Patents
Patents for C07D 405 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom (69,397)
03/2009
03/25/2009CN100471855C Oxetane compounds containing maleimide functional group
03/25/2009CN100471845C C 10 ester substituted taxadane
03/25/2009CN100471842C Quinolone derivative or its salt
03/25/2009CN100471832C Compound for preparing protease inhibitor
03/24/2009US7507839 e,g, 1,5-bis(5-acetyl-4,7-dimethoxybenzofuran-6-yloxy)pentane;potassium channel modulator; antiinflammatory agent, autoimmune diseases; immunosuppressant; multiple sclerosis, rejection of foreign organ transplants
03/24/2009US7507815 Succinoylamino lactams as inhibitors of a-β protein production
03/24/2009US7507762 Substituted 4H-chromene and analogs as activators of caspases and inducers of apoptosis and the use thereof
03/24/2009US7507761 Benzopyran derivatives, method of production and use thereof
03/24/2009US7507754 e.g. N-{4-[4-(5-Methoxy-pyridin-2-yl)-phenoxymethyl]-5-methyl-furan-2-carbonyl}-2-methyl-benzenesulfonamide; prostaglandin E4 receptor antagonist; analgesic, antiinflammatory agent; migraines and headache
03/24/2009US7507753 Biaryl compound and use thereof
03/24/2009US7507751 Biphenyl derivatives
03/24/2009US7507747 Muscarinic acetylcholine receptor antagonists
03/24/2009US7507741 Heterocyclic compounds
03/24/2009US7507734 Pyridazinone derivatives
03/24/2009US7507420 Peptidyl prodrugs and linkers and stabilizers useful therefor
03/24/2009CA2422380C Pyrazole compounds useful as protein kinase inhibitors
03/24/2009CA2224060C Manganese or iron complexes of nitrogen-containing macrocyclic ligands effective as catalysts for dismutating superoxide
03/19/2009WO2009035652A1 Synthesis of deuterated catechols and benzo[d][1,3] dioxoles and derivatives thereof
03/19/2009WO2009035067A1 Glucocorticoid receptor agonists consisting of 1,3,3-tri- methyl-7-phenyl-3,4-dihydro-1h-quinoxalin-2-one derivatives
03/19/2009WO2009034258A1 Tri-amino-pyrimidine cyclobutenedione derivatives used as phosphatase cdc25 inhibitors
03/19/2009WO2009033703A1 1,3-disubstituted-4-phenyl-1 h-pyridin-2-ones
03/19/2009WO2009002510A3 Crystalline polymorph of exemestane
03/19/2009WO2009002489A3 Crystalline polymorph of 7-ethyl-10-hydroxycamptothecin
03/19/2009WO2008157552A3 Invertebrate acetylcholinesterase inhibitors
03/19/2009WO2008116107A3 Piperazine derivatives as glucokinase activators
03/19/2009US20090076281 Process for the preparation of losartan and its salts
03/19/2009US20090076276 such as (R)-3-(3-hydroxypyrrolidin-1-yl)-N-methyl-N-methoxypropanamide; poly(ADP-ribose)polymerase inhibitors
03/19/2009US20090076274 Benzoxazinone derivatives, preparation thereof and uses in the treatment of cns and other disorders
03/19/2009US20090076103 Stem cell differentiating agents and uses therefor
03/19/2009US20090076091 Indazole-heteroaryl derivatives
03/19/2009US20090076088 Thrombin Receptor Antagonists
03/19/2009US20090076077 Methods and Compositions for Selectin Inhibition
03/19/2009US20090076030 Piperazine compounds
03/19/2009US20090076004 1-Aryl-or heteroaryl-3-aryl-or heteroarylindole-2-carboxylic acids or esters: e.g., 5-(4-tert-Butylphenyl)-1,3-bis(4-isopropoxyphenyl)-indole-2-carboxylic acid; inhibition of the activity of microsomal prostaglandin E synthase-1, leukotriene C4 and/or 5-lipoxygenase-activating protein; analgesics
03/19/2009US20090076003 Phthalazine Derivatives with Angiogenesis Inhibiting Activity
03/19/2009US20090075253 Bioreactive agents
