Patents
Patents for C07D 401 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom (107,979)
11/1998
11/26/1998WO1998052558A1 INHIBITION OF p38 KINASE ACTIVITY BY ARYL UREAS
11/26/1998WO1998052514A2 Treatment of hepatic cirrhosis
11/26/1998WO1998040357A3 Hiv protease inhibitors
11/26/1998DE19721031A1 Substituierte Pyridylpyrazole Substituted pyridylpyrazoles
11/26/1998CA2302438A1 Heteroarylcarboxamide compounds active against protein tyrosine kinase related disorders
11/26/1998CA2291115A1 Substituted pyrazoles as p38 kinase inhibitors
11/26/1998CA2291111A1 Quinoline-4-carboxamide derivatives as nk-2 and nk-3 receptor antagonists
11/26/1998CA2290789A1 Analogs of duocarmycin and cc-1065
11/26/1998CA2290475A1 Indoline derivatives as 5ht2c receptor antagonists
11/26/1998CA2290379A1 Substituted pyridylpyrazoles as herbicides, insecticides and acaricides
11/26/1998CA2289605A1 Cis-substituted substituted aminocycloalkylpyrrolidine derivatives
11/26/1998CA2288787A1 Pyrazole derivatives as p38 kinase inhibitors
11/26/1998CA2288741A1 4-aryl-3(5)-heteroaryl substituted pyrazoles as p38 kinase inhibitors
11/25/1998EP0879234A1 1-pyrazol-3-yl-ethyl-4-indol-3-yl-piperidine used as medicine acting on the central nervous system
11/25/1998EP0879233A1 Chinoline and benzimidazole derivatives as bradykinin agonists
11/25/1998EP0711291B1 N-(piperidinyl-1-alkyl)-substituted cyclohexane carboxylic acid amides as 5-ht1a receptor antagonists
11/25/1998EP0652866B1 Azacyclic compounds
11/25/1998EP0624159B1 Pyridyl substituted imidazoles
11/25/1998CN1200120A Piperazino derivatives as neurokinin antagonists
11/25/1998CN1199731A Propanolamine derivatives, processes for their preparation, pharmaceuticals comprising these compounds, and their use
11/25/1998CN1040873C Arylidene-1-azacycloalkanes and arylalkyl-1-azacycloalkanes, their salts, salts and composition and their application and producing process
11/25/1998CN1040829C Compositions containing pyridazinone derivatives for controlling and/or preventing insect pests and its application
11/24/1998US5840916 Quinoline carboxylic acid derivatives having 7-(4-amino-methyl-3-oxime) pyrrolidine substituent and processes for preparing thereof
11/24/1998US5840910 Pyridine derivatives having anti-ulcerative activity
11/24/1998US5840909 Pyrazole derivatives
11/24/1998US5840906 Forming anabaseine using nicotinyl piperidone salt
11/24/1998US5840892 Process for the preparation of substituted pyrimidines
11/24/1998US5840888 Useful in the diagnosis and treatment of anxiety, sleep and seizure disorders, overdose with benzodiazepine drugs and enhancement of memory
11/24/1998US5840745 Hydrosoluble 3-arylidene-2-oxindole derivatives as tyrosine kinase inhibitors
11/24/1998US5840738 Selective β-3 adrenergic agonists
11/24/1998US5840735 Estrogen
11/24/1998US5840727 (4-heteroaryl)-1- (2,3-dihydro-1H-isoindol-2-yl) alkyl! piperazines and related compounds and their therapeutic utility
11/24/1998US5840725 Substituted oximes, hydrazones and olefins as neurokinin antagonists
11/24/1998US5840722 Administering to inhibit endothelin receptors
11/24/1998US5840654 Herbicidal heterocyclic-substituted pyridines
11/24/1998US5840552 Using microorganisms or microbial enzyme system to produce stereospecific enantiomers; antiulcer agents
11/24/1998CA2108584C Substituted azetidinones as anti-inflammatory and antidegenerative agents
11/19/1998WO1998051687A1 Piperidino derivatives which promote growth hormone release
11/19/1998WO1998051686A1 N-triazolyl-2-indolecarboxamides and their use as cck-a agonists
11/19/1998WO1998051685A1 Method of manufacturing sertindole
11/19/1998WO1998051672A2 A method for the preparation of tertiary amines, a compound useful therefor and alpha-2-receptor active tetrahydroisoquinoline derivatives
11/19/1998WO1998051671A1 Substituted tetrahydroisoquinoline derivatives as modulators of dopamine d3 receptors
11/19/1998WO1998051665A2 Novel macrocyclic compounds as metalloprotease inhibitors
11/19/1998WO1998051311A2 Dihydropyrimidines and uses thereof
11/19/1998WO1998051298A1 Arylsubstituted piperazines useful in the treatement of benign prostatic hyperlasia
11/19/1998CA2300088A1 A method for the preparation of tertiary amines, a compound useful therefor and alpha-2-receptor active tetrahydroisoquinoline derivatives
11/19/1998CA2289573A1 N-triazolyl-2-indolecarboxamides and their use as cck-a agonists
