Patents
Patents for C07D 409 - Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms (52,226)
07/2005
07/20/2005CN1642907A Carbonylamino-derivatives as novel inhibitors of histone deacetylase
07/20/2005CN1642580A Radiolabelled quinoline and quinolinone derivatives and their use as metabotropic glutamate receptor ligands
07/20/2005CN1642551A Inhibitors of histone deacetylase
07/20/2005CN1642422A 4-aminopyrimidines and their use for the antimicrobial treatment of surfaces
07/20/2005CN1211373C 2,d-di (hetero-) arylamino (-oxy)-5-substituted pyrimidines as antineoplastic agents
07/20/2005CN1211367C Prostaglandin agonists and their use to treat bone disorders
07/20/2005CN1211362C New benzothiophene, benzofuran and indole compounds, process for their preparation and pharmaceutical compounds containing them
07/20/2005CN1211361C Fused-ring carboxylic acid derivatives
07/19/2005US6919375 Sulfonated amino acid derivatives and metalloproteinase inhibitors containing the same
07/19/2005US6919371 Antidiabetic agents; dietetics; gastrointestinal disorders
07/19/2005US6919367 Substituted thioacetamides
07/19/2005US6919359 Azabicyclic-substituted-heteroaryl compounds for the treatment of disease
07/19/2005US6919356 Antihistamines, antiallergens, autoimmune disease, antiinflammatory agents
07/19/2005US6919355 Amide derivatives as NMDA receptor antagonists
07/19/2005US6919354 1-aryl-or 1-alkylsulfonylbenzazole derivatives as 5-hydroxytryptamine-6 ligands
07/19/2005US6919347 Antidiabetic agents; antiinflammatory agents; analgesics; antiallergens
07/19/2005US6919339 ABCA-1 elevating compounds
07/19/2005US6919338 Antiproliferative agents; anticancer agents
07/14/2005WO2005063739A1 Novel quinoline derivatives
07/14/2005WO2005063734A2 Substituted thiophenes
07/14/2005WO2005063704A1 Azetidine ring compounds and drugs comprising the same
07/14/2005WO2005063241A1 Preventive and/or therapeutic agent for disease in which mitochondrial benzodiazepine receptor participates
07/14/2005WO2005063020A1 Plant growth regulation
07/14/2005WO2005037781A3 Derivatives of n-[heteroaryl(piperidine-2-yl)methyl]benzamide, preparation method thereof and application of same in therapeutics
07/14/2005WO2004108085A3 Methods for the protection of memory and cognition
07/14/2005US20050154229 Salt formation from the free base and maleic acid in the presence of an alcohol solvent to obtain the amorphous salt form, and then recrystallization; thrombin inhibitors with optimal solubility and no deliquescence
07/14/2005US20050154056 Inhibitors of HCV NS5B polymerase
07/14/2005US20050154048 cysteine proteases, cathepsin K; bone metabolic enzymes inhibitor; bone resorption process; anticarcinogenic; 5-[1-(hydroxyimino)ethyl]-2-thiophenecarboxylic acid 2-[[(9H-fluoren-9-yl)methoxy]carbonyl]hydrazide; esterification and coupling with diamine compounds of thiophenecarboxylic acid derivatives
07/14/2005US20050154039 5-Sulphanyl-4h-1,2,4-triazole derivatives and their use as medicine
07/14/2005US20050154038 bicyclo[2.2.2]-oct-1-yl-1,2,4-triazoles; type 2 diabetes, lipid disorders, obesity, atherosclerosis, metabolic syndrome, hyperglycemia, insulin resistance; increase insulin sensitivity in muscle, liver and adipose tissue by correction of the elevated plasma levels of glucose without causing hypoglycemia
07/14/2005US20050154023 1-(4-methoxynaphthalene-1-sulfonyl)-2,3-dihydro-1H-indole-3-carboxylic acid [2-(1-methyl-pyrrolidin-2-yl)-ethyl]amide; selective affinity for 5-HT6 receptor; psychosis, schizophrenia, depression, neurological disorders, cognitive enhancement, Parkinson's disease, ALS, Alzheimer's, Huntington's disease
