Patents for C07D 409 - Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms (52,226) |
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06/01/2005 | EP1534674A2 Cytotoxic agents containing novel potent taxanes and their therapeutic use |
06/01/2005 | EP1534391A1 Novel piperazinyl-pyrazinone derivatives for the treatment of 5-ht2a receptor-related disorders |
06/01/2005 | EP1534279A2 Prenylation inhibitors containing dimethyl-cyclobutane and methods of their synthesis and use |
06/01/2005 | EP1534277A1 Acylated, heteroaryl-condensed cycloalkenylamines and their use as pharmaceuticals |
06/01/2005 | EP1534276A2 Non-nucleoside reverse transcriptase inhibitors |
06/01/2005 | EP1534275A1 Acylamino-substituted heteroaromatic compounds and their use as pharmaceuticals |
06/01/2005 | EP1534268A2 Tyrosine kinase inhibitors |
06/01/2005 | EP1453820B1 Substituted 6h-dibenzo[c,h]chromenes as estrogenic agents |
06/01/2005 | EP1416936B1 Thiopyrane-4-ones as dna protein kinase inhibitors |
06/01/2005 | EP1254136A4 FACTOR Xa INHIBITORS WITH ARYL-AMIDINES AND DERIVATIVES, AND PRODRUGS THEREOF |
06/01/2005 | EP1095015B1 Sulfonylamino carboxylic acid n-arylamides as guanylate cyclase activators |
06/01/2005 | EP1009758B1 Meta-benzamidine derivatives as serine protease inhibitors |
06/01/2005 | EP0708756B1 Substituted 2-phenylpyridines with herbicidal action |
06/01/2005 | CN1622942A HIV protease inhibitors, compositions containing the same, their pharmaceutical uses and materials for their synthesis |
05/31/2005 | US6900230 Heterocyclo-alkylsulfonyl pyrazoles as anti-inflammatory/analgesic agents |
05/31/2005 | US6900226 Quinoline and quinazoline derivatives; prophylaxis or treatment of arthritis, cardiovascular diseases, diabetes, renal failure and particularly eating disorders and obesity. |
05/31/2005 | US6900214 Cyano-substituted dihydropyrimidine compounds and their use to treat diseases |
05/31/2005 | US6900211 CCR5 antagonists useful for treating aids |
05/31/2005 | US6900210 Pyridinyl, pyrimidinyl and pyrazinyl amides as potassium channel openers |
05/31/2005 | US6900196 Serine protease inhibitors |
05/31/2005 | US6900194 Use of substituted 4-biarylbutyric and 5-biarylpentanoic acid derivatives as matrix metalloprotease inhibitors for the treatment of respiratory diseases |
05/31/2005 | CA2158275C Taxanes having an amino substituted side-chain |
05/26/2005 | WO2005047282A1 Antiresorptive mutual salt of raloxifene and bisphosphonic acid |
05/26/2005 | WO2005047273A1 Thiazole and pyrazole derivatives as flt-3 kinase inhibitors |
05/26/2005 | WO2005047267A1 Process for the synthesis of imidazoles |
05/26/2005 | WO2005047266A1 Aryl imidazoles and their use as anti-cancer agents |
05/26/2005 | WO2005047258A2 Methods and compositions for selectin inhibition |
05/26/2005 | WO2005047257A2 Methods and compositions for selectin inhibition |
05/26/2005 | WO2005047255A1 Substituted nicotinoylcarbamates as pesticides |
05/26/2005 | WO2005047250A1 N-acylated-3- (benzoyl) - pyrrolidines as 11-beta-hsd1 inhibitors useful for the treatment of metabolic disorders. |
05/26/2005 | WO2005047247A1 Novel1,3-disubstituted azetidine derivatives for use as 5ht2a receptor ligands |
05/26/2005 | WO2005047246A1 Novel 1, 3-disubstituted azetidine deivatives for use as 5ht2a receptor ligands |
05/26/2005 | WO2005047244A2 Inhibition of fgfr3 and treatment of multiple myeloma |
05/26/2005 | WO2005046698A1 Fused heterocyclic compounds |
05/26/2005 | WO2005046685A1 Substituted piperidines for the treatment of metabolic syndrome |
05/26/2005 | WO2005046683A1 Amide derivatives as ion-channel ligands and pharmaceutical compositions and methods of using the same |
05/26/2005 | WO2005046604A2 Heteroaryl-hydrazone compounds |
