Patents for C07D 403 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group (62,587) |
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02/22/2005 | US6858628 Substituted cyclic amine metalloprotease inhibitors |
02/22/2005 | US6858609 Substituted diamino-1,3,5-triazine derivatives |
02/22/2005 | US6858606 Nitrogen compounds such as 1-(2-(4-(N'-(3-Methyl-benzylidene)-hydrazino)-6-morpholin-4-yl-pyrimidin-2 -yloxy)-ethyl)-1H-pyridin-2-one, used to control interleukin production; antiinflammatory agents |
02/22/2005 | US6858603 Acetindine derivatives, their preparation and medicaments containing them |
02/22/2005 | US6858594 Compounds and methods for treating urinary incontinence |
02/22/2005 | CA2218493C Benzimidazole compounds and their use as modulators of the gabaa receptor complex |
02/17/2005 | WO2005014602A1 Process for the preparation of tetrazole derivatives from organo boron and organo aluminium azides |
02/17/2005 | WO2005014584A1 3-(indol-1-yl)-4-(indol-3-yl)-pyrrole-2,5-diones,3-(benzimidazol-1-yl)-4-(indol-3-yl)-pyrrole-2,5-diones, and 3-(indolin-1-yl)-4-(indol-3-yl)-pyrrole-2,5-diones; their preparation and use as modulators of apoptosis |
02/17/2005 | WO2005014583A1 Antifungal azole derivatives having a fluorovinyl moiety and process for the preparation thereof |
02/17/2005 | WO2005014582A1 Quinazoline derivatives as angiogenesis inhibitors |
02/17/2005 | WO2005014573A1 Anthelmintic and insecticide pyrimidine derivatives |
02/17/2005 | WO2005014558A1 Condensed pyramidine compounds as inhibitors of voltage-gated ion channels |
02/17/2005 | WO2005014556A1 2-aminopyrimidine derivatives |
02/17/2005 | WO2005014554A1 1h-indazole-3-carboxamide compounds as mapkap kinase modulators |
02/17/2005 | WO2005014540A1 Cyclic amine base-1 inhibitors having a heterocyclic substituent |
02/17/2005 | WO2005014539A2 Pyrrole-based hmg-coa reductase inhibitors |
02/17/2005 | WO2005013997A1 Spiro-substituted tetrahydroquinazolines as corticotropin releasing factor (cfr) antagonists |
02/17/2005 | WO2005013982A1 Aminotriazole compounds useful as inhibitors of protein kinases |
02/17/2005 | WO2005013914A2 Heteroarylaminosulfonylphenyl derivatives for use as sodium or calcium channel blockers in the treatment of pain |
02/17/2005 | WO2005013909A2 Novel cathepsin k inhibitors |
02/17/2005 | WO2004110344A3 New azetidine compounds |
02/17/2005 | WO2004099131A3 Compounds having a fused, bicyclic moiety for binding to the minor groove of dsdna |
02/17/2005 | WO2004093829A3 (-)1-(4-sulfamylaryl)-3-substituted-5-heteroaryl-2 pyrazolines as inhibitors of cyclooxygenase-2 |
02/17/2005 | WO2004084813A3 Chemical compounds |
02/17/2005 | US20050038247 topoisomerase inhibitors such as [5-(4-Cyclopropylcarbamoyl-imidazol-1-yl)-7-pyrimidin-2-yl-1H-benzoimidazol-2-yl]-carbamic acid ethyl ester, used for prophylaxis of bacterial infections in mammals |
02/17/2005 | US20050038243 2, 4-pyrimidinediamine compounds and their uses |
02/17/2005 | US20050038236 Imidazolidinone derivatives |
02/17/2005 | US20050038099 3-Amido-5-substituted pyrazole derivatives and related compounds useful as bradykinin B1 receptor antagonists to relieve adverse symptoms in mammals mediated, at least in part, by bradykinin B1 receptor including pain, inflammation, septic shock, scarring process |
02/17/2005 | US20050038097 Modulate and/or inhibit tyrosine kinase signal transduction; antiproliferative agents; treating, prevention of cancer and other disease states associated with unwanted angiogenesis and/or cellular proliferation, such as diabetic retinopathy, neovascular glaucoma, rheumatoid arthritis |
02/17/2005 | US20050038095 Azolylbenzamides and analogues and their use for treating osteoporosis |
02/17/2005 | US20050038087 Derivatives of heterocycles with 5 members, their preparation and their use as medicaments |
02/17/2005 | US20050038085 Substituted benzimidazole antiviral agents |
