Patents
Patents for C07D 403 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group (62,587)
07/2006
07/05/2006EP1676575A2 Mucin production inhibitor
07/05/2006EP1675856A1 Novel tetraydrospiro{piperidine-2,7'-pyrrolo [3,2]pyridine} derivatives and novel indole derivatives useful in the treatment of 5-ht6 receptor -related disorders
07/05/2006EP1675852A1 7-amino alkylidenyl-heterocyclic quinolones and naphthyridones
07/05/2006EP1675849A1 Benzimidazolyl derivatives
07/05/2006EP1675838A1 1-benzoyl substituted diazepine derivatives as selective histamine h3 receptor agonists
07/05/2006EP1675836A1 Derivatives of 4-phenylthiazoles and 4-phenylimidazoles and the use thereof as medicaments for treating neurodegenerative diseases, pain and epilepsy
07/05/2006EP1675835A1 Methods of preparation of dehydro-diketopiperazines in liquid phase or of solid supported phase
07/05/2006EP1675826A1 Compounds having crth2 antagonist activity
07/05/2006EP1675585A2 Large conductance calcium-activated k channel opener
07/05/2006EP1399441B1 N-aroyl cyclic amine derivatives as orexin receptor antagonists
07/05/2006CN1798748A Inhibitors of cyclin-dependent kinases, compositions and uses related thereto
07/05/2006CN1798740A Nitrogen-containing heteroaryl derivatives
07/05/2006CN1798738A Biaryl substituted pyrazoles as sodium channel blockers
07/05/2006CN1798734A Novel compounds and compositions as protein kinase inhibitors
07/05/2006CN1798556A Fused indoles as dipeptidyl peptidase inhibitors for the treatment or prevention of diabetes
07/05/2006CN1796385A New method for prepraring Voriconazole intermediate of antifungal drug
07/05/2006CN1262547C Phenyl-and aminophenyl-alkyl sulfonamide and urea derivative
07/04/2006US7071332 Indolinone derivatives as protein kinase/phosphatase inhibitors
07/04/2006US7071224 Antihistamines; bronchodilator agents; respiratory system disorders
07/04/2006US7071213 Cannabinoid receptor ligands
07/04/2006US7071212 N-(4-carbamimidoyl-phenyl)-glycine derivatives
07/04/2006US7071201 Serotonin antagonism; muscle relaxant for myotonia; such as 1-(1-(2-(4-methoxyphenyl)ethyl)piperidin-4-yl)-7-methoxy-1,2,3,4 -tetrahydroquinoline
07/04/2006US7071196 Piperazine derivatives as antagonists of tachykinins, including substance P and other neurokinins.
07/04/2006US7071189 Heterocyclic compounds as antitumor agents with benzimidazole group and morpholine group, triazoline or pyrimidine heterocycles
07/04/2006US7071184 Protease inhibitors
07/04/2006US7071182 Antagonists of melanin concentrating hormone effects on the melanin concentrating hormone receptor
07/04/2006US7071180 Eating disorders; cognition activators; psychological disorders; anxiolytic agents; sexual disorders; incontinence; antidepressants
07/04/2006CA2332066C Tetrazole compounds as thyroid receptor ligands
07/04/2006CA2200579C Phenyl-oxo-alkyl-(4-piperidinyl)benzoate derivatives as colon motility enhancing agents
06/2006
06/29/2006WO2006068991A1 Cycloalkyl lactam derivatives as inhibitors of 11-beta-hydroxysteroid dehydrogenase 1
06/29/2006WO2006067976A1 Organic compound, charge-transporting material, and organic electroluminescent element
06/29/2006WO2006067529A1 Piperidine and azetidine derivatives as glyt1 inhibitors
06/29/2006WO2006067472A1 Parp inhibitors
06/29/2006WO2006067466A2 Pyrazines and pyridines and derivatives thereof as therapeutic compounds
06/29/2006WO2006067462A1 1,6 - substituted (3r,6r) -3- (2,3-dihydro-1h-inden-2-yl)-2,5-piperazinedione derivatives as oxytocin receptor antagonists for the treatment of pre-term labour, dysmenorrhea and endometriosis
06/29/2006WO2006067428A2 1, 2-diphenyl-imidazole derivatives and their use as cb1 receptor ligands
