Patents for C07D 405 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom (69,397) |
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11/07/2006 | US7132420 Aspartic protease inhibitors |
11/07/2006 | US7132417 2-phenyl-1-[4-(2-aminoethoxy)-benzyl]-indoles as estrogenic agents |
11/07/2006 | CA2416879C Methods of treating cancer and the pain associated therewith using endothelin antagonists |
11/07/2006 | CA2274093C Substituted pyrimidinone and pyridinone compounds and their use |
11/07/2006 | CA2200578C N-substituted piperidinyl bicyclic benzoate derivatives |
11/07/2006 | CA2146961C Heterobicyclic sulfonamide and sulfonic ester derivatives |
11/07/2006 | CA2132132C Process for the preparation of 3-arylbenzofuranones |
11/02/2006 | WO2006116713A1 Substituted amide derivatives as protein kinase inhibitors |
11/02/2006 | WO2006115134A1 Novel benzofuran derivative, pharmaceutical composition comprising the same, and use of the derivative or composition |
11/02/2006 | WO2006114966A1 Organic electroluminescent device, display and illuminating device |
11/02/2006 | WO2006114371A1 Novel compounds for treating inflammatory diseases |
11/02/2006 | WO2006114313A1 Pyrazole compounds as prostaglandin receptors ligands |
11/02/2006 | WO2006114272A1 FURAN COMPOUNDS USEFUL AS EPl RECEPTOR ANTAGONISTS |
11/02/2006 | WO2006114260A1 Phenylacetylene derivatives having mglur5 receptor affinity |
11/02/2006 | WO2006114202A1 Method for the production of 5-(4-[4-(5-cyano-3-indolyl)-butyl]-1-piperazinyl)-benzofuran-2-carboxamide |
11/02/2006 | WO2006091428A3 Heteroaryl substituted pyrazinyl-piperazine-piperidines with cxcr3 antagonist activity |
11/02/2006 | WO2006088921A3 Pyrazinyl substituted piperazine-piperidines with cxcr3 antagonist activity |
11/02/2006 | WO2006088919A3 Pyridyl and phenyl substituted piperazine-piperidines with cxcr3 antagonist activity |
11/02/2006 | US20060247448 zearalenone-like macrolides, used to to inhibit nuclear factor kappa-beta (NF- kappa B) activation, as sucnscreen agents and in the treatment of inflammatory or autoimmune disorders and disorders involving malignancy or increased angiogenesis |
11/02/2006 | US20060247442 Process for preparing isatins with control of side-product formation |
11/02/2006 | US20060247439 Mchir antagonists |
11/02/2006 | US20060247305 Chromen-4-one inhibitors of anti-apoptotic Bcl-2 family members and the uses thereof |
11/02/2006 | US20060247295 1,2,9,9a-tetrahydrocyclopropa[c]benz[e]indole-4-one (CBI) with incorporated alkylating domain; in vivo drug-cleavable substrate conjugates that are potent cytotoxins; antiproliferative, anticarcinogenic agent; leukemia; bone marrow and mucosal toxicity; chronic cardiac and neurological toxicity |
11/02/2006 | US20060247290 Derivatives of dioxan-2-alkyl carbamates, preparation thereof and application thereof in therapeutics |
11/02/2006 | US20060247283 5-(3,3-Dichloroprop-2-enyloxy)-2-[4-(2,2-dimethylbenzo[d]1,3-dioxolan-4-yloxy)butoxy]-1,3-dichlorobenzene; acaricides |
11/02/2006 | US20060247280 Non-peptide, reversible inhibitors of type 2 methionine aminopeptidase, useful in treating conditions mediated by angiogenesis, such as cancer, haemangioma, proliferative retinopathy, rheumatoid arthritis, atherosclerotic neovascularization, psoriasis; 3-Benzyl-5-(benzylthio)-1,2,4-triazole |
11/02/2006 | US20060247276 Benzofuranyl alkanamine derivatives and uses thereof |
11/02/2006 | US20060247273 Carbamoyl-type benzofuran derivatives |
11/02/2006 | US20060247262 2,4 Di (hetero) -arylamino-pyrimidine derivatives as ZAP-70 and/or syk inhibitors |
11/02/2006 | US20060247259 Urea derivatives containing aromatic or heteroaromatic rings; 4-(3-chloro-4-(cyclopropylaminocarbonyl)aminophenoxy)-7-methoxy-6-quinolinecarboxamide; prophylactic or therapeutic agent for a disease for which angiogenesis inhibition is effective |
