Patents
Patents for C07D 403 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group (62,587)
08/2006
08/31/2006US20060194865 G-lactam derivatives as prostaglandin agonists
08/31/2006US20060194863 e.g. [(4-Morpholinophenylamino)-methylene]-1,3-dihydro-indol-2-one;tyrosine kinase signal transduction modulators; antiproliferative agents; vision defects, atherosclerosis, restenosis, metabolic disorders, autoimmune diseases
08/31/2006US20060194858 Preparation of crude candesartan cilexetil
08/31/2006US20060194843 4-(2,6-Dichloro-benzoylamino)-1H-pyrazole-3-carboxylic acid piperidin-4-ylamide; anticancer agents; carcinoma of the colon; antifungal agents; antitumor agents; infections; 4-(2,6-difluoro-benzoylamino)-1H-pyrazole-3-carboxylic acid (1-methyl-piperidin-4-yl)-amide
08/31/2006US20060194842 Oxyindole derivatives
08/31/2006US20060194818 Inhibitors of macrophage migration inhibitory factor and methods for identifying the same
08/31/2006US20060194817 N-{(1S,2R)-1-(3,5-difluorobonzyl)-2-hydroxy-3-[(3-iodobonzyl)amino]propyl}-2-{4-[(methylsulfonyl)amino]phenyl}acetamide; inhibitors of the beta- secretase enzyme useful in the treatment of Alzheimer's disease and other diseases characterized by deposition of A beta peptide in a mamma
08/31/2006US20060194813 Indolinone derivatives substituted in the 6 position, the preparation thereof and their use as pharmaceutical compositions
08/31/2006US20060194811 Pyrimidine derivatives
08/31/2006US20060194807 Di-aryl substituted pyrazole modulators of metabotropic glutamate receptor-5
08/31/2006US20060194803 anti-dementia agent which uses a BEC 1 potassium channel inhibitor as the active ingredient; to improve learning disorder
08/31/2006US20060194798 Bicyclic-substituted amines as histamine-3 receptor ligands
08/31/2006US20060194793 Inhibitors of macrophage migration inhibitory factor and methods for identifying the same
08/31/2006US20060194787 substituted 1,1,4-1l6-trioxo[1,2]thiazepan-4-ylamide-derived protease inhibitors which inhibit the likes of cathepsin K; treating osteoporosis, osteo- and rheumatoid arthritis and periodontal disease; inhibiting excessive cartilage or matrix degradation
08/31/2006US20060194784 Analogs of clozapine; use with other neuropsychiatric agents; depression, anxiety, bipolar disorder, psychoses secondary to Alzheimer's or Huntington's disease
08/31/2006US20060194783 Cgrp receptor antagonists
08/31/2006US20060194779 1H-imidazole derivatives as cannabinoid CB2 receptor modulators
08/31/2006US20060194772 Triamide-substituted heterobicyclic compounds
08/31/2006US20060194073 Organic compound and organic electrolumiscent device
08/31/2006US20060193780 cyanine dyes and/or with lipophilic side chains; to detect stained cells both in vivo and in vitro; increased signal to noise ratio for rapidly labeling; improved solubility
08/31/2006CA2599348A1 Indole compound and use thereof
08/31/2006CA2599320A1 Hydrazinomethyl, hydr zonomethyl and 5-membered heterocylic compounds which act as mtor inhibitors and their use as anti cancer agents
08/31/2006CA2598853A1 Pyrrolidine and piperidine acetylene derivatives for use as mglur5 antagonists
08/31/2006CA2598518A1 5-phenyl-pentanoic acid derivatives as matrix metalloproteinase inhibitors for the treatment of asthma and other diseases
08/31/2006CA2586080A1 Novel compounds for treatment of cancer and disorders associated with angiogenesis function
08/30/2006EP1695967A1 Processes for production of pyrimidine derivatives and intermediates
08/30/2006EP1695960A1 Near-infrared fluorescent contrast medium
08/30/2006EP1695705A1 Compounds effecting glucokinase
08/30/2006EP1694799A2 Process for upgrading naphtha
08/30/2006EP1694686A1 Kinase inhibitors
08/30/2006EP1694671A2 Quinoxalines useful as inhibitors of protein kinases