06/29/2006WO2006067392A2 Indole derivatives for the treatment of tuberculosis
06/29/2006WO2006067391A1 Pyrazolylamino substituted quinazoles for the treatment of cancer
06/29/2006WO2006067139A1 Triazolone, tetrazolone and imidazolone derivatives for use as alpha-2c adrenoreceptor antagonists
06/29/2006WO2006066929A1 Quaternary ammonium salts as m3 antagonists
06/29/2006WO2006066928A1 Pyrrolinidium derivatives as m3 muscarinic receptors
06/29/2006WO2006066896A2 Pyrrolidine derivatives for the treatment of a disease depending on the activity of renin
06/29/2006WO2006066885A1 Substituted n-heterocyclic compounds and their use as dopamine d3 receptor ligands
06/29/2006US20060142579 crystallizing from a solvent selected from 1-propanol, 2-propanol, 1-butanol, ethyl acetate, acetonitrile
06/29/2006US20060142578 Novel process
06/29/2006US20060142577 4-Diethylamino-N-[4-methyl-3-[[4-(3-pyridinyl)-2-pyrimidinyl]amino]phenyl]-3-(trifluoromethyl)-benzamide; disease which responds to an inhibition of protein kinase activity, especially a neoplastic disease; leukemia
06/29/2006US20060142575 Hetereoaryl nitrile derivatives
06/29/2006US20060142572 Inhibitors of ERK protein kinase and uses thereof
06/29/2006US20060142571 improved ability to inhibit the replication of mutant strains of drug or multidrug resistant HIV strains; Indene/benzofuran Substituted Pyrimidines
06/29/2006US20060142553 Novel azo dye compound
06/29/2006US20060142506 Heterobifunctional poly(ethylene glycol) and uses thereof
06/29/2006US20060142365 Benzimidazole compounds and antiviral uses thereof
06/29/2006US20060142364 2-tert-Butyl-1-(cyclohexylmethyl)-N,N-bis(2,2,2-trifluoroethyl)-1H-benzimidazole-5-carboxamide; treating pain
06/29/2006US20060142361 Azole derivatives and methods for making the same
06/29/2006US20060142343 Pyrrolines
06/29/2006US20060142333 e.g. N-(1-Methyl-1,2,3,4-tetrahydroquinolin-7-yl)-1,1'-biphenyl-4-carboxamide; capsaicin recepor antagonist; analgesic; neuropathic, postoperative, postrheumatoid arthritic, back, cancer pain, neuralgia, dental pain, headache, migraine, diabetic and HIV-related neuropathy
06/29/2006US20060142329 Substituted fused N-heteroaryl compounds such as imidazo[1,5a]- or [1,2s]pyridines, e.g., 3-[3-(Pyrrolylphenoxy-2-hydroxypropyl)aminoalkyl]imidazo[1,5-a]pyridine derivatives, especially HCl salts; treating obesity and type 2 diabetes
06/29/2006US20060142328 Beta 3 adrenergic agonists
06/29/2006US20060142327 Beta 3 adrenergic agonists
06/29/2006US20060142325 Fused bicyclic-substituted amines as histamine-3 receptor ligands
06/29/2006US20060142318 eating disorders of disturbed fundus such as dyspepsia, early satiety, bloating, anorexia; fundic relaxation; 1-[1-[(2,3-dihydro[1,4]dioxino[2,3-b]pyridin-3-yl)methyl]-4-piperidinyl]-2-imidazolidinone; improved pharmacokinetics, less vasoconstriction, side effect reduction, sustain release
06/29/2006US20060142314 2-substituted-4-(indazol-5-ylamino)-6,7-dimethoxyquinazoline compounds; use treating hypertension, atherosclerosis, restenosis, cerebral ischemia or vasospasm, neurodegeneration, spinal cord injury, cancer, thrombotic disorders, asthma, glaucoma, osteoporosis or erectile dysfunction
06/29/2006US20060142313 2-substituted-4-(indazolamino)quinazoline compounds; use treating hypertension, atherosclerosis, restenosis, cerebral ischemia or vasospasm, neurodegeneration, spinal cord injury, cancer, thrombotic disorders, asthma, glaucoma, osteoporosis or erectile dysfunction
06/29/2006US20060142307 Controlling intraocular pressure
06/29/2006US20060142302 Chemical compounds
06/29/2006US20060142301 Substituted 1-benzyl-4-substituted piperazine analogues
