Patents
Patents for C07D 409 - Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms (52,226)
09/2003
09/04/2003US20030166690 Use of compounds for decreasing activity of hormone-sensitive
09/04/2003US20030166685 Acid derivatives of benzene useful as anticoagulants in treating and preventing cardiovascular diseases, as anti-inflammatory agents, and as metastasis inhibitors in treating cancer
09/04/2003US20030166684 3-phenyl-furan-(5H)-2-one and dihydrofuran-2-one derivatives as antibacterial agents
09/04/2003US20030166675 Substituted quinolin-2-one derivatives useful as antiproliferative agents
09/04/2003US20030166672 Derivatives of 4-(Thio- or Selenoxanthene-9-ylidene)-piperidine or acridine and its use as a selective 5-HT2B receptor antagonist
09/04/2003US20030166664 E.g. 3-(1-(2-(5-(acetylamino)-2-methylphenyl)ethyl)piperidin--4-yl)-6-chloro-1H -indole; potent dopamine D4 ligands, dopamine antagonists; antiseratonin agents; psychoses; anxiolytic agents; antidepressants; side effects reduction
09/04/2003US20030166663 E.g.,4-tert-butyl-N-(4-piperazin-1-yl-quinolin-6-yl)benzene-su lfonamide or 5-chloro-3-methyl-benzo(b)thiophene-2-sulfonic acid (4-piperazin-1-yl-quinolin-6-yl) amide; obesity; food intake reduction; bind to 5-HT6 receptors; antiseraton agents
09/04/2003US20030166655 Acyclic nucleotide phosphodiesterase of type 4 inhibitors; antiinflammatory agents; antiallergens; antiarthritis agents, rheumatic diseases; AIDS; gastrointestinal, respiratory, brain, urogenital disorders
09/04/2003US20030166652 Chemical compounds
09/04/2003US20030166649 E.g., 4-(2-(1-Benzhydryl-2-(2-((benzylsulfonyl)amino)ethyl)-5-chloro-1H-indol-3 -yl)ethoxy)benzoic acid; inhibitors of phospholipase enzymes, esp. phospholipase A2; antiarthritic and -inflammatory agents; analgesics; rheumatoid diseases
09/04/2003US20030166644 Compounds and uses thereof for decreasing activity of hormone-sensitive lipase
09/04/2003US20030166637 Amines such as 9-(4-(4-(benzothiazol-2-yl)-piperazin-1-yl)-butyl)-9H-fluorene-9-carboxylic acid (2,2,2-trifluoroethyl) amide, used as microsomal triglyceride transfer protein antagonists, to prevent atherosclerosis or hyperlipemia
09/04/2003US20030166633 Pyridinylimidazoles
09/04/2003US20030166590 Microsomal triglyceride transfer protein
09/04/2003US20030164173 Reduced ignition propensity smoking article
09/04/2003CA2477254A1 Methods and compounds useful in inhibiting oxidative and/or free radical damage and in the treatment and prevention of disease
09/04/2003CA2477224A1 Piperidine ouracil used as a medicament for treating bacterial infections
09/03/2003EP1341403A1 Luminescent element material and luminescent element comprising the same
09/03/2003EP1340744A2 Hiv protease inhibitors
09/03/2003EP1339699A1 Substituted amidoalkyl uracils and the use thereof
09/03/2003EP1339695A1 Farnesyltransferase inhibitors
09/03/2003EP1339692A1 Novel compounds for use as hiv protease inhibitors
09/03/2003EP1339691A1 Novel compounds
09/03/2003EP1339689A1 N-type calcium channel antagonists for the treatment of pain
09/03/2003EP1339683A2 Estrogen receptor modulators
09/03/2003EP1339678A2 Ep4 receptor selective agonists in the treatment of osteoporosis
09/03/2003EP1339677A1 Aminoalkylpyrrolidine serotonin receptor ligands and compositions, their pharmaceutical uses, and methods for their synthesis
09/03/2003EP0993454B1 Benzo(5,6)cyclohepta(1,2b)pyridine derivatives useful for inhibition of farnesyl protein transferase
09/03/2003EP0977741B1 Substituted phenyl derivatives, their preparation and use