08/30/2006EP1694670A1 Pyrazine derivatives as effective compounds against infectious diseases
08/30/2006EP1694669A2 Novel compounds which are modulators of the ppar-type receptors and their use in cosmetic or pharmaceutical compositions
08/30/2006EP1694654A2 Substituted triazoles as sodium channel blockers
08/30/2006EP1694410A2 Cyclopropane compounds and pharmaceutical use thereof
08/30/2006EP1490056B1 N-'4-(2-imino-pyrrolidin-1-yl)phenyl)-acetamide and corresponding piperidine derivatives as factor xa inhibitors for the treatment of thrombo-embolic diseases
08/30/2006EP1335722B1 Indolyl-sulfonyl- compounds useful in the treatment of cns disorders
08/30/2006EP1317429B1 Amidine inhibitors of serine proteases
08/30/2006CN1826336A Cyclohexanecarboxylic acid compound
08/30/2006CN1826334A Tetrahydropyranyl cyclopentyl heterocyclic amide modulators of chemokine receptor activity
08/30/2006CN1826328A Substituted pyridin-2-ylamine analogues
08/30/2006CN1826324A Indazole, benzisoxazole, and benzisothiazole kinase inhibitors
08/30/2006CN1826323A 3,4-disubstituted 1h-pyrazole compounds and their use as cyclin dependent kinase and glycogen synthase kinase-3 modulators
08/30/2006CN1826317A 酪氨酸激酶抑制剂 Tyrosine kinase inhibitor
08/30/2006CN1272324C Novel herbicides
08/30/2006CN1272316C Benzamides and related inhibitors of factor Xa
08/29/2006US7098345 Transamination of orndansetron preparing by Mannich reaction and isolation of product
08/29/2006US7098342 Dehydrohalogenation to form cilexetin trityl candesartan in the presence of phase transfer compounds
08/29/2006US7098331 Arylvinylazacycloalkane compounds and methods of preparation and use thereof
08/29/2006US7098330 Pyrazolylamine substituted quinazoline compounds useful as protein kinase inhibitors
08/29/2006US7098239 Dipeptidyl peptidase inhibitors for the treatment of diabetes
08/29/2006US7098236 3-(arylamino)methylene-1,3-dihydro-2H-indol-2-ones as kinase inhibitors
08/29/2006US7098234 Indole derivatives, process for preparation of the same and use thereof
08/29/2006US7098231 Viral polymerase inhibitors
08/29/2006US7098215 Nitrogenous compounds and antiviral drugs containing the same
08/29/2006US7098214 Dopamine D3 receptor ligands or antagonists for use in the treatment of renal function disorders
08/29/2006US7098213 three-ring saturated N-heterocyclic compounds in combination with one or more antiviral or other agents; in immunotherapy
08/29/2006US7098212 Piperazine derivatives
08/29/2006US7098201 Heteroaromatic derivatives having an inhibitory activity against HIV integrase
08/29/2006US7097706 non-calcined clay composite includes clay, lime, blast furnace slag, alkaline chemical, and water in specified amounts, and has high compression strength due to an ionic coagulation reaction, a pozzolan reaction, and a latent hydraulic reaction
08/29/2006CA2392271C Sulfonyl heteroaryl triazoles as anti-inflammatory/analgesic agents
08/29/2006CA2201785C New carboxylic acid derivatives, their preparation and their use
08/24/2006WO2006089060A1 Fungicidal pyrazine derivatives
08/24/2006WO2006088954A1 Dihydroindolyl methanones as alpha 1a/1d adrenoreceptor modulators for the treatment of benign prostatic hypertrophy and lower urinary tract symptoms
08/24/2006WO2006088711A1 AZOLYLACYLGUANIDINES AS β-SECRETASE INHIBITORS
08/24/2006WO2006088541A2 Quinoline derivatives and uses thereof
08/24/2006WO2006087538A1 Chemical compounds
08/24/2006WO2006087530A1 Chemical compounds
08/24/2006WO2006087355A1 1h-imidiazole derivatives as cannabinoid cb2 receptor modulators
08/24/2006WO2006071644A8 Selective inhibitors of erk protein kinases and uses therof
08/24/2006WO2006070195A8 Pyrazole compounds that modulate the activity of cdk, gsk and aurora kinases
