Patents
Patents for C07D 403 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group (62,587)
07/2006
07/12/2006EP1679308A1 Novel indazole derivative
07/12/2006EP1679073A1 2-(phenyl)-2h-pyrazole-3-carboxylic acid-n-4-(imino-heterocyclyl)-phenyl-amide derivatives and relates compounds for use as inhibitors of the coagulation factors xa and/or viia for treating thromboses
07/12/2006EP1678258A1 Cyanine dye labelling reagents
07/12/2006EP1678170A1 Use of a compound of formula (i) as an inhibitor of aromatase for therapeutic purposes and compounds of formula (1) thereas
07/12/2006EP1678167A1 Substituted cyclic hydroxamates as inhibitors of matrix metalloproteinases
07/12/2006EP1678163A1 Novel imidazole derivatives and their use as pharmaceutical agents
07/12/2006EP1678147A1 Pharmaceutically active 4,6-disubstituted aminopyrimidine derivatives as modulators of protein kinases
07/12/2006EP1678145A2 Benzimidazoles useful as modulators of ion channels
07/12/2006EP1678144A1 1,5,7-TRISUBSTITUTED BENZIMIDAZOLE DERIVATIVES AND THEIR USE FOR MODULATING THE GABA-a RECEPTOR COMPLEX
07/12/2006EP1678133A1 Sequence selective pyrrole and imidazole polyamide metallocomplexes
07/12/2006EP1677786A1 5-substituted 2-(phenylmethyl)thio-4-phenyl-4h-1,2,4-triazole derivatives and related compounds as gaba-agonists for the treatment of urinary incontinence and related diseases
07/12/2006CN1802368A Heteroaryl-substituted imdazole derivatives as glutamate receptor antagonists
07/12/2006CN1802357A Aminopyrimidine derivatives and their medical use
07/12/2006CN1802351A Substituted 3-alkyl and 3-alkenyl azetidine derivatives
07/12/2006CN1802159A 2-phenoxy- and 2-phenylsulfomamide derivatives with CCR3 antagonistic activity for the treatment of asthma and other inflammatory or immunological disorders
07/12/2006CN1800185A Substituted sulfonamide compounds, process for their use as medicament for the treatment of CNS disorders, obesity and type II diabetes.
07/12/2006CN1800179A Method for preparing candestartan
07/12/2006CN1800165A Cationic symmetric 2-imidazolium diazo compounds with a cationic linking group, compositions comprising them, a dying process and kit thereof
07/12/2006CN1263746C Pyridazinone derivatives
07/11/2006US7074921 Process for the preparation of 3,7-disubstituted-2,3,4,5-tetrahydro-1H-1,4-benzodiazepine compounds
07/11/2006US7074814 Antiinflammatory agents; cardiovascular disorders; anticancer agents; antiarthritic agents ; psoriasis
07/11/2006US7074810 Triazolone and triazolethione derivatives as inhibitors of matrix metalloproteinases and/or TNF-α converting enzyme
07/11/2006US7074801 Nitrogen-containing condensed cyclic compound having a pyrazolyl group as a substituent group and pharmaceutical composition thereof
07/11/2006US7074800 Quinazoline derivatives as angiogenesis inhibitors
07/11/2006US7074799 To treat one or more conditions responsive to capsaicin receptor modulation, such as pain, itch, urinary incontinence, cough, hiccup, and/or obesity
07/11/2006US7074796 High affinity for D4 receptors; treatment of psychological disorders such as schizophrenia, generalised anxiety disorder, panic disorder, and obsessive compulsive disorder.
07/11/2006US7074794 pyrrolo-2yl-carbonyl-amino compounds; dipeptidyl peptidase inhibitor
07/11/2006US7074793 KInase inhibitor; Alzheimer's disease; central nervous system disorders; antiinflamamtory agents; skin disorders; osteoporosis; atherosclerosis; restenosis; thrombosis; antidiabetic agents; viricides; fungicides
07/11/2006US7074789 Kinase inhibitors
07/11/2006US7074786 Histogranin-like peptides, processes for their preparation and uses thereof
07/11/2006US7074784 Medicaments against viral diseases
07/11/2006US7074782 Administering to a patient suffering from caspase mediated diseses, an effective amount of a mono,bi or tri-heterocyclic ring containing nitrogen atom attached to ester or thioester to form carbamate group, as caspase inhibitor
07/11/2006US7074781 E.g., 1-(2-methyl-4-(2,3,4,5-tetrahydro-1-benzazepin-1-ylcarbonyl)benzylcarbamoyl)-L-proline-N,N-dimethylamide; control of urinary incontinence and bleeding disorders.
