Patents for C07D 409 - Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms (52,226) |
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08/18/2005 | US20050182061 Phthalimide compounds useful as protein kinase inhibitors |
08/18/2005 | US20050182055 5-Chloro-N-({(5S)-2-oxo-3-[4-(3-oxo-4-morpholinyl)phenyl]-1,3-oxazolidin-5-yl}methyl)-2-thiophenecarboxamide formed by reacting 4-{4-[(5S)-5-(aminomethyl)-2-oxo-1,3-oxazolidin-3-yl]phenyl}-morpholin-3-one hydrochloride with 5-chlorothiophene-2-carbonyl chloride |
08/18/2005 | US20050182048 Paraciticides for use on or in animals, against insects, arachnids and nematodes; 1-(haloalkyl-substituted aryl)-3-cyano-4-alkylthio-5-(alkylthioalkylamino)pyrazoles or S-oxides thereof |
08/18/2005 | US20050179032 Octupolar molecules used as organic semiconductors |
08/18/2005 | US20050179013 Hyperpolarizable organic chromophores |
08/18/2005 | CA2554878A1 Bisarylurea derivatives |
08/18/2005 | CA2554796A1 Modulators of atp-binding cassette transporters |
08/17/2005 | EP1564210A1 4-oxoquinoline compounds and utilization thereof as hiv integrase inhibitors |
08/17/2005 | EP1562939A1 Carboxamides |
08/17/2005 | EP1562933A2 Substituted amine derivatives and methods of use in the treatment of angiogenesis related disorders |
08/17/2005 | EP1562931A2 Anti-infective biaryl compounds |
08/17/2005 | EP1562928A1 Aromatic sulfone hydroxamic acids and their use as protease inhibitors |
08/17/2005 | EP1562911A1 Compositions useful as inhibitors of jak and other protein kinases |
08/17/2005 | EP1562899A2 N-(indole-2-carbonyl)amides as anti-diabetic agents |
08/17/2005 | EP1562895A1 Substituted aryl acylthioureas and related compounds; inhibitors of viral replication |
08/17/2005 | EP1562595A1 Diaryl ethers as opioid receptor antagonists |
08/17/2005 | EP1499594B1 Process for the preparation of 7-substituted-3-quinoline and 3-quinol-4-one carbonitriles |
08/17/2005 | EP1282418B1 Use of pyrazole derivatives for treating infertility |
08/17/2005 | EP1266887B1 Indenoindoline derivatives, their process of preparation and pharmaceutical compositions containing them |
08/17/2005 | EP1202945B1 Methods for preparing perfluorinated [18 f]-radiolabelled nitroimidazole derivatives for cellular hypoxia detection |
08/17/2005 | CN1656089A Phenyl-thiophene type vitamin D receptor modulators |
08/17/2005 | CN1656087A Therapeutic ion channel blocking agents and methods of use thereof |
08/17/2005 | CN1656079A Pyrazole compounds and pharmaceutical compositions comprising the compound |
08/17/2005 | CN1656078A Aminoindazole derivatives as protein kinase inhibitor |
08/17/2005 | CN1656072A Phenyl heterocyclyl ether derivatives as serotonin re-uptake inhibitors |
08/17/2005 | CN1656071A New piperidine derivative |
08/17/2005 | CN1656069A 1-(aminoalkyl)-3-sulfonylindole and-indazole derivatives as 5-hydroxytryptamine-6 ligands |
08/17/2005 | CN1655785A N-acyl piperidine derivatives for use as melanocortin receptor ligands in the treatment of feeding disorders |
08/17/2005 | CN1655779A Substituted benzazoles and methods of their use as inhibitors of Raf kinase |
08/17/2005 | CN1654459A Substituted aminosalicylic acid amides with fungicidal effect and intermediate products for production thereof |
08/17/2005 | CN1215069C Sulfonamicles and derivatives thereof that moulate the activity of endothelin |
08/17/2005 | CN1215067C 哒嗪酮醛糖还原酶抑制剂 Pyridazinone aldose reductase inhibitors |
08/17/2005 | CN1215061C Process for preparing anticancer compound, and intermediate |
08/17/2005 | CN1215059C Novel heterocyclic compounds and salts thereof and medicinal use of same |
