Patents
Patents for C07D 405 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom (69,397)
02/2007
02/08/2007WO2007016292A2 Heterocyclic amides as biofilm modulators
02/08/2007WO2007015588A1 Piperidine derivative as tachykinin receptor antagonist
02/08/2007WO2007015412A1 Heterocyclic compound and organic electroluminescent device using same
02/08/2007WO2007015262A2 A process for the preparation of (-)-trans-4-(p-fluorophenyl)-3-[[3,4-(methylenedioxy)phenoxy]methyl)]piperidine
02/08/2007WO2007015162A1 Piperidinoyl-pyrrolidine and piperidinoyl-piperidine compounds
02/08/2007WO2007014885A1 Antibacterial quinoline derivatives
02/08/2007WO2007014851A2 Indol-3-yl-carbonyl-piperidin and piperazin derivatives
02/08/2007WO2007014619A1 Novelimidazolecarboxamide derivatives as fructose-1,6-bisphosphatase inhibitors, and pharmaceutical compositions comprising same
02/08/2007WO2007014412A1 Method for isolating 5-substituted tetrazoles
02/08/2007WO2006113704A3 Subtituted heteroaryl cb1 antagonists
02/08/2007WO2006071775A3 Novel compounds useful for bradykinin b1 receptor antagonism
02/08/2007WO2006045119A3 Improved inhibitors for the soluble epoxide hydrolase
02/08/2007US20070032664 Making intermediates such as ((4R,6R)-6-{2-[2-(4-fluorophenyl)-5-isopropyl-3-phenyl-4-phenylcarbamoyl-pyrrol-1-yl]-ethyl}-2-phenyl-[1,3]dioxan-4-yl)-acetic acid methyl ester for the synthesis of calcium atorvastatin (Lipitor(reg))
02/08/2007US20070032663 Intermediate in the synthesis of calcium atorvastatin (Lipitor(reg)) comprising an amine salt of a carboxylic acid, for example 2-(morpholinocarbonyl)ethylamine, phenylacetic acid salt
02/08/2007US20070032662 Novel process for the synthesis of 5-(4-fluorophenyl)-1-[2-((2R,4R-4-hydroxy-6-oxo-tetrahydro-pyran-2-yl)-ethyl]-2-isopropyl-4-phenyl-1H-pyrole-3-carboxylic acid and phenylamide
02/08/2007US20070032653 N-{1-(4-(3-bromophenyl)-1H-imidazol-2-yl)-5-methylhexyl}-N-cyclohexylamine; agonists or antagonists of somatostatin receptors; acromegaly, restenosis, Crohn's disease, systemic sclerosis, external and internal pancreatic pseudocysts and ascites, nesidoblastosis, hyperinsulinism, gastrinoma, etc.
02/08/2007US20070032541 monocyte chemotactic proteins (MCP)-1 receptor antagonist or agonist; 2-{1-[(1,2-cis)-2-(4-Methylsulfanyl-benzoylamino)-cyclohexyl]-2-oxo-pyrrolidin-3-ylcarbamoyl}-4-trifluoromethyl-phenyl)-carbamic acid tert-butyl ester; antiinflammatory agent, antiallergen; asthma, rheumatoid arthritis, atherosclerosis
02/08/2007US20070032526 Cyclic amide derivative as monocyte chemotactic protein modulator; prevention and treatment of rheumatoid arthritis, multiple sclerosis, atherosclerosis and asthma; antiinflammatory agents
02/08/2007US20070032525 e.g. (1H-benzoimidazol-2-yl)-[1-(3,4-dichloro-benzyl)-piperidin-4-ylmethyl]-amine; chemokine (C-C motif) receptor antagonist; antiallergen; asthma and allergic rhinitis, atopic dermatitis, urticaria, contact dermatitis, alleriric coniunctivitis, inflammatory bowel disease, AIDS, eosinqphilia
02/08/2007US20070032509 New capped pyrazinoylguanidine sodium channel blockers
02/08/2007US20070032497 Fused-ring compounds and use thereof as drugs
02/08/2007US20070032490 N-Phenyl-'(4-pyridyl)-azinyl!amine derivatives as plant protection agents
02/08/2007US20070032489 Substituted pyridones as inhibitors of poly(adp-ribose) polymerase (parp)
02/08/2007US20070032486 5Ht4-antagonistic 4-(aminomethyl)-piperidine benzamides
02/08/2007CA2617654A1 Piperidinoyl-pyrrolidine and piperidinoyl-piperidine compounds
02/08/2007CA2617282A1 Novel imidazolecarboxamide derivatives as fructose-1,6-bisphosphatase inhibitors, and pharmaceutical compositions comprising same
02/08/2007CA2616937A1 Indol-3-yl-carbonyl-piperidin and piperazin derivatives