07/11/2006US7074534 Polymeric charge transport compositions and electronic devices made with such compositions
07/11/2006CA2269810C N-substituted 2-cyanopyrrolidines
07/11/2006CA2260999C Heterocyclic compounds, their production and use in tyrosine kinase inhibition
07/11/2006CA2246783C Mcbi analogs of cc-1065 and the duocarmycins
07/11/2006CA2208630C 4-amino-2-ureidopyrimidine-5-carboxamides, processes for their preparation, pharmaceuticals comprising these compounds, and their use
07/11/2006CA2206532C Novel amidinonaphthyl derivative or salt thereof
07/06/2006WO2006071958A1 Compounds useful as chemokine receptor antagonists
07/06/2006WO2006071644A1 Selective inhibitors of erk protein kinases and uses therof
07/06/2006WO2006070284A1 Pyrrolidyl derivatives of heteroaromatic compounds as phosphodiesterase inhibitors
07/06/2006WO2006070202A1 Pyrazole derivatives having kinase modulating activity
07/06/2006WO2006070198A1 Pyrazole derivatives as that modulate the activity of cdk, gsk and aurora kinases
07/06/2006WO2006070195A1 Pyrazole compounds that modulate the activity of cdk, gsk and aurora kinases
07/06/2006WO2006069740A1 2, 5 and 2, 6-disubstituted benzazole analogues useful as protein kinase inhibitors
07/06/2006WO2006069525A1 Aminopyrimidine compounds and their salts, process for preparation and pharmaceutical use thereof
07/06/2006WO2006053274A3 2-amino-1-functionalized tetralin derivatives and related glycogen phosphorylase inhibitors
07/06/2006WO2006050389A3 Pyridazine compounds, compositions and methods
07/06/2006WO2006047415A3 FACTOR Xa COMPOUNDS
07/06/2006WO2006011859A3 Preparation of hydrochloride salts of tetrazole derivative
07/06/2006WO2005041867A8 2-(3,4-dimethylphenyl)-4-{[2-hydroxy-3’(1h-tetrazol-5-yl)biphenyl-3-yl]-hydrazono}-5-methyl-2,4-dihydropyrozol-3-one choline
07/06/2006US20060149080 Process for preparing optically active cyclic amines
07/06/2006US20060149078 Olmesartan medoxomil with reduced levels of impurities
07/06/2006US20060149072 Selective to alpha2B or alpha2C adrenergic receptors, minimal cardivascular or sedatory activity; treating visceral pain, neuropathic pain, corneal pain, glaucoma, elevated intraocular pressure, ischemic neuropathies, neurodegenerative diseases, diarrhea, nasal congestion
07/06/2006US20060149066 Imidazole derivatives
07/06/2006US20060149063 N-(4-Heptadecyl-6-oxo-1,6-dihydropyrimidin-2-yl)-N'-phenylguanidine; low viscosity values at the jetting temperature of a hot melt ink jet printer
07/06/2006US20060149062 Sulfanyl substituted phenyl methanones
07/06/2006US20060149061 2-chloro-4-(3-pyridyl)-pyrimidine is reacted with 2-amino-4-nitrotoluene to obtain N-(2-methyl-5-nitrophenyl)-4-(3-pyridyl)-2-pyrimidine-amine, hydrogenated to N-(5-amino-2-methyl)-4-(3-pyridyl)-pyrimidine-amine, reacted with 4-(4-methyl-piperazine-1-ylmethyl)-benzoyl chloride; avoids use of cyanamide
07/06/2006US20060149059 Phthalazinone derivatives
07/06/2006US20060148880 3-(Guanidinylcarbonylmethyl)-substituted; inhibit the cellular sodium-proton antiporter, in particular NHE1; antiarrhythmic agents;cardioprotective for infarction prophylaxis and treatment; preventing ischemia-induced damage
07/06/2006US20060148859 Substituted pyridyloxyalkylamides and their use as fungicides
07/06/2006US20060148858 1, 2-Azole derivatives with hypoglycemic and hypolipidemic activity
07/06/2006US20060148857 Tetrahydrocarbazole derivatives and their pharmaceutical use
07/06/2006US20060148856 Benzimidazole derivatives and their use for modulating the gabaa receptor complex
07/06/2006US20060148854 Chemical compounds
07/06/2006US20060148849 Quinoline derivatives, process of synthesis and medicaments containing these derivatives
07/06/2006US20060148845 In which a pyrrole ring is directly bonded to a 6,5-condensed ring system, such as a benzimidazole, imidazopyridine or imidazopyrimidine system; especially effective against drug resistant bacteria such as MRSA, PRSP, or VRE
