Patents
Patents for C07D 409 - Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms (52,226)
03/2004
03/03/2004EP1392641A1 Substituted cyclohexane-1,4-diamine derivatives
03/03/2004EP1392310A1 Combinations of aldose reductase inhibitors and cyclooxygenase-2 inhibitors
03/03/2004EP1392300A1 2,5-disubstituted pyridine, pyrimidine, pyridazine and 1, 2, 4-triazine derivatives for use as p38 inhibitors
03/03/2004EP1392283A1 Substituted coumarins and quinolines as caspases activators
03/03/2004EP1045839B1 Novel amines as pharmaceutical agents
03/03/2004EP1017692B1 4-heteroaryl-tetrahydroquinolines and their use as inhibitors of the cholesterin-ester transfer protein
03/03/2004EP0882714B1 Substituted vinylpyridine derivatives and drugs containing the same
03/03/2004EP0853617B1 Novel 2,3-dioxo-1,2,3,4-tetrahydro-quinoyxalinyl derivatives
03/03/2004EP0841916B9 Endothelin receptor antagonists
03/03/2004CN1479728A Pexoxisome proliferator activated receptor alpha agonists
03/03/2004CN1479727A Piperazinylpyrazine compounds as agonist or antagonist of 5-hydroxytryptamine 5HT-2 receptor
03/03/2004CN1479715A Amide for inhibition of IL-8-induced chemiotaxis of neutrophil leucocytes
03/03/2004CN1479703A Method for producing compounds having CF2O bridge
03/03/2004CN1479618A Treatment of sexual dysfunction using boonbesin antagonist
03/03/2004CN1478779A Tosylate and benzene sulfonate of pyrazolopy ridone compound
03/03/2004CN1478778A 抗真菌剂及其制备方法和中间体 Antifungal agent and its preparation method and intermediates
03/03/2004CN1478472A 细胞粘连抑制剂 Cell adhesion inhibitor
03/02/2004US6700013 O-bromophenylacetic acid derivative chemical intermediate; smooth muscle relaxants, antiinflammatory agents; respiratory system disorders
03/02/2004US6699887 Administering a therapeutically effective amount of a pyrrazole sulfide or ether compound to treat the human immunodeficiency virus infection
03/02/2004US6699881 Thiol compounds, their production and use
03/02/2004US6699870 Phthalazine compounds and therapeutic agents for erectile dysfunction
03/02/2004US6699860 Di-substituted aminomethyl-chroman derivative beta-3 adrenoreceptor agonists
03/02/2004US6699856 Pyrazinones, compositions containing such compounds and methods of use
03/02/2004US6699854 2-substituted 4-heteroaryl- pyrimidines, inhibitors of cyclin-dependent kinases (cdks)
03/02/2004US6699818 Trifluoromethylpyrrole carboxamides and trifluoromethylpyrrolethioamides as fungicides
03/02/2004CA2138289C N-substituted azabicycloheptane derivatives, the preparation and use thereof
02/2004
02/26/2004WO2004016741A2 Prenylation inhibitors containing dimethyl-cyclobutane and methods of their synthesis and use
02/26/2004WO2004016604A2 Azabicyclic compounds are central nervous system active agents
02/26/2004WO2004016597A2 Protein kinase inhibitors and uses thereof
02/26/2004WO2004016592A1 Prenylation inhibitors and methods of their synthesis and use
02/26/2004WO2004016576A1 Fused benzene derivative and use
02/26/2004WO2004016086A2 2,4,5-trisubstituted imidazoles and their use as anti-microbial agents
02/26/2004WO2003104217A3 Prodrugs of excitatory amino acids
02/26/2004WO2003057144A3 Change inhibitors of dipeptidyl peptidase iv
02/26/2004WO2003050261A3 (1-phenyl-2-heteroaryl)ethyl-guanidine compounds as inhibitors of mitochondrial f1f0 atp hydrolase
02/26/2004WO2003039549A8 Selective antibacterial agents
02/26/2004US20040039044 Coupling under reducing conditions aminoalkylpyrrolidine-n-alkyl with one equivalant of a aldehyde compound; useful for treating pain, schizophrenia, depression and sleep disorders
02/26/2004US20040039033 Administering (1-phenyl-2-heteroaryl)ethyl-guanidine compounds for treating ischemic conditions including myocardial infarction, congestive heart failure, and cardiac arrhythmias
02/26/2004US20040039028 Nitrogen compounds such as 3,5-dichloro-2-fluoro-4-(3-isoprop -yl-4-methoxyphenoxy)-6-methoxycarbonylmethylaminopyridine, administered for prophylaxis of metabolic disorders
02/26/2004US20040039016 HIV protease inhibitors
02/26/2004US20040038998 Aminopiperidine quinolines and their azaisosteric analogues with antibacterical activity
02/26/2004US20040038992 2-thio-(or oxy)-5-amino-1,3,4-thiadiazoles or oxadiazoles
02/26/2004US20040038991 Imidazolyl-cyclic acetals
02/26/2004US20040038979 Novel 6-heteroarylphenanthridines
02/26/2004US20040038977 Treating arthritis, pain and cancer
02/26/2004US20040038976 S,N-diarylsulfonamide derivatives; treating inflammatory diseases such as Celiac's disease, Crohn's disease or colitis.
02/26/2004US20040038973 Treating osteoarthritis or rheumatoid arthritis
02/26/2004US20040038969 Substituted aminopyrimidines and aminopyridazines; analgesics particularly for migraines, neuropathic pain and associated hyperalgesia and allodynia; antiinflammatory agents; treating asthma, gastrointestinal disorders, etc.
