Patents
Patents for C07D 403 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group (62,587)
02/2005
02/22/2005US6858628 Substituted cyclic amine metalloprotease inhibitors
02/22/2005US6858609 Substituted diamino-1,3,5-triazine derivatives
02/22/2005US6858606 Nitrogen compounds such as 1-(2-(4-(N'-(3-Methyl-benzylidene)-hydrazino)-6-morpholin-4-yl-pyrimidin-2 -yloxy)-ethyl)-1H-pyridin-2-one, used to control interleukin production; antiinflammatory agents
02/22/2005US6858603 Acetindine derivatives, their preparation and medicaments containing them
02/22/2005US6858594 Compounds and methods for treating urinary incontinence
02/22/2005CA2218493C Benzimidazole compounds and their use as modulators of the gabaa receptor complex
02/17/2005WO2005014602A1 Process for the preparation of tetrazole derivatives from organo boron and organo aluminium azides
02/17/2005WO2005014584A1 3-(indol-1-yl)-4-(indol-3-yl)-pyrrole-2,5-diones,3-(benzimidazol-1-yl)-4-(indol-3-yl)-pyrrole-2,5-diones, and 3-(indolin-1-yl)-4-(indol-3-yl)-pyrrole-2,5-diones; their preparation and use as modulators of apoptosis
02/17/2005WO2005014583A1 Antifungal azole derivatives having a fluorovinyl moiety and process for the preparation thereof
02/17/2005WO2005014582A1 Quinazoline derivatives as angiogenesis inhibitors
02/17/2005WO2005014573A1 Anthelmintic and insecticide pyrimidine derivatives
02/17/2005WO2005014558A1 Condensed pyramidine compounds as inhibitors of voltage-gated ion channels
02/17/2005WO2005014556A1 2-aminopyrimidine derivatives
02/17/2005WO2005014554A1 1h-indazole-3-carboxamide compounds as mapkap kinase modulators
02/17/2005WO2005014540A1 Cyclic amine base-1 inhibitors having a heterocyclic substituent
02/17/2005WO2005014539A2 Pyrrole-based hmg-coa reductase inhibitors
02/17/2005WO2005013997A1 Spiro-substituted tetrahydroquinazolines as corticotropin releasing factor (cfr) antagonists
02/17/2005WO2005013982A1 Aminotriazole compounds useful as inhibitors of protein kinases
02/17/2005WO2005013914A2 Heteroarylaminosulfonylphenyl derivatives for use as sodium or calcium channel blockers in the treatment of pain
02/17/2005WO2005013909A2 Novel cathepsin k inhibitors
02/17/2005WO2004110344A3 New azetidine compounds
02/17/2005WO2004099131A3 Compounds having a fused, bicyclic moiety for binding to the minor groove of dsdna
02/17/2005WO2004093829A3 (-)1-(4-sulfamylaryl)-3-substituted-5-heteroaryl-2 pyrazolines as inhibitors of cyclooxygenase-2
02/17/2005WO2004084813A3 Chemical compounds
02/17/2005US20050038247 topoisomerase inhibitors such as [5-(4-Cyclopropylcarbamoyl-imidazol-1-yl)-7-pyrimidin-2-yl-1H-benzoimidazol-2-yl]-carbamic acid ethyl ester, used for prophylaxis of bacterial infections in mammals
02/17/2005US20050038243 2, 4-pyrimidinediamine compounds and their uses
02/17/2005US20050038236 Imidazolidinone derivatives
02/17/2005US20050038099 3-Amido-5-substituted pyrazole derivatives and related compounds useful as bradykinin B1 receptor antagonists to relieve adverse symptoms in mammals mediated, at least in part, by bradykinin B1 receptor including pain, inflammation, septic shock, scarring process
02/17/2005US20050038097 Modulate and/or inhibit tyrosine kinase signal transduction; antiproliferative agents; treating, prevention of cancer and other disease states associated with unwanted angiogenesis and/or cellular proliferation, such as diabetic retinopathy, neovascular glaucoma, rheumatoid arthritis
02/17/2005US20050038095 Azolylbenzamides and analogues and their use for treating osteoporosis
02/17/2005US20050038087 Derivatives of heterocycles with 5 members, their preparation and their use as medicaments
02/17/2005US20050038085 Substituted benzimidazole antiviral agents