09/03/2003EP0977733B1 Arylsulfonylamino hydroxamic acid derivatives
09/03/2003EP0975588B1 Antipicornaviral compouds, compositions containing them, and methods for their use
09/03/2003EP0945445B1 1,5-benzodiazepine derivatives
09/03/2003EP0612318B1 Heteroarylpiperidines, pyrrolidines and piperazines and their use as antipsychotics and analgetics
09/03/2003CN1440404A Benzofuran derivatives and their use as antibacterial agents
09/03/2003CN1440402A N-ureidoheterocycloaklyl-piperidines as modulators of chemokine receptor activity
09/03/2003CN1440401A Amino substituted dibenzothiophene derivatives for treatmnt of disorders mediated by NP Y5 receptor
09/03/2003CN1440400A Bicyelyl or heterobicyclylmethanesulfonylamino-substituted N-hydroxyformamides
09/03/2003CN1440385A Pyrrole derivatives for treating AIDS
09/03/2003CN1439640A Lysotropic-photodiscolour diaryl ethylene and preparation and application thereof
09/03/2003CN1439639A Bipyridine diaryl ethylene compounds and preparation and application thereof
09/03/2003CN1439631A Substituted sulfamide (thio) carbonyl compounds
09/03/2003CN1120155C 2,6-dichloro-4-pyridinemethanol derivatives and agricultural chemicals
09/02/2003US6613942 Glucagon antagonists/inverse agonists
09/02/2003US6613905 Chemokine receptor antagonists and methods of use therefor
09/02/2003US6613888 Azo dyes, process for making the same, ink-jet printing ink, ink-jet recording method
09/02/2003US6613798 Small organic molecule regulators of cell proliferation
09/02/2003US6613795 Respiratory system disorders; muscle relaxants
09/02/2003US6613789 Heterocyclo-substituted imidazoles for the treatment of inflammation
09/02/2003US6613786 Thiophenyl triazol-3-one derivatives as smooth muscle relaxants
09/02/2003US6613781 Potential use in the treatment of a variety of central nervous system disorders such as anxiety, depression, epilepsy, obsessive-compulsive disorders, migraine, congnitive disorders, sleep disorders and schizophrenia
09/02/2003US6613776 Protein serine/threonine kinase inhibitors used for treating diseases such as cancer, diabetes and Alzheimer's disease
09/02/2003US6613773 Pyrimidinyloxyphenyl-3-alkoxypropenoates derivatives
09/02/2003US6613760 Indole derivatives and their use as MCP-1 receptor antagonists
08/2003
08/28/2003WO2003070731A2 Azabicyclic compounds for the treatment of disease
08/28/2003WO2003070726A1 Pyranones useful as atm inhibitors
08/28/2003WO2003070710A1 2-amino-4-bicyclyl amino-6h-1.3.5-triazines, method for the production and use thereof as herbicides and plant growth regulators
08/28/2003WO2003070707A1 Fused pyridazine derivative compounds and drugs containing the compounds as the active ingredient
08/28/2003WO2003070682A1 NON-COVALENT INHIBITORS OF AmpC ß-LACTAMASE
08/28/2003WO2003070673A1 Method for producing 1,2-dichloroethane by direct chlorination
08/28/2003WO2003070244A1 Antagonist of melanin concentrating hormone and their uses
08/28/2003WO2003070242A1 Piperidin-4-yl urea derivatives and related compounds as chemokine receptor inhibitors for the treatment of inflammatory diseases
08/28/2003WO2003028641A3 Mch receptor antagonists
08/28/2003WO2002102359A3 Alkylidene pyrazolidinedione derivatives and use for treating diabetes and obesity
08/28/2003US20030162979 Substituted sulphonylamino(thio)carbonyl compounds
08/28/2003US20030162972 Pyridyl alkane acid amides as cytostatics and immunosupressives
08/28/2003US20030162965 Process for the preparation of 3,7-disubstituted-2,3,4,5-tetrahydro-1H-1,4-benzodiazepine compounds
08/28/2003US20030162964 Benzene-fused heterocycle derivatives and drugs containing the same as the active ingredient