07/14/2005US20050154019 Substituted cyclic amine metalloprotease inhibitors
07/14/2005US20050154015 Substituted 4H-chromene and analogs as activators of caspases and inducers of apoptosis and the use thereof
07/14/2005US20050154014 Anticarcinogenic agents; antitumor agents treating cancer of breast, head, neck, gastrointestinal system or stomach, ovaries, bronchi, lungs or pancreas; leukemia
07/14/2005US20050154012 Substituted 3-aryl-5-aryl-[1,2,4]-oxadiazoles and analogs as activators of caspases and inducers of apoptosis and the use thereof
07/14/2005US20050154005 Administering to a subject in need of such treatment an effective amount of 1,1'-[1,4-(phenylenebis(methylene))]bis-1,4,8,11-tetraazacyclotetradecane or a pharmaceutical composition thereof, wherein the inhibition of CXCR4 receptor binding effects treatment or amelioration of said condition
07/14/2005US20050153997 Fredericamycin derivatives
07/14/2005US20050153987 Compounds
07/14/2005US20050153986 Psychiatric and mood disorders, Bipolar Disorder, Circadian rhythm disorders, sleep disorders, pain, Parkinson's disease, cognitive dysfunction, epilepsy, obesity, drug addiction, drug abuse, drug withdrawal; side effects reduction; 1-Methyl-3-[3-(5-pyridin-2-yl-2H-tetrazol-2-yl)phenyl]imidazolidin-2-one
07/14/2005US20050153966 2-hydroxy-1H-indol derivatives enzyme inhibitors for preventing or treating inflammation, inflammatory bowel disease, psoriasis, dementia related diseases Alzheimer's Disease, Cognitive Impairment, arthritis, neurodegenerative diseases, amyotrophic lateral sclerosis, Down syndrome, Huntington's Disease
07/14/2005US20050153965 Substituted polycyclic aryl and heteroaryl pyridines useful for selective inhibition of the coagulation cascade
07/14/2005US20050153960 Substituted arylamine derivatives and methods of use
07/14/2005US20050153958 Substituted aryl ketones
07/14/2005US20050153900 Novel inhibitors of hepatitis C virus NS3/NS4a serine protease
07/14/2005US20050151973 Optical device utilizing plasmon resonance
07/14/2005CA2550894A1 Plant growth regulation
07/14/2005CA2550428A1 Substituted thiophenes
07/13/2005EP1553179A1 Mouse-origin proteins forming domain or use thereof
07/13/2005EP1553091A1 Heteroaromatic pentacyclic compound and medicinal use thereof
07/13/2005EP1553085A1 Cyclic amine derivatives and their use as drugs
07/13/2005EP1553084A1 Piperidine derivative, process for producing the same, and use
07/13/2005EP1553074A1 Fused benzene derivative and use
07/13/2005EP1551827A1 Piperidine derivatives as ccr5 inhibitors
07/13/2005EP1551822A2 Pentacyclic oxepines and derivatives thereof, process for their preparation and pharmaceutical compositions containing them
07/13/2005EP1551811A1 Benzimidazole derivatives and their use as vanilloid receptor ligands
07/13/2005EP1551810A1 Diaryl-substituted cyclic urea derivatives having an mch-modulatory effect
07/13/2005EP1551809A1 Pyrazole compounds for treatment of neurodegenerative disorders
07/13/2005EP1551804A1 Substituted 1,4-di-piperidin-4-yl-piperazine derivatives and their use as neurokinin antagonists
07/13/2005EP1551404A2 Method of inhibiting angiogenesis
07/13/2005EP1551397A2 Guanidine compounds as anesthetics and for treatment of nervous system disorders
07/13/2005EP1551384A2 R-nsaid esters and their use
07/13/2005EP1235802B1 Carbamate derivatives having muscarinic receptor antagonist activity
