Patents for C07D 401 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom (107,979) |
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06/09/2005 | WO2005051300A2 Bicyclic inhibitors of mek and methods of use thereof |
06/09/2005 | WO2005051110A1 Corrective clothes with crotch |
06/09/2005 | WO2005035508A3 Method for producing acyl urea derivatives, salts of said acyl urea derivatives, and the use thereof as pesticides |
06/09/2005 | WO2003088897A3 Fab i inhibitors |
06/09/2005 | US20050124683 Viricides; immunomoderators |
06/09/2005 | US20050124682 Such as N-{2-[5-(methylthio)-1H-indol-3-yl]ethyl}acetamide for treatment of disorders of the melatoninergic system; hormone replacement therapy |
06/09/2005 | US20050124679 Alpha, beta-unsaturated hydroxamic acid derivatives and their use as histone deacetylase inhibitors |
06/09/2005 | US20050124672 Antineoplastic agents, analgesics, antipyretics; prostaglandin E2 receptor antagonists; 3-Methyl-4-[6-[N-isobutyl-N-(2-thiazolylsulfonyl)amino]indan-5-yloxymethyl]benzoic acid, a C1-4 alkyl ester, or a non-toxic salt |
06/09/2005 | US20050124671 Benzylcycloalkyl amines as modulators of chemokine receptor activity |
06/09/2005 | US20050124662 Indazole compounds and pharmaceutical compositions for inhibiting protein kinases, and methods for their use |
06/09/2005 | US20050124656 Substituted methylene amide derivatives as modulators of protein tyrosine phosphatases(ptps) |
06/09/2005 | US20050124655 Cyclization; solvent extraction; hydrolysis; phosphodiesterase (PDE IV) inhibitors |
06/09/2005 | US20050124652 Guanidino compounds |
06/09/2005 | US20050124640 Pyrimidine derivatives useful as inhibitors of PKC-theta |
06/09/2005 | US20050124638 Benzimidazoles and analogs thereof as antivirals |
06/09/2005 | US20050124631 For example, 2-amino-7-chloro-6-hydroxy-4-methylbenzothiazole; compounds that prevent the formation of polyglutamine containing protein aggregates; treatment of spinal and bulbar muscular atrophy, dentatorubal pallidoluysian atrophy, spinocerebellar ataxia, Alzheimers disease |
06/09/2005 | US20050124630 Bicyclic indolyl derivatives and methods for their use as serotonergic agents |
06/09/2005 | US20050124628 Quinoline and aza indole compounds having pharmacological activity, for example, 8-(4-Methyl-piperazin-1-yl)-3-phenylsulfonylquinoline; use in the treatment of CNS and other disorders |
06/09/2005 | US20050124625 For example, ((2R,5S)-4-(8-cyano-quinolin-5-yl)-2,5-dimethyl-piperazine-1-carboxylic acid(4-trifluoromethyl-pyridin-3-yl)-amide); use in treatment of nuclear hormone receptor-associated conditions such as cancer and immune disorders |
06/09/2005 | US20050124624 4-(4-methylpiperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl)pyrimidin-2-yl-amino)phenyl]-benzamide for threating ang ii-mediated diseases |
06/09/2005 | US20050124620 Indole derivatives having an acidic moiety that inhibit or modulate activity of p38 map kinase mediating a disease state; e.g., 3-(2-(4-pyridyl)ethyl)-5-(3-trifluoromethoxybenzamido)indole; enzyme inhibitors; antiarthritic, -inflammatory, and -carcinogenic agents; respiratory disorders; AIDS; Alzheimer's |
06/09/2005 | US20050124619 Medical devices employing triazine compounds and compositions thereof |
06/09/2005 | US20050124614 E. g., 3,5-bis-trifluoromethylphenyl)-4-[(furan-2-ylmethyl)-aminocarbonyl]-2-methyl-1-oxo-1,2,3,4-tetrahydroisoquinoline;anticarcinogenic agents; antitumor agents; antiproliferative agents; activators of the caspase cascades; enzyme inhibitors used in combination with radiation or chemotherapy |
06/09/2005 | US20050124611 Such as N-[4-[[4-(5-chloro-2-hydroxyphenyl)-1,2-dihydro-2-oxo-6-(trifluoromethyl)-3-quinolinyl]thio]phenyl]-4-morpholineacetamide; potassium channel modulators |
06/09/2005 | US20050124610 cyclin dependent kinase (CDK) inhibitors useful in treating or ameliorating a CDK mediated disorder consisting of cervical adenocarcinoma, colon carcinoma and malignant melanoma |