02/17/2005 | US20050038069 Tumor necrosis factor antagonist; antiinflammatory agents; such as 2-Cyclopropyl-4-(3,5-dimethyl-4-pyridylmethoxy)-7-methoxy-3H-benzimidazole |
02/17/2005 | US20050038067 A compound with azo containing mono and a bicyclic rings attached with an aryl or heteroaryl ring; both therapeutic and diagnostic |
02/17/2005 | US20050038066 Geometrically restricted 3-cyclopentylidene-1,3-dihydroindol-2-ones as potent protein tyrosine kinase inhibitors |
02/17/2005 | US20050038057 3-[2(R)-{hydroxycarbonylpropyl-amino}-2-phenylethyl]-5-(2-fluoro-3-methoxyphenyl)-1-[2-fluoro-6-(trifluoromethyl)benzyl]-6-methyl-pyrimidine-2,4(1H,3H)-dione; utility in treatment of a variety of sex-hormone related conditions in both men and women |
02/17/2005 | US20050038056 Gonadotropin-releasing hormone receptor antagonists and methods relating thereto |
02/17/2005 | US20050038055 Spiro tetrahydroquinazolines and dihydrocyclopentapyrimidines as CRF antagonists |
02/17/2005 | US20050038050 Therapeutic treatment of autoimmune disease, transplant rejection, rheumatoid arthritis, by administering 4-(6-chloro-2,3-methylenedioxyanilino)-7-[2-(4-methylpiperazin-1-yl)ethoxy]-5-tetrahydropyran-4-yloxyquinazoline |
02/17/2005 | US20050038041 Fungicide for agriculture, horticulture |
02/17/2005 | US20050038040 Corticotropin releasing factor antagonist; antiinflammatory agents; drug abuse; analgesics; antihistamines; skin disorders; neurodegenerative disease; eating disorders;eating disorders; antiepileptic agents; cardiovascular disorders |
02/17/2005 | US20050038035 Heterocyclic amide compounds as apolipoprotein b inhibitors |
02/17/2005 | US20050038032 Quinoxaline compounds |
02/17/2005 | US20050038027 Melanocortin-4 receptor agonists; obesity, type II diabetes; such as N-(2-(2-(2,4-dichlorophenyl)ethyl)-1-oxo-2,3-dihydro-1H-isoindol-5-yl) -3-methyl-N'-(2,6,6-trimethylbicyclo(3.1.1)hept-3yl)piperazine-1-carboximidamide |
02/17/2005 | US20050038023 Inhibitors of glycogen synthase kinase-3 (gsk-3) and aurora-2, both serine/threonine protein kinases; for treating diseases such as cancer, diabetes and alzheimer's disease |
02/17/2005 | US20050038016 Arylamine-substituted quinazolinone compounds useful as alpha 1A/B adrenergic receptor antagonists |
02/17/2005 | US20050037925 Mixture with other herbicides |
02/17/2005 | DE10328533A1 New 6-amino-substituted indolinone derivatives, useful e.g. for treating tumours and angiogenesis, are inhibitors of receptor tyrosine kinases |
02/17/2005 | DE10326918A1 Substituierte Alkylamide Substituted alkyl amides |
02/17/2005 | CA2554566A1 Condensed pyramidine compounds as inhibitors of voltage-gated ion channels |
02/17/2005 | CA2539227A1 Heteroarylaminosulfonylphenyl derivatives for use as sodium or calcium channel blockers in the treatment of pain |
02/17/2005 | CA2535249A1 Spiro-substituted tetrahydroquinazolines as corticotropin releasing factor (cfr) antagonists |
02/17/2005 | CA2534975A1 Anthelmintic and insecticide pyrimidine derivatives |
02/17/2005 | CA2534811A1 Quinazoline derivatives as angiogenesis inhibitors |
02/17/2005 | CA2534528A1 3-(indol-1-yl)-4-(indol-3-yl)-pyrrole-2,5-diones,3-(benzimidazol-1-yl)-4-(indol-3-yl)-pyrrole-2,5-diones, and 3-(indolin-1-yl)-4-(indol-3-yl)-pyrrole-2,5-diones; their preparationand use as modulators of apoptosis |
02/17/2005 | CA2534494A1 Pyrrole-based hmg-coa reductase inhibitors |
02/17/2005 | CA2534422A1 Quinazoline derivatives as inhibitors of vegf receptor tyrosine kinases |
02/17/2005 | CA2534057A1 Novel gamma-secretase inhibitors |
02/17/2005 | CA2532175A1 Process for the preparation of tetrazole derivatives from organo boron and organo aluminium azides |
02/16/2005 | EP1506204A2 1-oxa-dibenzoazulenes as inhibitors of tumor necrosis factor production and intermediates for the preparation thereof |