03/19/2009DE102007044277A1 Substituierte Nicotinamid-Verbindungen und deren Verwendung in Arzneimitteln Substituted nicotinamide compounds and their use in medicaments
03/19/2009CA2698929A1 1,3-disubstituted-4-phenyl-1h-pyridin-2-ones
03/19/2009CA2698808A1 Synthesis of deuterated catechols and benzo[d][1,3] dioxoles and derivatives thereof
03/19/2009CA2698792A1 Vegfr inhibitors containing a zinc binding moiety
03/19/2009CA2692702A1 Tri-amino-pyrimidine cyclobutenedione derivatives used as phosphatase cdc25 inhibitors
03/18/2009EP2036904A1 A process for the preparation of olmesartan medoxomil
03/18/2009EP2036889A2 Substituted indoles and a method for the production and use thereof
03/18/2009EP2035415A1 Azolylmethyloxiranes, their use for controlling phytopathogenic fungi and compositions comprising them
03/18/2009EP2035414A1 Azolylmethyloxiranes, their use for controlling phytopathogenic fungi and compositions comprising them
03/18/2009EP2035412A1 Muscarinic receptor agonists that are effective in the treatment of pain, alzheimer's disease and schizophrenia
03/18/2009EP2035411A1 Muscarinic receptor agonists that are effective in the treatment of pain, alzheimer's disease and schizophrenia.
03/18/2009EP2035407A1 Muscarinic receptor agonists that are effective in the treatment of pain, alzheimer's disease and schizophrenia
03/18/2009EP2035406A1 Novel substituted-1h-quinazoline-2,4-dione derivatives, preparation method thereof and pharmaceutical composition containing the same
03/18/2009EP2035396A2 Triazole compounds that modulate hsp90 activity
03/18/2009EP2035394A1 2-pyrazinecarboxamide derivatives
03/18/2009EP2035391A1 Indazole derivatives for treating hsp90-induced diseases
03/18/2009EP2035387A2 2-alkoxy-3,4,5-trihydroxy-alkylamide-benzazepines, the preparation and use thereof, and compositions containing the same
03/18/2009EP2035386A1 Isoquinoline derivatives and their use as inhibitors of cytokine mediated diseases
03/18/2009EP2035384A2 Process for synthesizing piperazine-piperidine compounds
03/18/2009EP2035380A2 Parp inhibitors
03/18/2009EP2035378A1 Substituted isoindoles as bace inhibitors and their use
03/18/2009EP2035377A1 Indole derivatives and their use as thyroid receptor ligands
03/18/2009EP2035375A1 1,3-disubstituted 4-methyl-1h-pyrrole-2-carboxamides and their use for the manufacture of medicaments
03/18/2009EP2035372A1 Modulators of the histamine h3-receptor useful for the treatment of disorders related thereto
03/18/2009EP2034996A2 Triazole compounds that modulate hsp90 activity
03/18/2009EP1824486B1 Benzdioxane piperazine derivatives with a combination of affinity for dopamine-d2 receptors and serotonin reuptake sites
03/18/2009EP1656346B1 1,2,3,4-tetrasubstituted indole for the treatment of respiratory diseases
03/18/2009EP1567493B1 Phenyl substituted piperidine compounds for use as ppar activators
03/18/2009EP1558603A4 Oxyge-containing heterocyclic fused naphthopyrans
03/18/2009EP1539151B1 Biaryl compounds having anti-infective activity
03/18/2009EP1453810B1 Substituted 4-phenyltetrahydroisoquinolines, method for the production thereof, the use thereof as medicaments, in addition to a medicament containing same
03/18/2009EP1386912B1 Cyclic amidine derivative
03/18/2009EP0963984B1 Heteroarylpiperidines and piperazines and their use as antipsychotics and analgetics
03/18/2009CN101389622A Pyrimidine derivatives used as pi-3 kinase inhibitors
03/18/2009CN101389608A 5-HT7 receptor antagonists
03/18/2009CN100469779C Inhibitors of interleukin-1beta converting enzyme
03/18/2009CN100469776C Amelioration of the development of cataracts and other ophthalmic diseases
