Patents for C07D 409 - Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms (52,226) |
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12/20/2005 | CA2176962C N-substituted azabicycloheptane derivatives, their preparation and use |
12/20/2005 | CA2114007C Substituted beta-lactam compounds useful as hypocholesterolemic agents and processes for the preparation thereof |
12/15/2005 | WO2005119315A2 Non-linear optically active molecules, their synthesis, and use |
12/15/2005 | WO2005118578A1 Mercaptoimidazoles as ccr2 receptor antagonists |
12/15/2005 | WO2005118575A1 Non nucleoside reverse transcriptase inhibitors |
12/15/2005 | WO2005118556A1 Propane-1,3-dione derivative or its salt |
12/15/2005 | WO2005118547A1 Tetrahydroisoquinoline sulfonamide derivatives, the preparation thereof, and the use of the same in therapeutics |
12/15/2005 | WO2005118543A1 Kinase inhibitor and use thereof |
12/15/2005 | WO2005118537A2 Arylpiperazine derivatives as adrenergic receptor antagonists |
12/15/2005 | WO2005118535A1 Substituted pyrrolidine-2-ones |
12/15/2005 | WO2005117908A2 Triheterocyclic compounds compositions, and methods for treating cancer or viral diseases |
12/15/2005 | WO2005117876A1 Dual small molecule inhibitors of cancer and angiogenesis |
12/15/2005 | WO2005117543A2 N-sulfonylcarboximidamide apoptosis promoters |
12/15/2005 | WO2004098590A8 4-bromo-5- (2-chloro-benzoylamino)-1h-pyrazole-3-carboxylic acid (1-(aminocarbonyl) eth-1-yl) amide derivatives and related compounds as bradykinin b1 receptor antagonists for the treatment of inflammatory diseases |
12/15/2005 | US20050277686 Benzimidazole compounds for regulating IgE |
12/15/2005 | US20050277678 5-(4-Fluorophenyl)-1-(4-methylsulfoximinylphenyl)-3-trifluoromethyl-1H-pyrazole; prostaglandin and cyclooxygenase inhibitor; antiinflammatory, analgesic, and antipyretic agent |
12/15/2005 | US20050277663 3-Aryl-3-hydroxy-and 3-aryl-3-oxopropionic acid esters as fungicides |
12/15/2005 | US20050277652 Hepatocyte growth factor receptor inhibitors; Antitumor agents, anticarcinogenic agents, angiogenesis inhibitors; pyrimidine derivatives like Pyrrolidine-1-carboxylic acid [6-(2-fluoro-4-{3-[2-(4-fluorophenyl)acetyl]thioureido}phenoxy)pyrimidin-4-yl]amide |
12/15/2005 | US20050277646 N-[4-({5-(4-fluorophenyl)-4-[4-(trifluoromethyl)phenyl]pyridin-2-yl}oxy)-1,3-benzothiazol-2-yl]acetamide; vanilloid (capsaicin) receptor antagonist/agonist; antiinflammatory, analgesic, antiarthritis, antirheumatic; diseases involving sensory nerve function |
12/15/2005 | US20050277640 Pyrimidine derivatives for treatment of hyperproliferative disorders |
12/15/2005 | US20050277638 Antagonists of melanin concentrating hormone effects on the melanin concentrating hormone receptor |
12/15/2005 | US20050277637 Arylindenopyridines and related therapeutic and prophylactic methods |
12/15/2005 | US20050277631 Vanilloid receptor ligands and their use in treatments |
12/15/2005 | US20050277628 Substituted thiophene carboxamides |
12/15/2005 | DE102004026026A1 New 2-(hetero)aryl-tetrahydroquinoline derivatives and 1,2,3,4-tetrahydro-1,5-naphthyridine derivatives are mitotic motor protein Eg5 inhibitors used as anticancer agents for treating carcinoma or leukemia |
12/15/2005 | CA2568622A1 Dual small molecule inhibitors of cancer and angiogenesis |
12/15/2005 | CA2567831A1 N-sulfonylcarboximidamide apoptosis promoters |
12/15/2005 | CA2566187A1 Mercaptoimidazoles as ccr2 receptor antagonists |
