Patents
Patents for C07D 405 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom (69,397)
09/2006
09/13/2006CN1274675C Novel cyclobutene diketone compound and its producing process, and pharmaceutical composition containing the same compound
09/12/2006US7105682 Substituted amine derivatives and methods of use
09/12/2006US7105671 2-Substituted phenyl,3-polar ring,N-heroaromatic propion-amides, e.g., 1-(2-(3,4-Dichlorophenyl)-3-(tetrahydro-furan-2-yl)-propionyl)-3- methylurea; antidiabetic agents; increase the flux of glucose metabolism in beta-cells and hepatocytes
09/12/2006US7105669 Quinazoline derivatives
09/12/2006US7105668 Methods and compositions utilizing quinazolinones
09/12/2006US7105563 5-ureido-3-[(4-(3-methoxyphenyl)pyrrol-2-yl)methylene]indolin-2-one and derivatives; inhibition of phosphoinositide-dependent kinase-1 (PDK-1).
09/12/2006US7105549 Aryl substituted pyridines and the use thereof
09/12/2006US7105544 N-{3-[1-(3-{[BIS(4-FLUOROPHENYL)ACETYL]AMINO}PROPYL)-4-PIPERIDINYL]PHENYL}-2-METHYLPROPANAMIDE; antagonists for melanin concentrating hormone-1 (MCH1) receptors; treating depression, anxiety, obesity
09/12/2006US7105543 4-, 5-, 6- and 7-indole derivatives useful for the treatment of CNS disorders
09/12/2006US7105542 Chromone compound; also viricide, antiinflammatory agents
09/12/2006US7105537 For enhancing bone formation; for therapy of diseases or disorders associated with abnormal bone or mineral homeostasis
09/12/2006US7105529 A novel compound for treating alopecia induced by cancer chemotherapy or radiotherapy
09/12/2006US7105527 such as beta-D-N4-p-bromobenzoyl-2',3'-didehydro-2',3'-dideoxy-5-fluorocytidine; for treating human immunodeficiency virus (HIV) and hepatitis B virus (HBV) infections
09/12/2006US7105526 Benzimidazole derivatives
09/12/2006US7105522 Aids therapy; viricides
09/12/2006US7105519 Inhibitors of macrophage migration inhibitory factor and methods for identifying the same
09/12/2006US7105513 Cardiovascular disorders; strokes; hypotensive agents
09/12/2006US7105509 Benzodiazepine derivatives as APP modulators
09/12/2006US7105507 Cyclohexane derivatives and their use as therapeutic agents
09/12/2006US7105505 Benzimidazole derivatives useful as histamine H3 antagonists
09/12/2006US7105503 Pyrazole compounds
09/12/2006US7105482 Administering {(3R, 4S, 5S, 6R)-5-Methoxy-4-[(2R, 3R)-2-methyl-3-(3-methyl-but-2-enyl)-oxiranyl]-1-oxa-spiro[2.5]oct-6-yloxycarbonylamino}-3-methyl-butyric acid methyl ester; parasitic infections, thymoma, and lymphoid malignancies; prevents the metabolic degradation of the angiogenesis inhibitor
09/12/2006US7105471 Arylphenyl-substituted cyclic ketoenols
09/12/2006CA2315110C Pellets having a core coated with an antifungal and a polymer
09/12/2006CA2235986C Inhibitors of protein isoprenyl transferases
09/12/2006CA2140929C Hydroxyethylamino sulfonamides useful as retroviral protease inhibitors
09/11/2006CA2500676A1 Preparation of acid addition salts of amine bases by solid phase-gas phase reactions
09/08/2006WO2006094237A2 Acridine and quinoline dervatives as sirtuin modulators
09/08/2006WO2006093853A1 Crystalline and amorphous 4-cyano-n{(2r)-2-[4-(2,3-dihydro-benzo[1,4]dioxin-5-yl)-piperazin-1-yl]-propyl}-n-pyridin-2-yl-benzamide hydrochloride
09/08/2006WO2006093339A1 Use of cinnamoyl compound
09/08/2006WO2006093336A1 Use of cinnamoyl compound
09/08/2006WO2006092731A1 1, 2, 4-triazole derivatives and their use as oxytocin antagonists