11/02/2006 | US20060247249 Carboximide derivatives as useful uro-selective alpha-1a adrenoceptor blockers |
11/02/2006 | US20060247247 Pyrazole-amine compounds useful as kinase inhibitors |
11/02/2006 | US20060247242 Pesticidal compositions |
11/02/2006 | US20060247241 2,4-Di (phenylamino) pyrimidines useful in the treatment of neoplastic diseases, inflammatory and immune system disorders |
11/02/2006 | US20060247230 chemokines receptor modulators such as 4-(2-ethyl-6-fluoro-3-{1-[3-(4-fluoro-phenylsulfanyl)-propyl]-piperidin-4-yl}-indol-1-yl)-benzoic acid ethyl ester, used for treating inflammatory diseases such as asthma and allergic diseases, autoimmune pathologies such as rheumatoid arthritis and atherosclerosis |
11/02/2006 | US20060247228 Phenylazole compounds production process and antioxidants |
11/02/2006 | US20060247225 e.g. (1 alpha ,5 alpha ,6 alpha )-N-[3-(4-methyl-3-pentenyl)-3-azabicyclo[3.1.0]hex-6-yl]-2-hydroxy-2-cyclopentyl-2-(4-methoxy)phenylacetamide; respiratory, urinary and gastrointestinal systems disorder; antidiabetic agent |
11/02/2006 | US20060247224 Melanocortin receptor ligands |
11/02/2006 | US20060247212 Heterocyclic compounds having inhibitory activity against HIV integrase |
11/02/2006 | EP1717229A1 Novel cyclic compound having 4-pyridylalkylthio group having (un)substituted amino introduced therein |
11/02/2006 | EP1717227A1 Substituted indole compounds, their preparation and use in medicaments |
11/02/2006 | EP1717226A1 2,7-substituted 5-amino-4-hydroxy-8-(1h-indol-5-yl)-octan amide derivatives as renin inhibitors for the treatment of hypertension |
11/02/2006 | EP1717225A1 Bicyclic amide derivatives |
11/02/2006 | EP1717220A2 Vanilloid receptor ligands and their use in treatments |
11/02/2006 | EP1716141A1 Benzopyran derivatives, method of production and use thereof |
11/02/2006 | EP1716140A1 Coupling reactions useful in the preparation of (1h-tetrazol-5-yl)-biphenyl derivatives |
11/02/2006 | EP1716134A1 Amino heterocyclic modulators of chemokine receptor activity |
11/02/2006 | EP1716133A1 2-(piperidin-4-yl)-4,5-dihydro-2h-pyridazin-3-one derivatives as pde4 inhibitors |
11/02/2006 | EP1716130A1 Acetylinic piperazine compounds and their use as metabotropic glutamate receptor antagonists |
11/02/2006 | EP1716122A1 Modulators of atp-binding cassette transporters |
11/02/2006 | EP1716100A2 Therapeutic amide derivatives |
11/02/2006 | EP1715867A1 Bipyridyl amides as modulators of metabotropic glutamate receptor-5 |
11/02/2006 | EP1715862A1 Kinase inhibitors |
11/02/2006 | EP1406620B1 Vinyl phenyl derivatives as glk activators |
11/02/2006 | EP1395568B1 4-aminopyrimidine derivatives |
11/02/2006 | EP1244446B1 Thrombopoietin mimetics |
11/02/2006 | EP1202976B1 Pyrazinones, compositions containing such compounds |
11/02/2006 | EP1194144B1 Antibacterial compounds |
11/02/2006 | EP1192133B1 N-cyclopentyl modulators of chemokine receptor activity |
11/02/2006 | EP1143959B1 Antifungal activity of dicationic molecules |
11/02/2006 | EP1058686B1 2'-fluoronucleosides |
11/02/2006 | EP1003721B1 Benzylidene-1,3-dihydro-indol-2-one derivatives as receptor tyrosine kinase inhibitors, particularly of raf kinases |
11/02/2006 | EP0885883B1 Fused heterocyclic compounds and pharmaceutical applications thereof |
11/02/2006 | EP0821683B1 Benzimidazole compounds and their use as modulators of the gaba a receptor complex |
11/02/2006 | DE102005020331A1 New 5-substituted quinoline and isoquinoline derivatives are glucocorticoid receptor binders useful for treating inflammatory diseases e.g. alveolitis, Sjogren's syndrome, atopic dermatitis, acute lymphatic leukemia, rhinitis and emesis |
11/02/2006 | DE102005019670A1 Preparation of 5-(4-(4-(5-cyano-3-indolyl)-butyl)-1-piperazinyl)-benz ofuran-2-carboxamide, comprises reacting a heterocyclic compound with a carbonitrile compound; and/or converting the obtained benzofuran compound to its salt |
