Patents
Patents for C07D 405 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom (69,397)
10/2006
10/26/2006WO2006111858A2 Bis-(coumarin) compounds with anti-inflammatory activity
10/26/2006WO2006111662A2 4h-1,2,4-triazin-5-one derivatives, their preparation and their use as alpha 7 nicotinic acetylcholine receptors
10/26/2006WO2006111371A1 Pharmaceutically active diazepanes
10/26/2006WO2006094237A3 Acridine and quinoline dervatives as sirtuin modulators
10/26/2006WO2006090268A3 Processes for the preparation of alfuzosin and salts thereof and novel crystalline forms of alfuzosin
10/26/2006WO2006083271A3 Substituted aryl acylthioureas and related compounds; inhibitors of viral replication
10/26/2006WO2006036941A3 Specific kinase inhibitors
10/26/2006WO2005105778A3 4-amino-5-cyanopyrimidine derivatives
10/26/2006WO2005095384A8 Pyrazine derivatives and pharmaceutical use thereof as adenosine antagonists
10/26/2006US20060241259 for photopolymerization; photography, relief imaging; color filters
10/26/2006US20060241171 Novel physiologically active substances
10/26/2006US20060241168 administering a protein kinase B activating agent comprising (R)-5,6-dimethoxy-2-[2,2,4,6,7-pentamethyl-3-(4-methylphenyl)-2,3-dihydro-1-benzofuran-5-yl]isoindoline; treating depression, posttraumatic stress disorder, Parkinson's disease, Alzheimer's diseases
10/26/2006US20060241155 TNF-alpha production inhibitors
10/26/2006US20060241147 Pyridine derivatives useful for inhibiting sodium/calcium exchange system
10/26/2006US20060241146 2-cyano-1-[t-4-(4-acetyl-1-piperazinyl)-1-methyl-r-1-cyclohexylamino]acetylpyrrolidine; dipeptidylpeptidase IV (DPPIV) inhibitor; antidiabetic, insulin resistance, hyperglycemia, obesity; antiproliferative agent for T-cell, HIV, AIDS; arthritis, osteoporosis
10/26/2006US20060241137 Triazole compounds and the therapeutic use thereof
10/26/2006US20060241126 Phospholipase inhibitors perticularly phospholipase A2 enzyme Lipoprotein Associated Phospholipase A2; N-(1-Methylpiperidin-4-yl)-(2-(2-(2,3-difluorophenyl)ethyl)-4-oxo-4H-pyrido[2,3-d]pyrimidin-1-yl)-N-(4-(4-trifluoromethylphenyl)phenyl)methylacetamide; amidation
10/26/2006US20060241123 Substituted piperidine and piperazine derivatives as melanocortin-4 receptor modulators
10/26/2006US20060241119 Thio-substituted tricyclic and bicyclic aromatic methanesulfinyl derivatives
10/26/2006US20060241115 2,3-Dihydro-4H-1,4-benzoxazine derivatives containing an optionally fused pyridine or pyrimidine ring; 7-((6,7-bis(methyloxy)-4-quinolinyl)oxy)-N-phenyl-2,3-dihydro-4H-1,4-benzoxazine-4-carboxamide; kinase inhibitors; inflammation, angiogenesis and cancer
10/26/2006US20060241111 inhibitors of coagulation factor Xa such as 1-(5-chlorothien-2-ylcarbonyl)-4-[4-(3-oxomorpholin-4-yl)phenyl]-2-propylsemicarbazide, used for preventing thrombosis, infarction, arteriosclerosis, inflammation, bleeding, angina pectoris, restenosis, intermittent claudication and treatment of tumors
10/26/2006US20060241110 2-(Imidazol-1-ylalkyl)-3H-quinazolin-4-one derivatives; mitotic kinesin KSP inhibitors; anticarcinogenic, antiinflammatory, and antiproliferative agents
10/26/2006US20060241105 To control arthropods (including insects and arachnids) and helminths (including nematodes) also valuable to protect timber from sawflies, beetles or termites or use in veterinary medicine; 1-(2,6-Dichloro-4-trifluoromethylphenyl)-3-(N-benzyloxy-2-amidino)-5-methylamino-4-trifluoromethylsulfonylpyrazole
10/26/2006US20060241103 Inhibiting polymerization of FtsZ in a bacterium by contactng with 2,3-diphenyl-6-(ethoxycarbonylamino)-8-(4-(diethylamino)-1-methylbutylamino)pyrido[2,3-b]pyrazine, optionally linked to a permeability enhancer to allow the compound to cross the bacterium's cell envelope
