Patents
Patents for C07D 401 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom (107,979)
03/2004
03/17/2004CN1483029A Sodium channel modulators derived from 2-piperidylimidazoles
03/17/2004CN1483028A Quinolinone derivatives as tyrosine kinase inhibitors
03/17/2004CN1483024A Vla-4 inhibitors
03/17/2004CN1483019A Method for the regioselective preparation of substituted benzo[g]quinoline-3-carbonitriles and benzo[g]quinazolines
03/17/2004CN1482912A Heteroaryl urea neuropeptide yy5 receptor antagonists
03/17/2004CN1482127A Quinacridone derivant and application in organic electroluminescent device thereof
03/17/2004CN1142164C Optically active quinoline carboxylic acid derivatives having 7-pyrrolidine substituent causing optical activity and process for preparing thereof
03/17/2004CN1142159C Prearation method of [(substituted pyridyl) methyl] sulfinyl-IH-benzimidazole compound magnesium salt
03/17/2004CN1142153C Benzoylpyridazines
03/17/2004CN1142151C 2,4,6-trisubstituted striazine compound and its synthesizing process
03/17/2004CN1142149C Novel pyridazine derivatives and drugs containing same as active ingredient
03/17/2004CN1142148C Pyridazine derivatives and drugs containing the same as the active ingredient
03/17/2004CN1142144C 4-phenyl pyridine derivatives
03/16/2004US6706885 Process for preparing integrin antagonist intermediates
03/16/2004US6706883 Separating atropisomer by liquid chromatography; heating in dimethylformamide, toluene, or o-dichlorobenzene solvent; chemical reduction
03/16/2004US6706882 Process for the preparation of (pyridinylidene)-phthalides
03/16/2004US6706749 Substituted phenyl derivatives, their preparation and use
03/16/2004US6706743 β3 adrenergic receptor agonists and uses thereof
03/16/2004US6706740 Controlling, prevention fungi infections
03/16/2004US6706739 Treating enterovirus infection
03/16/2004US6706738 Substituted bicyclic heteroaryl compounds and their use as integrin antagonists
03/16/2004US6706737 Inhibiting gastric acid secretion are known in the art and include a class of benzimidazole- substituted compounds, one of which is omeprazole
03/16/2004US6706735 Nitrogen compounds such as n-(3-(4-benzyl-2-piperidinyl)propyl )-n'-(3-cyanophenyl)urea, used as chemotactic cytokine controllers administered for prophylaxis of asthma, allergies and autoimmune diseases
03/16/2004US6706731 With isoquinoline derivatives as antitumor agents
03/16/2004US6706723 Pyrimidine-2,4,6-trione metalloproteinase inhibitors
03/16/2004US6706716 Compounds specific for the human α1d adrenergic receptor and uses thereof
03/16/2004US6706711 Substituted diaminopyrazoles; treating diseases, such as cancer, inflammatory disorders, restenosis, and cardiovascular disease. coatings for implantable medical devices, such as prostheses, artificial valves, etc.
03/16/2004US6706709 Treating, for example, proliferative disorders including cancer
03/16/2004US6706703 Bis(5-aryl-2-pyridyl) compound having excellent immunoglobulin (ige) antibody production inhibiting activity, useful for the prevention or treatment of allergic immune diseases
03/16/2004US6706215 Coating compositions stabilized against damage by light, heat and oxygen
03/16/2004US6706021 Anticoagulant for catheters, dialysis machines, syringes, tubes, blood lines and stents; trypsin-like serine proteases such as thrombin; 3-benzylsulfonylamino-6-methyl-1-((2-guanidinooxyethyl) aminocarbonylmethyl)-2-pyridinone
03/16/2004CA2294399C Farnesyl transferase inhibitors in combination with hmg coa reductase inhibitors for the treatment of cancer
03/11/2004WO2004020448A1 Neutral metallic dendrimer complexes
03/11/2004WO2004020441A1 Hetereoaryl nitrile derivatives
03/11/2004WO2004020437A1 S-(+)-3-{1-[2-(2,3-dihydro-1h-indol-3-yl)ethyl]-3,6-dihydro-2h-pyridin-4-yl}-6-chloro-1h-indole and acid addition salts thereof
03/11/2004WO2004020436A1 Amorphous hydrates of esomeprazole magnesium and process for the preparation thereof
03/11/2004WO2004020435A1 Piperidinyl compounds that selectively bind integrins
03/11/2004WO2004020434A1 Azaarene derivatives
03/11/2004WO2004020433A1 Novel crystals
03/11/2004WO2004020432A1 Arylamides
03/11/2004WO2004020431A2 Novel benzoimidazole derivatives useful as antiproliferative agents
03/11/2004WO2004020415A1 2,5-dioxoimidazolidin-4-yl acetamides and analogues as inhibitors of metalloproteinase mmp12.
