Patents
Patents for C07D 401 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom (107,979)
04/2004
04/28/2004EP1411984A2 Combination medicament for treatment of neoplastic diseases which contains cyanoguanidine ikk inhibitors and a second anti-neoplastic drug
04/28/2004EP1411949A2 8/17 heterocyclic compounds and uses thereof as d-alanyl-d-alanine ligase inhibitors
04/28/2004EP1411948A1 Tetrahydroquinoxalines acting as bradykinin antagonists
04/28/2004EP1411945A1 Substituted pyridin-4-ones and their use as gonadotropin-releasing hormone receptor antagonists
04/28/2004EP1411944A1 Sulfonamide derivatives as gamma secretase inhibitors
04/28/2004EP1411942A1 Substituted anilinic piperidines as mch selective antagonists
04/28/2004EP1411941A2 Pyridinone and pyridazinone derivatives as gonadotropin-releasing hormone receptor antagonists
04/28/2004EP1411940A1 Bridged piperidine derivatives as melanocortin receptor agonists
04/28/2004EP1411933A1 Alpha-ketoamide derivatives as cathepsin k inhibitors
04/28/2004EP1411929A2 Malonyl-coa decarboxylase inhibitors useful as metabolic modulators
04/28/2004EP1411928A1 Viral polymerase inhibitors
04/28/2004EP1244642B1 Substituted oxazoles and thiazoles derivatives as hppar alpha activators
04/28/2004EP1230237B1 Magnesium omeprazole
04/28/2004EP1228062B1 Herbicidal 2-aryloxy-6-fluoroalkylthioalk(en)yloxy-pyridines
04/28/2004EP1208096B1 Substituted pyridazines and fused pyridazines with angiogenesis inhibiting activity
04/28/2004EP1042313B1 Benzopyran and benzothiopyran derivatives having retinoid antagonist like activity
04/28/2004EP0946544B1 Heterocyclyluracil
04/28/2004EP0888271B1 Benzamidine derivatives substituted by amino acid and hydroxy acid derivatives and their use as anti-coagulants
04/28/2004CN1492863A Heterocyclylalkylindole or azaindole compounds as 5-hydroxytryptamine-6 ligands
04/28/2004CN1492860A 喹唑啉衍生物 Quinazoline derivatives
04/28/2004CN1492856A Pyridone derivative having affinity for cannabinoid 2-type receptor
04/28/2004CN1491945A Process for preparing human immunodeficiency virus (HIV) proteinase inhibitor
04/28/2004CN1491944A 5-amino-8-methoxy quinolone carboxylic acid derivatives and its preparation
04/28/2004CN1491941A Heterobicyclic sulfonamide derivative and sulfonic ester derivative
04/28/2004CN1147486C 4-and 5-alkynyloxindoles and 4-and 5-alkenyloxindoles
04/28/2004CN1147485C Indoline derivatives useful as 5-HT-2C receptor antagonists
04/28/2004CN1147476C Pyrazole derivatives as P-38 MAP kinase inhibitors
04/28/2004CN1147471C Renin inhibitors
04/27/2004US6727364 Antiinflammatory agents
04/27/2004US6727275 Pyrrolidinone derivatives
04/27/2004US6727273 Therapy for osteoporosis, anticancer agents
04/27/2004US6727264 Substituted anilinic piperidines as MCH selective antagonists
04/27/2004US6727257 Hypotensive agents for intraocular pressure; anticholesterol agents; relaxing urinary tract tissue; benign prostatic hyperplasia, impotency, and cardiovascular disorders; antiarrhythmia agents
04/27/2004US6727255 Brain, nervous system and psychological disorders
04/27/2004US6727251 Inhibitors of glycogen synthase kinase-3 (gsk-3) and aurora-2, both serine/threonine protein kinases; for treating diseases such as cancer, diabetes and alzheimer's disease
04/27/2004US6727248 Substituted quinolinecarboxamides as antiviral agents
04/27/2004US6727239 Inhibitory activity on no- synthase enzymes producing nitrogen monoxide no and/or an activity which traps the reactive oxygen species (ros)
04/27/2004US6727237 Alkylating 5-nitroindole with 6-bromohexyl acetate to form a 6-(N-(5-nitroindolyl)) hexyl acetate, hydrolyzing to form alcohol of above ester, estrifying with nicotinic acid, and methylating the intermediate
04/27/2004US6727041 Optical recording media
04/27/2004CA2136745C Heterocyclically disubstituted sulphonylamino(thio)carbonyl compounds
04/23/2004CA2445817A1 Novel derivatives of imidazoline, process for their preparation and pharmaceutical compositions containing them
04/22/2004WO2004033632A2 Hydantoin derivatives as inhibitors of matrix metalloproteinases and/or tnf-alpha converting enzyme (tace)
04/22/2004WO2004033446A1 Protein tyrosine kinase inhibitors
04/22/2004WO2004033445A1 4-amino-azepan-3-one compounds as cathepsin k inhibitors useful in the treatment of osteoporosis
04/22/2004WO2004033444A1 Dihydropyridine compounds having simultaneous ability to block l-type calcium channels and to inhibit phosphodiesterase type 3 activity
04/22/2004WO2004033436A1 Sulfonylbenzodiazepinone acetamides as bradykinin antagonists
04/22/2004WO2004033434A1 Pyrazole compounds for treatment of neurodegenerative disorders
04/22/2004WO2004033432A1 Novel pyrazole compounds having antifungal activity
04/22/2004WO2004033431A2 Hydroxypyrazoles for use against metabolic-related disorders