02/16/2005 | EP1506196A2 Pyrazolopyrimidines |
02/16/2005 | EP1506190A1 (imidazol-1-yl-methyl)-pyridazine as nmda receptor blocker |
02/16/2005 | EP1506189A1 Pyrrole derivatives as inhibitors of erk2 and uses thereof |
02/16/2005 | EP1506176A1 Aminoindazole derivatives active as kinase inhibitors, process for their preparation and pharmaceutical compositions comprising them |
02/16/2005 | EP1506175A1 N-substituted tricyclic 3-aminopyrazoles as pdgf receptor inhibitors |
02/16/2005 | EP1505979A1 Phenyl substituted imidazopyridines and phenyl substituted benzimidazoles |
02/16/2005 | EP1505963A1 Hepatitis c virus inhibitors |
02/16/2005 | EP1401832B1 High molecular weight hydroxyphenylbenzotriazole uv-absorbers for thin film applications |
02/16/2005 | EP1281709B1 Novel heterocyclic compounds with anti-inflammatory activity |
02/16/2005 | CN1582285A Heteroaryl amines as glycogen synthase kinase 3beta inhibitors (GSK3 inhibitors) |
02/16/2005 | CN1582284A Aminopyrimidines and pyridines |
02/16/2005 | CN1582281A Mch受体拮抗剂 Mch receptor antagonist |
02/16/2005 | CN1582280A 3, 4-di-substituted pyridazinediones as CXC chemokine receptor antagonists |
02/16/2005 | CN1582279A Peroxisome proliferator activated receptor agonists |
02/16/2005 | CN1582277A Amide derivatives as glycogen synthase kinase 3-beta inhibitors |
02/16/2005 | CN1582274A Inhibitors of factor Xa and other serine proteases involved in the coagulation cascade |
02/16/2005 | CN1189466C New direct chain or cyclic urea, its preparing method and medicinal composition containing them |
02/15/2005 | US6855730 3-methylidenyl-2-indolinone modulators of protein kinase |
02/15/2005 | US6855726 Heterocyclic amides such as 3-(1-5-((2R,6S)-2,6-dimethyltetra-hydro-1(2H)-pyridinyl)pentyl-2-oxo-1,2 -dihydro-3-quinolinyl) benzenecarboximidamide, administered as anticoagulants or for prophylaxis of cardiovascular disorders |
02/15/2005 | US6855722 Substituted indoles and their use as integrin antagonists |
02/15/2005 | US6855715 Drugs such as 1-(3-Amino-4-chlorobenzoyl-D-phenylglycinyl)-4-(4-fluoro-2 -methylsulphonylphenyl)piperazine, used as anticoagulants |
02/15/2005 | US6855714 For therapy of inflammatory, allergic, infectious or autoimmune diseases |
02/15/2005 | US6855710 Antiproliferative agents; antitumor agents |
02/10/2005 | WO2005012914A2 Method for characterising polypeptides by maldi-tof mas spectrometry |
02/10/2005 | WO2005012294A1 2,4-pyrimidinediamine compounds for use in the treatment or prevention of autoimmune diseases |
02/10/2005 | WO2005012292A1 Gyrase inhibitors and uses thereof |
02/10/2005 | WO2005012288A1 Bicyclic imidazol derivatives against flaviviridae |
02/10/2005 | WO2005012262A1 2-aminophenyl-4-phenylpyrimidines as kinase inhibitors |
02/10/2005 | WO2005012256A1 3, 4-disubstituted 1h-pyrazole compounds and their use as cyclin dependent kinases (cdk) and glycogen synthase kinase-3 (gsk-3) modulators |
02/10/2005 | WO2005012228A1 O-coordinated metal chelates and their use in optical recording media having high storage capacity |
02/10/2005 | WO2005011700A1 INHIBITORS OF Akt ACTIVITY |
02/10/2005 | WO2005011699A1 Phenylahistin and the phenylahistin analogs, a new class of anti-tumor compounds |
02/10/2005 | WO2005011681A1 Chemical compounds |
02/10/2005 | WO2005011657A2 Piperazine derivatives and their use as therapeutic agents |
02/10/2005 | WO2005011646A2 Nitrooxy derivatives of losartan, valsatan, candesartan, telmisartan, eprosartan and olmesartan as angiotensin-ii receptor blockers for the treatment of cardiovascular diseases |
02/10/2005 | WO2004060305A3 Anti-cancer medicaments |
02/10/2005 | WO2003099793A9 1,2-azole derivatives with hypoglycemic and hypolipidemic activity |
02/10/2005 | US20050033055 Edg receptor agonists |
02/10/2005 | US20050032874 Indole derivatives |
02/10/2005 | US20050032871 Sulfonylated pyrrole-2-indolinone derivatives as kinase inhibitors |