Patents
Patents for C07D 403 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group (62,587)
08/2006
08/24/2006CA2598897A1 Fungicidal pyrazine derivatives
08/24/2006CA2598076A1 Chemical compounds
08/24/2006CA2597896A1 1h-imidazole derivatives as cannabinoid cb2 receptor modulators
08/24/2006CA2597813A1 Chemical compounds
08/24/2006CA2597594A1 Azolylacylguanidines as beta-secretase inhibitors
08/24/2006CA2597033A1 1,5-diarylpyrrole derivatives, preparation method thereof and application of same in therapeutics
08/23/2006EP1693372A1 Novel Sulfamides and their use as endothelin receptor antagonists
08/23/2006EP1693365A1 Inhibitors of dipeptidyl peptidase IV
08/23/2006EP1692129A1 Keto lactam compounds and use thereof
08/23/2006EP1692128A1 Indazole compounds and methods of use thereof as protein kinase inhibitors
08/23/2006EP1692116A1 1,2,3-triazole amide derivatives as inhibitors of cytokine production
08/23/2006EP1692114A1 Novel benzimidazole and imidazopyridine derivatives and use thereof as a medicament
08/23/2006EP1692113A1 Aryl imidazoles and their use as anti-cancer agents
08/23/2006EP1691810A1 Substituted piperazines
08/23/2006EP1691803A1 N-alkyl pyrroles as hmg-coa reductase inhibitors
08/23/2006EP1633346B1 Pyrrolidin-1, 2- dicarboxylic acid- 1- (4- ethinyl- phenyl) - amid|- 2- (phenyl)- amid| derivative as inhibitors of coagulation factor xa and viia for the treatment of thrombosis
08/23/2006CN1823063A Quinoline derivatives as phosphodiesterase inhibitors
08/23/2006CN1823060A Improved process for preparing alpha-polymorphic eletriptan hydrobromide
08/23/2006CN1823059A Selective D1/dD receptor antagonists for the treatment of obesity and CNS disorders
08/23/2006CN1823057A Biaryl piperazinyl-pyridine analogues
08/23/2006CN1823056A Trisubstituted aryl and heteroaryl derivatives as modulatorsof metabolism and the prophylaxis and treatment of disorders related thereto
08/23/2006CN1823048A Substituted pyrimidin-4-ylamina analogues as vanilloid receptor ligands
08/23/2006CN1823043A Hydroxypyridine cgrp receptor antagonists
08/23/2006CN1271068C Novel method for preparing olmesartan
08/23/2006CN1271052C Sulphonamide derivatives, the preparation thereof and the application of same as medicaments
08/22/2006US7094904 Process for preparing monohydrate and crystal modifications of fluconazole
08/22/2006US7094869 Animal growth regulators
08/22/2006US7094808 Antineoplastic polyamines capable of uptake by a target cell upon administration to a human or non-human animal, and upon uptake bind via an electrostatic interaction between positively charged nitrogen and biological counter- anions
08/22/2006US7094796 Coupling product between tryptamine and an alpha-amino acid, process for its preparation as well as its application in the neurocosmetic field
08/22/2006US7094794 used for lowering the blood glucose and for the prevention and treatment of diabetes
08/22/2006US7094790 containing a pyrrole ring, e.g., 4-{2-[2-(2-(R)-Methyl-pyrrolidin-1-yl)-ethyl]-benzothiazol-5-yl}-benzonitrile; useful for treating conditions and disorders related to memory and cognition processes, neurological processes, cardiovascular function, and body weight.
08/22/2006US7094781 Sulfamides and their use as endothelin receptor antagonists
08/22/2006US7094780 3-aminoquinazolin-2,4-dione antibacterial agents
08/22/2006US7094779 2-(3-indolylmethyl)-1-benzoyl-4-oxime-piperazine derivatives, e.g., 1-{(2R)-1-[3,5-bis(trifluoromethyl)benzoyl]-2-(1H-indol-3-ylmethyl)-piperazin-4-yl}-2-propanone O-[2-(dimethylamino)-ethyl]oxime, used for treatment of CNS disorders.