09/08/2006WO2006092599A2 Pyrrole derivatives as dna gyrase and topoisomerase inhibitors
09/08/2006WO2006092493A1 $g(b) crystalline form of ivabradine hydrochloride, preparation method thereof and pharmaceutical compositions containing same
09/08/2006WO2006092037A1 Process for producing atorvastatin hemicalcium
09/08/2006WO2005086700A3 Hiv integrase inhibitors
09/08/2006CA2600933A1 Amide derivatives as ion-channel ligands and pharmaceutical compositions and methods of using the same
09/08/2006CA2600287A1 Use of cinnamoyl compound
09/08/2006CA2599992A1 Acridine and quinoline dervatives as sirtuin modulators
09/08/2006CA2599588A1 Crystalline and amorphous 4-cyano-n{(2r)-2-[4-(2,3-dihydro-benzo[1,4]dioxin-5-yl)-piperazin-1-yl]-propyl}-n-pyridin-2-yl-benzamide hydrochloride
09/07/2006US20060199966 Indol-2-amides as glycogen phosphorylase inhibitors
09/07/2006US20060199964 preparation of 6-haloalkyl-3-nicotinic acid esters and also to novel enamine intermediates
09/07/2006US20060199827 Inhibitors of macrophage migration inhibitory factor and methods for identifying the same
09/07/2006US20060199825 4-Aminating a 4-chloro-2-hydroxy-3-nitrodihydroquinoline with a N-(hetero)cyclylpiperazine, and alkylating the remaining amine group in the quinoline ring to produce a 4-(4-(hetero)cyclylpiperazinyl)-3-nitro-1-alkyldihydroquinolinone
09/07/2006US20060199822 Bis-sulfonamide hydroxyethylamino retroviral protease inhibitors
09/07/2006US20060199821 Heterocyclic amides and sulfonamides
09/07/2006US20060199818 Inhibiting the activity of a 5-hydroxytryptamine 2A by administering a N-heterocyclyl (preferably 1,3-dioxan-5-yl)-4-[(N-substituted)(hetero)arylamino]piperidine in which the N-substituant is arylalkanoyl, arylthioalkanoyl, arylalkylaminocarbonyl or arylalkylaminothiocarbonyl group
09/07/2006US20060199789 medical composition
09/07/2006DE102005010000A1 Indane Indanes
09/06/2006EP1698628A1 Hydroxypyrimidinone derivative having hiv integrase inhibitory activity
09/06/2006EP1698627A1 Pyrazole compounds useful as protein kinase inhibitors
09/06/2006EP1698626A1 Amidopyrazole derivative
09/06/2006EP1698620A1 Benzene compounds disubstituted with cyclic groups at the 1- and 2-positions
09/06/2006EP1698375A1 Azetidine ring compounds and drugs comprising the same
09/06/2006EP1697375A2 Heterocyclic protein kinase inhibitors and uses thereof
09/06/2006EP1697352A2 4-azole substituted imidazole compositions useful as inhibitors or c-met receptor tyrosine kinase
09/06/2006EP1697351A1 2,6-bisheteroaryl-4-aminopyrimidines as adenosine receptor antagonists
09/06/2006EP1697350A1 Tricyclic steroid hormone nuclear receptor modulators
09/06/2006EP1697349A1 Doxepin analogs and methods of use thereof
09/06/2006EP1697348A1 Hiv protease inhibiting compounds
09/06/2006EP1697347A1 5- or 6-substituted benzimidazole derivatives as inhibitors of respiratiory syncytial virus replication
09/06/2006EP1697343A1 Aminobenzimidazoles and benzimidazoles as inhibitors of respiratory syncytial virus replication
09/06/2006EP1697327A1 Insecticidal spiroindane derivatives
09/06/2006EP1697312A2 Hydroxamic acid esters and pharmaceutical use thereof
09/06/2006EP1697307A1 Opioid receptor antagonists
09/06/2006EP1696931A2 Amino substituted diaryl [a,d]cycloheptene analogs as muscarinic agonists and methods of treatment of neuropsychiatric disorders
09/06/2006EP1696924A1 Acidic quinoline derivatives and their use for the prevention and/or treatment of hyperglycaemia-related pathologies
