Patents
Patents for C07D 409 - Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms (52,226)
01/2004
01/29/2004WO2004009555A1 5-substituted isoquinoline derivative
01/29/2004WO2004009552A1 Phosphodiesterase 4 inhibitors, including n-substituted aniline and diphenylamine analogs
01/29/2004WO2004009551A1 Process for producing 2-substituted pyridine derivative
01/29/2004WO2004009549A2 Piperidines useful for the treatment of central nervous system disorders
01/29/2004WO2004009548A1 1-heterocyclylalkyl-3-sulfonylindole or -indazole derivatives as 5-hydroxytryptamine-6 ligands
01/29/2004WO2004009547A1 Indoline derivatives substituted in position 6, production and use thereof as medicaments
01/29/2004WO2004009546A1 Indoline derivatives substituted in position 6, production and use thereof as medicaments
01/29/2004WO2004009544A1 2-cyano-4-fluoropyrrolidine derivative or its salt
01/29/2004WO2004009543A2 1-carbonyl-4-cyano-pyrrolidine-2-carboxylic acid derivatives as hepatitis c virus inhibitors
01/29/2004WO2003053366A3 Pyrimidine a2b selective antagonist compounds, their synthesis and use
01/29/2004WO2003000180A3 Dipeptidyl peptidase inhibitors for the treatment of diabetes
01/29/2004US20040019216 Copper-catalyzed formation of carbon-heteroatom and carbon-carbon bonds
01/29/2004US20040019208 5-Aryltetrazole Compounds, compositions thereof, and uses therefor
01/29/2004US20040019190 Thrombopoietin mimetics
01/29/2004US20040019106 Cyano and carboxy derivatives of substituted styrenes; inhibitors of tumor necrosis factor alpha, nuclear factor kappa B, and phosphodiesterase
01/29/2004US20040019103 Method of enhancing cellular production of molecular chaperon, hydroxylamine derivatives useful for enhancing the chaperon production and the preparation thereof
01/29/2004US20040019099 Treating inflammatory diseases, allergic conditions and central nervous system disorders
01/29/2004US20040019084 Nitric oxide synthase inhibitors; antioxidant regenerants
01/29/2004US20040019078 Substituted tetrahydroisoquinoline compounds, methods of making, and their use
01/29/2004US20040019065 Indolyl-urea derivatives of thienopyridines useful as antiangiogenic agents, and methods for their use
01/29/2004US20040019050 Selective NPY (Y5) antagonists (triazines)
01/29/2004US20040019039 Substituted piperazines and diazepanes
01/29/2004US20040019038 Compounds useful as anti-inflammatory agents
01/29/2004US20040018956 Aporphine esters and their use in therapy
01/29/2004US20040018192 Integrin expression inhibitors
01/29/2004CA2493721A1 Indoline derivatives substituted in position 6, production and use thereof as medicaments
01/29/2004CA2493458A1 Ureido substituted benzoic acid compounds, their use for nonsense suppression and the treatment of diseases caused by such mutations
01/29/2004CA2493339A1 2-cyano-4-fluoropyrrolidine derivative or salt thereof
01/29/2004CA2493234A1 4-(substituted aryl)-5-hydroxyisoquinolinone derivative
01/29/2004CA2493230A1 5-substituted isoquinoline derivative
01/29/2004CA2492907A1 Phosphodiesterase 4 inhibitors, including n-substituted aniline and diphenylamine analogs
01/29/2004CA2492847A1 5-aryltetrazole compounds, compositions thereof, and uses therefor
01/29/2004CA2491248A1 1-heterocyclylalkyl-3-sulfonylindole or -indazole derivatives as 5-hydroxytryptamine-6 ligands
01/28/2004EP1384713A1 4-amino-azepan-3-one derivatives as protease inhibitors
01/28/2004EP1383761A1 Phenyl- and pyridyl-piperidines with tnf activity
01/28/2004EP1383760A1 Biarylcarboxamide compounds as apolipoprotein b inhibitors
01/28/2004EP1383759A1 Triazole compounds useful in treating diseases associated with unwanted cytokine activity
01/28/2004EP1383757A1 Antagonists of mcp-1 function and methods of use thereof
01/28/2004EP1383751A1 Novel azoles having an insecticidal action
01/28/2004EP1204714B1 Bi-or terthienyl substituted photochromic naphtho 2,1-b]pyran compounds
01/28/2004EP0794947B1 N-substituted hydrazinophenylsulphonyl ureas used as herbicides and plant-growth regulators
01/28/2004CN1471536A Chemokine receptor antagonsis and method of use thereof
01/28/2004CN1471524A Novel farnesyl protein transferase inhibitors as antitumor
01/28/2004CN1471522A Cholesterol lowering benzo [b] thiophenes and benzo[d] isothiazoles
01/28/2004CN1471521A Amino alkoxybenzoyl-benzofuran or benzothiophene derivatives, methods for preparing same and compositions containing same
01/28/2004CN1471520A Aminoalkyl benzoyl-benzofuran or benzothiophene derivatives, method for preparing same and compositions containing same
01/28/2004CN1471519A Amino alkyenylbenzoyl-benzofuran or benzothiophene derivatives, method for preparing same and compositions containing same
01/28/2004CN1470512A Asymmetric diaryl ethylene photochromic compound, and its preparing method and use
01/28/2004CN1136218C Process for preparing 3-(substituted phenyl)-5-(thienyl or fully)-1,2,4-triazoles and novel intermediates utilized therein
01/28/2004CN1136217C 4-aryloxindoles as inhibitor of JNK protein kinases
01/28/2004CN1136213C New benzothiophene, benzofuran and indole compounds, preparation method there for and medicine composition containing them
