Patents
Patents for C07D 403 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group (62,587)
02/2004
02/26/2004WO2003101444A8 Diarylurea compounds and derivatives as chk-1 inhibitors for the treatment of cancer
02/26/2004WO2003099211A3 Mitotic kinesin inhibitors
02/26/2004WO2003086271A3 Azole derivatives as antifungal agents
02/26/2004WO2003076398A3 Pyrrole-2, 5-dione derivatives and their use as gsk-3 inhibitors
02/26/2004WO2003057144A3 Change inhibitors of dipeptidyl peptidase iv
02/26/2004WO2003050261A3 (1-phenyl-2-heteroaryl)ethyl-guanidine compounds as inhibitors of mitochondrial f1f0 atp hydrolase
02/26/2004WO2003047517A3 Novel-n-[4-(1h-imidazol-1-yl)-2-fluorophenyl]-3-(trifluoromethyl)-1-h-pyrazole-5-carboxamides as factor xa
02/26/2004WO2003039549A8 Selective antibacterial agents
02/26/2004WO2002041910A8 Methods and compositions for the treatment of diseases of the eye
02/26/2004US20040039196 (2-Oxindol-3-ylidenyl) acetic acid derivatives and their use as protein kinase inhibitors
02/26/2004US20040039040 Urea derivative and adhesive-molecule inhibitor containing the same as active ingredient
02/26/2004US20040039033 Administering (1-phenyl-2-heteroaryl)ethyl-guanidine compounds for treating ischemic conditions including myocardial infarction, congestive heart failure, and cardiac arrhythmias
02/26/2004US20040039007 Nitrogen compounds such as (6-(3-Methylaminopropyl)-2-(2-tri-fluoromethylphenyl)pyrimidin-4-yl)-(1H -pyrazolo(3,4-b)pyridin-3-yl)-amine, use as glycogen synthase kinase-3 (GSK-3) antagonists
02/26/2004US20040039005 HIV replication inhibiting pyrimidines
02/26/2004US20040038991 Imidazolyl-cyclic acetals
02/26/2004US20040038973 Treating osteoarthritis or rheumatoid arthritis
02/26/2004US20040038969 Substituted aminopyrimidines and aminopyridazines; analgesics particularly for migraines, neuropathic pain and associated hyperalgesia and allodynia; antiinflammatory agents; treating asthma, gastrointestinal disorders, etc.
02/26/2004US20040038962 Treatment of nocturnal enuresis, nocturia, polyuria resulting from central diabetes insipidus, urinary incontinence or bleeding disorders such a hemophilia
02/26/2004US20040038961 Azaisoquinoline derivatives as matrix metalloproteinase inhibitors
02/26/2004CA2495589A1 Azabicyclic compounds are central nervous system active agents
02/25/2004EP1391457A1 Substituted 2-Phenylbenzimidazoles and their use as PARP inhibitors
02/25/2004EP1391456A1 2-iminoimidazole derivative (2)
02/25/2004EP1391451A1 2-iminopyrrolidine derivates
02/25/2004EP1391203A1 Antitumor agents
02/25/2004EP1390361A2 Melanocortin receptor ligands
02/25/2004EP1390354A1 Triazinyl acrylamide derivatives as kinase inhibitors
02/25/2004EP1390353A1 Triazole-derived kinase inhibitors and uses thereof
02/25/2004EP1390350A1 Novel compounds
02/25/2004EP1390347A1 Pyrrolidine ester derivatives with oxytocin modulating activity
02/25/2004EP1390029A1 Phenylindoles for the treatment of hiv
02/25/2004EP1211246B1 Pyrimidine derivatives and herbicides containing the same
02/25/2004EP1181269B1 Cell proliferation inhibitors
02/25/2004CN1478087A Indolylmaleimide derivatives as protein kinase C inibitors
02/25/2004CN1478080A Phenylethenyl or phenylethinyl derivatives as glutamate receptor antagonists
02/25/2004CN1478079A Diaminopyrazole derivatives and their use for oxidation dyeing of keratinous fibres
02/25/2004CN1477960A EPA receptor inhibitors to treat rheumatoid arthritis
02/25/2004CN1139577C Improved process for preparation of unsymmetrical 4,6-bis(aryloxy) pyrimidine compounds
