Patents for C07D 409 - Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms (52,226) |
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10/26/2005 | EP1129071B1 Phenyl-substituted cyclic enaminones |
10/26/2005 | EP1098870B1 Nitrate salt of Cetirizine |
10/26/2005 | CN1688576A Thiophene compounds |
10/26/2005 | CN1688571A Substituted heterocyclylpyrimidines |
10/26/2005 | CN1688552A Pyrimidine derivatives and their use as CB2 modulators |
10/26/2005 | CN1688550A 2, 5-dioxoimidazolidin-4-yl acetamides and analogues as inhibitors of metalloproteinase MMP12 |
10/26/2005 | CN1688545A Phosphodiesterase 4 inhibitors, including n-substituted phenylamine and diphenylamine analogs |
10/26/2005 | CN1688527A Fused benzene derivative and use |
10/26/2005 | CN1688194A 2, 4, 5-trisubstituted imidazoles and their use as anti-microbial agents |
10/26/2005 | CN1224622C Method for preparing 2-alkyl-3-aminothiophene derivative and 3-aminothiophene derivative |
10/25/2005 | US6958358 Inhibitors of cruzipain and other cysteine proteases |
10/25/2005 | US6958353 Imidazole derivatives or salts thereof and drugs containing the derivatives or the salts |
10/25/2005 | US6958349 Heteroaryl alkylamide derivatives useful as bradykinin receptor modulators |
10/25/2005 | US6958346 4-heteroaryl-tetrahydroquinolines and their use as inhibitors of the cholesterin-ester transfer protein |
10/25/2005 | US6958339 Pyrazole derivative |
10/25/2005 | US6958333 N'-(isoindolino[3,2-b]perhydro-1,3-oxazin-5-on-9-yl)-N-(pyridin-2-yl) urea, for example; cyclin-dependent kinase inhibitors; colon cancer treatment |
10/25/2005 | US6958328 5H-indeno(1,2-b)pyridine-3-carboxylic acid,4-phenyl-2-amino-5-oxo-, ethyl ester; adenosine receptor antagonists, phosphodiesterase inhibitors; neurodegenerative disorders, AIDS; antiinflammatory agent |
10/25/2005 | CA2332461C New benzenesulfonamide derivatives, their method of preparation and the pharmaceutical compositions containing them |
10/25/2005 | CA2304974C 1-substituted-1-aminomethyl-cycloalkane derivatives (=gabapentin analogues), their preparation and their use in the treatment of neurological disorders |
10/25/2005 | CA2261725C Piperidine and piperazine derivatives and their use as muscarinic antagonists |
10/25/2005 | CA2059882C Sulfonylureas |
10/20/2005 | WO2005097791A1 Inhibitors of iap |
10/20/2005 | WO2005097782A1 Piperidine derivative |
10/20/2005 | WO2005097781A1 Quinines-4-substituted derivatives, method and intermediates for the preparation thereof and pharmaceutical compositions containing said derivatives |
10/20/2005 | WO2005097780A1 [4-(5-aminomethyl-2-fluoro-phenyl)-piperidin-1-yl]-(4-bromo-3-methyl-5-propoxy-thiophen-2-yl)-methanone hydrochloride as an inhibitor of mast cell tryptase |
10/20/2005 | WO2005097774A1 Substituted 4-alkyl- and 4-alkanoyl-piperidine derivatives and their use as neurokinin antagonists |
10/20/2005 | WO2005097758A1 Certain triazole-based compounds, compositions, and uses thereof |
10/20/2005 | WO2005097750A1 Substituted pyridones as inhibitors of poly(adp-ribose) polymerase (parp) |
10/20/2005 | WO2005097746A2 2-propene-1-ones as hsp 70 inducers |
10/20/2005 | WO2005097136A1 Biaryl substituted pyrazinones as sodium channel blockers |
10/20/2005 | WO2005097116A1 Composition comprising a jnk inhibitor and cyclosporin |