08/24/2006WO2006065726A3 Process for preparing voriconazole
08/24/2006WO2006017822A3 Quinazoline derivatives and their use in the treatment of thrombocythemia
08/24/2006WO2005090333A8 3-‘4-heterocyclyl -1,2,3,-triazol-1-yl!-n-aryl-benzamides as inhibitors of the cytokines production for the treatment of chronic inflammatory diseases
08/24/2006US20060189812 Regioselective halogenation of nicotine and substituted nicotines
08/24/2006US20060189811 Process for producing 1,2,4-triazole compound and intermediate therefor
08/24/2006US20060189810 Novel sulfonamide inhibitors of aspartyl protease
08/24/2006US20060189804 Synthetic method for the preparation of quinazolin-4-one derivative
08/24/2006US20060189674 Deacetylase inhibitors
08/24/2006US20060189672 2-Heterocyclyl- indole, pyrrolopyridine, pyrrolopyrimidine, or pyrrolopirazine substituted with an N-(amino)sulfonyl(thio)carboxamide: 3-Cyclohexyl-2-furan-3-yl-7-methyl-1H-indole-6-(N-methylsulfonyl)carboxamide; treating a hepatitis virus infection
08/24/2006US20060189671 Compounds, compositions, and methods
08/24/2006US20060189663 Pyrrole-2,5-dithione derivatives as liver x receptor modulators
08/24/2006US20060189658 Substituted pyrazoline compounds, their preparation and use as medicaments
08/24/2006US20060189630 Mitotic kinesin inhibitors
08/24/2006US20060189629 N-(2-morpholin-4-ylethyl)-1-(4-{[4-(trifluoromethoxy)benzyl]oxy}phenyl)-1H -benzimidazole-5-carboxamide; c-Kit proto-oncogene (stem cell factor receptor) anhibitor; tyrosine kinase inhibitor; antiproliferative, anticarcinogenic agent;
08/24/2006US20060189628 Compounds useful as chemokine receptor antagonists
08/24/2006US20060189627 RAF inhibitor compounds and methods
08/24/2006US20060189626 For example, 2-methyl-6'-(4-methyl-piperazin-1-yl)-[3,4']bipyridinyl-3'-carboxylic acid (3,5-bis-trifluoromethyl-benzyl)-methyl-amide; treatment of certain depressive disorders or emesis
08/24/2006US20060189622 Pyridazinone and triazinone compounds and use thereof as pharmaceutical preparations
08/24/2006US20060189618 6-{4-[2-(4-tert-butyl-phenyl)-1H-imidazo[4,5-c]pyridin-4-yl]-piperazin-1-ylmethyl}quinoxaline; controls biosynthesis and release of sex steroids in the gonads; contraceptive; anticarcinogenic agent; prostate, uterine, breast, ovarian cancer, endometriosis, uterine fibroids, primary hirsutism
08/24/2006US20060189614 preparing 4-[[4-amino-6-[(2,6-dichlorophenyl)methyl]-1,3,5-triazin-2-yl]amino]benzonitrile by reacting 2,6-dichlorobenzeneethanimidamide with phenyl N'-cyano-N-(4-cyanophenyl)-carbamimidate in a reaction-inert solvent; HIV (Human Immunodeficiency Virus) infection
08/24/2006US20060189607 e.g. 8-(2-{3-[3-(4-fluoro-phenyl)-5-methyl-[1,2,4]triazol-1-yl]-1,1-dimethyl-propylamino}-1-hydroxy-ethyl)-6-hydroxy-4h-benzo[1,4]oxazin-3; mimetics of beta-adrenergic substances; beta 2-adrenoceptor modulator; antiinflammatory agent; chronic obstructive respiratory diseases; longer duration of activity
08/24/2006US20060189606 comprising administering compounds that affect viral internal ribosome entry site (IRES) activity, such as [4-(3-cyano-1-ethyl-6-methoxy-1H-indol-2-yl)-phenyl]-carbamic acid ethyl ester
08/24/2006US20060189600 Benodiazepine spirohydantoin cgrp receptor antagonists
08/24/2006US20060189593 Aryl spirohydantoin cgrp receptor antagonists
08/24/2006US20060189591 Five-membered heterocyclic derivative
08/24/2006US20060189590 Alkaline salts of proton pump inhibitors
08/24/2006US20060189577 Tyrosine kinase inhibitors
08/24/2006US20060189484 Pyridone compounds useful for producing pyridine compounds
08/24/2006DE19639859B4 1-Arylpyrazole, Zusammensetzungen, besonders giftige Köder zur Schädlingsbekämpfung 1 arylpyrazoles compositions, particularly toxic bait for pest control