Patents
Patents for C07D 405 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom (69,397)
07/2009
07/29/2009EP2081892A1 Compounds and methods for treating protein folding disorders
07/29/2009EP2081572A1 Benzimidazole cannabinoid agonists bearing a substituted heterocyclic group
07/29/2009EP1807407B1 Aromatic amides as inhibitors of c-fms kinase
07/29/2009EP1701944B1 2-(amino-substituted)-4-aryl pyramidines and related compounds useful for treating inflammatory diseases
07/29/2009EP1678166B1 Protein kinase inhibitors
07/29/2009EP1513527B1 Prodrugs of imidazole derivatives, for use as proton pump inhibitors in the treatment of e.g. peptic ulcers
07/29/2009EP1397357B1 Polymorphic forms of 1-[4-(5-cyanoindol-3-yl)butyl]-4-(2-carbamoylbenzofuran-5-yl)piperazine hydrochloride
07/29/2009CN101495473A Azolylmethyloxiranes, use thereof for controlling plant pathogenic fungi, and agents containing the same
07/29/2009CN101492444A Nitrogenous heterocyclic compounds with insecticidal activity, preparation and uses thereof
07/29/2009CN101492416A Compounds effecting glucokinase
07/29/2009CN101492383A Process for making chiral 1,4-disubstituted piperazines
07/29/2009CN100519573C Novel chemical substance having morphogenetic and growth-accelerating activities
07/29/2009CN100519556C Method of synthesizing Itraconazole
07/29/2009CN100519550C 2-oxo-indole compound having a functtion of inhibiting glycogen synthase kinase-3
07/29/2009CN100519549C Pyrimidine derivatives and pharmaceutical compositions containing the compounds
07/29/2009CN100519539C N3 alkylated benzimidazole derivatives as MEK inhibitors
07/29/2009CN100519528C Compounds with analgesic effect
07/29/2009CN100519527C Inhibitors of histone deacetylase
07/29/2009CN100519526C Azabicyclo derivatives as muscarinic receptor antagonists
07/28/2009US7566786 enzyme inhibitor 4-[(3-methylphenyl)amino]-6-(methylsulfonyl)-3-quinolinecarboxamide; antiinflammatory agents for treatment, prophylaxis of inflammatory or allergic diseases such as chronic obstructive pulmonary disease (COPD), asthma, rheumatoid arthritis or allergic rhinitis
07/28/2009US7566734 Imidazolyl derivatives
07/28/2009US7566718 Amine-linked pyridyl and phenyl substituted piperazine-piperidines with CXCR3 antagonist activity
07/28/2009US7566710 4-((7-chloroquinolin-4-yl)aminoalkyleneamino-)-spiro(cyclohexane-1.5'-1H-4,5,6-trioxaindene )dicitrate; malaria; paraciticides; antiprotozoa agents; Plasmodium; synergistic; chloroquine-resistant; cost efficiency; industrial scale; penetration and activity of artemisine
07/28/2009US7566709 4-(3-(2-Fluorophenyl)-1-phenyl-1H-pyrazol-4-ylmethyl)morpholine; 5HT2A/5HT2C receptors; central nervous system; schizophrenia; antidepressants; dementia; Parkinson's disease; Azheimer's disease; Huntington's disease; Tourette's syndrome; anxiolytic agents; congnition activators; analgesics
07/28/2009US7566444 Versatile hydrophilic dyes
07/23/2009WO2009091634A1 Crystalline 2-(4-cyclopropanesulphonyl-phenyl)-n-pyrazin-2-yl-3-(tetrahydropyran-4-yl)-propionamide
07/23/2009WO2009091433A2 Spiro and dispiro 1,2,4-trioxolane antimalarials
07/23/2009WO2009091324A1 Quinoline, naphthalene and conformationally constrained quinoline or naphthalene derivates as anti-mycobacterial agents
07/23/2009WO2009091014A1 Phenyl acetamide derivative
07/23/2009WO2009090548A2 3-azabicyclo [3.1.0] hexane derivatives as vanilloid receptor ligands
07/23/2009WO2009063061A3 Aryl- and heteroarylcarbonyl derivatives of benzomorphanes and related scaffolds, medicaments containing such compounds and their use
07/23/2009WO2009050352A3 Imidazolone derivatives, preparation method thereof and biological use of same
07/23/2009WO2009013348A3 Pyrimidine derivatives useful for the treatment of inflammatory or allergic conditions
