Patents
Patents for C07D 405 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom (69,397)
05/2009
05/06/2009CN101426486A Compounds for the treatment of inflammatory disorders and microbial diseases
05/06/2009CN101423497A 6-amino-1H-indazole and 4-aminobenzofuran compounds as phosphodiesterase 4 inhibitors
05/06/2009CN101423491A Acenaphtho-heterocycles compounds and application thereof in preparation of BH3 analogue Bcl-2 family protein inhibitor
05/06/2009CN101423489A Indoline-2-one derivates and uses thereof
05/06/2009CN101423481A Diketohydrazine derivative compound and medicine containing the compound as active ingredient
05/05/2009US7528258 Trityl olmesartan medoxomil is reacted with an acid in a water miscible organic solvent, separating the precipitate of triphenyl carbinol from the solution of olmesartan medoxomil; solution of olmesartan medoxomil is treated with a base to obtain a precipitate of olmesartan medoxomil
05/05/2009US7528167 Inhibitors of papilloma virus
05/05/2009US7528165 Treatment of peroxisome proliferation activated receptor diseases such as diabetes, skin disorders or high blood pressure
05/05/2009US7528157 EP4 receptor antagonists
05/05/2009US7528137 Compounds, compositions, and methods
05/05/2009US7528134 Acetamides and benzamides that are useful in treating sexual dysfunction
05/05/2009CA2513549C Capture compounds, collections thereof and methods for analyzing the proteome and complex compositions
05/05/2009CA2386230C Modulators of cytokine mediated signalling pathways and integrin .alpha.v.beta.3 receptor antagonists for combination therapy
05/05/2009CA2322953C Pyridine derivative and pharmaceutical containing the same
04/2009
04/30/2009WO2009055519A1 Synthesis of quaternary salt compounds
04/30/2009WO2009055516A1 Synthesis of quaternary salt compounds
04/30/2009WO2009054984A1 Heterocycle phenyl amide t-type calcium channel antagonists
04/30/2009WO2009025839A3 Phosphodiesterase 10 inhibitors
04/30/2009WO2009015037A3 5-pyridinone substituted indazoles
04/30/2009WO2009012482A3 5-membered heterocyclic amides and related compounds
04/30/2009WO2008141119A3 Modulators of cftr
04/30/2009WO2008140553A4 Mapk/erk kinase inhibitors
04/30/2009WO2008126106A8 Novel and improved processes for the preparation of intermediates of darifenacin, darifenacin and its pharmaceutically acceptable salts
04/30/2009US20090111992 Alkyl ether derivatives or salts thereof
04/30/2009US20090111986 Novel crystals of pyrimidine compound and process for producing the same
04/30/2009US20090111809 Inhibitors of 11-beta-hydroxysteroid dehydrogenase 1
04/30/2009US20090111151 Production of Polyketides
04/30/2009US20090110662 Modification of biological targeting groups for the treatment of cancer
04/30/2009CA2704040A1 Synthesis of quaternary salt compounds
04/30/2009CA2703717A1 Synthesis of quaternary salt compounds
04/30/2009CA2702126A1 Heterocycle amide t-type calcium channel antagonists
04/30/2009CA2701594A1 Heterocycle phenyl amide t-type calcium channel antagonists
04/30/2009CA2701292A1 Process for making thienopyrimidine compounds
04/29/2009EP2053041A2 1,3,5-Trisubstituted 2(1H)-pyridones as AMPA receptor inhibitors useful for the treatment of eg Parkinson's disease
04/29/2009EP1828127A4 INSECTICIDAL BIS(SUBSTITUTED PHENYL)-1-äÝ4-(SATURATED HETEROCYCLYL-SUBSTITUTED)PHENYLMETHYL¨-(4-PIPERIDYL)üMETHANE DERIVATIVES
04/29/2009EP1786475B1 1,4-bis(carboxymethyl)-6-[bis(carboxymethyl)amino]-6-methyl-perhydro-1,4-diazepine (aazta) derivatives as ligands in high relaxivity contrast agents for use in magnetic resonance imaging (mri)
04/29/2009EP1765812B1 Contrast agents endowed with high relaxivity for use in magnetic resonance imaging (mri) which contain a chelating moiety with polyhydroxylated substituents
