Patents
Patents for C07D 401 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom (107,979)
01/2004
01/22/2004WO2004007510A1 Novel chemical substance having activity for morphogenesis and growth promotion
01/22/2004WO2004007481A2 Substituted amine derivatives and methods of use in the treatment of angiogenesis relates disorders
01/22/2004WO2004007480A1 3-guanidinocarbonyl-1-heteroaryl-indole derivatives, preparation process, their use as medicaments, and pharmaceutical compositions comprising them
01/22/2004WO2004007479A1 3-guanidinocarbonyl-1-heteroaryl-indole derivatives, preparation process, their use as medicaments, and pharmaceutical compositions comprising them
01/22/2004WO2004007478A2 Derivatives of 3-guanidinocarbonyl-1-heteroaryl-pyrrole, process for their preparation and their pharmaceutical use
01/22/2004WO2004007472A1 Ccr4 antagonist and medicinal use thereof
01/22/2004WO2004007463A1 Cck-1 receptor modulators
01/22/2004WO2004007461A1 8-hydroxy quinoline derivatives
01/22/2004WO2004007459A2 Naphthol, quinoline and isoquinoline-derivatives as modulators of vanilloid vr1 receptor
01/22/2004WO2004007458A1 Substituted 2-alkylamine nicotinic amide derivatives and use there of
01/22/2004WO2004007457A2 Substituted benzylamine derivatives and methods of use
01/22/2004WO2004007454A1 Piperidinetriol derivatives as inhibitors of glycosylceramidsynthase
01/22/2004WO2004007453A1 Piperidinetriol derivatives as inhibitors of glycosylceramide synthase
01/22/2004WO2004007449A1 Process for conversion of phenols to carboxamides via the succinimide esters
01/22/2004WO2004007407A2 Fluorous tagging and scavenging reactants and methods of synthesis and use thereof
01/22/2004WO2004006934A2 1,4,7,10-tetraazacyclododecanes as modulators of the guanine-binding protein for treating tumours
01/22/2004WO2004006928A1 Crystalline 2,5-dione-3-(1-methyl-1h-indol-3-yl)-4-[1-(pyridin-2-ylmethyl)piperidin-4-yl]-1h-indol-3-yl]-1h-pyrrole mono-hydrochloride
01/22/2004WO2004006927A2 Sulphonylpiperidine derivatives containing an alkenyl or alkynly moiety for use as matrix metalloproteinase inhibitors
01/22/2004WO2004006926A1 Sulphonylpiperidine derivatives containing an aryl or heteroaryl group for use as matrix metalloproteinase inhibitors
01/22/2004WO2004006925A1 N-sulfonylpiperidines as metalloproteinase inhibitors (tace)
01/22/2004WO2004006923A1 Aryl piperidine derivatives as inducers of ldl-receptor expression for the treatment of hypercholesterolemia
01/22/2004WO2004006922A1 Aryl piperidine derivatives as inducers of ldl-receptor expression for the treatment of hypercholesterolemia
01/22/2004WO2004006920A1 Topical treatment of skin diseases
01/22/2004WO2004006846A2 Receptor-type kinase modulators and methods of use
01/22/2004WO2003055447A3 Heterocyclic acridone inhibitors of impdh enzyme
01/22/2004WO2002092573A3 Heterocyclic substituted pyrazoles as inhibitors of src and other protein kinases
01/22/2004US20040015037 Radioactive member and method of making
01/22/2004US20040014978 Such as (4S,7R,8S,9S,13(Z),16S(Z))-4,8-Dihydroxy-16-(1-fluoro-2-(2-methyl-4 -thiazolyl)ethenyl)-1-oxa-5,5,7,9,13-pentamethyl-cyclohexadec-13-ene-2,6 -dione
01/22/2004US20040014973 Pyridin-4-YL or pyrimidin-4-YL substituted pyrazines