08/16/2005 | US6930107 treating obesity, overweight condition, hyperlipidemia, thyroid disease, hypothyroidism, thyroid cancer and related disorders |
08/16/2005 | US6930104 beta -amyloid precursor protein secretory stimulators; treating neurodegenerative disorders; n-carbamoyl- quinoxaline or quinoline derivatives |
08/16/2005 | CA2323707C New substances derived from benzothiophenes, benzofurans and indolics, processes for preparing them and pharmaceutical compounds containing them |
08/11/2005 | WO2005073216A2 Hcv ns-3 serine protease inhibitors |
08/11/2005 | WO2005073206A1 Selective estrogen receptor modulators |
08/11/2005 | WO2005073205A1 Selective estrogen receptor modulators |
08/11/2005 | WO2005073198A1 Heterocyclic sulfonamide inhibitors of beta amyloid production containing an azole |
08/11/2005 | WO2005073197A1 Derivatives of n-` (1,5-diphenyl-1h-pyrazol-3-yl) sulphonamide with cb1 receptor affinity |
08/11/2005 | WO2005073196A1 OPTICALLY ACTIVE QUATERNARY AMMONIUM SALT HAVING AXIAL ASYMMETRY AND PROCESS FOR PRODUCING α-AMINO ACID AND DERIVATIVE THEREOF WITH THE SAME |
08/11/2005 | WO2005073195A2 Hcv ns-3 serine protease inhibitors |
08/11/2005 | WO2005072733A1 Dyarylurea compounds as chk-1 inhibitors |
08/11/2005 | WO2005072681A2 Vanilloid receptor ligands and their use in treatments of inflammatory and neurotic pain. |
08/11/2005 | WO2005053663A3 Norepinephrine reuptake inhibitors useful for treatment of cognitive failure |
08/11/2005 | WO2005007635A3 Combretastatin derivatives with cytotoxic action |
08/11/2005 | US20050177011 ethylene, chlorine, catalyst; solvent is ECD; prevents formation of an interface that promotes side reactions; undissolved gases removed by centrifugal separator |
08/11/2005 | US20050176964 Nicotinamide derivatives useful as p38 inhibitors |
08/11/2005 | US20050176958 Rhodium and iridium complexes |
08/11/2005 | US20050176813 Modulating the potassium ion channel activity of T-cells; autoimmune and inflammatory diseases such as multiple sclerosis, rheumatoid arthritis or transplant rejection; synthesis by reaction of an acetophenone such as khellinone with an aryl aldehyde |
08/11/2005 | US20050176799 drugs such as 1-Benzyl-3-(2-furyl)-5-trifluoromethylpyrazole, capable of modulating biosynthesis of cyclic guanosine monophosphate, used for therapy and prophylaxis of cardiovascular disorders such as hypertension, angina pectoris, cardiac insufficiency, thrombosis or atherosclerosis |
08/11/2005 | US20050176780 2,5-disubstituted 3-mercaptopentanoic acid |
08/11/2005 | US20050176775 Substituted pyridinones |
08/11/2005 | US20050176771 4-fluoro-1-({[1-(methanesulfonyl)piperidin-4-yl]amino}acetyl)pyrrolidine-2-carbonitrile; insulin-dependent diabetes (type 1 diabetes), non insulin-dependent diabetes (type 2 diabetes), insulin-resistant disorders, obesity; dipeptidyl peptidase IV-inhibiting activity |
08/11/2005 | US20050176767 Pyridine carboxamide and methods for inhibiting HIV integrase |
08/11/2005 | US20050176765 For therapy of glaucoma, dementia such as Alzheimer's disease and vascular dementia, depression, attention deficit disorder, sleep disorder, schizophrenia, pain, ischemia; -[1-[1-(3-Thienoyl)piperidin-4-yl]piperidin-4-yl]-1,3-dihydro-2H-benzimidazol-2-one |
08/11/2005 | US20050176762 Tachykinin receptor subtypes NK3 and NK2 (NK neurokinin); various diseases including respiratory system disorders, autoimmune disorders, psychological disorders, skin disorders |
08/11/2005 | US20050176758 2-(hydroxy or methoxymethoxy)-4-(carboxy or alkoxycarbonyl)-5-(fluoro or hydrogen)-7-oxabicyclo(4.1.0)hept-3-ene chemical intermediates to neuraminidase inhibitors |
08/11/2005 | US20050176733 Chk-1 inhibitors |