04/29/2009EP1670769B1 Benzimidazole derivatives, compositions containing them, preparation thereof and uses thereof
04/29/2009EP1651592B1 Novel dibenzo[b,f]oxepine-10-carboxamides and pharmaceutical uses thereof
04/29/2009EP1446379B1 Aryl aniline beta-2 adrenergic receptor agonists
04/29/2009EP1345910B1 Quinazoline derivatives, medicaments containing said compounds, their utilization and method for the production thereof
04/29/2009CN101421624A Methods for detecting substances which bind to the amyloid precursor protein or beta amyloid fragments, and binding compounds
04/29/2009CN101421258A Sulfonyl-substituted bicyclic compounds as modulators of ppar
04/29/2009CN101421250A 4-aryl-2-amino-pyrimidines or 4-aryl-2-aminoalkyl-pyrimidines as jak-2 modulators and pharmaceutical compositions containing them
04/29/2009CN101421240A Aminomethyl pyridine derivatives, method for preparing same and therapeutic use thereof
04/29/2009CN100482659C Benzimidazolone compounds having 5-HT4 receptor agonistic activity
04/29/2009CN100482229C Substituted 1-piperidin-3-yl-4-piperidin-4-yl-piperazine derivatives and their use as neurokinin antagonists
04/28/2009USRE40703 N-(2-aminophenyl)-4-(N-benzoylaminomethyl)benzamide hydrochloride; differentiation-inducing activity, for malignant tumors, autoimmune diseases, dermatologic diseases and parasitism, hematologic malignancy, a solid carcinoma
04/28/2009US7524959 Biphenyl-2-ylcarbamic acid 1-[2-(2-chloro-4-{[(R)-2-hydroxy-2-(8-hydroxy-2-oxo-1,2-dihydroquinolin-5-yl)ethylamino]methyl}-5-methoxyphenyl-carbamoyl)ethyl]piperidin-4-yl ester; beta 2 adrenergic receptor agonist and muscarinic receptor antagonist; bronchodilator agent; pulmonary disorders, asthma
04/28/2009US7524957 Compounds effecting glucokinase
04/28/2009US7524883 Eponemycin and epoxomicin analogs and uses thereof
04/28/2009US7524874 Vanilloid receptor ligands and their use in treatments
04/28/2009US7524873 Substituted N-phenylmethyl ethanamines; N-((6-(methyloxy)-4'-(trifluoromethyl)-1,1'-biphenyl-3-yl)methyl)-1-(1-naphthalenyl)ethanamine; parathyroid hormone inhibitors; antisecretory agents; osteoporosis
04/28/2009US7524869 Taxanes having a C10 ester substituent
04/28/2009US7524864 Methods of treating sleep disorders
04/28/2009US7524862 Melanin-concentrating hormone (MCH); for the treatment of metabolic disorders and/or eating disorders, such as obesity and diabetes, also drug dependencies, and urinary incontinence
04/28/2009US7524861 Process for the preparation of a hydrate of an anthranilic acid derivative
04/28/2009US7524855 (4-Chloro-2-{[4-(2,4-diamino-pyrimidin-5-ylmethyl)-6,7-dimethoxy-benzofuran-2-ylmethyl]-amino}-phenyl)-pyrrolidin-1-yl-methanone; dihydrofolate reductase; bactericide; grampositive (Staphylococcus aureusand, Enterococcus faecalis) and and gramnegative pathogens (Escherichia coli, Haemophilus influenzae)
04/28/2009US7524854 Trimethoprim derivative; 5-[6,7-Dimethoxy-2-(7-methoxy-1H-indol-3-ylmethyl)-benzofuran-4-ylmethyl]-pyrimidine-2,4-diamine; potent activity against dihydrofolate reductase, mutated enzyme; superior bioavailability, antibacterial activity; gram positive and negative pathogens
04/28/2009US7524849 5-arylpyrimidines as anticancer agents
04/28/2009US7524848 Diaza heterocyclic amide compounds and their uses
04/28/2009US7524846 heterocylcyclic amines used for treating or preventing conditions ameliorated by monoamine reuptake such as vasomotor symptoms, sexual dysfunction, gastrointestinal and genitourinary disorders, chronic fatigue syndrome, fibromylagia syndrome, nervous system disorders