10/26/2006US20060240048 Pyridine derivatives as cb2 receptor modulators
10/26/2006US20060239927 Drug for airway administration
10/26/2006DE102005018026A1 New substituted styrol stereoisomers are glucocorticoid receptor ligands useful for the treatment of e.g. inflammatory diseases, lung diseases, rheumatic diseases, autoimmune diseases, joint disorders and gastrointestinal disorders
10/26/2006CA2610446A1 Nitrogen-containing heterocyclic compound
10/26/2006CA2606288A1 Subtituted heteroaryl cb1 antagonists
10/26/2006CA2605059A1 Oxindole compounds and their uses as therapeutic agents
10/26/2006CA2604920A1 Novel compounds useful for bradykinin b1 receptor antagonism
10/26/2006CA2602610A1 Benzimidazole compound
10/26/2006CA2601979A1 2,3 substituted pyrazine sulfonamides
10/26/2006CA2600774A1 Pharmaceutically active diazepanes
10/25/2006EP1713823A2 Hcv ns-3 serine protease inhibitors
10/25/2006EP1713822A2 Hcv ns-3 serine protease inhibitors
10/25/2006EP1713797A1 1-ISOPROPYL-2-OXO-1,2-DIHYDROPYRIDINE-3-CARBOXAMIDE DERIVATIVES HAVING 5-HT sb 4 /sb RECEPTOR AGONISTIC ACTIVITY
10/25/2006EP1713796A1 Process for preparing substituted benzopyran compounds
10/25/2006EP1713790A2 Method of preparation of benzofuran-2-carboxylic acid (s)-3-methyl-1- ((4s, 7r)-7methyl-3-oxo-1-(pyridine-2-sulfonyl)-az epan-4-ylcarbamoyl-butyl)-amide
10/25/2006EP1713782A1 Pth agonists
10/25/2006EP1713780A2 Novel inhibitors of glutaminyl cyclase
10/25/2006EP1713778A1 Benzazepine derivatives as histamine h3 antagonists
10/25/2006EP1713484A2 Compounds and methods of use
10/25/2006EP1590346B1 4- {'3-(sulfonylamino) phenyl] '1-(cyclymethyl) piperidin-4-ylidene] methyl} benazmide derivatives as delta opioid receptor ligands for the treatment of pain, anxiety and functional gastrointestinal disorder
10/25/2006EP1554272B1 Benzimidazoles and benzothiazoles as inhibitors of map kinase
10/25/2006EP1409525B1 Human papillomavirus e2 transactivation domain/inhibitor co-crystal and x-ray coordinates defining the inhibitor-binding pocket
10/25/2006EP1265606B1 Cell adhesion inhibitors
10/25/2006EP1089998B1 Epothilone derivatives and their synthesis and use
10/25/2006EP1016866B1 Novel compound 2-amino-3-[2-(alpha-mannopyranosyl) indol-3-yl] propionic acid, process for preparing the same, and method for inspecting function of living body with the novel compound
10/25/2006CN1852906A Novel compounds
10/25/2006CN1852905A N-substituted benzimidazolyl c-kit inhibitors
10/25/2006CN1852900A 2,4-di (phenylamino) pyrimidines useful in the treatment of proliferative disorders
10/25/2006CN1852897A Gabanergic modulators
10/25/2006CN1852896A Quinoline and quinazoline derivatives having affinity for 5HT1-type receptors
10/25/2006CN1852710A Pyrazolines as PAR-1 antagonists for treatment of cardiovascular diseases
10/25/2006CN1850820A Coumarin derivatives, and their preparing method and use as alpha, receptor agonist
10/25/2006CN1281604C Substituted pyrazole compounds
10/25/2006CN1281598C Compounds and methods for modulation of estrogen receptors
10/25/2006CN1281597C New compounds, which are potent inhibitors of Na<+>/Ca<2+> exchange mechanism and are useful in the treatment of arrhythmias
10/25/2006CN1281585C Cyclic diamine compounds having fused-ring groups
10/24/2006US7126012 Has affinity for melatonin receptors and/or selectivity for melatoninergic receptors; antiinflammatory and anticarcinogic agents
10/24/2006US7126010 Benzylcycloalkyl amines as modulators of chemokine receptor activity
10/24/2006US7125997 Differential tumor cytotoxicity compounds and compositions
10/24/2006US7125996 Fluorescent probes for use in protein kinase inhibitor binding assay
10/24/2006US7125995 Substituted amidoalkyl uracils and their use as inhibitors of the poly(adp-ribose) synthetase (PARS)