03/11/2004WO2004020414A1 Oxytocin inhibitors
03/11/2004WO2004020412A1 Dihydropyridine derivatives for use as human neutrophil elastase inhibitors
03/11/2004WO2004020410A2 Dihydropyridinone derivatives as hne inhibitors
03/11/2004WO2004020409A1 Indoles having anti-diabetic activity
03/11/2004WO2004020408A1 Indoles having anti-diabetic activity
03/11/2004WO2004020371A1 Condensed polycyclic compound and organic light-emitting device using the same
03/11/2004WO2004019943A1 Anabaseine derivatives useful in the treatment of neurodegenerative diseases
03/11/2004WO2004019935A1 -3 (sulfonamidoethyl) -indole derivaties for use as glucocorticoid mimetics in the treatment of inflammatory, allergic and proliferative diseases
03/11/2004WO2004019889A2 Inhibitors of post-amadori advanced glycation end products
03/11/2004WO2004019868A2 N-biarylmethyl aminocycloalkanecarboxamide derivatives
03/11/2004WO2004005279A3 Substituted anthranilic amide derivatives and methods of use
03/11/2004WO2003101452A8 Process for the preparation of highly pure rabeprazole sodium salt
03/11/2004WO2003091264A3 Non nucleoside reverse transcriptase inhibitors
03/11/2004WO2003078420A3 Process for making chiral 1,4-disubstituted piperazines
03/11/2004WO2003009845A9 Substituted urea neuropeptide y y5 receptor antagonists
03/11/2004WO2003006444A3 Substituted amides, sulfonamides and ureas useful for inhibiting kinase activity
03/11/2004WO2002076404A3 Fatty alcohol drug conjugates
03/11/2004US20040049083 Arylpiperazines having activity at the serotonin 1A receptor
03/11/2004US20040049046 Small molecule inhibitors of rotamase enzyme activity
03/11/2004US20040049045 Process for the crystallization of (r)-or (s)-lansoprazole
03/11/2004US20040049044 Process for the preparation of pantoprazole and intermediates therefor
03/11/2004US20040049039 Treating neurodegenerative, psychotropic, and drug and alcohol induced central and peripheral nervous system disorders.
03/11/2004US20040049035 Pyrrolecarboxamides and pyrrolethioamides as fungicides
03/11/2004US20040049032 Inhibitors of protein kinases, especially Aurora kinase; anticancer agents
03/11/2004US20040049020 Especially for dyeing paper; red dyeings with good fastness
03/11/2004US20040048903 Nicotinamide biaryl derivatives useful as inhibitors of PDE4 isozymes
03/11/2004US20040048901 Increased water solubility and bioabsorption; treatment of CNS disorders such as depression and emesis
03/11/2004US20040048898 Benzimidazole compound crystal
03/11/2004US20040048896 Treating gastric acid disorders by orally administering a proton pump inhibitor and a mixture of buffers
03/11/2004US20040048891 Aniline derivatives or salts thereof and cytokine production inhibitors containing the same
03/11/2004US20040048884 3-aminoalkyluracil derivatives, e.g., 1-(2,6-Difluorobenzyl)-5-(3-methoxyphenyl)-6-methyl-3-(N-methyl-N-(2 -pyridylethyl)-aminoethyl)uracil; contraceptives; treating lupus, sex hormone related cancer, benign prostatic hypertrophy, etc.
03/11/2004US20040048882 4-phenyl-6-alpha-(imidazolyl-, 1,2,4-triazolyl- or pyridyl)-benzyl substituted
03/11/2004US20040048881 Quinazoline derivatives with anti-tumour activity
03/11/2004US20040048880 Bicyclic heterocyclic compounds, pharmaceutical compositions containing these compounds, their use and process for preparing them
03/11/2004US20040048875 Compounds and methods for treatment of asthma, allergy and inflammatory disorders
03/11/2004US20040048873 Pyrimidine compounds
03/11/2004US20040048872 Sedatives, anticonvulsants, hypnotics and general anesthetics.
03/11/2004US20040048868 Benzimidazoles
03/11/2004US20040048867 Especially quinoline carbonyl pyrrolidines with binding selectivity to benzodiazepine site of GABAA receptor to treatanxiety, depression, a sleep disorder, or cognitive impairment.
03/11/2004US20040048866 3-substituted with an oxy-, thio- or amino- group; increasing cGMP levels
03/11/2004US20040048864 Fungicidal heterocyclic aromatic amides and their compositions, methods of use and preparation
03/11/2004US20040048863 Treating osteoarthritis or rheumatoid arthritis
03/11/2004US20040048862 Chemical compounds
03/11/2004US20040048853 Compounds, compositions, and methods
03/11/2004US20040048852 Aromatic sulfone hydroxamic acid metalloprotease inhibitor
03/11/2004US20040048850 Activators of soluble guanylate cyclase.
03/11/2004US20040048848 Novel gamma secretase inhibitors
03/11/2004US20040048844 Acylsemicarbazides as cyclin dependent kinase inhibitors useful as anti-cancer and anti-proliferative agents
03/11/2004US20040048843 And aza- and diaza-derivatives thereof; especially treating allergy or nasal congestion
03/11/2004US20040048797 Regulation of TNF-alpha
03/11/2004DE10238865A1 New carboxamides are melanin-concentrating hormone receptor antagonists, useful for treating e.g. metabolic diseases, diabetes, eating disorders, cardiovascular disease, emotional disorders, reproductive and memory disorders
03/11/2004DE10236910A1 Substituierte 1,2,3,4-Tetrahydrochinolinderivate Substituted 1,2,3,4-tetrahydroquinoline
03/11/2004CA2501424A1 Amorphous hydrates of esomeprazole magnesium and process for the preparation thereof
03/11/2004CA2496887A1 Oxytocin inhibitors
03/11/2004CA2496580A1 3-(sulfonamidoethyl)-indole derivaties for use as glucocorticoid mimetics in the treatment of inflammatory, allergic and proliferative diseases
03/11/2004CA2496452A1 Inhibitors of post-amadori advanced glycation end products
03/11/2004CA2495914A1 N-biarylmethyl aminocycloalkanecarboxamide derivatives
03/11/2004CA2495853A1 2,5-dioxoimidazolidin-4-yl acetamides and analogues as inhibitors of metalloproteinase mmp12