08/28/2003US20030162814 Amines such as 2-(3-(N-hydroxyamidino)phenylamino)-N-(2'-sulfamoylbiphenyl-4-yl)-2 -methylpropionamide, used as anticoagulants or for prophylaxis of arteriosclerosis, angina pectoris, restinosis or metastasis
08/28/2003US20030162811 Heterocyclic amines such as 4-(3'-Thienyl)-alpha, alpha, 1-trimethyl-4-piperidinemethanol and/or prodrugs, used as analgesics for prophylaxis of neuropathic pain
08/28/2003US20030162808 Acetindine derivatives, their preparation and medicaments containing them
08/28/2003US20030162784 Pyridazinone aldose reductase inhibitors
08/28/2003US20030162780 Administering to a patient with a disease treatable with a muscarinic receptor antagonist a 1,2,3,4-tetrahydro-naphthalene-2-yl-alkylaminoalkyl-piperidine derivative
08/28/2003US20030162777 Administering a biheterocyclic compounds containing aminocarbonyl, aminothiocarbonyl or aminosulfonyl group for treating neuromuscular dysfunction of the lower urinary tract in a mammal in need of such treatment
08/28/2003US20030162775 Heterocyclic substituted pyrazolones
08/28/2003US20030162774 Derivatives of sulfonylurea, sulfonylthiourea, sulfonylguanidine, thioacylsufonamide and acylsulfonamide; useful for treating thromobis
08/28/2003US20030162766 Aminomethylene substituted non-aromatic heterocycles and use as substance P antagonists
08/28/2003US20030162764 Pyrimidine A2b selective antagonist compounds, their synthesis and use
08/28/2003US20030162690 Bood anticoagulant
08/28/2003CA2476624A1 Azabicyclic compounds for the treatment of disease
08/28/2003CA2476406A1 Fused pyridazine derivative compounds and drugs containing the compounds as the active ingredient
08/28/2003CA2473100A1 Pyranones useful as atm inhibitors
08/28/2003CA2473089A1 Piperidin-4-yl urea derivatives and related compounds as chemokine receptor inhibitors for the treatment of inflammatory diseases
08/27/2003EP1337529A2 Heterocyclylalkyl piperidine derivatives, their preparation and compositions containing same
08/27/2003EP1337528A2 Benzothiophene derivative compounds, process of preparation and use thereof
08/27/2003EP1337524A1 Substituted quinolines as antitumor agents
08/27/2003EP1337523A2 2,4-substituted pyridine derivatives
08/27/2003EP1337520A1 Substituted 5-aryl and 5-heteroaryl-2-(2-hydroxyphenyl)-2h-benzotriazole derivatives as uv absorbers
08/27/2003EP1337517A1 Pyrimidinone derivatives and their use in the treatment of atherosclerosis
08/27/2003EP1337515A1 (dihydro)isoquinoline derivatives as phosphodiesterase inhibitors
08/27/2003EP1337513A1 4-substituted quinolines as antitumor agents
08/27/2003EP1337510A2 Synthesis and antimicrobial activityof novel dicationic "reversed amidines"
08/27/2003EP1337251A1 Monocyclic or bicyclic carbocycles and heterocycles as factor xa inhibitors
08/27/2003EP1337247A1 Gaba enhancers in the treatment of diseases relating to reduced neurosteroid activity
08/27/2003EP1337150A2 Substituted 4,5-dihydro-1,2,4-triazin-6-ones, 1,2,4-triazin-6-ones, and their use as fungicides and insecticides
08/27/2003EP1140889B1 Compounds and methods for modulation of estrogen receptors
08/27/2003EP1109560B1 Compounds useful as aicarft inhibitors
08/27/2003EP1095039B1 New pharmaceutically active compounds
08/27/2003EP0901469B1 Arylalkylpiperazine compounds as antioxidants
08/27/2003EP0846111B1 Syntheses of optically pure compounds useful as garft inhibitors and their intermediates
08/27/2003CN1439006A Novel compounds possessing antibacterial, antifungal or antitumor activity