Patents
Patents for C07D 401 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom (107,979)
04/2004
04/15/2004WO2004031158A1 Indazolecarboxamide derivatives, preparation and use thereof as cdk1, cdk2 and cdk4 inhibitors
04/15/2004WO2004031153A2 Enantioselective alkylation of tricyclic compounds
04/15/2004WO2004031150A1 Oxoammonium salts of 1-oxy-2,2,6,6-tetramethyl-1-piperidine (tempo) and their use as oxidizing agents
04/15/2004WO2004031145A2 Lactam-containing diaminoalkyl, beta-aminoacids, alpha-aminoacids and derivatives thereof as factor xa inhibitors
04/15/2004WO2004030637A2 Treatment of obesity and other disorders associated with excessive food intake
04/15/2004WO2004030635A2 Vasculostatic agents and methods of use thereof
04/15/2004WO2004030620A2 Novel tyrosine kinase inhibitors
04/15/2004WO2004030611A2 Non-nucleoside reverse transcriptase inhibitors
04/15/2004WO2004018436A3 Compounds derived from aryl carbamates, preparation thereof and uses of same
04/15/2004WO2004016607B1 Inhibition of phosphoinositide 3-kinase beta
04/15/2004WO2004014859A3 Process for preparing quinolin antibiotic intermediates
04/15/2004WO2004009558A3 Ureido substituted benzoic acid compounds, their use for nonsense suppression and the treatment of diseases caused by such mutations
04/15/2004WO2004005262A3 New neuropeptide y y5 receptor antagonists
04/15/2004WO2003106381A3 Human adam-10 inhibitors
04/15/2004WO2002083111A3 Imidazole, thiazole and oxazole derivatives and their use for the manufacture of a medicament for the treatment and/or prevention of pollakiuria or urinary incontinence
04/15/2004US20040073054 Using a fluorinated phenyl compound containing electrophilic and nucleophilic groups
04/15/2004US20040073039 Blocking neurotransmitter
04/15/2004US20040073036 Substituted alkyl amido piperidines
04/15/2004US20040073025 Thrombin inhibitors
04/15/2004US20040072892 Dipeptidyl aminopeptidase inhibitors; kidney and liver disorders; autoimmune diseases; antiarthritic agents; psoriasis; anticancer agents
04/15/2004US20040072889 Method of using a COX-2 inhibitor and an alkylating-type antineoplastic agent as a combination therapy in the treatment of neoplasia
04/15/2004US20040072888 Administering pyrazoloanthrone compound
04/15/2004US20040072881 Dietetics; osteoporosis; muscular disorders
04/15/2004US20040072874 N-substituted-2-oxodihydropyridine derivatives
04/15/2004US20040072869 Bipolar disorders; psychological diseases
04/15/2004US20040072867 Antiemetics, antidepressants, anxiolytic agents, antitussive agents
04/15/2004US20040072865 Anticholesterol agents; antidiabetic agents; antilipemic agents
04/15/2004US20040072862 Compositions for treating ischemia-related neuronal damage
04/15/2004US20040072860 Piperazin-2-one amides as inhibitors of factor xa
04/15/2004US20040072844 2,4-Substituted indoles and methods of use
04/15/2004US20040072843 Novel sulfonamide substituted chroman derivatives useful as beta 3 adrenoreceptor agonists
04/15/2004US20040072830 Squalene synthetase inhibitors; antilipemic agents; antiischemic agents; cardiovascular disorders; anticholesterol agents
04/15/2004US20040072829 Piperazinyltriazines as estrogen receptor modulators
04/15/2004US20040072823 Central nervous system disorders; analgesics; antiinflammatory agents
04/15/2004US20040072818 Antiinflammatory agents; autoimmune disease; anticancer agents
04/15/2004US20040072816 Dysmenorrhea; congestive heart failure; liver disorders; vision defects
04/15/2004US20040072802 Antiarthritic agents; antiulcer agents; bone disorders; antitumor agents; oral diseases
04/15/2004US20040072692 4-trifluoromethylpyrazolyl-substituted pyridines and pyrimidines
04/15/2004US20040072309 Method for producing 2-azetidinone derivative
04/15/2004DE10257188B3 Preparation of meso-substituted cyanine dye, for radiation-sensitive coating, e.g. for making printing plate, printed circuit boards or DVD, from 2-halo-cyclo-pentene or -hexene-dianil involves 1-stage introduction of end and meso-groups
04/15/2004DE10248067A1 New N-diaminophenylpropyl- or N-heteroarylpropyl-piperazine or piperidine derivatives, useful as dopaminergic and/or serotoninergic agents for e.g. treating Parkinson's disease or schizophrenia
04/15/2004CA2726754A1 N-substituted-2-oxodihydropyridine derivatives
04/15/2004CA2501292A1 Enantioselective alkylation of tricyclic compounds
04/15/2004CA2501243A1 Piperidine derivatives as ccr5 inhibitors
04/15/2004CA2500977A1 2-thiohydantoine derivative compounds and use thereof in therapeutics
04/15/2004CA2500815A1 Method and intermedia used to obtain derivatives of 1-(1h-benzimidazole-2-il)-4-(2-aminopyrimidine)piperidine
04/15/2004CA2500727A1 Vasculostatic agents and methods of use thereof
04/15/2004CA2499732A1 Piperazine derivatives and methods of use
04/15/2004CA2496565A1 Non-nucleoside reverse transcriptase inhibitors
04/15/2004CA2495698A1 Imidazol-1-ylmethyl pyridazine derivatives