07/23/2009WO2008061796A3 Compounds for the treatment of diseases associated with amyloid or amyloid-like proteins
07/23/2009WO2008059130A9 Thionucleosides and pharmaceutical applications
07/23/2009US20090186932 Pesticidal N-Phenylpyrazole Derivatives
07/23/2009US20090186927 Trans-9,10-dehydroepothilone c and d, analogs thereof and methods of making the same
07/23/2009US20090186921 Azacyclic compounds
07/23/2009US20090186914 Ethyl (2S)-2-[(4,4-dimethyl-3-oxo-1-cyclobutenyl)amino]-3-[(4-([2,7]naphthyridin-1-yloxy)phenyl]propanoate; compounds can inhibit the binding of integrins to their ligands and are of use in the prophylaxis and treatment of immuno or inflammatory disorders
07/23/2009US20090186906 N-((S)-4,4-dimethyl-1-oxo-1-((3aS,6aR)-3-oxo-dihydro-2H-furo[3,2-b]pyrrol-4(5H6H, 6aH)-yl)pentan-2-yl)-4-(4-methylpiperazin-1-yl)benzamide; treatment of a disease selected from osteoporosis, Paget's disease, Chagas's disease, malaria, gingival diseases, hypercalaemia, metabolic bone disease, bone cancer
07/23/2009US20090186895 Ethers, secondary amines and derivatives thereof as modulators of the 5-ht2a serotonin receptor useful for the treatment of disorders related thereto
07/23/2009US20090186871 Tyrosine kinase inhibitors
07/23/2009US20090186834 Diphenylheterocycle cholesterol absorption inhibitors
07/23/2009US20090186373 Pyrimidines reacting with O6-Alkylguanine-DNA alkyltransferase
07/23/2009CA2712948A1 Phenylacetamide derivative
07/23/2009CA2712245A1 Crystalline (r)-2-(4-cyclopropanesulphonyl-phenyl)-n-pyrazin-2-yl-3-(tetrahydropyran-4-yl)-propionamide
07/23/2009CA2711912A1 Quinoline, naphthalene and conformationally constrained quinoline or naphthalene derivates as anti-mycobacterial agents
07/22/2009EP2080754A2 Organic compounds
07/22/2009EP2079732A1 3- (1, 3-benz0di0x0l-5-yl) -6- (4-cyclopropylpiperazin-1-yl) -pyridazine, its salts and solvates and its use as histamine h3 receptor antagonist
07/22/2009EP2079729A1 Compounds and compositions as protein kinase inhibitors
07/22/2009EP2079701A1 Sulfonamide substituted pyrazoline compounds, their preparation and use as cb1 modulators
07/22/2009EP2079693A1 Ether derivatives dual modulators of the 5-ht2a and d3 receptors
07/22/2009EP2079690A2 3-aza-bicyclo[3.1.0]hexane derivatives
07/22/2009EP1896460B1 Benzofuranyl derivatives as 5-ht6-receptor inhibitors
07/22/2009EP1750704B1 Urea antagonists of p2y1 receptor useful in the treatment of thrombotic conditions
07/22/2009EP1745039A4 3-aryl-5,6-disubstituted pyridazines
07/22/2009EP1644337B1 Melanocortin-4 receptor binding compounds and methods of use thereof
07/22/2009EP1503988B1 Fredericamycin derivatives
07/22/2009EP1392680B1 Selective anthranilamide pyridine amides as inhibitors of vegfr-2 and vegfr-3
07/22/2009EP1391456B1 2-iminoimidazole derivatives
07/22/2009CN101490043A Azolylmethyloxiranes, use thereof for controlling plant pathogenic fungi, and agents containing the same
07/22/2009CN101490042A Fungicide hydroximoyl-tetrazole derivatives
07/22/2009CN101486682A N3 alkylated benzimidazole derivatives as MEK inhibitors
07/22/2009CN101486675A 2- and 2,5-substituted phenylketoenols
07/22/2009CN100515419C Substituted benzazoles and its application as inhibitors of Raf kinase
07/21/2009US7563910 Heterocyclic cannabinoid receptor antagonists
07/21/2009US7563907 Fluorophores with a large Stokes shift, high photostability, long storage life and a high fluorescent quantum yield, and that can be excited by white light or lasers in the ultraviolet, visible or near-infrared spectral region; immunoassays, receptor binding assays, DNA sequencing, electrophoresis
07/21/2009US7563905 Triazole derivatives and method of using the same to treat HIV infections