07/06/2006US20060148830 Lpa receptor antagonist
07/06/2006US20060148824 Administering compounds such as 6-Chloro-N-[(1R)-1-phenylethyl]pyrazin-2-amine for inhibiting a protein kinase
07/06/2006US20060148823 Tricyclic delta -opioid modulators; 10-(1-Benzyl-piperidin-4-yl)-6-hydroxy-10H-phenoxazine-3-carboxylic acid diethylamide; immunosuppressants, antiinflammatory agents, depression, Parkinson's disease; reduced side effects; veterinary composition to treat mild to severe pain in warm-blooded animals
07/06/2006US20060148819 Chemical compounds
07/06/2006US20060148818 Novel tetraydrospiro(piperdine-2,7'- pyrrolo{3,2-b}pyridine derivatives and novel in-dole derivatives useful in the treatment of 5-ht6 receptor-related disorders
07/06/2006US20060148817 Pyrazole compounds
07/06/2006US20060148816 17Beta-hydroxysteroid dehydrogenase type 3 inhibitors for the treatment of androgen dependent diseases
07/06/2006US20060148815 4-Phenyl-1-piperazinyl, -piperidinyl and-tetrahydropyridyl derivatives
07/06/2006US20060148814 4-(2-Pyridyl)-1-amino(thio)carbonylpiperazine derivatives are antagonists of the mGluR5 receptor
07/06/2006US20060148811 Aralkyl-ketone piperazine derivatives and their uses as new antalgic or ataractic agent
07/06/2006US20060148809 For the therapy of deleterious neurological complaints; anxiolytic agents;cognitive disorders; good affinity as ligands for the alpha 2 and or alpha 3 and or alpha 5 subunit of the human GABAA receptor; 3-(6-Phenylpyridazin-4-yl)thiophene-2-carboxylic Acid Methyl Ester
07/06/2006US20060148798 Antiinflammatory agents; cardiovascular disorders; antidiabetic agents;central nervous system diosrders ; anticancer agents
07/06/2006US20060148794 Neuropeptide Y antagonist; antiarthritic agents; cardiovascular disorders; antidiabetic agents; kidney disorders; eating disorders; obesity
07/06/2006US20060148792 Substituted 1,4-benzodiazepines and uses thereof
07/06/2006US20060148791 Glutamate receptor antagonists
07/06/2006US20060148790 Benzodiazepine cgrp receptor antagonists
07/06/2006US20060148779 Calcitonin Gene-Related Peptide (CGRP) antagonists for migraine and cluster headaches; 5'-acylamino-spiro[imidazolidine-4,2'-indane]-2,5-dione derivatives
07/06/2006US20060148764 5-phenypyrimidines their preparation compositions comprising them and their use
07/06/2006US20060148649 Substituted n-aryl nitrogen heterocycles
07/06/2006US20060147948 bioassay with compounds having dimaleimide groups attached directly to fluorescent cores, whose latent fluorescence is quenched until maleimide groups undergo thiol addition reaction, for detecting target proteins having sterically unhindered sulfhydryl groups; fluorescence resonance energy transfer
07/06/2006US20060145145 Tertiary amine compounds, organic semiconductor devices using the same and organic electroluminescence devices using the same
07/06/2006DE112004001603T5 TGF-β-Genexpressionsinhibitor TGF-β gene expression inhibitor
07/06/2006DE102004061751A1 Cyanoguanidin-substituierte Pyrazoline Cyanoguanidino substituted pyrazolines
07/06/2006DE102004061748A1 Azetidin-substituierte Pyrazoline Azetidine-substituted pyrazolines
07/06/2006CA2594345A1 Compositions and methods of treating cell proliferation disorders
07/06/2006CA2594251A1 Pyrrolidyl derivatives of heteroaromatic compounds as phosphodiesterase inhibitors
07/06/2006CA2593993A1 Pyrazole compounds that modulate the activity of cdk, gsk and aurora kinases
07/06/2006CA2592514A1 Glucocorticoid mimetics, methods of making them, pharmaceutical compositions, and uses thereof
07/06/2006CA2592509A1 Benzazole analogues and uses thereof
07/06/2006CA2590586A1 Substituted biaryl analogues
07/05/2006EP1676846A2 Hydantoin derivatives as MMP inhibitors
07/05/2006EP1676837A1 Process for producing aminopyrrolidine derivative and intermediate compound