01/28/2004CN1136198C Novel benzyl pyrimidines
01/28/2004CN1136197C Novel pyridajinone derivatives
01/28/2004CN1136191C Carboxy substituted carboxamide derivatives as tachykinin receptor antagonists
01/27/2004US6683196 Reacting racemic beta-lactam with lithium- 7-protected baccatin iii- complex to form 3'desphenyl-3'-(1-napthyl)taxol; antitumor agents
01/27/2004US6683192 Substituted benzo(b)thien compounds useful for modulating proliferation or differentiation of a cell, agonizes hedgehog mediated signal trasnduction with an ed50 of 1mm or less
01/27/2004US6683191 Preparing a azole compound on a solid support resin, cleaving the compound from the solid support resin by nucleophilic substitution to further substituting by alkylation reaction
01/27/2004US6683108 Agonists of hedgehog signaling pathways and uses related thereto
01/27/2004US6683107 Furans, benzofurans, and thiophenes useful in the treatment of insulin resistance and hyperglycemia
01/27/2004US6683103 Sulfonamides containing oxazole and substituted thiophene rings, useful for treating hypertension, cardiovascular disease, asthma, pulmonary hypertension, inflammatory diseases, vision defects, menstrual disorders, renal failure
01/27/2004US6683093 Enzyme inhibitors; cardiovascular disorders; antiinflammatory agents; autoimmune disease
01/27/2004US6683091 Heterocyclic sulfanamides; alzheimer's disease; preventing deposition of amyloid protein
01/27/2004US6683079 Reverse transcriptase inhibitors
01/27/2004US6683078 Use of sulfonyl aryl or heteroaryl hydroxamic acids and derivatives thereof as aggrecanase inhibitors
01/27/2004US6683074 Cyclic amine derivatives-CCR-3 receptor antagonists
01/27/2004CA2256247C New naphtalene compounds, their preparation and pharmaceutical compositions containing them
01/22/2004WO2004007481A2 Substituted amine derivatives and methods of use in the treatment of angiogenesis relates disorders
01/22/2004WO2004007477A1 Novel thiophene acyl hydrazino derivatives, method for preparing same, use thereof as medicines, pharmaceutical compositions and novel use
01/22/2004WO2004007472A1 Ccr4 antagonist and medicinal use thereof
01/22/2004WO2004007463A1 Cck-1 receptor modulators
01/22/2004WO2004007461A1 8-hydroxy quinoline derivatives
01/22/2004WO2004007459A2 Naphthol, quinoline and isoquinoline-derivatives as modulators of vanilloid vr1 receptor
01/22/2004WO2004007458A1 Substituted 2-alkylamine nicotinic amide derivatives and use there of
01/22/2004WO2004007457A2 Substituted benzylamine derivatives and methods of use
01/22/2004WO2004007449A1 Process for conversion of phenols to carboxamides via the succinimide esters
01/22/2004WO2004006926A1 Sulphonylpiperidine derivatives containing an aryl or heteroaryl group for use as matrix metalloproteinase inhibitors
01/22/2004WO2004006923A1 Aryl piperidine derivatives as inducers of ldl-receptor expression for the treatment of hypercholesterolemia
01/22/2004WO2004006922A1 Aryl piperidine derivatives as inducers of ldl-receptor expression for the treatment of hypercholesterolemia
01/22/2004WO2002092573A3 Heterocyclic substituted pyrazoles as inhibitors of src and other protein kinases
01/22/2004US20040014995 Chromene compounds
01/22/2004US20040014979 For use as antitumor agents
01/22/2004US20040014803 Antilipemic agents; anticholesterol agents; cardiovascular disorders
01/22/2004US20040014802 Aminoindazole derivatives and intermediates, preparation thereof, and pharmaceutical compositions thereof
01/22/2004US20040014801 Thio semicarbazone and semicarbazone inhibitors of cysteine proteases and methods of their use
01/22/2004US20040014798 Skin disorders; hormone replacement therapy
01/22/2004US20040014784 Substituted propargylamines
01/22/2004US20040014783 Antiinflammatory agents; autoimmune diseases; rheumatic diseases; anticholesterol agents; cardiovascular disorders
01/22/2004US20040014775 2,5-substituted pyrimidine derivatives-CCR-3 receptor antagonists
01/22/2004US20040014774 Aryl and heteroaryl quinazoline compounds which inhibit CSF-1R receptor tyrosine kinase
01/22/2004US20040014767 Central nervous system diosrders; antidepressants, anxiolytic agents, anxiolytic agents
01/22/2004US20040014758 Benzylcycloalkyl amines as modulators of chemokine receptor activity
01/22/2004US20040014744 Anticancer, antitumor agents
01/22/2004US20040014740 Compound containing sulfur containing ring; parasiticides
01/22/2004DE10228132A1 Amide cyclischer Aminosäuren als PDE 4 Inhibitoren Amides of cyclic amino acids as PDE 4 inhibitors
01/22/2004CA2492164A1 Substituted benzylamine derivatives and methods of use
01/22/2004CA2492100A1 Substituted 2-alkylamine nicotinic amide derivatives and use there of
01/22/2004CA2492086A1 Sulphonylpiperidine derivatives containing an aryl or heteroaryl group for use as matrix metalloproteinase inhibitors
01/22/2004CA2492045A1 Substituted amine derivatives and methods of use
01/22/2004CA2491213A1 Cck-1 receptor modulators
01/22/2004CA2490468A1 Novel thiophene acyl hydrazino derivatives, method for preparing same, use thereof as medicines, pharmaceutical compositions and novel use