02/08/2007CA2616510A1 Cycloalkyl amino-hydantoin compounds and use thereof for .beta.-secretase modulation
02/08/2007CA2615574A1 Multicyclic sulfonamide compounds as inhibitors of histone deacetylase for the treatment of disease
02/08/2007CA2614981A1 Antibacterial quinoline derivatives
02/07/2007EP1749817A1 Neurogenic pain control agent composition
02/07/2007EP1749002A1 Pyrrole or imidazole amides for treating obesity
02/07/2007EP1749001A1 3-piperidinylisochroman-5-ols as dopamine agonists
02/07/2007EP1749000A2 Bicyclic, substituted triazoles as modulators of ppar and methods of their preparation
02/07/2007EP1748995A1 Arylsulfonyl benzodioxanes useful for modulation the 5-ht6 receptor, the 5-ht2areceptor or both
02/07/2007EP1748991A1 Morpholinylanilinoquinazo- line derivatives for use as antiviral agents
02/07/2007EP1748989A2 Aryl sulfonamides
02/07/2007EP1748987A2 2-propene-1-ones as hsp 70 inducers
02/07/2007EP1748984A1 Piperidine derivatives as nk1 and nk3 antagonists
02/07/2007EP1748980A1 Pyrrolidine derivatives as cb1-receptor antagonists
02/07/2007EP1656348B1 Acetylene derivatives as inhibitors of histone deacetylase
02/07/2007EP1606255A4 Cyclic derivatives as modulators of chemokine receptor activity
02/07/2007EP1501504B1 1-substituted imidazole derivatives as nos inhibitors
02/07/2007EP1017680B1 Tricyclic compounds, preparation method and said method intermediates, application as medicines and pharmaceutical compositions containing same
02/07/2007EP0998474B1 Piperazine derivatives
02/07/2007CN1910176A Crystalline polymorph of a bisulfate salt of a thrombin receptor antagonist
02/07/2007CN1910175A 组织蛋白酶半胱氨酸蛋白酶抑制剂 Cathepsin cystatin
02/07/2007CN1910159A 2,4-diaminopyrimidines and their use for inducing cardiomyogenesis
02/07/2007CN1910151A Cyclic amine derivative with heteroaryl ring
02/07/2007CN1909909A 1-benzyl-5-piperazin-1-yl-3,4-dihydro-1H- quinazolin-2-one derivatives and the respective 1H-benzo(1,2,6)thiadiazine-2,2-dioxide and 1,4-dihydro-benzene as modulators of the 5-hydroxytryptamine recept
02/07/2007CN1909907A Quinoline derivatives and use thereof as mycobacterial inhibitors
02/07/2007CN1907985A N,N-dimethylaminoacyl-2,3-difuryl-6-aminoquinoxaline, preparation method and application thereof
02/07/2007CN1907984A Compound for preparing intermediate for synthesis of atorvastatin calcium
02/07/2007CN1907982A New compounds useful for the treatment of obesity,type II diabetes and CNS disorders
02/07/2007CN1298715C Non-imidazole compounds as histamine H3 antagonists
02/07/2007CN1298714C Process to produce 4-hydroxy-2-oxo-pyrone derivates useful as protease inhibitors
02/07/2007CN1298711C Processes for producing epoxytriazole derivative and intermediate therefor
02/07/2007CN1298705C Novel piperidine-4-sulfamide compound, its preparing method and medicinal composition containing them
02/06/2007US7173136 3-Cyano-quinoline derivatives
02/06/2007US7173135 Substituted 3-cyanoquinolines as MEK inhibitors
02/06/2007US7173134 retinoid X receptors ("RXRs"); useful for the treatment of diabetes (NIDDIM) and obesity; for example, 3-{4-[(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-2-naphthalenyl)methyl]-2-furyl}-2-propenoic acid
02/06/2007US7173133 cCs-rac-4-phenyl-8-(2-phenyl-cyclohexyl)-2,8-diaza-spiro[4.5]decan-1-one; treating diseases related to activation of NMDA receptors via Glyt-1 inhibition
02/06/2007US7173129 Sulfonamide-substituted chalcone derivatives and their use to treat diseases
02/06/2007US7173128 Benzoxazinone, oxanilide, benzylidene malonate, quinazoline and benzotriazole derivatives; polymer and photographic stabilizers
02/06/2007US7173054 Respiratory syncytial virus replication inhibitors
