Patents
Patents for C07D 403 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group (62,587)
08/2008
08/14/2008WO2008039087A3 Indoline derivatives and uses thereof
08/14/2008WO2008010984A3 Acridine activation of p53 and uses thereof
08/14/2008US20080194839 Synthesis of porphyrins designed for attachment to electroactive surfaces via one or more carbon tethers
08/14/2008US20080194661 1-(5-(4-trifluoromethyl-benzylamino)-1H-indazol-1-yl)-2-(2,4-difluorophenyl)-3-(1H-1,2,4-triazol-1-yl)propan-2-ol; 2-(2,4-difluorophenyl)-1-(1H-indazol-1-yl)-3-(1H-1,2,4-triazol-1-yl)propan-2-ol
08/14/2008US20080194627 Aryl substituted pyridines and the use thereof
08/14/2008US20080194617 Fused ring compound
08/14/2008US20080194607 Modulation of pathogenicity
08/14/2008US20080194606 Pyrazolyl-Amino-Substituted Pyrimidines and Their Use in the Treatment of Cancer
08/14/2008US20080194597 Platelet adp receptor inhibitors
08/14/2008US20080194588 Modulation of pathogcnicity
08/14/2008US20080194585 Fungicidal Pyrazine Derivatives
08/14/2008US20080194583 Tubulin Inhibitors
08/14/2008US20080194582 3,5-Diphenyl-4,5-dihydro-1H-dipyrazole derivatives such as {2-[1-acetyl-3-(2,5-difluorophenyl)-5-phenyl-4,5-dihydro-1H-pyrazol-5-yl]ethyl}(dimethyl)silanol that are useful for treating cancer
08/14/2008US20080194581 Pyrrole derivatives, intermediates therefor, preparation and therapeutic use thereof
08/14/2008US20080194578 Quinazoline based egfr inhibitors containing a zinc binding moiety
08/14/2008US20080194577 Antiallergens; asthma; autoimmune disease; pruritius; antiarthritic agents
08/14/2008US20080194576 Pyrimidine Derivatives and Their Use as P2Y12 Receptor Antagonists
08/14/2008US20080194574 Pyrazine Derivatives As Effective Compounds Against Infectious Diseases
08/14/2008US20080194565 5-Phenyl-Pentanoic Acid Derivatives as Matrix Metalloproteinase Inhibitors for the Treatment of Asthma and Other Diseases
08/14/2008US20080194556 Quinazolines and Their Use as Aurora Kinase Inhibitors
08/14/2008US20080194549 Organic Compounds
08/14/2008US20080194545 Antimicrobial compositions and methods of use
08/14/2008US20080194539 Phenyl Diazepane Carboxamides and Annelated Phenyl Piperazine Carboxamides Containing Oxygen and Used as Dopamine D3 Antagonists
08/14/2008US20080193411 Anti-viral Compounds
08/14/2008US20080193384 having chemical exchange saturation transfer (CEST)-active paramagnetic complexes linked to carriers selected from liposomes, particles, micelles and polypropylenimine dendrimers, used for mapping local pH, temperature, oxygen concentration or metabolites, detection of cancer lesions and inflammation
08/14/2008CA2677995A1 Acylguanidine derivative
08/14/2008CA2677661A1 Tricyclic compounds
08/14/2008CA2677481A1 Triazole compounds that modulate hsp90 activity
08/14/2008CA2677241A1 Compounds that inhibit cholinesterase
08/14/2008CA2677015A1 Hcv inhibiting macrocyclic phenylcarbamates
08/14/2008CA2676268A1 5 -amido- (ih- indol- 2 -yl) piperazin-1-yl-methanone derivatives as histamine h3 receptor ligands
08/13/2008EP1956020A2 1-[2-(heterocyclyl-aminomethyl)-piperidin-1-YL]-1-(2-methyl-5-phenyl-heterocyclyl)-methanone derivatives and related compounds as orexin-1 antagonists for the treatment of obesity
08/13/2008EP1956013A1 Diagnostic and remedy for disease caused by amyloid aggregation and/or deposition
08/13/2008EP1956008A1 Organic compound, charge-transporting material, composition for charge-transporting material and organic electroluminescent device
08/13/2008EP1955697A1 2-aminobenzamide derivative
08/13/2008EP1954692A1 Heterocycle-substituted 3-alkyl azetidine derivatives
08/13/2008EP1954682A1 Novel 2-amino-imidazole-4-one compounds and their use in the manufacture of a medicament to be used in the treatment of cognitive impairment, alzheimer s disease, neurodegeneration and dementia