04/28/2009US7524843 N-methyl-N-(1-methyl-1H-indol-3-ylmethyl)-3-(7-oxo-5,6,7,8-tetrahydro-1,8-naphthyridin-3-yl)acrylamide as an enzyme inhibitor for both Fab I and Fab K which are used in the biosynthesis of fatty acids; enoyl-acyl-carrier protein renamed Fab 1; bactericides; fungicides; Staphylococcus aureus; antibiotics
04/28/2009US7524837 Benzotriazapinone salts and methods for using same
04/28/2009CA2555258C 1-isopropyl-2-oxo-1,2-dihydropyridine-3-carboxamide derivatives having 5-ht4 receptor agonistic activity
04/28/2009CA2525437C Benzamide inhibitors of the p2x7 receptor
04/28/2009CA2507465C Phenyl substituted piperidine compounds for use as ppar activators
04/28/2009CA2425704C Tissue-specific exogenous optical agents
04/28/2009CA2375259C Bicyclic heterocycles, pharmaceutical compositions containing these compounds, their use and processes for preparing them
04/28/2009CA2273328C 5-cyclo indole compounds as 5-ht1d receptor ligands
04/28/2009CA2227762C Substituted aminouracils
04/23/2009WO2009052237A1 Inhibitors of c-fms kinase
04/23/2009WO2009052065A1 Substituted n-phenyl-bipyrrolidine carboxamides and therapeutic use thereof
04/23/2009WO2009052063A1 Substituted n-phenyl-pyrrolidinylmethylpyrrolidine amides and therapeutic use thereof as histamine h3 receptor modulators
04/23/2009WO2009052062A1 Substituted n-phenyl-bipyrrolidine carboxamides and therapeutic use thereof
04/23/2009WO2009051660A2 Compounds for activating tgf-beta signaling
04/23/2009WO2009051112A1 Amide compounds and use of the same
04/23/2009WO2009050999A1 Indolium compound and optical recording material using the compound
04/23/2009WO2009050352A2 Imidazolone derivatives, preparation method thereof and biological use of same
04/23/2009WO2009050232A1 Cgrp antagonists
04/23/2009WO2009050220A1 Indazoles as glucocorticoid receptor ligands
04/23/2009WO2009050201A2 4-phenyl-5-oxo-imidazole derivatives, pharmaceutical compositions and uses therof
04/23/2009WO2009050200A1 Imidazolidine-2,4-dione (hydantoin) derivatives useful as npy y2 receptor modulators
04/23/2009WO2009050197A2 Substituted piperazines and piperidines as modulators of the neuropeptide y2 receptor
04/23/2009WO2009050185A1 1,3,5-trisubstituted triazole derivative
04/23/2009WO2009049837A1 Process for preparing 8-hydrazino-8-aryloctanoyl derivatives and their use
04/23/2009WO2009024342A3 Novel microbiocides
04/23/2009WO2009015164A3 Piperidinyl derivatives as modulators of chemokine receptor activity
04/23/2009WO2009010230A3 Process and intermediate for the production of a tertiary alcohol as an intermediate in the synthesis of montelukast
04/23/2009WO2009004383A3 Aza-bicyclohexane compounds useful as anticoagulants
04/23/2009WO2009004171A3 1-benzylpyrazole derivatives, preparation thereof and therapeutic use thereof
04/23/2009WO2009001060A3 Use of compounds for preparing anti-tuberculosis agents
04/23/2009WO2008152094A3 Substituted acetamides as modulators of the ep2 receptor
04/23/2009WO2008152014A3 3-hetrocyclylidene-indolinone derivatives as inhibitors of specific cell cycle kinases
04/23/2009WO2008131501A3 New anti-viral nucleoside analogs
04/23/2009US20090105306 Novel compounds as cannabinoid receptor ligands
04/23/2009US20090105296 Inhibitors of c-fms kinase
04/23/2009US20090105291 Ethyl (2S)-2-[(4,4-dimethyl-3-oxo-1-cyclobutenyl)amino]-3-[(4-([2,7]naphthyridin-1-yloxy)phenyl]propanoate; compounds can inhibit the binding of integrins to their ligands and are of use in the prophylaxis and treatment of immuno or inflammatory disorders
04/23/2009US20090105286 Low-molecular inhibitors of cytohesin-family guanine nucleotide exchange factors
04/23/2009US20090105279 Tetrahydrofuro[2,3-b]furyl carbamates containing an (oxy)hydrazide group; these compounds target the HIV protease in both wild type and mutant strains of HIV.