08/11/2005 | US20050176719 An enzyme inhibitors of cyclin-dependent kinases, antitumor agents; chemical intermediate synthesis |
08/11/2005 | US20050176712 Integrin expression inhibitor |
08/11/2005 | US20050176709 Selective NPY (Y5) antagonists |
08/11/2005 | US20050176708 Piperidine derivatives useful as modulators of chemokine receptor activity |
08/11/2005 | US20050176705 5-Chloro-1-(3,5-dichloro-2-methoxy benzenesulfonyl)-4-piperazin-1-yl-1H-indole trifluoroacetic acid salt; 5-hydroxytryptamine (serotonin) HT6 receptor antagonists; antidepressant, anxiolytic agent, cognition activator; ADHD, Alzheimer's and Parkinson's disease, drug and nicotine abuse |
08/11/2005 | US20050176701 Inhibitors of hepatitis C virus RNA-dependent RNA polymerase, and compositions and treatments using the same |
08/11/2005 | US20050176699 Benzodiazepine derivatives, preparation thereof and use thereof |
08/11/2005 | US20050176698 Neuropeptide Y antagonists |
08/11/2005 | CA2553968A1 Vanilloid receptor ligands and their use in treatments of inflammatory and neuropathic pain |
08/11/2005 | CA2553089A1 Novel piperidines as chemokine modulators (ccr) |
08/11/2005 | CA2553084A1 Novel benzofuran derivative, medicinal composition containing the same, and uses of these |
08/11/2005 | CA2552558A1 Heterocyclic sulfonamide inhibitors of beta amyloid production containing an azole |
08/11/2005 | CA2552317A1 Hcv ns-3 serine protease inhibitors |
08/10/2005 | EP1561749A1 TNF-Alpha production inhibitors for the treatment of autoimmune diseases |
08/10/2005 | EP1560825A1 Novel 2,3-dihydro-4(1h)-pyridinone derivatives, method for production thereof and pharmaceutical composition comprising the same |
08/10/2005 | EP1560817A1 Methods and compositions of novel triazine compounds |
08/10/2005 | EP1560815A1 Novel pyrimidine-4,6-dicarboxamides for the selective inhibition of collagenases |
08/10/2005 | EP1560580A1 Sulfonamides, sulfamates and sulfamides as gamma-secretase inhibitors |
08/10/2005 | EP1392674B1 Furan and thiophene derivatives that activate human peroxisome proliferator activated receptors |
08/10/2005 | EP1368340B1 Piperazine derivatives as melanocortin receptor agonists |
08/10/2005 | EP1194425B1 Substituted benzimidazole |
08/10/2005 | CN1653062A (imidazol-1-yl-methyl)-pyridazine as NMDA receptor blocker |
08/10/2005 | CN1653050A Opioid and opioid-like compounds and uses thereof |
08/10/2005 | CN1653048A Pyridine carboxamide derivatives and their use as pesticides |
08/10/2005 | CN1653047A Monocyclic aroylpyridinones as antiinflammatory agents |
08/10/2005 | CN1653046A 8-azaprostaglandin derivative compounds and drugs containing the compounds as the active ingredient |
08/10/2005 | CN1652779A Treatment of chemokine mediated diseases |
08/10/2005 | CN1652775A Peptide deformylase inhibitors |
08/10/2005 | CN1651430A Synthesis method of saijiabin, its racemate and S-configuration, and preparation method of its amorphous powder |
08/10/2005 | CN1651426A Synthesis method of Gabitril and its racemate and S-configuration |
08/10/2005 | CN1651392A 2-and 2, 5-substituted phenylketoenols |
08/10/2005 | CN1214026C Indol-3-yl derivatives |
08/10/2005 | CN1214017C 四唑衍生物 Tetrazole derivatives |
08/10/2005 | CN1214014C HIV inhibiting pyrimidine derivatives |
08/10/2005 | CN1214007C Cyclopentanoindoles, compositions containing such compounds and methods of treatment |
08/09/2005 | US6927225 Fungicidal 2-pyridyl alkyl amides and their compositions, methods of use and preparation |
08/09/2005 | US6927216 Treatment of inflammatory disorders |
08/09/2005 | CA2105518C Condensed heterocyclic compounds, their production and use |
08/04/2005 | WO2005070920A1 Amino-benzazoles as p2y1 receptor inhibitors |