10/24/2006US7125994 PNA monomer and precursor
10/24/2006US7125904 Cardiovascular disorders; hypotensive agents; congestive heart failure
10/24/2006US7125898 Kinase inhibitors to mediate disease and as antiinflammatory agents
10/24/2006US7125895 Arylalkylamine compounds as chemokine receptor antagonists for therapy and prevention of diseases such as arthritis or rheumatic diseases
10/24/2006US7125893 Compounds useful for treatment of tumors or cancer of the stomach, colon, neck or used in angiogenesis and forming the compound with cyclization
10/24/2006US7125892 Aryl aniline β2 adrenergic receptor agonists
10/24/2006US7125887 Pyrrolidine modulators of CCR5 chemokine receptor activity
10/24/2006US7125883 alpha v beta 3 integrin receptor modulators; treating variety of diseases including cardiovascular disorders, retinopathy, strokes, cancer, osteoporosis, tumor metastasis, high blood pressure, psoriasis, antiviral, antimycotic, antiparasitic or antibacterial therapy; 1,2-dihydropyrimidin-2-one moiety
10/24/2006US7125881 Use of pyrimidine—or triazine—2 carbonitiles for treating diseases associated with cysteine prostease activity and novel pyrimidine-2-carbonitile derivatives
10/24/2006US7125879 Prevention reproduction of virus
10/24/2006US7125877 Brain disorders; psychological disorders; central nervous system disorders; antidiabetic agents; hypotensive agents
10/24/2006CA2261848C Cell adhesion inhibitors
10/24/2006CA2249402C Benzopyran derivatives having leukotriene-antagonistic action
10/24/2006CA2246678C Substituted 2-aryl-1,2,4-triazine-3,5-di(thi)ones as herbicides
10/24/2006CA2223094C Phenylpyridazinones
10/24/2006CA2214752C Herbicidal or fungicidal sulphonylaminocarbonyltriazolinones with halogenated alk(en)oxy substituents
10/24/2006CA2211411C Sulphonyl amino(thio)carbonyl-1,2,4-triazolin(thi)one derivatives, the production thereof and the use thereof as herbicides
10/24/2006CA2195663C Dihydrobenzofuranes
10/24/2006CA2168023C Vasoconstrictive substituted aryloxyalkyl diamines
10/19/2006WO2006110804A2 Synthesis of nitrodibenzylfuran chromophore for photodeprotection of organic molecules
10/19/2006WO2006110476A2 Cytotoxic compounds and conjugates comprising duocarmycins with cleavable substrates
10/19/2006WO2006109846A1 Triazole derivative and the use thereof
10/19/2006WO2006109084A1 Dna-pk inhibitors
10/19/2006WO2006109081A1 Dna-pk inhibitors
10/19/2006WO2006108837A1 Aminoalkyl-amidomethyl-substituted 2- (4-sulphonylamino) -3-hydroxy-3 , 4-dihydro-2h-cromen-6-yl derivatives and their use as potassium channel blockers
10/19/2006WO2006108791A2 Heterocyclylethylheterocyclylcarboxamide derivatives as fungicides
10/19/2006WO2006108699A1 Indazoles as glucocorticoid receptor ligands
10/19/2006WO2006108591A1 1h-quinaz0line-2,4-diones and their use as ampa-receptor ligands
10/19/2006WO2006050476A3 Pyrimidine derivatives as ion channel modulators and methods of use
10/19/2006WO2005103041A3 Treatment of cns disorders using cns target modulators
10/19/2006US20060235225 Having a diffraction peak at a diffraction angle (2 theta +-0.2 degrees ) of 12.8 degrees, 18.1 degrees and/or 23.5 degrees in a powder X-ray diffraction; stable against exposure to light
10/19/2006US20060235222 Indole-derivative modulators of steroid hormone nuclear receptors
10/19/2006US20060235054 e.g. 3-substituted 5-(4-fluorophenyl)-4-(4-pyridyl)imidazole-2-thione; immunomodulating and cytokine-release-inhibiting action; antiinflammatory agent
10/19/2006US20060235032 Substituted quinazolines as antiviral agents, especially against cytomegaloviruses
10/19/2006US20060235024 Acetylinic piperazine compounds and their use as metabotropic glutamate receptor antagonists