11/19/1998CA2288850A1 Substituted tetrahydroisoquinoline derivatives as modulators of dopamine d3 receptors
11/19/1998CA2287923A1 Novel macrocyclic compounds as metalloprotease inhibitors
11/18/1998EP0877744A1 Substituted aza- and diazacycloheptane and cyclooctane compounds and their use
11/18/1998EP0877737A1 Novel n-(arylsulphonyl)amino acid derivatives having bradykinin receptor affinity
11/18/1998EP0877736A1 Benzazepine derivatives with vasopressin agonistic activity
11/18/1998EP0877734A1 Quinoline and quinazoline compounds useful in therapy
11/18/1998EP0717734B1 Pyridazinone derivatives or their salts, processes for their production, and anti-shock agents containing them
11/18/1998EP0706514B1 Compounds and methods for inhibition of hiv and related viruses
11/18/1998EP0537201B1 1-[4-(imidazol-1-yl)benzoyl]piperidine derivatives as antiarrhythmic agents
11/18/1998CN1199397A Pyrimidin derivatives
11/18/1998CN1199394A Didepsipeptide-based endoparasiticides, new didepsipeptides and process for preparing same
11/18/1998CN1040754C 3-(substd. ketone and alcohol)-2-(2-imidazolin-2-yl)-pyridine and quinoline,their preparing process and herbicidal agents contg. same
11/18/1998CN1040752C Novel piperidine derivs. and process for preparation thereof
11/18/1998CN1040748C Benzazepine deriv., pharmaceutical composition contg. same, and intermediate for same
11/17/1998US5837873 Intermediates of retroviral protease inhibiting compounds
11/17/1998US5837720 N-2-(pyrrolidinyl-1)-1-phenethyl) acetamides as kappa receptor antagonists
11/17/1998US5837719 2,5-substituted aryl pyrroles, compositions containing such compounds and methods of use
11/17/1998US5837718 Antihistamines
11/17/1998US5837716 Analgesics
11/17/1998US5837710 Enzyme inhibitors for treatment of aids
11/17/1998US5837708 Sulphonamides
11/17/1998US5837707 Dimeric piperidine, tetrahydropyridine and piperazine derivatives
11/12/1998WO1998050534A1 Protease inhibitors
11/12/1998WO1998050394A1 Nitric oxide carriers based on polyazamacrocycle complexes
11/12/1998WO1998050366A1 Substituted 4-(3-alkenyl-benzoyl)-pyrazoles
11/12/1998WO1998050364A1 Tetrahydroisoquinoline derivatives as modulators of dopamine d3 receptors
11/12/1998WO1998050363A1 Substituted tetrahydro isoquinolines as modulators of dopamine d3 receptors
11/12/1998WO1998050360A1 Light-stabilized organic polymers
11/12/1998WO1998050358A1 Indole derivatives having combined 5ht1a, 5ht1b and 5ht1d receptor antagonist activity
11/12/1998WO1998050356A1 2-indolinone derivatives as modulators of protein kinase activity
11/12/1998WO1998050348A1 Metalloproteinase inhibitors, pharmaceutical compositions containing them and their pharmaceutical uses
11/12/1998WO1998050346A2 Acetamide and urea derivatives, process for their preparation and their use in the treatment of cns disorders
11/12/1998WO1998050342A1 Protease inhibitors
11/12/1998WO1998049897A1 Beta lactams as antiproliferative agents
11/12/1998CA2289705A1 Beta lactams as antiproliferative agents
11/12/1998CA2289602A1 Protease inhibitors
11/12/1998CA2289552A1 Light-stabilized organic polymers
11/12/1998CA2289112A1 Substituted 4-(3-alkenylbenzoyl)-pyrazoles
11/12/1998CA2289102A1 2-indolinone derivatives as modulators of protein kinase activity
11/12/1998CA2289010A1 Protease inhibitors
11/12/1998CA2289001A1 Novel heterocyclic compounds
11/12/1998CA2288899A1 Tetrahydroisoquinoline derivatives as modulators of dopamine d3 receptors
11/12/1998CA2288662A1 Indole derivatives having combined 5ht1a, 5ht1b and 5ht1d receptor antagonist activity
11/12/1998CA2287981A1 Nitric oxide carriers based on polyazamacrocycle complexes
11/12/1998CA2287913A1 Substituted tetrahydro isoquinolines as modulators of dopamine d3 receptors
11/11/1998EP0877022A1 Synthesis of the sulfonylpyrimidine derivatives with anticancer activity
11/11/1998EP0877019A1 Substituted diaminocarboxylic acid
11/11/1998EP0877018A1 Sulfonylaminocarboxylic acids
11/11/1998EP0876365A1 Substituted quinolylmethylen-oxindole analogues as tyrosine kinase inhibitors
11/11/1998EP0876363A1 Polymer-bound fluorophores as optical ion sensors
11/11/1998EP0876357A1 New quinoxalindione derivatives, their preparation and use in medicaments
11/11/1998EP0876353A1 Retroviral protease inhibiting compounds
11/11/1998EP0876346A1 Antimalarial quinolin derivatives