04/14/2004EP1408037A1 Novel diarylmethylpiperazine and diarylmethylphenyl compounds with analgesic effect
04/14/2004EP1407774A1 2-Amino-4-quinazolinones as LXR nuclear receptor binding compounds
04/14/2004EP1406983A1 Tertiary diamines containing heterocyclic groups and their use in organic electroluminescent devices
04/14/2004EP1406897A2 Compounds
04/14/2004EP1406894A1 Piperazine oxime derivatives having nk-1 receptor antagonistic activity
04/14/2004EP1406893A1 Pyrrolidine bicyclic compounds
04/14/2004EP1406892A1 Phenyl pyrazole derivatives as soluble epoxide hydrolase inhibitors
04/14/2004EP1406884A1 Arylsusfonamide compounds for the treatment of obesity, type ii diabetes and cns-disorders
04/14/2004EP1406878A1 4-(benzylidene-amino)-3-(methylsulfanyl)-4h-(1, 2, 4) triazin-5-one derivatives having a pde-iv inhibiting and tnf-antagonistic effect for the treatment of cardiac diseases and allergies
04/14/2004EP1406877A1 Heterocyclic amines for the treatment of conditions associated with gsk-3
04/14/2004EP1406875A1 N-heterocyclic inhibitors of tnf-alpha expression
04/14/2004EP1406873A2 Fluoropyrrolidines as dipeptidyl peptidase inhibitors
04/14/2004EP1406872A2 Dipeptidyl peptidase inhibitors for the treatment of diabetes
04/14/2004EP1406696A1 Use of compositions comprising cyclooxygenase-2 selective inhibitors in combination with radiation for inhibition or prevention of cardiovascular disease
04/14/2004EP1406628A1 Tetrahydroquinoline derivatives
04/14/2004EP1406627A1 Pyridin-2-yl-methlyamine derivatives for treating opioid dependence
04/14/2004EP1406626A2 Sulphonyl aryl hydroxamates and their use as mmp inhibitors
04/14/2004EP1406622A2 Dipeptidyl peptidase inhibitors for the treatment of diabetes
04/14/2004EP1406620A1 Vinyl phenyl derivatives as glk activators
04/14/2004EP1406619A1 Antiviral and antimicrobial guanidine or biguanidine derivatives
04/14/2004EP1406618A2 Use of nk-1 receptor antagonists with pyridinic structure for the treatment of brain, spinal or nerve injury
04/14/2004EP1406602A2 Use of sulfonyl aryl or heteroaryl hydroxamic acids and derivatives thereof as aggrecanase inhibitors
04/14/2004EP1406572A2 Pediatric formulation of gatifloxacin
04/14/2004EP1375465A9 Cyclooctanone derivative and cyclodecanone derivative, and use thereof
04/14/2004EP1305270B1 Kinetic resolutions of chiral 2- and 3-substituted carboxylic acids
04/14/2004EP1214312B1 5-aminoalkyl and 5-aminocarbonyl substituted indoles
04/14/2004EP1214299B1 Muscarinic antagonists
04/14/2004EP1155012B1 Anti-cancer dihydroquinazoline derivatives
04/14/2004EP1131297B1 Certain substituted caprolactams, pharmaceutical compositions containing them and their use in treating tumors
04/14/2004EP1042315B1 Cyclic imide-substituted pyridylalkane, alkene, and alkine carboxamides useful as cytostatic and immunosuppressive agents
04/14/2004EP0948495B1 Aryl and heteroaryl substituted fused pyrrole antiinflammatory agents
04/14/2004EP0935465B1 Novel substituted imidazole compounds
04/14/2004EP0912565B1 Process for preparing imidazoquinolinamines
04/14/2004EP0892790B1 New quinazoline-4-amino-2-(piperidine-1-yl-4-substituted) derivatives having anti-hypertensive activity, a method for their preparation and their pharmaceutical use
04/14/2004EP0706515B1 Intercalators having affinity for dna and methods of use
04/14/2004CN1489591A Benzensulfonic acid indol-5-yl esters and antigonists of the 5-HT6 receptor
04/14/2004CN1489586A Indazolyl-substituted pyrroline compounds as kinase inhibitor
04/14/2004CN1489585A Process for producing substituted 2-(2-pyridylmethye)sulfinye-1H-benzinmidazoles
04/14/2004CN1489584A Method for carbamoylating alcohols
04/14/2004CN1489581A 喹唑啉酮衍生物 Quinazolinone derivatives
04/14/2004CN1489580A Imidazole derivatives
04/14/2004CN1145624C New Process
04/14/2004CN1145623C Imidazole derivatives
04/14/2004CN1145616C Novel amino-triazole compound, its preparation method and drug composition containing them
04/14/2004CN1145612C New 1-aza-2-alkyl-6-aryl-cyclanes compound, its producing process and medical composition containing them
04/14/2004CN1145609C Piperazine compounds and medical use thereof
04/14/2004CN1145485C 8-chloro-6,11-dihydro-11-(4-piperidy lidene)-5H-benzo[5,6] cyclohepta [1,2,-b] pyridine oral compositions
04/13/2004US6720351 1h-indole-2-carboxylic acid (2-(benzyl(methyl)amino) -2-oxo-1-phenylethyl)amides; triamide microsomal triglyceride transfer protein (mtp) and apolipoprotein b (apo b) inhibitors; obesity; antilipemic agents
04/13/2004US6720344 Methods and compositions for stimulating osteoblast proliferation or treating malignant cell proliferation and methods for selecting osteoblast proliferation stimulants
04/13/2004US6720339 Such as n-phenyl-4-oxo-6,6-dimethyl-4,5,6,7-tetrahydro-1h-indole-3-carboxamide; for diagnosis and treatment of anxiety, sleep and seizure disorders, overdose with benzodiazepine drugs, and for memory enhancement