02/17/2005US20050038069 Tumor necrosis factor antagonist; antiinflammatory agents; such as 2-Cyclopropyl-4-(3,5-dimethyl-4-pyridylmethoxy)-7-methoxy-3H-benzimidazole
02/17/2005US20050038067 A compound with azo containing mono and a bicyclic rings attached with an aryl or heteroaryl ring; both therapeutic and diagnostic
02/17/2005US20050038066 Geometrically restricted 3-cyclopentylidene-1,3-dihydroindol-2-ones as potent protein tyrosine kinase inhibitors
02/17/2005US20050038057 3-[2(R)-{hydroxycarbonylpropyl-amino}-2-phenylethyl]-5-(2-fluoro-3-methoxyphenyl)-1-[2-fluoro-6-(trifluoromethyl)benzyl]-6-methyl-pyrimidine-2,4(1H,3H)-dione; utility in treatment of a variety of sex-hormone related conditions in both men and women
02/17/2005US20050038056 Gonadotropin-releasing hormone receptor antagonists and methods relating thereto
02/17/2005US20050038055 Spiro tetrahydroquinazolines and dihydrocyclopentapyrimidines as CRF antagonists
02/17/2005US20050038050 Therapeutic treatment of autoimmune disease, transplant rejection, rheumatoid arthritis, by administering 4-(6-chloro-2,3-methylenedioxyanilino)-7-[2-(4-methylpiperazin-1-yl)ethoxy]-5-tetrahydropyran-4-yloxyquinazoline
02/17/2005US20050038041 Fungicide for agriculture, horticulture
02/17/2005US20050038040 Corticotropin releasing factor antagonist; antiinflammatory agents; drug abuse; analgesics; antihistamines; skin disorders; neurodegenerative disease; eating disorders;eating disorders; antiepileptic agents; cardiovascular disorders
02/17/2005US20050038035 Heterocyclic amide compounds as apolipoprotein b inhibitors
02/17/2005US20050038032 Quinoxaline compounds
02/17/2005US20050038027 Melanocortin-4 receptor agonists; obesity, type II diabetes; such as N-(2-(2-(2,4-dichlorophenyl)ethyl)-1-oxo-2,3-dihydro-1H-isoindol-5-yl) -3-methyl-N'-(2,6,6-trimethylbicyclo(3.1.1)hept-3yl)piperazine-1-carboximidamide
02/17/2005US20050038023 Inhibitors of glycogen synthase kinase-3 (gsk-3) and aurora-2, both serine/threonine protein kinases; for treating diseases such as cancer, diabetes and alzheimer's disease
02/17/2005US20050038016 Arylamine-substituted quinazolinone compounds useful as alpha 1A/B adrenergic receptor antagonists
02/17/2005US20050037925 Mixture with other herbicides
02/17/2005DE10328533A1 New 6-amino-substituted indolinone derivatives, useful e.g. for treating tumours and angiogenesis, are inhibitors of receptor tyrosine kinases
02/17/2005DE10326918A1 Substituierte Alkylamide Substituted alkyl amides
02/17/2005CA2554566A1 Condensed pyramidine compounds as inhibitors of voltage-gated ion channels
02/17/2005CA2539227A1 Heteroarylaminosulfonylphenyl derivatives for use as sodium or calcium channel blockers in the treatment of pain
02/17/2005CA2535249A1 Spiro-substituted tetrahydroquinazolines as corticotropin releasing factor (cfr) antagonists
02/17/2005CA2534975A1 Anthelmintic and insecticide pyrimidine derivatives
02/17/2005CA2534811A1 Quinazoline derivatives as angiogenesis inhibitors
02/17/2005CA2534528A1 3-(indol-1-yl)-4-(indol-3-yl)-pyrrole-2,5-diones,3-(benzimidazol-1-yl)-4-(indol-3-yl)-pyrrole-2,5-diones, and 3-(indolin-1-yl)-4-(indol-3-yl)-pyrrole-2,5-diones; their preparationand use as modulators of apoptosis
02/17/2005CA2534494A1 Pyrrole-based hmg-coa reductase inhibitors
02/17/2005CA2534422A1 Quinazoline derivatives as inhibitors of vegf receptor tyrosine kinases
02/17/2005CA2534057A1 Novel gamma-secretase inhibitors
02/17/2005CA2532175A1 Process for the preparation of tetrazole derivatives from organo boron and organo aluminium azides
02/16/2005EP1506204A2 1-oxa-dibenzoazulenes as inhibitors of tumor necrosis factor production and intermediates for the preparation thereof