07/13/2005EP1161415B1 N-cyanomethylamides as protease inhibitors
07/13/2005EP1042291B1 Aryl-substituted pyridylalkane, alkene, and alkine carboxamides useful as cytostatic and immunosuppressive agents
07/13/2005CN1639154A Pyranones useful as ATM inhibitors
07/13/2005CN1639146A Fused tricyclic heterocycles useful for treating hyper-proliferative disorders
07/13/2005CN1639145A Benzofuran and benzothiophene derivatives useful in the treatment of hyper-proliferative disorders
07/13/2005CN1639132A N-pyrazinyl-phenylsulphonamides and their use in the treatment of chemokine mediated diseases
07/13/2005CN1639128A O-cyclopropyl-carboxanilides and their use as fungicides
07/13/2005CN1639125A New inhibitors of histone deacetylase
07/13/2005CN1639124A Aminotetralin derivatives as muscarinic receptor antagonists
07/13/2005CN1639123A 4-(phenyl-(piperidin-4-yl)-amino)-benzamide derativatives and their use for the treatment of pain, anxiety or gastrointestinal disorders
07/13/2005CN1639120A Indolamid derivatives which possess glycogenphosphorylase inhibitory activity
07/13/2005CN1639119A Substituted 2-amino-cycloalkanecarboxamides and their use as cysteine protease inhibitors
07/13/2005CN1638810A Near infrared fluorescent contrast agent and method for fluorescence imaging
07/13/2005CN1638776A Substituted 3-aryl-5-aryl-[1, 2, 4]-oxadiazoles and analogs
07/13/2005CN1638763A Antidepressant
07/13/2005CN1638761A Azetidine derivatives as CCR-3 receptor antagonists
07/13/2005CN1637624A Organophotoreceptor with charge transport material having a thiiranyl group
07/13/2005CN1636994A Process of preparing alkali metal salys of hydrophobic sulfonamides and alkali metal salt produced thereby
07/13/2005CN1636986A Benzophenones as inhibitors of reverse transcriptase
07/13/2005CN1636985A Benzophenones as inhibitors of reverse transcriptase
07/13/2005CN1636984A Benzophenones as inhibitors of reverse transcriptase
07/13/2005CN1636565A Modified form of the r(-)-n-(4, 4-di(3-methylthien-2-yl)but-3-enyl)-nipecotic acid hydrochloride
07/13/2005CN1210274C Piperazine and piperidine derivatives
07/13/2005CN1210273C Substituted 3-pyridyl-4-arylpyrroles, and related therapeutic and prophylactic methods
07/13/2005CN1210268C (Cyclo) alkyl substituted-gamma-aminobutyric acid derivatives (=GABA analogurs), their preparation and their use in the treatment of neurolog disorders
07/13/2005CN1210265C Phthalazine derivatives and remedies for erectile dysfunction
07/13/2005CN1210263C N-hydroxy-2-(alkyl, aryl or heteroaryl sulfanyl, sulfinyl or sulfonyl)-3-substituted alkyl, aryl or heteroarylamides as matrix metalloproteinase inhibitors
07/12/2005US6916940 Oxidation, fluorination, desulfurization
07/12/2005US6916931 Tridentate ligands and relative complexes with transition metals
07/12/2005US6916841 Inhibitors of phospholipase enzymes
07/12/2005US6916819 Benzimidazole and pyridylimidazole derivatives
07/12/2005US6916817 Inhibitors of metalloproteinases
07/12/2005US6916813 (1-phenyl-2-heteoaryl)ethyl-guanidine compounds as inhibitors of mitochondrial F1F0 ATP hydrolase
07/12/2005US6916812 Dietetic agents
07/12/2005US6916804 Pyrimidine A2b selective antagonist compounds, their synthesis and use
07/12/2005US6916798 Inhibitors of glycogen synthase kinase-3 (GSK-3), a serine/threonine protein kinase; for treatment and prevention of diabetes and Alzheimer's disease
07/07/2005WO2005061519A1 Kinase inhibitors
07/07/2005WO2005061487A1 Hiv protease inhibiting compounds