12/15/2005 | CA2565705A1 Non-linear optically active molecules, their synthesis, and use |
12/15/2005 | CA2565689A1 Substituted pyrrolidine-2-ones |
12/14/2005 | EP1604988A1 Pyridazinone derivatives, methods for producing them and their use as pharmaceuticals |
12/14/2005 | EP1604979A1 2-oxo-1-pyrrolidine derivative and its pharmaceutical uses |
12/14/2005 | EP1603897A1 Pyrazole compounds useful in the treatment of inflammation |
12/14/2005 | EP1603893A1 Ep4 receptor antagonists |
12/14/2005 | EP1603885A1 Fused tri and tetra-cyclic pyrazole kinase inhibitors |
12/14/2005 | EP1603883A2 Quinoline-derived amide modulators of vanilloid vr1 receptor |
12/14/2005 | EP1603881A2 Substituted thiophenes with antibacterial activity |
12/14/2005 | EP1603874A2 G-lactam derivatives as prostaglandin agonists |
12/14/2005 | EP1603572A1 Lactam-containing cyclic diamines and derivatives as factor xa inhibitors |
12/14/2005 | EP1603570A2 Aminoheteroaryl compounds as protein kinase inhibitors |
12/14/2005 | EP1603562A2 Sulfonyl-amidino containing and tetrahydropyrimidino containing compounds as factor xa inhibitors |
12/14/2005 | EP1326858B1 Piperidine compounds as anti-allergic |
12/14/2005 | EP1119562B1 2,3-dihydro-1h-isoindole derivatives useful as modulators of dopamine d3 receptors (antipsychotic agents) |
12/14/2005 | EP1112255B1 4,4-biarylpiperidine derivatives with opioid receptor activity |
12/14/2005 | CN1708496A Cyclopropyl-thienyl-carboxamide as fungicides |
12/14/2005 | CN1708479A Novel compounds useful in treating PPAR mediated diseases |
12/14/2005 | CN1708306A Quinazolinone compounds as calcilytics |
12/14/2005 | CN1706841A 1-(4,4-diaryl-3-butene)-piperidine formic acid or its medicine salt, prepn process and application |
12/14/2005 | CN1231762C Method for directly identifying candidate compound |
12/14/2005 | CN1231476C Substd. pyridine herbicides |
12/14/2005 | CN1231473C Substituted arylpyrazines |
12/14/2005 | CN1231467C High affinity ligands for nociceptin receptor ORL-1 |
12/14/2005 | CN1231465C Biphenylsulfonyl cyanamides, method for the production thereof and their utilization as a medicament |
12/13/2005 | US6974831 sPLA2 inhibitors |
12/13/2005 | US6974827 For use as pesticides and herbicides |
12/13/2005 | US6974813 For therapy of perioperative myocardial ischemic injury in mammals, including humans |
12/13/2005 | US6974810 4,5-Dihydro-1H-pyrazole derivatives having potent CB1-antagonistic activity |
12/13/2005 | CA2250930C 4-[(thien-3-yl)methyl] imidazole derivatives having .alpha.2-adrenoceptor agonistic activity |
12/08/2005 | WO2005117242A1 Method and installation means for installing an electrical machine |
12/08/2005 | WO2005116012A1 Pyrrolidine derivative |
12/08/2005 | WO2005116010A1 Ep4 receptor agonist, compositions and methods thereof |
12/08/2005 | WO2005116009A1 Substituted 2-quinolyl-oxazoles useful as pde4 inhibitors |
12/08/2005 | WO2005115992A1 Theramutein modulators |
12/08/2005 | WO2005115990A1 Cinnamide compound |
12/08/2005 | WO2005115984A2 Large conductance calcium-activitated k channel opener |
12/08/2005 | WO2005115977A1 Pyrrolidine derivatives as cb1-receptor antagonists |
12/08/2005 | WO2005115976A1 3-amino-2-phenylpyrrolidine derivatives |
12/08/2005 | WO2005115975A1 Arylalkylamines and process for production thereof |
12/08/2005 | WO2005115148A1 3-aryl-3-hydroxy-2-methylenepropionic acid esters as fungicides |
12/08/2005 | WO2005115145A2 Quinone substituted quinazoline and quinoline kinase inhibitors |
12/08/2005 | WO2005087724A3 Sulphonylpyrroles as hdac inhibitors |