11/02/2006 | DE102005018025A1 New heterocyclic compounds which are cytokine interleukin-8 inhibitors useful for treating e.g., chronic obstructive lung disease, bronchitis, rheumatoid arthritis, psoriasis, gastrointestinal disease and Crohn's disease |
11/02/2006 | CA2605758A1 Process for the preparation of 5-(4-(4-(5-cyano-3-indolyl)butyl)-1-piperaz-lnyl)benzofuran-2-carboxamide |
11/02/2006 | CA2605262A1 Phenylacetylene derivatives having mglur5 receptor affinity |
11/01/2006 | CN1856488A Carbamoyl-type benzofuran derivatives |
11/01/2006 | CN1856478A Bicyclic imino acid derivatives as inhibitors of matrix metalloproteinases |
11/01/2006 | CN1856477A 异喹啉钾通道抑制剂 Isoquinoline potassium channel inhibitors |
11/01/2006 | CN1856474A Isoquinolinone potassium channel inhibitors |
11/01/2006 | CN1856249A Pyridyl pyrimidines for use as pesticides |
11/01/2006 | CN1854135A Heteronuclear compound with dicyandiamide connection and its medicinal use |
11/01/2006 | CN1854134A Piperazine derivatives and their use as serotonin reuptake inhibitors or as neurokinin antagonists |
11/01/2006 | CN1854128A Copper-catalyzed formation of carbon-heteroatom and carbon-carbon bonds |
11/01/2006 | CN1853630A Heteropolycyclic compounds and their use as metabotropic glutamate receptor antagonists |
10/31/2006 | US7129359 for treating infection by enterovirus of the Picornaviridae family ; exemplified by: 1-[2-(4'-Chloro-biphenyl-4-yloxymethyl)-benzyl]-3-pyridin-4-yl-imidazolidin-2-one |
10/31/2006 | US7129350 Coupling process and intermediates useful for preparing cephalosporins |
10/31/2006 | US7129261 Cytotoxic agents |
10/31/2006 | US7129260 Isoindolinone kinase inhibitors |
10/31/2006 | US7129255 Substituted 2-carba-3,5-dicyano-4-aryl-6-aminopyridines and the use of the same as selective ligands of the adenosine receptor |
10/31/2006 | US7129254 highly active active agents from the structural class of the epothilones and epothilone derivatives with suitable linkers; to link these epothilone-linker conjugates to recognition units, such as, for example, monoclonal antibodies or fragments thereof, to form immune conjugates |
10/31/2006 | US7129253 Compounds |
10/31/2006 | US7129247 Aryl phenylheterocyclyl sulfide derivatives and their use as cell adhesion-inhibiting anti-inflammatory and immune-suppressive agents |
10/31/2006 | US7129245 Anticoagulants which act selectively on factor Xa; fast acting; oral; do not interfere with lysis of blood clots |
10/31/2006 | US7129242 Such as 4-((4-chlorophenyl)pyrimidin-2-yl)amino)benzamide; for treatment of inflammation/autoimmune conditions |
10/31/2006 | US7129240 1,3-dihydro-2H-indol-2one derivatives, process for preparing them and pharmaceutical compositions containing them |
10/31/2006 | US7129236 For therapy of immune related responses, tumor growth, glomerulonephritis, inflammation, malarial anemia, septic shock, tumor associated angiogenesis, vitreoretinopathy, psoriasis, graft versus host disease, atopic dermatitis |
10/31/2006 | US7129235 Amides useful for treating pain |
10/31/2006 | US7129228 Heterocyclic analgesic compounds and methods of use thereof |
10/31/2006 | CA2355886C Substituted oximes and hydrazones as neurokinin antagonists |
10/31/2006 | CA2276455C Phthalazinones |
10/31/2006 | CA2276310C Process for the production of tetrazolylbenzopyrans |
10/31/2006 | CA2191759C Formylaminophenylsulfonylureas, preparation processes and use as herbicides and plant growth regulators |
10/26/2006 | WO2006113864A2 Oxindole compounds and their uses as therapeutic agents |
10/26/2006 | WO2006113704A2 Subtituted heteroaryl cb1 antagonists |
10/26/2006 | WO2006112479A1 Nitrogen-containing heterocyclic compound |
10/26/2006 | WO2006112442A1 Benzimidazole compound |