02/26/2004US20040038943 Indole and benzimidazole 15-lipoxygenase inhibitors
02/26/2004US20040038858 Carboxamide derivatives and their use in the treatment of thromboembolic diseases and tumours
02/26/2004CA2495589A1 Azabicyclic compounds are central nervous system active agents
02/26/2004CA2495383A1 Fused benzene derivative and use
02/25/2004EP1391952A2 Salts of pentacyclic or tetrapentaline derived anions, and their uses as ionic conductive materials
02/25/2004EP1391456A1 2-iminoimidazole derivative (2)
02/25/2004EP1391451A1 2-iminopyrrolidine derivates
02/25/2004EP1390362A1 Substituted benzofurans and benzothiophenes, methods of making and methods of use as integrin antagonists
02/25/2004EP1390352A1 Pyrimidine derivatives
02/25/2004EP1390350A1 Novel compounds
02/25/2004EP1390349A1 Aminoquinoline and aminopyridine derivatives and their use as adenosine a3 ligands
02/25/2004EP1390348A1 5-cyano-1h-indole derivatives as antagonists of the interleukine-8 receptors
02/25/2004EP1390340A1 Copper-catalyzed formation of carbon-heteroatom and carbon-carbon bonds
02/25/2004EP1390034A1 N-substituted nonaryl-heterocyclo amidyl nmda/nr2b antagonists
02/25/2004EP1283837B1 New thiochromane derivatives and their use as thrombin inhibitors
02/25/2004EP1263756B1 Beta-amino acid derivatives as inhibitors of matrix metalloproteases and tnf-alpha
02/25/2004EP1230232B1 Substituted 4h-chromene and analogs as activators of caspases and inducers of apoptosis and the use thereof
02/25/2004EP1222171B1 Pyridinium derivatives for the management of aging-related and diabetic vascular complications, process for their preparation and therapeutic uses thereof
02/25/2004EP1211246B1 Pyrimidine derivatives and herbicides containing the same
02/25/2004EP1200426B1 Substituted thiene-3-yl-sulfonyl amino(thio)carbonyl-triazolin(thi)ones
02/25/2004EP1200409B1 Substituted isoquinoline derivatives and their use as anticonvulsants
02/25/2004EP1178986B1 Furanone derivatives as inhibitors of cathepsin s
02/25/2004EP1042296B1 Substituted isoquinoline derivatives and their use as anticonvulsants
02/25/2004EP1040108B1 Ortho-anthranilamide derivatives as anti-coagulants
02/25/2004CN1478089A Substituted derivatives of aminofuran-2-Y1-acetic acid and aminothien-2-Y1-acetic acid and use thereof for treating migraines and pain
02/25/2004CN1478088A Benzothiophene derivative compounds, process of preparation and use thereof
02/25/2004CN1478085A ABCA-1 elevating compounds against coronary artery disease or atherosclerosis
02/25/2004CN1478078A Nitrogenous aromatic ring compounds
02/24/2004US6696540 Episulfide compound, method for producing the same and optical product comprising the same
02/24/2004US6696470 Pyridylthiophene compounds
02/24/2004US6696467 Quinoline derivatives
02/24/2004US6696452 Glycogen synthase kinase-3 and aurora-2 a serine/threonine protein kinase inhibitors; antidiabetic and anticancer agents and alzheimer's disease treatments
02/24/2004US6696449 Control degradation of conencting tissue; cardiovascular disorders
02/24/2004US6696447 Hydroxyphenyl-piperazinyl-methyl-benzamide derivatives for the treatment of pain
02/24/2004US6696437 Polymerase inhibitors comprising heterocyclic amides such as 2-pyridin-2-ylbenzimidazole-4-carboxamide, used for prophylaxis of neurodegenerative disorders, damage to hearts or brains, and as anticarcinogenic agents
02/24/2004US6696182 Organic electroluminescent device comprising dipyridylthiophene derivative
02/24/2004CA2279186C Sulfonyl urea derivatives and their use in the control of interleukin-1 activity
02/19/2004WO2004014905A1 Substituted benzimidazole compounds
02/19/2004WO2004014900A1 Benzimidazoles and benzothiazoles as inhibitors of map kinase
02/19/2004WO2004014899A1 Thiophene compounds
02/19/2004WO2004014891A1 Pyridazine derivatives as ligands for gaba receptors
02/19/2004WO2004014873A1 4-substituted quinazoline-8-carboxyamide derivative and pharmaceutically acceptable addition salt thereof
02/19/2004WO2004014871A1 Vanilloid receptor ligands and their use in treatments
02/19/2004WO2004014867A2 Matrix metalloproteinase inhibitors and methods for identification of lead compounds
02/19/2004WO2004014865A1 Phenylpyridazine derivatives as ligands for gaba receptors
02/19/2004WO2004014864A1 1h-indazole-3-carboxamide compounds as cyclin dependent kinases (cdk) inhibitors
02/19/2004WO2004014860A2 Fused heterocyclic compounds as peptidase inhibitors
02/19/2004WO2004014851A2 Tyrosine kinase inhibitors
02/19/2004WO2004014844A2 Aryl and heteroaryl compounds and methods to modulate coagulation
02/19/2004WO2004014842A1 Acylated arylcycloalkylamines and their use as pharmaceuticals
02/19/2004WO2004014425A1 Activators of small conductance calcium activated potassium channels and use thereof
02/19/2004WO2004014381A2 Matrix metalloproteinase inhibitors and methods for identification of lead compounds