08/22/2006US7094778 Nervous system disorders; muscular disorders; urogenital disorders; gastrointestinal disorders; repiratory system disorders; antiallergens; side effect reduction
08/22/2006US7094777 5-HT2A receptor ligands
08/22/2006CA2270301C Hydroxyindoles, their use as inhibitors of phosphodiesterase 4, and processes for their preparation
08/22/2006CA2242102C Quinazoline derivatives as antitumor agents
08/17/2006WO2006086657A1 Process for preparing 2,3-disubstituted indoles
08/17/2006WO2006085685A1 Pyrazole compound
08/17/2006WO2006084882A2 Substituted 4-(indol-3-yl)quinazolines and their use
08/17/2006WO2006084854A2 [1,2,4]-dithiazoli(di)ne derivatives, inducers of gluthathione-s-transferase and nadph quinone oxido-reductase, for prophylaxis and treatment of adverse conditions associated with cytotoxicity in general and apoptosis in particular
08/17/2006WO2006076646A3 Heteroaryl substituted quinolin-4-ylamine analogues
08/17/2006WO2006060122A9 Cardiotonic compounds with inhibitory activity against beta-adrenergic receptors and phosphodiesterase
08/17/2006WO2006055734A3 3-phenyl-pyrazole derivatives as modulators of the 5-ht2a serotonin receptor useful for the treatment of disorders related thereto
08/17/2006WO2005107762A3 Certain chemical entities, compositions, and methods
08/17/2006WO2005086895A3 Ion channel modulators
08/17/2006US20060183917 Processes and compounds for the preparation of substituted naphthylindole derivatives
08/17/2006US20060183916 By direct ortho-metallation of (tetrazol-5- gamma l)benzene; useful intermediates for the preparation of angiotensin II antagonists used, for example, in the treatment of hypertension, anxiety, glaucoma and heart failure; provides high yields, is less costly than known procedures
08/17/2006US20060183902 Dihydroindolyl methanones as alpha 1a/1d adrenoreceptor modulators for the treatment of benign prostatic hypertrophy and lower urinary tract symptoms
08/17/2006US20060183901 Crystalline form of an indazole-carboxamide compound
08/17/2006US20060183897 Biaryl substituted triazoles as sodium channel blockers
08/17/2006US20060183785 For the treatment of pain; epilepsy, manic depression, bipolar disorder, depression, anxiety and diabetic neuropathy; 5-Methyl-1-[2'-(trifluoromethoxy)-1,1'-biphenyl-3-yl]-1H-pyrazole-3-carboxamide
08/17/2006US20060183784 Human growth hormone antagonists
08/17/2006US20060183780 Lipoxygenase (e.g. 15-lipoxygenase) inhbitors; less toxic; longer acting; more potent; fewer side effects; easily absorbed; higher oral bioavailability and/or lower clearance; 4-Methyl-1-(pyridine-2-sulfonyl)pyrazole-3-carboxylic acid (2-chloro-4-fluorophenyl)amide
08/17/2006US20060183772 To inhibit tumor growth in an animal; to induce apoptosis
08/17/2006US20060183763 Novel pyrrolidyl derivatives of heteroaromatic compounds
08/17/2006US20060183762 3-aminoquinazolin-2,4-dione antibacterial agents
08/17/2006US20060183752 Process for preparing 2, 3-disubstituted indoles
08/17/2006US20060183745 Vanilloid receptor ligands and their use in treatments
08/17/2006US20060183742 Pyrazolidine-1,2-dicarboxyldiphenylamide derivatives as coagulation factor xa inhibitors for the treatment of thromboses
08/17/2006US20060183741 Treatment of associated conditions and disorders such as gastrointestinal reflux disorders, eating disorders leading to obesity and irritable bowel syndrome
08/17/2006US20060183694 Serine protease inhibition via 1-{[1-(2-Methoxycarbonylamino-3,3-dimethyl-butyryl)-4-(7-methoxy-2-phenyl-quinolin-4-yloxy)-pyrrolidine-2-carbonyl]-amino}-2-vinyl-cyclopropanecarboxylic acid