09/06/2006EP1696915A1 Benzenesulfonylamino-pyridin-2-yl derivatives and related compounds as inhibitors of 11-beta-hydroxysteroid dehydrogenase type 1 (11-beta-hsd-1) for the treatment of diabetes and obesity
09/06/2006EP1562935B1 Heteroaryloxy-substituted phenylaminopyrimidines as rho-kinase inhibitors
09/06/2006EP1455579B1 Pyrazoles-pyrimidine fungicides
09/06/2006EP1406609B1 Substituted aryl compounds as novel cyclooxygenase-2 selective inhibitors, compositions and methods of use
09/06/2006EP1223933B1 5-membered heterocycle derivatives and use thereof as monoaminoxidase inhibitors
09/06/2006EP1135374B1 Benzimidazole compounds that are vitronectin receptor antagonists
09/06/2006CN1829711A Novel heterocyclic compounds useful for the treatment of inflammatory and allergic disorders: process for their preparation and pharmaceutical compositions containing them
09/06/2006CN1829709A Bicyclic imidazol derivatives against flaviviridae
09/06/2006CN1829701A Piperazine derivatives and their use as therapeutic agents
09/06/2006CN1829698A Pyridazine derivatives and their use as therapeutic agents
09/06/2006CN1829695A Aminoquinoline derivatives and their use as adenosine A3 ligands
09/06/2006CN1829688A Process and intermediate compounds useful in the preparation of statins, particularly atorvastatin
09/06/2006CN1829516A S 2-'4(phenylamino)-piperidin-1-yl!-n-phenyl-acetamine derivatives and related compounds as neuropeptide y5 (npy5) ligands for the treatement of obesity
09/06/2006CN1829512A Medicinal composition containing triazole compound
09/06/2006CN1829507A 酪氨酸激酶抑制剂 Tyrosine kinase inhibitor
09/06/2006CN1829506A Novel coumarin-amide derivatives and its preparation, its drug composition and use
09/06/2006CN1827617A Antivirus use of 17-(tetrahydrofuryl-2'-yl) methyl amine-17-demethoxy geldanamycin
09/06/2006CN1827616A Synthesis and uses of indole analogs of 1-benzyl-3-(5'-hydroxymethy 1-2' -furyl) indazole
09/06/2006CN1827600A Crystalline form beta of the chlorhydrate of ivabradine, process for its preparation and pharamcetuical composition containing it
09/06/2006CN1827108A Use of cytosine derivative for preparing drug for treating cancer
09/06/2006CN1273468C One step preparation method of paluxitin hydrochloride A crystal type crystal molecule assembly
09/06/2006CN1273467C Beta-lactam compounds, process for producing the same and serum cholesterol-lowering agents containing the same
09/06/2006CN1273454C New pyrimidine-2,4,6-trione derivatives, processes for their production and pharmaceutical agents containing these compounds
09/06/2006CN1273451C Piperidine MCH antagonists and their use in treatment of obesity
09/06/2006CN1273450C 1-aryl-or 1-alkylsulfonylbenzazole derivatives as 5-hydroxytryptamine-6ligands
09/06/2006CN1273444C Dipeptide nitriles
09/05/2006USRE39265 Heteroarylpiperidines, and their use as antipsychotics and analgetics
09/05/2006USRE39263 2-2-fluoro-5-ethylsulphonylamino-4-thiocarbamoyl-phenyl)-5,6,7,8-tetrahydro-1,2,4triazolo[4,3-a]pyridin-3(2H)-one; post or preemergent
09/05/2006US7102009 For treating cancer and angiogenesis-related disorders
09/05/2006US7102008 Hydantoin derivatives as inhibitors of matrix metalloproteinases and/or TNF-α converting enzyme
09/05/2006US7101902 2-guanidinylimidazolidinedione compounds and methods of making and using thereof
09/05/2006US7101898 Amides of aminoalkyl-substituted azetidines, pyrrolidines, piperidines and azepanes
09/05/2006US7101896 Pharmaceutical compositions and methods for use