05/26/2005 | WO2005046590A2 Methods for synthesizing quinolinone compounds |
05/26/2005 | WO2005046589A2 Pharmaceutically acceptable salts of quinolinone compounds having improved pharmaceutical properties |
05/26/2005 | WO2005019168A8 Fluorinated lysine derivatives as dipeptidyl peptidase iv inhibitors |
05/26/2005 | WO2004112719A8 Chemical compounds |
05/26/2005 | US20050113566 Inhibitors of C-FMS kinase |
05/26/2005 | US20050113450 method of sterilization, sanitation, antisepsis, and disinfection, includes applying antimicrobial compounds to a surface; e.g. 2-[(3-{[4-chloro(methyl)anilino]sulfonyl}benzoyl)amino]-5-(trifluoromethyl)benzoic acid |
05/26/2005 | US20050113438 Indolecarboxylic acid derivatives as plasminogen activator inhibitor inhibitors; anticoagulant, antiischemic, and anticarcinogenic agents; noninsulin-dependent diabetes, polycystic ovarian syndrome, cardiovascular disorders, atherosclerosis, alzheimer*s disease, chronic obstructive pulmonary disease |
05/26/2005 | US20050113423 Modulators of ATP-binding cassette transporters |
05/26/2005 | US20050113414 1-[1-((E)-1-Cyclooct-1-enyl)methylpiperidin-4-yl]-3-(3,4-dichlorophenyl)-urea; potent and selective modulators of CXCR3, a chemokine receptor; antagonists; treatment of conditions involving inappropriate T-cell trafficking; antiinflammatory, -arthritic agents, autoimmune diseases; antiallergens |
05/26/2005 | US20050113399 Platelet ADP receptor inhibitors; ADP (adenosine 5'-diphosphate); thrombosis; contain thien-2-yl-sulfonylurea groups; 1-(thiophen-2-ylsulfonyl)-3-(4-(7-fluoro-6-(sec or tert-amino)-1-oxo-(3,4-dihydro)isoquinolin-2(1H)-yl)aryl)urea |
05/26/2005 | US20050113396 Na+/H++exchanger-3 (NHE-3) inhibitors; antiischemic agents |
05/26/2005 | US20050113387 Pyrazine derivatives and pharmaceutical use thereof |
05/26/2005 | US20050113383 For therapy of allergy, allergy-induced airway responses, congestion, hypotension, cardiovascular disease, hypotension, diseases of the GI tract, hyper and hypo motility and acidic secretion of the gastrointestinal tract, obesity, sleep |
05/26/2005 | US20050113373 medicine to inhibit proliferative conditions, such as cancer and psoriasis; detecting or identifying a histone deactylase (HDAC) in a biological sample |
05/26/2005 | US20050113369 Small molecule modulators of hepatocyte growth factor (scatter factor) activity |
05/26/2005 | US20050113361 Amide derivatives as NMDA receptor antagonists |
05/26/2005 | US20050113360 NMDA (N-methyl-D-aspartate) receptors; eg 6-(4-benzylpiperidin-1-carbonyl)-1,5-dihydro-oxazolo[4,5-f]indole-2-one |
05/26/2005 | US20050113359 NMDA (N-methyl-D-aspartate) receptors; eg 1-[4-(4-fluoro-benzyl)-piperidin-1-yl]-1-(6-hydroxy-1H-indole-2-yl)methanone |
05/26/2005 | US20050113357 Cholinergic agents such as 3-[3-(4-methoxypiperidine)-1-yl-propyl]-1H-indole; for therapy of cognitive dysfunction, forgetfulness, confusion, memory loss, attention deficits, deficits in visual perception, depression, pain, sleep disorders, and psychosis |
05/26/2005 | US20050113341 Stent with a disposed traiazine compound such as 6-(3-Chloro-4-methoxy-phenoxy)-N-cycloheptyl-N'-methyl-N'-(1-methyl-piperidin-4-yl)-[1,3,5]triazine-2,4-diamine for inhibiting smooth muscle proliferation; restenosis and atherosclerosis |
05/26/2005 | US20050113309 Useful as thrombin inhibitors |
05/26/2005 | US20050112490 Electrophotographic organophotoreceptors with novel charge transport compounds |
05/26/2005 | CA2545742A1 Process for the synthesis of imidazoles |
05/26/2005 | CA2545373A1 Novel 1,3-disubstituted azetidine derivatives for use as 5ht2a receptor ligands |
05/26/2005 | CA2545350A1 Thiazole and pyrazole derivatives as flt-3 kinase inhibitors |
05/26/2005 | CA2545340A1 Fused heterocyclic compounds |