08/13/2008EP1954673A1 Hydroxy-substituted diphenylazetidinones for the treatment of hyperlipidaemia
08/13/2008EP1954317A2 Heterocyclic-substituted bis-1,8 naphthalimide compounds, antibody drug conjugates, and methods of use
08/13/2008EP1954276A2 Indole orexin receptor antagonists
08/13/2008EP1453501B1 N- aryl-n'-arylcycloalkyl-urea derivatives as mch antagonists for the treatment of obesity
08/13/2008EP1322309B1 High affinity small molecule c5a receptor modulators
08/13/2008CN101243075A Novel 2,3-dihydroindole compounds
08/13/2008CN101243071A Novel 2,4-dianilinopyrimidine derivatives, the preparation thereof, their use as medicaments, pharmaceutical compositions and, in particular, as ikk inhibitors
08/13/2008CN101243070A Trombin inhibiting 2,4-dioxo-3,4-dihydropyrimidine derivatives
08/13/2008CN101243068A Compounds for the treatment of multi-drug resistant bacterial infections
08/13/2008CN101243055A Dihydropyrimidone multimers and their use as human neutrophil elastase inhibitors
08/13/2008CN101243052A Helix 12 directed non-steroidal antiandrogens
08/13/2008CN101242848A Pyrimidine compounds
08/13/2008CN101242844A Aminopyrimidines as kinase modulators
08/13/2008CN101242843A Aminopyrimidines as kinase modulators
08/13/2008CN101242834A Inhibitors of AKT activity
08/13/2008CN101239975A Synthesis of 2-butyl-3-(2'-(1-trityl-1h-tetrazol-5-yl)biphenyl-4-yl)methyl-1,3-diazaspirol[4,4]-non-ene-4-one
08/13/2008CN101239974A Synthesis of 2-butyl-3-(2'-(1-trityl-1h-tetrazol-5-yl)biphenyl-4-yl)methyl-1,3-diazaspirol[4,4]-non-ene-4-one
08/13/2008CN101239972A Heterocyclic n-aryl carboxamides as cytokine inhibitors
08/13/2008CN101239930A Synthesis of 2-butyl-3-(2'-(1-trityl-1h-tetrazol-5-yl)biphenyl-4-yl)methyl-1,3-diazaspirol[4,4]-non-ene-4-one
08/13/2008CN100410253C Highly effective environment friendly triazine amino stilbene fluorescent bleachng agent
08/13/2008CN100410250C Spiroheterocyclic compoundsus reversible inhibitors of cysteine proteases
08/12/2008US7411098 Aldol condensation of citral with acetone and subsequent hydrogenation; using tetrahydrogeranylacetone for preparing phytol, isophytol, tocopherol and/or tocopherol derivatives
08/12/2008US7411073 cyclopent[f]pyrazole derivatives; antiinflammatory agent; autoimmune diseases; side effect reduction, advantages over steroidal glucocorticoid ligands with respect to undesireable side-effects, efficacy, toxicity or metabolism
08/12/2008US7411072 e.g. 5-(10,11-Dihydro-dibenzo[a,d]cyclohepten-5-ylidenemethyl)-3H-benzooxazol-2-one; antiinflammatory, antidiabetic agent; electrolytes and water retention modulator; hypotensive, hypoglycemic agent; arrhythmias, myocardial fibrosis, osteoporosis, polyuria, polydipsia, Crohn's disease
08/12/2008US7411065 Peptide nucleic acid monomers: diphenylmethyl, benzyl, alkylthioalkyl, or phenylthioalkyl esters of N-(1-[4-(2-benzothiazolyl-, 2-benzoxazolyl-, 2-benzofuranyl- or 2-benzothiophenyl-sulfonyl)-3-piperazinon-1-ylcarbonylmethyl]pyrimidon-4-yl)carbamic acids
08/12/2008US7410989 intravenous or oral administration of viricides against the Flaviviridae family of viruses; e.g. 2-[5(6)-Amidino-2-benzimidazoyl]-5-(4-nitrophenyl)furan
08/12/2008US7410972 Compounds
08/12/2008US7410970 Substituted 1,4,-di-piperidin-4-yl-piperazine derivatives and their use as neurokinin antagonists
08/12/2008US7410968 N-(3,5-diamino-6-chloropyrazine-2-carbonyl)-N'-(4-{4-[3-(1H-tetrazol-5-yl)propoxy]phenyl}butyl)guanidine hydrochloride; hydrates mucosal surfaces; are absorbed less rapidly, thus have a prolonged pharmacodynamic half-life; skin and respiratory disorders, vision deffects
08/12/2008CA2420461C Preparations for oral administration
08/07/2008WO2008094909A2 Quinazolinone and fused pyrimidinone compounds and their use in treating sodium channel-mediated diseases or conditions
