Patents
Patents for C07D 403 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group (62,587)
01/2004
01/06/2004US6673817 Anticoagulants
01/06/2004US6673807 Administering compound possessing inhibitory activity on production of nitric oxide and tricyclic macrolide or salt, solvate or hydrate thereof to increase graft survival time in transplantation subject
01/06/2004US6673803 Quinazoline derivatives and pharmaceutical compositions containing them
01/06/2004US6673797 Cyclooxygenase-2 inhibitors; treating inflammatory disease induced by cyclooxygenase-2
01/06/2004US6673790 Indolin-2-one derivatives, preparation and their use as ocytocin receptor ligands
01/06/2004US6673787 Pyrimidinesulfonamide containing indole compounds used as antiangiogenic and antitumor agents
01/06/2004CA2285891C Triazole antifungal agents
01/02/2004EP1375486A1 Nitrogen-containing heteroaryl compounds having hiv integrase inhibitory activity
01/02/2004EP1375482A1 Benzamidine derivative
01/02/2004EP1373271A1 Indole derivatives having an inhibitory effect on protein kinases
01/02/2004EP1373259A1 Pyridazinone aldose reductase inhibitors
01/02/2004EP1373257A1 Inhibitors of c-jun n-terminal kinases (jnk) and other protein kinases
01/02/2004EP1373256A1 Ccr5 antagonists useful for treating aids
01/02/2004EP1373255A1 Process for the preparation of imidazole compounds
01/02/2004EP1373254A1 New process
01/02/2004EP1373253A1 Inhibitors of cyclin dependent kinases as anti-cancer agent
01/02/2004EP1373224A1 New spirotricyclic derivatives and their use as phosphodiesterase-7 inhibitors
01/02/2004EP1373223A1 Cyano-substituted dihydropyrimidine compounds and their use to treat diseases
01/02/2004EP1373222A2 5-phenylpyrimidine, methods and intermediate products for the production thereof and use of the same for controlling pathogenic fungi
01/02/2004EP1373221A2 Novel cyano-substituted dihydropyrimidine compounds and their use to treat diseases
01/02/2004EP1373219A1 Thiohydantoins and use thereof for treating diabetes
01/02/2004EP1373218A1 Imidazolyl derivatives useful as histamine h3 receptor ligands
01/02/2004EP1373217A1 2-mercapto-4,5-diarylimidazole derivatives and the use thereof as cyclooxygenase inhibitors
01/02/2004EP1373204A2 Heterocyclic compounds
01/02/2004EP1373203A1 Cyclopropylindole derivatives as selective serotonin reuptake inhibitors
01/02/2004EP1373194A1 BENZAMIDE INHIBITORS OF FACTOR Xa
01/02/2004EP1373191A1 Acylated indanyl amines and their use as pharmaceuticals
01/02/2004EP1372692A2 Asymmetric synthesis of (s, s, r)-(-)-actinonin and its analogs and uses therefor
01/02/2004EP1372657A2 A method of treating proliferative diseases using eg5 inhibitors
01/02/2004EP0836595B1 Triazoline and isoxazoline bis-oxime derivatives and their use as pesticides
01/01/2004US20040002608 Central nervous system disorders
01/01/2004US20040002539 Enzyme inhibitors; anticoagulants; blood collecting device
01/01/2004US20040002535 Methods of treating hormone-related conditions using thio-oxindole derivatives
01/01/2004US20040002534 Stem cell factor; signal transduction passageways; anticancer agents
01/01/2004US20040002531 Imidazolyl derivatives
01/01/2004US20040002527 Indolylalkylidenehydrazine-carboximidamide derivatives as 5-hydroxytryptamine-6 ligands
01/01/2004US20040002525 Obesity; osteoporosis
01/01/2004US20040002524 Cardiovascular disorders; osteoporosis; central nervous system disorders
01/01/2004US20040002508 Antitumor agents; anticancer agents; sexual disorders; cardiovascular disorders
01/01/2004US20040002495 Lactam glycogen phosphorylase inhibitors and method of use
01/01/2004US20040002487 Bone disorders; osteoporosis; oral diseases; antiarthritic agents
01/01/2004US20040002485 Enzyme inhibitors; viricides
01/01/2004US20040002424 2-Amino-4-bicyclylamino-6H-1,3,5-triazines, processes for their preparation and their use as herbicides and plant growth regulators
12/2003
12/31/2003WO2004000833A1 Processes for preparing substituted pyrimidines and pyrimidine derivatives as inhibitors of protein kinase
12/31/2003WO2004000832A1 1-[(indol-3-yl)carbonyl] piperazine derivatives
12/31/2003WO2004000819A1 New use of pyrimidine - or triazine- 2-carbonitiles for treating diseases associated with cysteine protease activity and novel pyrimidine-2-carbonitile derivatives
12/31/2003WO2004000817A2 Benzimidazole compounds and their use as estrogen agonists/antagonists
12/31/2003WO2004000814A1 8-(biaryl) quinoline pde4 inhibitors
12/31/2003WO2004000804A1 Ring-substituted diphenyl azetidinones, method for the production thereof, medicaments containing said compounds, and use thereof
12/31/2003WO2004000227A2 Use of thio-oxindole derivatives in treatment of skin disorders
12/31/2003WO2004000225A2 Use of thio-oxindole derivatives in treatment of hormone-related conditions
12/31/2003WO2004000210A2 Indole, azaindole and related heterocyclic sulfonylureido piperazine derivatives