05/26/2005 | CA2545259A1 Heteroaryl-hydrazone compounds |
05/26/2005 | CA2544693A1 Methods and compositions for selectin inhibition |
05/26/2005 | CA2544492A1 Pharmaceutically acceptable salts of quinolinone compounds having improved pharmaceutical properties |
05/26/2005 | CA2544186A1 Inhibition of fgfr3 and treatment of multiple myeloma with benzimidazole quinolinones |
05/26/2005 | CA2543765A1 Methods and compositions for selectin inhibition |
05/26/2005 | CA2541949A1 Amide derivatives as ion-channel ligands and pharmaceutical compositions and methods of using the same |
05/25/2005 | EP1533310A1 Isonipecotamides for the treatment of integrin-mediated disorders |
05/25/2005 | EP1533303A1 Substituted Aminosalicylacid Amides ( intermediates ) |
05/25/2005 | EP1533294A1 Beta-alanine derivative and use thereof |
05/25/2005 | EP1532209A2 Charge transport compositions and electronic devices made with such compositions |
05/25/2005 | EP1532140A1 Thienylhydrazon with digitalis-like properties ( positive inotropic effects ) |
05/25/2005 | EP1532136A1 Pyridazine derivatives as ligands for gaba receptors |
05/25/2005 | EP1532134A1 Novel thiophene acyl hydrazino derivatives, method for preparing same, use thereof as medicines, pharmaceutical compositions and novel use |
05/25/2005 | EP1532128A1 Inhibitors of hcv ns5b polymerase |
05/25/2005 | EP1532120A1 Phenylpyridazine derivatives as ligands for gaba receptors |
05/25/2005 | EP1532118A2 Imidazole compounds for the treatment of hepatitis c virus infections |
05/25/2005 | EP1532113A2 Substituted hihydroquinolines as glucocorticoid mimetics, methods of making them, pharmaceutical compositions, and uses thereof |
05/25/2005 | EP1532111A1 2,5-disubstituted 3-mercaptopentanoic acid |
05/25/2005 | EP1531824A2 Cyclothiocarbamative derivatives as pr modulators and use thereof for treatment of skin disorders |
05/25/2005 | EP1531822A1 1-aryl-4-substituted piperazine derivatives for use as ccr1 antagonists for the treatment of inflammation and immune disorders |
05/25/2005 | EP1531820A1 Anabaseine derivatives useful in the treatment of neurodegenerative diseases |
05/25/2005 | EP1531816A1 Spirocyclic piperidines as mch1 antagonists and uses thereof |
05/25/2005 | EP1531812A1 Fused heteroaryl derivatives for use as p38 kinase inhibitors in the treatment of i.a. rheumatoid arthristis |
05/25/2005 | EP1531811A2 Derivatives of 3-hydroxy-4-(cyclyl-alkylaminoalkyl)-5-phenyl-1h-pyrazole as antagonists of the gonadotropin releasing hormone (gnrh) for use in the treatment of sex hormone related conditions, such as prostatic of uterine cancer |
05/25/2005 | EP1531674A2 2,4,5-trisubstituted imidazoles and their use as anti-microbial agents |
05/25/2005 | EP1341742B1 Method for producing compounds having a cf2o bridge |
05/25/2005 | EP1286673B1 Ligands of integrin receptors |
05/25/2005 | EP1064281B1 Benzoheterocyclic distamycin derivatives, process for preparing them, and their use as antitumor agents |
05/25/2005 | EP1056724B1 Substituted cycloalkyl-4-oxonicotinic carboxamides; gaba brain receptor ligands |
05/25/2005 | EP0946511B1 Novel compounds with analgesic effect |
05/25/2005 | DE10349587A1 Benzimidazolylderivate Benzimidazolylderivate |
05/25/2005 | CN1620452A 3, 4-dihydro-1h-isoquinoloin-2-yl-derivatives |
05/25/2005 | CN1620447A Isochroman compounds for treatment of cns disorders |
05/25/2005 | CN1620439A Pancreatic lipase inhibitor compounds, their synthesis and use |
05/25/2005 | CN1620435A 4-(phenyl-(piperidin-4-yl)-amino)-benzamide derivatives and their use for the treatment of pain, anxiety or gastrointestinal disorders |
05/25/2005 | CN1620434A Pyrrolidine-2-ones as factor Xa inhibitors |
05/25/2005 | CN1620433A Pyrrolidine derivatives as inhibitors of endothelin-converting enzyme |