10/20/2005 | WO2005097107A2 Diphenyl - indol-2-on compounds and their use in the treatment of cancer |
10/20/2005 | WO2005070891A3 Compounds and methods of use |
10/20/2005 | WO2005061450A3 Hiv protease inhibiting sulfonamides |
10/20/2005 | WO2005046590A3 Methods for synthesizing quinolinone compounds |
10/20/2005 | WO2004071460A3 Cyclic derivatives as modulators of chemokine receptor activity |
10/20/2005 | US20050234244 Synthesis of COX-2 and FAAH inhibitors |
10/20/2005 | US20050234238 8-(Biaryl)quinoline pde4 inhibitors |
10/20/2005 | US20050234118 Novel aryllimidazole derivatives, preparation and therapeutic used thereof |
10/20/2005 | US20050234106 1-aryl-1-heteroarylaminoalkylene-substituted, e.g., 1-[fluorophenylcyclohexylmethyl]isoquinolin-1-ylamine; antiarrhythmia agents; cardiovascular disorders |
10/20/2005 | US20050234101 Alkyne compounds with MCH antagonistic activity and medicaments comprising these compounds |
10/20/2005 | US20050234098 antitumor, anticarcinogenic agents; cytotoxic activity and angiogensis inhibitors; leukemia, colorectal cancer; orally |
10/20/2005 | US20050234083 Diamino-pyrimidines and their use as angiogenesis inhibitors |
10/20/2005 | US20050234082 Gonadotropin-releasing hormone receptor antagonists and methods relating thereto |
10/20/2005 | US20050234081 for inhibiting the enzyme C1s, a protease in the classical pathway of the complement system; and the use of this inhibition to treat or ameliorate acute or chronic disorders in mammals |
10/20/2005 | US20050234061 N-[3-(4-chlorophenyl)-2-(3-pyridyl)-1-methylpropyl]-2-(5-trifluoromethyl-2-pyridyloxy)-2-methylpropanamide; obesity; antipsychotic agents; synergistic; cannabinoid receptor antagonists |
10/20/2005 | US20050234057 1-Phenylpiperidin-3-one derivatives and processes for the preparation thereof |
10/20/2005 | US20050234055 Pyrazole derivative |
10/20/2005 | US20050234048 substituted 4,5-dihydro-1H-benzo[b][1,4]-diazepin-2-one; amidation of a substituted monoprotected 1,2-diaminobenzene with an ester, deprotecting, cyclization; chronic neurological disorders, psychosis, schizophrenia, Alzheimer's disease |
10/20/2005 | US20050234044 Cyclic amine derivatives and methods of use |
10/20/2005 | US20050234042 Organic compounds |
10/20/2005 | US20050234030 Modulators of CRTH2, COX-2 and FAAH |
10/20/2005 | CA2567574A1 Benzotriazine inhibitors of kinases |
10/20/2005 | CA2562399A1 Diphenyl - indol-2-on compounds and their use in the treatment of cancer |
10/20/2005 | CA2561967A1 Substituted 4-alkyl- and 4-alkanoyl-piperidine derivatives and their use as neurokinin antagonists |
10/20/2005 | CA2561907A1 Composition comprising a jnk inhibitor and cyclosporin |
10/20/2005 | CA2561280A1 Substituted pyridones as inhibitors of poly(adp-ribose) polymerase (parp) |
10/20/2005 | CA2560954A1 Certain triazole-based compounds, compositions, and uses thereof |
10/20/2005 | CA2560796A1 Biaryl substituted pyrazinones as sodium channel blockers |
10/20/2005 | CA2560649A1 [4-(5-aminomethyl-2-fluoro-phenyl)-piperidin-1-yl]-(4-bromo-3-methyl-5-propoxy-thiophen-2-yl)-methanone hydrochloride as an inhibitor of mast cell tryptase |
10/20/2005 | CA2560162A1 Inhibitors of iap |
10/19/2005 | EP1586571A1 Dipeptidyl peptidase inhibitors |
10/19/2005 | EP1586565A1 Substituted polycyclic aryl and heteroaryl pyrazinones useful for selective inhibition of the coagulation cascade |