02/24/2004US6696574 Processes and intermediates for preparing glycogen phosphorylase inhibitors
02/24/2004US6696469 For treatment of diseases or pathological conditions in which endothelial dysfunction is known; atherosclerosis, dyslipidaemia, diabetes
02/24/2004US6696456 Carbocyclic acids and salts such as (2s,3r)-3-ethylsulfanyl-2-(4'-fluoro-biphenyl-4-sulfonylamino)-3- phenylpropionic acid, used as metalloenzyme antagonists for the prophylaxis of degenerative joint disease and as wound healing agents
02/24/2004US6696452 Glycogen synthase kinase-3 and aurora-2 a serine/threonine protein kinase inhibitors; antidiabetic and anticancer agents and alzheimer's disease treatments
02/24/2004US6696447 Hydroxyphenyl-piperazinyl-methyl-benzamide derivatives for the treatment of pain
02/24/2004US6696443 Piperidine/piperazine-type inhibitors of p38 kinase
02/24/2004US6696438 Cyclic amino acid compounds, pharmaceutical compositions comprising same, and methods for inhibiting β-amyloid peptide release and/or its synthesis by use of such compounds
02/24/2004US6696437 Polymerase inhibitors comprising heterocyclic amides such as 2-pyridin-2-ylbenzimidazole-4-carboxamide, used for prophylaxis of neurodegenerative disorders, damage to hearts or brains, and as anticarcinogenic agents
02/24/2004US6696434 Quinoline and quinoxaline compounds which inhibit platelet-derived growth factor and/or p56lck tyrosine kinases
02/24/2004CA2114542C Benzimidazolone derivatives as 5-ht1a and 5-ht2 antagonists
02/19/2004WO2004014900A1 Benzimidazoles and benzothiazoles as inhibitors of map kinase
02/19/2004WO2004014895A1 Piperazine substituted aryl benzodiazepines
02/19/2004WO2004014892A1 Monocyclic derivatives as matrix metalloproteinase inhibitors
02/19/2004WO2004014891A1 Pyridazine derivatives as ligands for gaba receptors
02/19/2004WO2004014878A1 1,2,4-triazole derivative, method for preparing the same, and pharmaceutical composition containing the same
02/19/2004WO2004014877A1 Process for preparing rizatriptan
02/19/2004WO2004014871A1 Vanilloid receptor ligands and their use in treatments
02/19/2004WO2004014869A2 5,6-fused 3,4-dihydropyrimidine-2-one derivatives as matrix metalloproteinase inhibitors
02/19/2004WO2004014868A2 Pyrimidine-2,4-dione derivatives as matrix metalloproteinase inhibitors
02/19/2004WO2004014867A2 Matrix metalloproteinase inhibitors and methods for identification of lead compounds
02/19/2004WO2004014866A1 Azaisoquinoline derivatives as matrix metalloproteinase inhibitors
02/19/2004WO2004014865A1 Phenylpyridazine derivatives as ligands for gaba receptors
02/19/2004WO2004014864A1 1h-indazole-3-carboxamide compounds as cyclin dependent kinases (cdk) inhibitors
02/19/2004WO2004014863A1 Benzoylpyrazolones substituted by 3-aminocarbonyl
02/19/2004WO2004014851A2 Tyrosine kinase inhibitors
02/19/2004WO2004014844A2 Aryl and heteroaryl compounds and methods to modulate coagulation
02/19/2004WO2004014381A2 Matrix metalloproteinase inhibitors and methods for identification of lead compounds
02/19/2004WO2004014372A1 Acylated, heteroaryl-condensed cycloalkenylamines and their use as pharmaceuticals
02/19/2004WO2004014369A1 Acylamino-substituted heteroaromatic compounds and their use as pharmaceuticals
02/19/2004WO2004014368A1 3-pyrrolyl-pyridopyrazoles and 3-pyrrolyl-indazoles as novel kinase inhibitors
02/19/2004WO2004014366A1 Hetero biaryl derivatives as matrix metalloproteinase inhibitors
02/19/2004WO2004014365A1 Phthalimide derivatives as matrix metalloproteinase inhibitors
02/19/2004WO2004014364A1 Substituted phenylindoles for the treatment of hiv