01/22/2004US20040014971 N-(4-(4-(2-oxo-1-phenyl-2-((2,2,2-trifluoroethyl)amino)ethyl)-1 -piperazinyl)-phenyl)-4'-(trifluoromethyl)-(1,1'-biphenyl)-2-carboxamide for treatment of obesity, diabetes, and cardiovascular disorders; decreases apoplioprotein secretion
01/22/2004US20040014964 Vitronectin receptor antagonist pharmaceuticals
01/22/2004US20040014802 Aminoindazole derivatives and intermediates, preparation thereof, and pharmaceutical compositions thereof
01/22/2004US20040014793 Stability in blood
01/22/2004US20040014790 Tartrate salt of thiazolidinedione derivative
01/22/2004US20040014784 Substituted propargylamines
01/22/2004US20040014783 Antiinflammatory agents; autoimmune diseases; rheumatic diseases; anticholesterol agents; cardiovascular disorders
01/22/2004US20040014776 Anticancer agents; cyclin-dependent kinase inhibitor
01/22/2004US20040014775 2,5-substituted pyrimidine derivatives-CCR-3 receptor antagonists
01/22/2004US20040014774 Aryl and heteroaryl quinazoline compounds which inhibit CSF-1R receptor tyrosine kinase
01/22/2004US20040014767 Central nervous system diosrders; antidepressants, anxiolytic agents, anxiolytic agents
01/22/2004US20040014765 Chk-1 inhibitors
01/22/2004US20040014758 Benzylcycloalkyl amines as modulators of chemokine receptor activity
01/22/2004US20040014748 Cardiovascular disorders, central nervous susyem disorders
01/22/2004US20040014745 Amide compounds
01/22/2004US20040014744 Anticancer, antitumor agents
01/22/2004DE10231711A1 Bicyclische Heterocyclen, diese Verbindungen enthaltende Arzneimittel, deren Verwendung und Verfahren zu ihrer Herstellung Bicyclic heterocycles, pharmaceutical compositions containing them, their use and process for their preparation
01/22/2004DE10228132A1 Amide cyclischer Aminosäuren als PDE 4 Inhibitoren Amides of cyclic amino acids as PDE 4 inhibitors
01/22/2004CA2492427A1 3-guanidinocarbonyl-1-heteroaryl-indole derivatives, preparation process, their use as medicaments, and pharmaceutical compositions comprising them
01/22/2004CA2492421A1 3-guanidinocarbonyl-1-heteroaryl-indole derivatives, preparation process, their use as medicaments, and pharmaceutical compositions comprising them
01/22/2004CA2492330A1 Derivatives of 3-guanidinocarbonyl-1-heteroaryl-pyrrole, process for their preparation and their pharmaceutical use
01/22/2004CA2492251A1 Sulphonylpiperidine derivatives containing an alkenyl or alkynly moiety for use as matrix metalloproteinase inhibitors
01/22/2004CA2492164A1 Substituted benzylamine derivatives and methods of use
01/22/2004CA2492100A1 Substituted 2-alkylamine nicotinic amide derivatives and use there of
01/22/2004CA2492093A1 Topical treatment of skin diseases
01/22/2004CA2492086A1 Sulphonylpiperidine derivatives containing an aryl or heteroaryl group for use as matrix metalloproteinase inhibitors
01/22/2004CA2492083A1 N-sulfonylpiperidines as metalloproteinase inhibitors (tace)
01/22/2004CA2492045A1 Substituted amine derivatives and methods of use
01/22/2004CA2491213A1 Cck-1 receptor modulators
01/22/2004CA2491191A1 Receptor-type kinase modulators and methods of use
01/21/2004EP1382604A1 Quinoline derivative having azolyl group and quinazoline derivative
01/21/2004EP1382603A1 NITROGENOUS FUSED−RING COMPOUND HAVING PYRAZOLYL GROUP AS SUBSTITUENT AND MEDICINAL COMPOSITION THEREOF
01/21/2004EP1382598A1 Novel heterocyclic derivatives
01/21/2004EP1382597A2 Steroid receptor modulator compounds and methods