02/16/2005EP1506196A2 Pyrazolopyrimidines
02/16/2005EP1506190A1 (imidazol-1-yl-methyl)-pyridazine as nmda receptor blocker
02/16/2005EP1506189A1 Pyrrole derivatives as inhibitors of erk2 and uses thereof
02/16/2005EP1506176A1 Aminoindazole derivatives active as kinase inhibitors, process for their preparation and pharmaceutical compositions comprising them
02/16/2005EP1506175A1 N-substituted tricyclic 3-aminopyrazoles as pdgf receptor inhibitors
02/16/2005EP1505979A1 Phenyl substituted imidazopyridines and phenyl substituted benzimidazoles
02/16/2005EP1505963A1 Hepatitis c virus inhibitors
02/16/2005EP1401832B1 High molecular weight hydroxyphenylbenzotriazole uv-absorbers for thin film applications
02/16/2005EP1281709B1 Novel heterocyclic compounds with anti-inflammatory activity
02/16/2005CN1582285A Heteroaryl amines as glycogen synthase kinase 3beta inhibitors (GSK3 inhibitors)
02/16/2005CN1582284A Aminopyrimidines and pyridines
02/16/2005CN1582281A Mch受体拮抗剂 Mch receptor antagonist
02/16/2005CN1582280A 3, 4-di-substituted pyridazinediones as CXC chemokine receptor antagonists
02/16/2005CN1582279A Peroxisome proliferator activated receptor agonists
02/16/2005CN1582277A Amide derivatives as glycogen synthase kinase 3-beta inhibitors
02/16/2005CN1582274A Inhibitors of factor Xa and other serine proteases involved in the coagulation cascade
02/16/2005CN1189466C New direct chain or cyclic urea, its preparing method and medicinal composition containing them
02/15/2005US6855730 3-methylidenyl-2-indolinone modulators of protein kinase
02/15/2005US6855726 Heterocyclic amides such as 3-(1-5-((2R,6S)-2,6-dimethyltetra-hydro-1(2H)-pyridinyl)pentyl-2-oxo-1,2 -dihydro-3-quinolinyl) benzenecarboximidamide, administered as anticoagulants or for prophylaxis of cardiovascular disorders
02/15/2005US6855722 Substituted indoles and their use as integrin antagonists
02/15/2005US6855715 Drugs such as 1-(3-Amino-4-chlorobenzoyl-D-phenylglycinyl)-4-(4-fluoro-2 -methylsulphonylphenyl)piperazine, used as anticoagulants
02/15/2005US6855714 For therapy of inflammatory, allergic, infectious or autoimmune diseases
02/15/2005US6855710 Antiproliferative agents; antitumor agents
02/10/2005WO2005012914A2 Method for characterising polypeptides by maldi-tof mas spectrometry
02/10/2005WO2005012294A1 2,4-pyrimidinediamine compounds for use in the treatment or prevention of autoimmune diseases
02/10/2005WO2005012292A1 Gyrase inhibitors and uses thereof
02/10/2005WO2005012288A1 Bicyclic imidazol derivatives against flaviviridae
02/10/2005WO2005012262A1 2-aminophenyl-4-phenylpyrimidines as kinase inhibitors
02/10/2005WO2005012256A1 3, 4-disubstituted 1h-pyrazole compounds and their use as cyclin dependent kinases (cdk) and glycogen synthase kinase-3 (gsk-3) modulators
02/10/2005WO2005012228A1 O-coordinated metal chelates and their use in optical recording media having high storage capacity
02/10/2005WO2005011700A1 INHIBITORS OF Akt ACTIVITY
02/10/2005WO2005011699A1 Phenylahistin and the phenylahistin analogs, a new class of anti-tumor compounds
02/10/2005WO2005011681A1 Chemical compounds
02/10/2005WO2005011657A2 Piperazine derivatives and their use as therapeutic agents
02/10/2005WO2005011646A2 Nitrooxy derivatives of losartan, valsatan, candesartan, telmisartan, eprosartan and olmesartan as angiotensin-ii receptor blockers for the treatment of cardiovascular diseases
02/10/2005WO2004060305A3 Anti-cancer medicaments
02/10/2005WO2003099793A9 1,2-azole derivatives with hypoglycemic and hypolipidemic activity
02/10/2005US20050033055 Edg receptor agonists
02/10/2005US20050032874 Indole derivatives
02/10/2005US20050032871 Sulfonylated pyrrole-2-indolinone derivatives as kinase inhibitors