl group) |
12/04/2003 | US20030225150 Method of using a COX-2 inhibitor and a topoisomerase II inhibitor as a combination therapy in the treatment of neoplasia |
12/04/2003 | US20030225148 Biological methods of use of 4-amino-3-mercapto-triazoles |
12/04/2003 | US20030225121 Treatment of a disorder of the central nervous system related to or affected by the 5-HT6 receptor |
12/04/2003 | US20030225115 Anticoagulants |
12/04/2003 | US20030225109 Inducing contraception, treat progesterone-related carcinomas and adenocarcinomas; hormone replacement therapy |
12/04/2003 | US20030225106 Prophylaxis and treatment of angiogenesis mediated diseases such as cancer |
12/04/2003 | US20030225100 Aminoalkoxybenzoyl-benzofuran or benzothiophene derivatives, method of preparing same and compositions containing same |
12/04/2003 | US20030225097 Amino substituted dibenzothiophene derivatives for the treatment of disorders mediated by np y5 receptor |
12/04/2003 | US20030225085 For reducing neuronal cell death in response to a traumatic event |
12/04/2003 | US20030225084 Have an affinity for the gabapentin binding site and can be used to treat conditions such as pain, epilepsy, migraine and others. |
12/04/2003 | US20030225077 Naphthylamines used to chronic inflammatory diseases. |
12/04/2003 | US20030225071 N-heterocyclic amides and carbamates |
12/04/2003 | US20030225061 Protease inhibitors |
12/04/2003 | US20030225057 3-Benzoazepine derivatives |
12/04/2003 | US20030225053 N-arylcarboxamides of fused ring systems including naphthalenes, benzothiophenes, benzofurans and indoles |
12/04/2003 | US20030225043 Especially for inhibiting type IV collagenase |
12/04/2003 | US20030224442 Comprises nucleotide sequences coding g-protein coupled receptor for use in treatment of anxiety, depression, obsessive-compulsive, schizophrenia autism, migraine, emesis, alcoholism and neurodegenerative disorders |
12/04/2003 | US20030224288 Stimulation sensitive composition and compound |
12/04/2003 | CA2784937A1 Ccr9 inhibitors and methods of use thereof |
12/04/2003 | CA2486962A1 Compounds |
12/04/2003 | CA2486564A1 Acetamides and benzamides that are useful in treating sexual dysfunction |
12/04/2003 | CA2486376A1 Amino-pyridine, -pyridine and pyridazine derivatives for use as vanilloid receptor ligands for the treatment of pain |
12/04/2003 | CA2484822A1 Novel thiophene amidines, compositions thereof, and methods of treating complement-mediated diseases and conditions |
12/03/2003 | EP1367055A1 Isoquinolinyl carboxamides and their use as anticonvulsants |
12/03/2003 | EP1366043A1 2-heteroaryl-3,4-dihydro-2h-pyrrole derivatives and the use thereof as pesticides |
12/03/2003 | EP1366038A1 Cdk-1 inhibitor oxindoles and the application thereof in therapeutics |
12/03/2003 | EP1366028A1 Diaminoquinazoline esters for use as dihydrofolate reductase inhibitors |
12/03/2003 | EP1119557B1 Indeno-, naphto- and benzocyclohepta dihydrothiazole derivatives, the production thereof and their use as anorectic medicaments |
12/03/2003 | EP1117659B1 Substituted 3-cyanoquinolines as protein tyrosine kinases inhibitors |
12/03/2003 | EP0937070B1 Benzoheterocyclic distamycin derivatives, process for preparing them, and their use as antitumor and antiviral agents |
12/03/2003 | EP0786455B1 Imidazole derivative |
12/03/2003 | CN1129605C Modified aminoacids, pharmaceuticals containing these compounds and mehtod for their prodn |
12/03/2003 | CN1129596C Synthetic intermediate of cephalo olefine compound |
12/03/2003 | CN1129591C O-substituted hydroxycumaranone derivatives as antitumor and antimetastatic agents |
12/03/2003 | CN1129584C Pyrimidinyloxyalkanoic amide derivatives and fungicides for agricultural and horiticultural use |
12/03/2003 | CN1129583C Compound as intermediates for use in preparation of optically active 2-imidazoline-5-one or 2-imidazoline-5-thionone derivatives |
12/03/2003 | CN1129578C Tetrahydrobenzindole derivs |
12/03/2003 | CN1129576C Phenyl heterocyclic compound used as epoxy enzyme-2 inhibitor |
12/02/2003 | US6657070 Production of chirally pure α-amino acids and N-sulfonyl α-amino acids |
12/02/2003 | US6657060 Neuropeptide Y antagonists; treatment of eating disorders such as obesity and hyperphagia |
12/02/2003 | US6656966 Nitrosated and nitrosylated taxanes, compositions and methods of use |
12/02/2003 | US6656957 Pyridine derivatives |
12/02/2003 | US6656954 Such as N-hydroxy-2-(((4-phenoxyphenyl)-sulfonyl)methyl) benzamide which inhibits matrix metalloprotease activity |
12/02/2003 | US6656939 Pyrazole compounds useful as protein kinase inhibitors |
12/02/2003 | US6656933 Novel compounds which inhibit production of cytokines involved in inflammatory processes |