06/29/2006US20060142300 Anhydrous crystalline forms of I and II of 1-cyclopropyl-6-fluoro-8-methoxy-7-(3-methyl-1- piperazinyl) 4-oxo-1, 4-dihydroquinoline-3-carboxylic acid (gatifloxacin)
06/29/2006US20060142299 Crystalline aripiprazole solvates
06/29/2006US20060142293 e.g. 4-[5-(Piperidine-1-carbonyl)-furan-2-ylmethyl]-2H-phthalazin-1-one; enzyme poly(ADP-ribose)polymerase (synthase)-1 or poly ADP-ribosyltransferase (PARP-1) inhibitor; anticarcinogenic agent with BRCA2 deficient phenotype; septic shock; ischemic injury; hemorrhagic shock; multiple sclerosis
06/29/2006US20060142292 Water-soluble phenylpyridazine derivative and medicine containing the same
06/29/2006US20060142281 Indolinone derivatives
06/29/2006US20060142264 Novel amide derivatives
06/29/2006US20060142263 Such as 5-bromo-thiophene-2-carboxylic acid-{1-[3-chloro-4-(2-oxo-[1,3]oxazinan-3-yl)-phenyl]-5-oxo-pyrrolidin-3-yl}-amide
06/29/2006US20060138408 Multifunctional linker molecules for tuning electronic charge transport through organic-inorganic composite structures and uses thereof
06/29/2006CA2591827A1 1,6 - substituted (3r,6r) -3- (2,3-dihydro-1h-inden-2-yl)-2,5-piperazinedione derivatives as oxytocin receptor antagonists for the treatment of pre-term labour, dysmenorrhea and endometriosis
06/29/2006CA2591208A1 Pyrazines and pyridines and derivatives thereof as therapeutic compounds
06/29/2006CA2589648A1 Fused pyrazole derivatives and methods of treatment of metabolic-relateddisorders thereof
06/29/2006CA2589331A1 Pyrrolidine derivatives for the treatment of a disease depending on the activity of renin
06/29/2006CA2589133A1 Quaternary ammonium salts as m3 antagonists
06/29/2006CA2588220A1 Heteroaromatic derivatives useful as anticancer agents
06/29/2006CA2588028A1 Triazolone, tetrazolone and imidazolone derivatives for use as alpha-2c adrenoreceptor antagonists
06/29/2006CA2587664A1 Compounds with kv4 ion channel activity
06/28/2006EP1674466A1 2,5- and 2,6-disubstituted benzazole analogues useful as protein kinase inhibitors
06/28/2006EP1674097A1 Compounds effecting glucokinase
06/28/2006EP1673369A1 Benzimidazole derivatives, compositions containing them, preparation thereof and uses thereof
06/28/2006EP1673357A2 Heteroarylaminosulfonylphenyl derivatives for use as sodium or calcium channel blockers in the treatment of pain
06/28/2006EP1673355A1 Substituted triazole derivatives as oxytocin antagonists
06/28/2006EP1673353A1 Transition state structure and inhibitors of thymidine phosphorylases
06/28/2006EP1673350A2 Method for producing acyl urea derivatives, salts of said acyl urea derivatives, and the use thereof as pesticides
06/28/2006EP1673348A2 Benzoimidazole compounds
06/28/2006EP1673082A2 Dual alanyl aminopeptidase and dipeptidyl peptidase iv inhibitors for functionally influencing different cells and for treating immunological, inflammatory, neuronal and other diseases
06/28/2006EP1673081A1 Indoles and azaindoles as antiviral agents
06/28/2006EP1255536B1 Indolinone derivatives for modulation of c-kit tyrosine protein kinase
06/28/2006CN1795193A N-acyl nitrogen heterocyles as ligands of peroxisome proliferator-activated receptors
06/28/2006CN1795188A Inhibitors of serine proteases, particularly hcv ns3-ns4a protease
06/28/2006CN1795187A Novel ido inhibitors and methods of use
06/28/2006CN1795179A Novel imidazole derivatives, the production thereof, and the use of the same as a medicament
06/28/2006CN1795177A 1,2,4-substituerte 1,2,3,4-tetrahydro-and 1,2 dihydro-quinoline and 1,2,3,4-tetrahydro-quinoxaline derivatives as cetp inhibitors for the treatment of atherosclerosis and obesity
06/28/2006CN1795176A Azabicyclo derivatives as muscarinic receptor antagonists
06/28/2006CN1795174A Novel substituted 3-sulfur indoles