01/21/2004EP1382336A1 Abc expression promoters
01/21/2004EP1382333A2 Use of beta 3 adrenergic receptor agonists in the treatment of dysuria
01/21/2004EP1381602A1 Heterocyclyldicarbamides as caspase inhibitors
01/21/2004EP1381598A1 Novel tyrosine kinase inhibitors
01/21/2004EP1381594A1 Urea compounds useful as anti-inflammatory agents
01/21/2004EP1381592A1 1,4-disubstituted benzo-fused compounds
01/21/2004EP1381590A1 3,4-di-substituted cyclobutene-1,2-diones as cxc-chemokine receptor ligands
01/21/2004EP1381382A2 Methods and compositions for the treatment of diseases of the eye
01/21/2004EP1381370A1 N-biphenylcarbonyl- and n-phenylpyridylcarbonyl substituted bi- and tricyclic azepines and diazepines as vasopressing agonists
01/21/2004EP1381360A1 Compounds and methods for inhibiting metap2 in mammals
01/21/2004EP1305028A4 Antimicrobial biaryl compounds
01/21/2004EP1280799B1 Ortho-substituted anthranilic acid amides and their use as medicaments
01/21/2004EP1126852B1 Pyridin-4-yl or pyrimidin-4-yl substituted pyrazines
01/21/2004EP1044198B1 Morpholino end-capped, hindered amine substituted aminotriazine and their use as light stabilizers
01/21/2004EP0937048B1 HETEROCYCLE DERIVATIVES WHICH INHIBIT FACTOR Xa
01/21/2004EP0811002B1 Benzylpiperidines and piperazines as muscarinic antagonists
01/21/2004CN1469876A Alpha-aryl ethanolamines and their use as beta-3 adrenergic receptor agonists
01/21/2004CN1469875A Pyrazole compounds useful as protein kinase inhibitors
01/21/2004CN1469874A Pyrazole compounds useful as protein kinase inhibitors
01/21/2004CN1469873A Piperidine compounds as anti-allergic
01/21/2004CN1469867A Novel phenylalanine derivatives
01/21/2004CN1469866A New derivatives of cyano-aryl (or cyanoheteroaryl)-carbonyl-piperazinyl- pyrimidines, their preparation and application as medication
01/21/2004CN1469865A Pyrazole derivatives for the treatment of viral diseases
01/21/2004CN1469864A Process for preparing cilostazol
01/21/2004CN1135227C 2,6-twice substituted pyridine and 2,4 twice substituted pyrimidine for berbicide
01/21/2004CN1135224C Benzimidazole derivatives
01/20/2004US6680338 Matrix metalloproteinase and tumor necrosis factor inhibitors; anticarcinogenic agents; rheumatoid arthritis
01/20/2004US6680335 Methods of modulating protein tyrosine kinase function with substituted indolinone compounds
01/20/2004US6680333 Imidazolidine derivatives, their preparation, their use and pharmaceutical preparations comprising them
01/20/2004US6680329 N-(heterocyclyl)benzene or pyridinesulphonamides as antithrombotic agents and anticoagulants
01/20/2004US6680323 Dihydropyrimidines and uses thereof
01/20/2004US6680321 4-((1-piperazinylmethyl)-benzamide derivatives; hypotensive agents; immunomodulators
01/20/2004US6680316 Pyridazin-3-one derivatives and medicines containing the same
01/20/2004US6680315 Compounds that down-regulate interleukin-12 production used for treating inflammatory diseases: rheumatoid arthritis, sepsis, chrohn's disease, multiple sclerosis, psoriasis or insulin-dependent diabetes
01/20/2004US6680314 Azacyclooctane and heptane derivatives, their preparation and use in therapy
01/20/2004US6680312 Sulfonamide derivatives, their production and use
01/20/2004CA2284795C Novel pyrimidine derivatives and processes for the preparation thereof