02/19/2004WO2004014300A2 Tyrosine kinase inhibitors
02/19/2004WO2004007478A3 Derivatives of 3-guanidinocarbonyl-1-heteroaryl-pyrrole, process for their preparation and their pharmaceutical use
02/19/2004WO2003086306A3 5ht2c receptor modulators
02/19/2004WO2003057213A3 Cyclohexano- and cycloheptapyrazole derivative compounds, for use in diseases associated with the 5-ht2c receptor
02/19/2004WO2002080869A3 Novel dyeing composition for dyeing keratinous fibres comprising a particular dicationic monoazo dye
02/19/2004WO2002006219A3 1-alkyl-3-[1-(substituted phenyl) benzotriazol-6-yl] uracils
02/19/2004US20040034251 Such as 2-(4,6-dimethoxypyrimidine-2-ylcarbonyl)acetanilide; for use as intermediate in production of agricultural chemicals and medicines
02/19/2004US20040034231 Amidinophenyl-4-aminoacetic acid derivative is useful for treating diseases such as thrombosis, apoplexy, cardiac infarction, inflammation and arteriosclerosis, which are associated with coagulation factors xa, IXa and thrombin
02/19/2004US20040034229 3,4-Di-substituted maleimide compounds as CXC chemokine receptor antagonists
02/19/2004US20040034222 Phenyloxyalkylamino substituted triazine compound, useful for applying to the parts of the plants, to plant seed or to the area under cultivation as plant growth regulator
02/19/2004US20040034218 Farnesyl transferase inhibiting benzoheterocyclic derivatives
02/19/2004US20040034089 Such as (1-((2,3-dihydro-2-(4-propyl-1H-imidazol-2-yl)-1H-indol-1 -yl)carbonyl)propyl)-carbamate; for inactivation of cholecystokinins
02/19/2004US20040034084 Side effect reduction; for treatment of AIDS, cancer and arthritis
02/19/2004US20040034081 Estrogen receptor modulators
02/19/2004US20040034078 Such as 2-(2-butylamino-ethylsulfanylmethyl)-1H-benzimidazole-4-carboxylic acid amide for treatment of cancer, strokes, head trauma, and neurodengenerative diseases; solid phase synthesis
02/19/2004US20040034077 Processes for preparing losartan and losartan an potassium
02/19/2004US20040034076 Such as methyl-3-azido-2-((4,6-dimethoxy-2-pyrimidinyl)oxy) 3,3-diphenylpropionate; for treatment of high blood pressure
02/19/2004US20040034063 Antiallergens for treating and prevention of asthma
02/19/2004US20040034052 Antitumor agents
02/19/2004US20040034037 Heteroaryl compounds useful as inhibitors of GSK-3
02/19/2004US20040034034 Novel piperazine derivatives
02/19/2004US20040034032 Quinoline and quinazoline compounds useful in therapy
02/19/2004US20040034018 2-amino-trihydroindole or tetrahydronapthalene-2-yl derivatives, useful for disease state associated with smooth muscle disorders, such as gastrointestinal and urogenital disorders
02/19/2004DE10236340A1 New heteroar(alkan)oyl-substituted phenyl-beta-alaninamide derivatives, useful as broad-spectrum antibacterial agents in human or veterinary medicine
02/19/2004DE10235945A1 New 4-(3-substituted benzoyl)-pyrazol-5-one derivatives, useful as broad-spectrum, pre- and post-emergence herbicides especially for selective weed control in crops e.g. wheat, maize and rice
02/19/2004CA2497656A1 Pyrimidine-2,4-dione derivatives as matrix metalloproteinase inhibitors
02/19/2004CA2495293A1 Azaisoquinoline derivatives as matrix metalloproteinase inhibitors
02/19/2004CA2495285A1 Phenylpyridazine derivatives as ligands for gaba receptors
02/19/2004CA2495216A1 3-pyrrolyl-pyridopyrazoles and 3-pyrrolyl-indazoles as novel kinase inhibitors
02/19/2004CA2494298A1 Acylamino-substituted heteroaromatic compounds and their use as pharmaceuticals