08/17/2006US20060182751 Heterocyclic-substituted bis-1,8 naphthalimide compounds, antibody drug conjugates, and methods of use
08/17/2006US20060179586 Cationic direct dyes
08/17/2006CA2597680A1 Process for preparing 2,3-disubstituted indoles
08/17/2006CA2597523A1 [1,2,4]-dithiazoli(di)ne derivatives, inducers of gluthathione-s-transferase and nadph quinone oxido-reductase, for prophylaxis and treatment of adverse conditions associated withcytotoxicity in general and apoptosis in particular
08/16/2006EP1689740A1 Pyrazolyl and imidazolyl pyrimidines
08/16/2006EP1689739A1 Azole-based kinase inhibitors
08/16/2006EP1689729A1 Tetronic and tetramic acids as inhibitors of beta-secrease
08/16/2006EP1689722A2 4-aminopyrimidine derivatives for treatment of hyperproliferative disorders
08/16/2006EP1689720A1 Pyrazolyl derivatives in the form of drugs for treating acute or chronic neuronal regressions
08/16/2006EP1689715A1 Tubulin inhibitors
08/16/2006EP1689710A1 Indole derivatives for use as chemical uncoupler
08/16/2006EP1689709A1 N-sulfonyldicarboximide containing tethering compounds
08/16/2006EP1689406A2 Heterocyclic inhibitors of mek and methods of use thereof
08/16/2006EP1689403A2 Heteroaryl-hydrazone compounds
08/16/2006EP1689392A1 N-heteroaryl indole carboxamides and analogues thereof, for use as glucokinase activators in the treatment of diabetes
08/16/2006EP1689387A2 Bicyclic inhibitors of mek and methods of use thereof
08/16/2006EP1689376A2 Diaryl urea derivatives in the treatment of protein kinase dependent diseases
08/16/2006EP1689233A2 Bicyclic inhibitors of mek and methods of use thereof
08/16/2006EP1487437B1 Use of selective ep4 receptor agonists for the treatment of diseases
08/16/2006EP1259234B1 3-heteroarylidenyl-2-indolinone compounds for modulating protein kinase activity and for use in cancer chemotherapy
08/16/2006EP1019075B9 Beta 2-adrenergic receptor agonists
08/16/2006CN1820003A Pyrrole-2, 5-dithione derivatives as liver X receptor modulators
08/16/2006CN1820002A Novel benzimidazole compound
08/16/2006CN1819829A Pyrimidine-2, 4-dione derivatives as gonadotropin-releasing hormone receptor antagonists
08/16/2006CN1817868A Group of ornidazole deriative for preventing anaerobe infection and production thereof
08/16/2006CN1269813C Imidazolo-5-yl-2-anilino-pyrimidines as agents for inhibition of cell proliferation
08/16/2006CN1269807C Aryl substituted piperazine for curing benign prostatauxe
08/16/2006CN1269804C Metalloproteinase inhibitors
08/15/2006US7091380 Bradykinin B1 antagonists or inverse agonists, for prophylaxis and therapy of pain and inflammation
08/15/2006US7091350 Produce powerful, particularly chromatic and bright colorations, in red tones, and which are relatively unselective and are stable to outside factors
08/15/2006US7091343 Compositions useful as inhibitors of protein kinases
08/15/2006US7091247 urotensin antagonists; vasoactive agents
08/15/2006US7091220 Substituted indole Mannich bases
08/15/2006US7091204 Sulfonamides
08/15/2006US7091201 Arylalkane-sulfonamides having endothelin-antagonist activity
08/15/2006US7091200 adrenoceptor or G-protein coupled receptors inhibitors such as 3-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)-6,7-dimethoxy-2H-benzo[1,2,4]-thiadiazine-1,1-dioxide and carriers, used for prophylaxis of urogenital disorders, or as analgesics
08/15/2006US7091199 Thienoisoxazole phenoxy unsubstituted ethyl and propyl derivatives useful as d4 antagonists