07/21/2009US7563900 Reacting 4-cyclopentyloxy-3-hydroxy-benzaldehyde with 3-bromo-4-fluoro nitrobenzene
07/21/2009US7563811 3-(2-Cyanophenyl)-5-(2-methoxyphenyl)-1-phenyl-1,2-dihydropyridin-2-one; antagonists of AMPA and kainate receptors; neuroprotectants; neurodegenerative diseases; Alzheinmer's disease; antiepileptic agents; antispasmodic agents; anxiolytic agents; ddrug abuse; nervous sytem disorders; antihypoxic agents
07/21/2009US7563808 administering a cholinesterase inhibitor ( a dimethoxyindanone derivative) to treat dementia associated with or caused by vascular diseases
07/21/2009US7563784 substituted 1,1,4-1l6-trioxo[1,2]thiazepan-4-ylamide-derived protease inhibitors which inhibit the likes of cathepsin K; treating osteoporosis, osteo- and rheumatoid arthritis and periodontal disease; inhibiting excessive cartilage or matrix degradation
07/21/2009CA2495943C Indoles having anti-diabetic activity
07/21/2009CA2379972C Prodrug of an ice inhibitor
07/16/2009WO2009089057A1 Amide derivatives as ion-channel ligands and pharmaceutical compositions and methods of using the same
07/16/2009WO2009088531A1 6-substituted indole-3-carboxylic acid amide compounds having sphingosine-1-phosphate (s1p) receptor antagonist biological activity
07/16/2009WO2009088103A1 Pyridylamidine compound or salt thereof, and agricultural or horticultural fungicide composition containing the same as active ingredient
07/16/2009WO2009088070A1 (heterocyclic methyl)azolylmethylcyclopentanol derivative and intermediate thereof, process for production of the derivative, and agricultural or horticultural preparation and protective agent for industrial material each comprising the derivative
07/16/2009WO2009087212A2 Pyridine derivatives
07/16/2009WO2009086835A1 Novel cyanoguanidines
07/16/2009WO2009058800A3 Synthesis of nucleosides
07/16/2009WO2008079787A8 Glucokinase activators
07/16/2009US20090182150 Deblocking, deprotecting via hydrogenation
07/16/2009US20090182149 Salt of sulfinylbenzimidazole compound, and crystal and amorphous form thereof
07/16/2009US20090182143 Novel heterocyclic compounds useful for the treatment of inflammatory and allergic disorders: process for their preparation and pharmaceutical compositions containing them
07/16/2009US20090182140 Alicyclic Heterocyclic Compound
07/16/2009US20090182028 Plant Components and Extracts and Uses Thereof
07/16/2009US20090182011 Chimeric Nitrate Esters and Use of the Same in a Treatment for Depression
07/16/2009US20090182007 Organic compounds
07/16/2009US20090181994 Triazole derivatives as inhibitors of 11-beta-hydroxysteroid dehydrogenase-1
07/16/2009US20090181993 Hiv inhibiting 5-heterocyclyl pyrimidines
07/16/2009US20090181981 Crystalline (r)-2-(4-cyclopropanesulphonyl-phenyl)-n-pyrazin-2-yl-3-(tetrahydropyran-4-yl)-propionamide
07/16/2009US20090181979 Pharmaceutically acceptable salts of quinolinone compounds having improved pharmaceutical properties
07/16/2009US20090181968 Novel 3-Bicyclocarbonylaminopyridine-2-Carboxamides or 3-Bicyclocarbonylaminopyrazine-2-Carboxamides
07/16/2009US20090181966 PGD2 receptor antagonists for the treatment of inflammatory diseases
07/16/2009US20090181958 Substituted nitrogen-containing heterobicycles, the preparation thereof and their use as pharmaceutical compositions
07/16/2009US20090181949 1h-imidazole derivative having cb1, agonistic, cb1 partial agonistic or cb1 antagnistic activity
07/16/2009US20090181939 Azetidinecarboxamide Derivatives And Their Use In The Treatment Of CB1 Receptor Mediated Disorders
07/16/2009CA2711815A1 6-substituted indole-3-carboxylic acid amide compounds having sphingosine-1-phosphate (s1p) receptor antagonist biological activity
07/16/2009CA2711803A1 Pyridine derivatives