02/06/2007US7173042 Quinoline inhibitors of cGMP phosphodiesterase
02/06/2007US7173040 4-phenyl-6-alpha-(imidazolyl-, 1,2,4-triazolyl- or pyridyl)-benzyl substituted
02/06/2007US7173039 Compounds that modulate or inhibit enzymes for occular diseases
02/06/2007US7173036 Therapeutic treatment of diabetes with a 4-[piperazine-1-yl]-1,2-dihydro-quinolines; treating tumor growth, glomerulonephritis, inflammation, malarial anemia, septic shock, tumor associated angiogenesis, vitreoretinopathy, psoriasis, graft versus host disease, atopic dermatitis
02/06/2007US7173034 Drugs for treatment of viral diseases such as Respiratory syncytial virus
02/06/2007US7173032 Antiproliferative agents for smooth muscle cells; antiinflammatory agents for endothelial cells; restenosis, atherosclerosis
02/06/2007US7173028 Pyrimidine derivatives
02/06/2007CA2214320C Novel taxoids, preparation thereof, and pharmaceutical compositions containing same
02/01/2007WO2007014198A1 1, 2, 3 -triazoles inhibitors of tubulin polymerization for the treatment of poliferative disorders
02/01/2007WO2007013694A1 Phenoxyalkanoic acid compound
02/01/2007WO2007013421A1 Novel nitrogenated heterocyclic compound
02/01/2007WO2007012900A1 Quinoline derivatives as neurokinin receptor antagonists
02/01/2007WO2006129120A3 Benzotriazepinone derivatives
02/01/2007WO2005112919A3 Self-immolative linkers and drug conjugates
02/01/2007WO2005090329A9 New compounds for the inhibition of angiogenesis and use of thereof
02/01/2007US20070027321 Bipyridyl amines and ethers as modulators of metabotropic glutamate receptor-5
02/01/2007US20070027310 Novel ligands and methods for preparing same
02/01/2007US20070027196 Activator of peroxisome proliferator-activated receptor delta
02/01/2007US20070027190 Antibacterial fab i inhibitors
02/01/2007US20070027185 inhibitor of factor Xa and/or thrombin; anticoagulantsto treat thromboembolic disorders, myocardial ischemia, myocardial infarction and cerebral thrombosis; N-(5-chloropyridin-2-yl)-3-[2-(piperidin-4-yloxy)-4-(pyrrolidin-1-yl)benzoylamino]pyridine-4-carboxamide; high bioavailability; acylation
02/01/2007US20070027174 Phenylalanine Enamide Derivatives
02/01/2007US20070027170 Process for preparing amino crotonyl compounds
02/01/2007US20070027162 Crystalline and amorphous 4-cyano-N-{(2R)-2-[4-(2,3-dihydro-benzo[1,4]dioxin-5-yl)-piperazin -1-yl]-propyl}-N-pyridin-2-yl-benzamide hydrochloride
02/01/2007US20070027159 Therapeutic agents useful for treating pain
02/01/2007US20070027158 High affinity small molecule C5a receptor modulators
02/01/2007US20070027126 E.g., N-[4-(5-cyano-1-methyl-1H-pyrrol-2-yl)phenyl]propane-1-sulfonamide and tert-butyl 2-cyano-5-{4-{(ethylsulfonyl)amino]phenyl}-1H-pyrrole-1-carboxylate; useful for contraception and hormone replacement therapy
02/01/2007US20070027125 Cyanopyrrole-phenyl progesterone receptor modulators and uses thereof
02/01/2007DE102005035395A1 Preparation of optically active 2,3-diarylepoxide compounds comprises epoxidizing diaryl compounds and optionally separating the obtained enantiomeric mixture
02/01/2007DE102005034264A1 4-Chromenonyl-1,4-dihydropyridincarbonitrile und ihre Verwendung 4-Chromenonyl-1,4-dihydropyridincarbonitrile and their use
02/01/2007CA2616547A1 Quinoline derivatives as neurokinin receptor antagonists
02/01/2007CA2614919A1 1, 2, 3 -triazoles inhibitors of tubulin polymerization for the treatment of proliferative disorders
01/2007
01/31/2007EP1748045A1 Light-emitting device material and light-emitting device
01/31/2007EP1747210A1 3- or 4-monosubstituted phenol and thiophenol derivatives useful as h3 ligands
01/31/2007EP1747206A1 Amino-tetrazoles analogues and methods of use
01/31/2007EP1747204A1 Tri-substituted ureas as cytokine inhibitors