04/22/2004WO2004033428A1 Substituted 1,4-di-piperidin-4-yl-piperazine derivatives and their use as neurokinin antagonists
04/22/2004WO2004033427A1 1,4-disubstituted piperidine derivatives and their use as 11-betahsd1 inhibitors
04/22/2004WO2004033426A2 Heteroaryl propyl-piperazines and heteroaryl propyl-piperidines serving as dopaminergic and serotoninergic agents
04/22/2004WO2004033418A2 Sulfonylamino-acetic derivatives and their use as orexin receptor antagonists
04/22/2004WO2004032929A2 Dual binding site acetylcholinesterase inhibitors for the treatment of alzheimer’s disease
04/22/2004WO2004032908A2 Method of inhibiting angiogenesis
04/22/2004WO2004032848A2 Pgd2 receptor antagonists for the treatment of inflammatory diseases
04/22/2004WO2004032846A2 Triazolone and triazolethione derivatives
04/22/2004WO2004032834A2 Thrombin inhibitors
04/22/2004WO2004022544A8 Novel aminoindazole derivatives as medicines and pharmaceutical compositions containing same
04/22/2004WO2004020410A3 Dihydropyridinone derivatives as hne inhibitors
04/22/2004WO2004018431A3 Novel phenanthridines
04/22/2004WO2004016597A3 Protein kinase inhibitors and uses thereof
04/22/2004WO2004014300A3 Tyrosine kinase inhibitors
04/22/2004WO2004005407A3 Tetra-azapentamethine and use thereof for dyeing keratinous fibers
04/22/2004WO2004002984A3 Marked maleimide compounds, method for preparing same and use thereof for marking macromolecules
04/22/2004WO2003078403A3 Derives d’aminoindazoles comme inhibiteurs de proteine-kinase
04/22/2004WO2003072106A3 Use of tyrosine kinase inhibitors for treating substance use disorders
04/22/2004WO2003005999A8 Methods of treating cytokine mediated diseases
04/22/2004WO2002098857A8 New indole derivatives with 5-ht6 receptor affinity
04/22/2004WO2002074767A8 Metalloproteinase inhibitors
04/22/2004WO2002074752A8 Metalloproteinase inhibitors
04/22/2004WO2002074748A8 Metalloproteinase inhibitors
04/22/2004US20040077877 Jun n-terminal kinase inhibitors
04/22/2004US20040077869 Process for preparation of optically pure or optically enriched sulfoxide compounds, including amorphous esomeprazole and salts thereof
04/22/2004US20040077865 Making 1-amino-6-nitroisoquinoline by reacting beta-(dimethylamino)-2-cyano-5-nitro-styrene with lithium hexamethyldisilazane or reacting said styrene compound with 2,4-dimethoxybenzylamine and then with anisole
04/22/2004US20040077860 Quinoxaline derivative; light-emitting diode, light-emitting electrochemical cell, or a photodetector
04/22/2004US20040077853 2-amino-6-(2,4,5-substituted-phenyl)-pyridines
04/22/2004US20040077851 Receptor selective cannabimimetic aminoalkylindoles
04/22/2004US20040077798 Thermosetting resin compositions containing maleimide and/or vinyl compounds
04/22/2004US20040077709 Neuronal death inhibitors
04/22/2004US20040077707 Pyrrole based inhibitors of glycogen synthase kinase 3
04/22/2004US20040077706 Piperidine and azepine derivatives; anxiolytic, analgesic, antidepressant, antiemetic, antiinflammatory, and hypotensive agents; sexual and psychological disorders; Alzheimer*s, Parkinson*s, Lesche-Nyhane, Wilson*s, and Tourette*s syndrome
04/22/2004US20040077701 Pyrazole derivates for treatment of osteoporosis, breast and endometrial cancers, atherosclerosis, and Alzheimer*s disease
04/22/2004US20040077699 Substituted triazole diamine derivatives as kinase inhibitors
04/22/2004US20040077690 Anticoagulants; cardiovascular and brain disorders
04/22/2004US20040077689 Abc expression promoters
04/22/2004US20040077688 Treating psoriasis, gastroesophageal reflux, Zollinger-Ellison Syndrome; antiulcer and antisecretory agents
04/22/2004US20040077686 Inhibition of cyclooxygenase-2 activity
04/22/2004US20040077685 Analogs of thalidomide as potential angiogenesis inhibitors
04/22/2004US20040077684 Piperidinyl compounds that selectively bind integrins
04/22/2004US20040077671 Sorbitol dehydrogenase inhibitors
04/22/2004US20040077670 Novel sulfamides and their use as endothelin receptor antagonists
04/22/2004US20040077668 Compounds, compositins, and methods
04/22/2004US20040077667 Quinazolinone derivatives
04/22/2004US20040077656 Quinolines and nitrogenated derivatives thereof substituted in 4-position by a piperazine-containing moiety and their use as antibacterial agents
04/22/2004US20040077655 Piperazine derivatives for treatment of bacterial infections
04/22/2004US20040077654 Anticholesterol agents; cardiovascular disorders
04/22/2004US20040077653 GABAA (gamma-aminobutyric acid) receptor modulators; anxiolytic, antidepresant agents; attention deficit disorder, Alzheimer*s disease treatment; central nervous systmem disorders
04/22/2004US20040077650 Cannabinoid receptor ligands and uses thereof
04/22/2004US20040077648 Antiproliferative agents for smooth muscle cells; antiinflammatory agents for endothelial cells; restenosis, atherosclerosis