10/19/2005 | EP1586564A1 8-azaprostaglandin derivatives and medicinal uses thereof |
10/19/2005 | EP1586559A1 Biaryl-methanethio-, -sulphinyl- and sulphonyl derivatives |
10/19/2005 | EP1585745A1 Fc receptor modulating compounds and compositions |
10/19/2005 | EP1585735A1 Hydroxamid acid derivatives as histone deacetylase (hdac) inhibitors |
10/19/2005 | EP1585728A1 Imino acid derivatives for use as inhibitors of matrix metalloproteinases |
10/19/2005 | EP1585727A1 Indoles useful in the treatment of androgen-receptor related diseases |
10/19/2005 | EP1585521A2 Derivatives of aryl-quinazoline/aryl-2amino-phenyl methanone which promote the release of parathyroid hormone |
10/19/2005 | EP1585517A1 Use of substituted 2-phenylbenzimidazoles as medicaments |
10/19/2005 | EP1463714A4 Vanilloid receptor ligands and their use in treatments |
10/19/2005 | EP1337523B1 2,4-substituted pyridine derivatives |
10/19/2005 | EP1255740B1 Substituted arylpyrazines |
10/19/2005 | EP0966446B1 Bicyclic inhibitors of protein farnesyl transferase |
10/19/2005 | CN1685232A Novel fluorescent label compounds |
10/19/2005 | CN1684960A Delta1 pyrrolines used as pesticides |
10/19/2005 | CN1684957A Substituted thienyl-hydroxamic acids as histone deacetylase inhibitors |
10/19/2005 | CN1684955A Dehydrophenylahistins and analogs thereof and the synthesis of dehydrophenylahistins and analogs thereof |
10/19/2005 | CN1684948A Cytotoxic agents containing novel potent taxanes and their therapeutic use |
10/19/2005 | CN1223593C Preparation process of Leiliqusai |
10/19/2005 | CN1223592C Bipyridine diaryl ethylene compounds and preparation and application thereof |
10/19/2005 | CN1223591C Piperazine oxime derivatives having Nk-1 receptor antagonistic activity |
10/19/2005 | CN1223348C N-(aryloxy group alkyl) heteroaromatic guadine and heteroaromatic guazine used as medicines |
10/18/2005 | US6956052 treatment of cancer and inflammation-associated disorders, such as arthritis; for example,1-[4-(aminosulfonyl)phenyl]-8-{[(trifluoromethyl)sulfonyl]amino}-4,5-dihydro-1H-benzo[g]indazole-3-carboxamide |
10/18/2005 | US6956033 3,4-dihydroisoquinoline derivative compound and a pharmaceutical agent comprising it as active ingredient |
10/18/2005 | CA2329075C Carboxy substituted carboxamide derivatives as tachykinin receptor antagonists |
10/18/2005 | CA2295063C Indole compounds as anti-inflammatory/analgesic agents |
10/18/2005 | CA2294171C N-hydroxyformamide derivatives as inhibitors of matrix metalloproteinases |
10/18/2005 | CA2125730C Novel sulfonylamino pyrimidines |
10/18/2005 | CA2117511C N-cyanoaryl-nitrogen heterocycles |
10/13/2005 | WO2005095440A1 BETA-AMINOACID-DERIVATIVES AS FACTOR Xa INHIBITORS |
10/13/2005 | WO2005095392A1 Silylated carboxamides |
10/13/2005 | WO2005095387A1 Tricyclic pyrazole kinase inhibitors |
10/13/2005 | WO2005095386A1 Substituted thiophene derivatives as anti-cancer agents |
10/13/2005 | WO2005095384A1 Pyrazine derivatives and pharmaceutical use thereof as adenosine antagonists |
10/13/2005 | WO2005095381A1 Dipeptidyl peptidase inhibitors |
10/13/2005 | WO2005095359A1 Diaminopyrimidines as p2x3 and p2x2/3 antagonists |
10/13/2005 | WO2005095357A2 Pyrimidine derivatives and methods of treatment related to the use thereof |
10/13/2005 | WO2005095354A1 Therapeutic agents |