12/31/2003WO2004000204A2 Labelled somatostatin analogs backbone cyclized through metal complexation
12/31/2003WO2003060475A3 Melanin concentrating hormone receptor ligands: substituted 2-(4-benzyl-piperazin-1-ylmethyl)- and 2-(4-benzyl-diazepan-1-ylmethyl)-1h-benzoimidazole analogues
12/31/2003CN1132817C Process for preparation of heteroarylcarboxamides
12/31/2003CN1132814C 含有磺酰胺的吲哚化合物 Sulfonamide-containing indole compound
12/31/2003CA2490109A1 Ring-substituted diphenyl azetidinones, method for the production thereof, medicaments containing said compounds, and use thereof
12/31/2003CA2490043A1 8-(biaryl) quinoline pde4 inhibitors
12/31/2003CA2489813A1 Use of thio-oxindole derivatives in treatment of hormone-related conditions
12/31/2003CA2489810A1 Use of thio-oxindole derivatives in treatment of skin disorders
12/31/2003CA2487266A1 Benzimidazole compounds and their use as estrogen agonists/antagonists
12/31/2003CA2445515A1 Transcription factor modulating compounds and methods of use thereof
12/30/2003US6670473 Inhibitors of nitric oxide synthase (nos)
12/30/2003US6670383 Pyranocoumarin compounds as a novel pharmacophore with anti-TB activity
12/30/2003US6670362 Pyridazine endothelin antagonists
12/30/2003CA2052884C Angiotensin 11 antagonists in the treatment of hyperuricemia
12/29/2003CA2433983A1 Aryl- and heteroarylcarbonylpiperazines and their use for the treatment of benign and malignant oncoses
12/25/2003WO2003105853A1 1-aryl-4-substituted piperazines derivatives for use as ccr1 antagonists for the treatment of inflammation and immune disorders
12/25/2003WO2003105846A1 2-ureido-6-heteroaryl-3h-benzoimidazole-4-carboxylic acid derivatives and related compounds as gyrase and/or topoisomerase iv inhibitors for the treatment of bacterial infections
12/25/2003US20030236420 Pharmaceuticals
12/25/2003US20030236402 A caspase-3 enzyme inhibitors, 3-(3-alkyl-amino-2-oxo-1,2-dihydro-1-pyrazinyl-alkanoylamino) -4-oxopentanoic acid; treating cardiac or cerebral ischemia or reperfusion injury, diabetes, AIDS
12/25/2003US20030236294 Anticancer agents
12/25/2003US20030236277 Viricides; immunomoderators
12/25/2003US20030236267 Benzimidazole derivatives
12/25/2003US20030236262 Dietetics; antidiabetic agents; sexual disorders
12/25/2003US20030236260 Antiarthritic agents; autoimmune diseases; anticholesterol agents; cardiovascular disorders; antiinflammatory agents
12/25/2003US20030236258 Heterocyclo-alkylsulfonyl pyrazole derivatives as anti-inflammatory/analgesic agents
12/25/2003US20030236251 Hepatitis virus viricides
12/25/2003US20030236250 Antidepressants, anxiolytic agents, analgesics, antiinflammatory agents, reduce concentration of tachykinins
12/25/2003US20030236248 Kappa agonist compounds and pharmaceutical formulations thereof
12/25/2003US20030236198 For treatment of infections by drug resistant bacteria
12/24/2003WO2003106628A2 Benzodiazepine inhibitors of mitochondial f>10< atp hydrolase and methods of inhibiting f>10< atp hydrolase
12/24/2003WO2003106452A2 Antagonists of melanin concentrating hormone receptor
12/24/2003WO2003106435A1 Fused-ring pyrimidin-4(3h)-one derivatives, processes for the preparation and uses thereof
12/24/2003WO2003106431A2 Novel hexahydro-pyridazine-3-carbocylic acid hydrazide or hydrazone derivatives, combinatorial libraries containing same, use thereof as medicines, pharmaceutical compositions containing same and methods for preparing same
12/24/2003WO2003106430A1 Benzimidazole inhibitors of poly(adp-ribosyl) polymerase
12/24/2003WO2003106416A2 Chemical process
12/24/2003WO2003105855A1 Mitotic kinesin inhibitors
12/24/2003WO2003105854A2 Substituted dihydropyrimidines, dihydropyrimidones and dihydropyrimidinethiones as calcium channel blockers
12/24/2003WO2003105847A1 Ophthalmic compositions for treating ocular hypertension
12/24/2003WO2003084940B1 Thiazolidine-4-carbonitriles and analogues and their use as dipeptidyl-peptidas inhibitors
12/24/2003WO2003061653A9 3-(imidazolyl)-2-aminopropanoic acids for use as tafi-a inhibitors for the treatment of thrombotic diseases
12/24/2003WO2002028829A3 Peptide deformylase inhibitors
12/24/2003CN1131860C 依来曲普坦氢溴酸盐一水合物 According to eletriptan hydrobromide monohydrate
12/24/2003CA2489648A1 Chemical process
12/24/2003CA2489447A1 Novel hexahydro-pyridazine-3-carbocylic acid hydrazide or hydrazone derivatives, combinatorial libraries containing same, use thereof as medicines, pharmaceutical compositions containing same and methods for preparing same
12/24/2003CA2488802A1 Ophthalmic compositions for treating ocular hypertension
12/23/2003US6667335 NMDA (N-methyl-D-aspartate)-receptor subtype selective blockers
12/23/2003US6667332 Benzisoxazolyl-pyrazole derivatives formed by salt formation with maleic acid and hydrochloric acid and cyclization with acetohydroxamic acid
12/23/2003US6667330 Cytoprotective; neuroinflammation and neurodegenerative disorders; oxidative stress related conditions