08/07/2008WO2008093639A1 Pyrazole compound
08/07/2008WO2008092844A1 Piperidin-acetamide derivatives for the treatment of inflammatory or allergic diseases
08/07/2008WO2008092231A1 Compounds for the prevention and treatment of cardiovascular diseases
08/07/2008WO2008092199A1 Thiopyrimidine-based compounds and uses thereof
08/07/2008WO2008061792A3 Tricarbonyl complexes with tridentate chelators for myocardium imaging
08/07/2008WO2008054748A3 Indazole derivatives as modulators of the 5-ht2a serotonin receptor useful for the treatment of disorders related thereto
08/07/2008WO2007138351A3 Pyridinone and pyridazinone derivatives as inhibitors of poly(adp-ribose)polymerase (parp)
08/07/2008US20080188655 Monomer With Anti-Microbial Character, Polymer Using The Same, And Manufacturing Method Thereof
08/07/2008US20080188652 Salt forms of [R-(R*,R*)]-2-(4-fluorophenyl)-beta, delta-dihydroxy-5-(1-methylethyl)-3-phenyl-4-[(phenylamino)carbonyl]-1H-pyrrole-1-heptanoic acid
08/07/2008US20080188536 2-thiophenecarboxylic acid-5-nitro-2-(2-thienylcarbonyl)hydrazide; antibacterial agent; inhibition of formation of biofilms in personal hygiene articles, toileteries, cosmetics and in industrial setting; bacterial damage or disease; Pseudomonas aeruginosa or Burkholderia cepacia
08/07/2008US20080188535 2-thiophenecarboxylic acid-5-nitro-2-(2-thienylcarbonyl)hydrazide; antibacterial agent; inhibition of formation of biofilms in personal hygiene articles, toileteries, cosmetics and in industrial setting; bacterial damage or disease; Pseudomonas aeruginosa or Burkholderia cepacia
08/07/2008US20080188521 Novel pharmaceutical compounds
08/07/2008US20080188501 retrovirus inhibor; anticarcinogenic, antidiabetic agent, immunosuppressant, autoimmune diseases; 2-{6-[3(R)-Amino-piperidin-1-yl]-3-methyl-2,4-dioxo-3,4-dihydro-2H-pyrimidin-1-ylmethyl}-4-fluoro-benzonitrile; type 2 diabetes mellitus, impaired glucose tolerance, obesity, multiple sclerosis
08/07/2008US20080188491 Modulation of pathogenicity
08/07/2008US20080188487 5-amido-(1h-indol-2-yl)-piperazin-1-yl-methanone derivatives
08/07/2008US20080188474 Substituted triazoles useful as axl inhibitors
08/07/2008US20080188472 Indole-2-Carboxylic Acid Hydrazides
08/07/2008US20080188454 angiogenesis and/or cell proliferation, carcinoma, myeloid leukemia, endometriosis; inhibitors of the receptor protein tyrosine kinase; N3-(3-cyclopentyl-1,2,3,4,5,6-hexahydrobenzo[d]azocin-8-yl)-1-(6-fluoroquinazolin-4-yl)-1H-1,2,4-triazole-3,5-diamine
08/07/2008US20080188452 Macrocyclic Benzofused Pyrimidine Derivatives
08/07/2008US20080188451 4-Methyl-3-[[4-(3-pyridinyl)-2-pyrimidinyl]amino]-N-[5-(4-methyl-1H-imidazol1yl)-3-(trifluoromethyl)phenyl]benzamide or an N-oxide or salts; anticarcinogenic agent (leukaemia)
08/07/2008US20080187978 Anti-inflammatory medicaments
08/07/2008US20080187575 Pyrimidine Derivatives
08/07/2008CA2702647A1 Thiopyrimidine-based compounds and uses thereof
08/07/2008CA2676984A1 Compounds for the prevention and treatment of cardiovascular diseases
08/07/2008CA2675348A1 Piperidin-acetamide derivatives for the treatment of inflammatory or allergic diseases
08/06/2008EP1953152A1 Process for preparing quinazoline RHO-kinase inhibitors and intermediates thereof
08/06/2008EP1953148A1 Heterocyclic amide compound and use thereof
08/06/2008EP1953147A1 Heterocyclic compound and medicinal application thereof
08/06/2008EP1953146A1 Methods of making 6-[(4,5-Dihydro-1H-imidazol-2-yl) amino-]-7-methyl-1H-benzimidazole-4-carbonitrile and its preferred salt form
08/06/2008EP1953145A1 Heterocyclic compound having inhibitory activity on 11- -hydroxysteroid dehydrogenase type i
08/06/2008EP1951719A2 Certain chemical entities, compositions, and methods
08/06/2008EP1951716A1 Aminopyrimidines useful as kinase inhibitors