03/18/2009CN100469769C Benzyl-pyridazinons as reverse transcriptase inhibitors
03/18/2009CN100469767C Bipiperidinyl-derivatives and their use as chemokine receptor inhibitors
03/17/2009USRE40667 [R-(R*R*)]-2-(4-fluorophenyl)-β,δ-dihydroxy-5-(1-methylethyl-3-phenyl-4-[(phenylamino)carbonyl]-1H-pyrrole-1-heptanoic acid, its lactone form and salts thereof
03/17/2009US7504537 osteoarthritis or rheumatoid arthritis
03/17/2009US7504522 e.g. 3-(2,4,4'-trichlorobenzhydryloxy)-N-(tert-butyl)azetidine-1-carboxamide; cannabinoid receptor antagonist; antidiabetic agent, antidepressant; eating disorders, obesity, nicotine addiction
03/17/2009US7504511 e.g. N-[4-(5-Butyl-2-methoxyphenyl)-1,3-thiazol-2-yl]-4((4-[2-(S)-(hydroxymethyl)pyrrolidin-1-yl]piperidin-1-yl)carbonyl)benzamide; antiinflammatory, anticarcinogenic, antidiabetic, analgesic agent
03/17/2009US7504508 PGD2 receptor antagonists for the treatment of inflammatory diseases
03/17/2009US7504489 enzyme inhibitors such as beta-1'-nicotinamide-2'-deoxyribose, used for treating diseases and conditions associated with CD38, related enzymes and cyclic-adenosine-diphosphate-ribose (cADPR)
03/17/2009US7504436 Bioisosteres of actinonin
03/17/2009US7504429 Receptor or non-receptor types; 1H-pyrrole-3-carboxylates; anticarcinogenic, antidiabetic, antiproliferative agents; autoimmune and Crohn's diseases, acromegaly, aging resistance; coadminister tamoxifen, raloxifene, taxol, trastuzumab, tirofiban or a COX-2 inhibitor
03/17/2009US7504421 Substituted 2-thio-3,5-dicyano-4-aryl-6-aminopyridines and their use
03/17/2009US7504416 4-substituted quinolines as antitumor agents
03/17/2009US7504414 Useful as adjuvants to chemotherapy or radiation therapy to treat cancer; as inhibitors of checkpoint kinase Cds1 (in man also known as Chk2); 2-[4-(3,4-dichloro-phenoxy)-phenyl]-1H-imidazo[4,5-b]pyridine-5-carboxylic acid amide
03/17/2009US7504411 2,3,6-Trisubstituted-4-pyrimidone derivatives
03/17/2009US7504410 such as N-[3-[[5-bromo-4-[[3-[[[1-(trifluoromethyl)cyclobutyl]carbonyl]amino]propyl]amino]-2-pyrimidinyl]amino]phenyl]-1-pyrrolidinecarboxamide; Chks (checkpoint kinases), Akts (protein kinases B) and Pdks (phosphoinositide-dependent kinases) inhibitors; antiproliferative agents
03/17/2009US7504408 Quinzoline derivatives for use in the treatment of cancer
03/17/2009US7504402 bicyclo[2.2.2]-oct-1-yl-1,2,4-triazoles; type 2 diabetes, lipid disorders, obesity, atherosclerosis, metabolic syndrome, hyperglycemia, insulin resistance; increase insulin sensitivity in muscle, liver and adipose tissue by correction of the elevated plasma levels of glucose without causing hypoglycemia
03/17/2009US7504392 2,3,4,5-tetrahydro-1H-3-benzazepines and their medical use
03/17/2009US7504362 Pesticidal compositions
03/17/2009US7504360 Containing crystalline compounds which produce color when thermally converted to liquid or amorphous form time-independent
03/17/2009US7504243 Methods for the production of biliverdin
03/17/2009US7504087 Receptor-avid exogenous optical contrast and therapeutic agents
03/17/2009CA2717039A1 Catalytic process for asymmetric hydrogenation
03/17/2009CA2360668C The use of 4-h-1-benzopyran-4-one derivatives as inhibitors of smooth muscle cell proliferation
03/17/2009CA2337849C Piperazinone derivatives and applications thereof
03/17/2009CA2328234C Compounds that inhibit the binding of integrins to their receptors
03/17/2009CA2316351C Benzopyran and benzothiopyran derivatives having retinoid antagonist-like activity