12/08/2005 | WO2005077932A3 Chemokine receptor antagonists |
12/08/2005 | WO2004099126A8 N-(2-PHENYLETHYL)SULFAMIDE DERIVATIVES AS INTEGRIN α4 ANTAGONISTS |
12/08/2005 | WO2004098589A8 4- bromo - 5 - (2- chloro - benzoylamino) - 1h - pyrazole - 3 - carboxylic acid amide derivatives and related compounds as bradykinin b1 receptor antagonists for the treatment of inflammatory diseases |
12/08/2005 | WO2004093798A3 Quinoxalinyl macrocyclic hepatitis c serine protease inhibitors |
12/08/2005 | US20050272931 Vanilloid receptor ligands and their use in treatments |
12/08/2005 | US20050272803 Phosphodiesterase 4 inhibitors |
12/08/2005 | US20050272791 Lung melanoma metastasis, rheumatoid arthritis, 1-isopropylsulfonyl-2-amino-6-(2-(2,6-difluorophenyl)-5-(phenyl)-imidazol-4-yl)-benzimidazole |
12/08/2005 | US20050272785 Amidobiphenyloxime derivatives, useful as fungicide or bactericide for protection of crops and materials |
12/08/2005 | US20050272780 Small molecule inhibitors of rotamase enzyme activity |
12/08/2005 | US20050272777 Vanilloid receptor ligands and their use in treatments |
12/08/2005 | US20050272753 signal transducer and activator of transcription-6 inhibitors; asthma, COPD, respiratory, inflammatory and allergic diseases; compounds have less suppressive effect on immunological functions; 4-[(2,5 -difluorobenzyl) amino]-2-[(4-morpholin-4-ylphenyl)amino]pyrimidine-5 -carboxamide |
12/08/2005 | US20050272744 N-((4-((( 1R)-3 -(dimethylamino)-1-((phenylsulfanyl)methyl)propyl)amino)-3-nitrophenyl)sulfonyl)-4-(4-(2-fluorobenzyl)-4-methoxy-1-piperidinyl)benzenecarboximidamide; trigger apoptosis through the inhibition of the Bcl family of proteins |
12/08/2005 | US20050272740 Benzimidazole derivatives |
12/08/2005 | US20050272728 Bicyclic-substituted amines having cyclic-substituted monocyclic substituents |
12/08/2005 | US20050272709 tert-butyl-[5-methyl-4-(phenylhydrazono)-4H-pyrazol-3-yl]amine; 4-(3-fluorophenylhydrazono)-5-methyl-2H-pyrazol-3-ylamine; demonstrate anti-proliferative activity, and may promote apoptosis in cells lacking normal regulation of cell cycle and death |
12/08/2005 | US20050272699 1- and 2-substituted with carbo- or heterocyclic groups, e.g., 3-[4-(5-Difluoromethoxy-3-trifluoromethyl-pyrazol-1-yl)-phenyl]-2-(2-fluoro-phenyl)-acrylonitrile; inhibit the production of IL-2. |
12/08/2005 | US20050272663 Novel substituted prolines as inhibitors of hepatitis C virus NS3 serine protease |
12/08/2005 | US20050272036 Ketones |
12/08/2005 | CA2568046A1 3-amino-2-phenylpyrrolidine derivatives |
12/08/2005 | CA2567813A1 Theramutein modulators |
12/08/2005 | CA2566094A1 Cinnamide compound |
12/08/2005 | CA2564668A1 Pyrrolidine derivatives |
12/07/2005 | EP1602656A1 Pyrazole derivatives having affinity for cb1 and/or cb2 receptors |
12/07/2005 | EP1602642A1 Imino ether derivative compounds and drugs containing the compounds as the active ingredient |
12/07/2005 | EP1601664A1 Biaryltetrahydroisoquinoline piperidines as selective mch receptor antagonists for the treatment of obesity and related disorders |
12/07/2005 | EP1601659A1 Pyrimidin-2-one compounds and their use as dopamine d3 receptor ligands |
12/07/2005 | EP1601657A1 Pyrazole modulators of atp-binding cassette transporters |
12/07/2005 | EP1601654A1 Heterocyclic amides, method for the production thereof, substances containing said heterocyclic amides, and use thereof as pesticides |
12/07/2005 | EP1601653A1 Process for the production of substituted nicotinic acid esters |