06/09/2005 | US20050124607 5-Substituted quinazolinone compounds useful as alpha 1A/B adrenergic receptor antagonists |
06/09/2005 | US20050124605 E.g., substituted 2,3,5,10b-tetraaza-benzo[e]azulen-6-yl)-acetic acids, 2,3,4,5-tetrahydro-1H-benzo[e][1,4]diazepin-5-yl)-(4,6-dimethoxy-pyrimidin-2-yloxy)-acetic acids and 2,3,4,5-tetrahydro-benzo[e][1,4]diazepin-1-ylmethyl}-benzoates; treating circulatory, inflammatory, and proliferative disorders |
06/09/2005 | US20050124603 Heterocyclylindazole and -azaindazole compounds as 5-hydroxytryptamine-6 ligands |
06/09/2005 | US20050124602 1-(3-chlorophenyl)-7-oxo-6-[4-(2-oxo-1(2H)pyridinyl)phenyl]-4,5,6,7-tetrahydro-1H-pyrazolo[3,4-c]pyridine-3-carboxamide; treating a thromboembolic disorder such as deep vein thrombosis or pulmonary embolism |
06/09/2005 | US20050124600 And thiones, 1-substituted with a (hetero)aryl)carbonyl group, e.g., 6-Bromo-1-[[3-bromo-1-(3-chloro-2-pyridinyl)-1H-pyrazol-5-yl]carbonyl]-8-methyl-3-(1-methylethyl)-2,4(1H,3R)-quinazolinedione; especially for use in growing and stored agronomic crops |
06/09/2005 | US20050124599 Novel benzoimidazole derivatives useful as antiproliferative agents |
06/09/2005 | US20050124562 Using Dna polymerase inhibitor as bactericide |
06/09/2005 | US20050124497 Pesticide, 5-tert-butyl-2-{4-[5-(2,6-difluorophenyl)-3,4-dihydro-2H-pyrrol-2-yl]phenyl}-1,3-benzoxazole; chemical intermediates, N-(5-tert-butyl-2-hydroxyphenyl)-4-[5-(2,6-difluorophenyl)-3,4-dihydro-2H-pyrrol-2-yl]benzamide; applying on plants, animals |
06/09/2005 | US20050124209 Illuminated electrical cords and outlets |
06/09/2005 | DE10352499A1 Substituierte Dihydrochinazoline II Substituted dihydroquinazolines II |
06/09/2005 | CA2547472A1 Cyclic amine derivative having heteroaryl ring |
06/09/2005 | CA2546932A1 Quinazolinone compounds as anticancer agents |
06/09/2005 | CA2546709A1 Amino substituted pyridinyl methanone compounds useful in treating kinase disorders |
06/09/2005 | CA2546673A1 Diaryl urea derivatives in the treatment of protein kinase dependent diseases |
06/09/2005 | CA2546493A1 Indazole compounds and methods of use thereof as protein kinase inhibitors |
06/09/2005 | CA2546486A1 Heterocyclic inhibitors of mek and methods of use thereof |
06/09/2005 | CA2546360A1 Methods of treating diseases and disorders by targeting multiple kinases |
06/09/2005 | CA2546353A1 Bicyclic inhibitors of mek and methods of use thereof |
06/09/2005 | CA2546264A1 4-phenylpiperidine derivatives as renin inhibitors |
06/09/2005 | CA2546142A1 Benzylether and benzylamino beta-secretase inhibitors for the treatment of alzheimer's disease |
06/09/2005 | CA2545660A1 Heterocyclic inhibitors of mek and methods of use thereof |
06/09/2005 | CA2545659A1 Bicyclic inhibitors of mek |
06/09/2005 | CA2545601A1 Quinazolinone compounds with reduced bioaccumulation |
06/09/2005 | CA2545262A1 Quinazoline derivatives |
06/09/2005 | CA2544519A1 Pyrazolyl derivatives in the form of drugs for treating acute or chronic neuronal regressions |
06/08/2005 | EP1538159A1 Substituted N-benzyl-lactam derivatives as melanocortin-4 receptor agonists |
06/08/2005 | EP1538150A1 Novel pleuromutilin derivatives |
06/08/2005 | EP1538145A1 Process for production of phenoxy-substituted 2-pyridone compounds |
06/08/2005 | EP1537870A2 Methods and compositions for treating cancer |
06/08/2005 | EP1537111A1 Hetereoaryl nitrile derivatives |
06/08/2005 | EP1537102A1 Inhibition of phsphoinostide 3-dinase beta |
06/08/2005 | EP1537100A1 Pyrrolidinedione substituted piperidine-phthalazones as pde4 inhibitors |
06/08/2005 | EP1537099A1 Pyrrole based inhibitors of glycogen synthase kinase 3 |
06/08/2005 | EP1537098A1 Monocyclic derivatives as matrix metalloproteinase inhibitors |
06/08/2005 | EP1537097A2 Method for preparing 3-halo-4,5-dihydro-1 i h /i -pyrazoles |
06/08/2005 | EP1537089A2 Compounds compositions and methods |
06/08/2005 | EP1537087A1 Novel aminoindazole derivatives as medicines and pharmaceutical compositions containing same |
06/08/2005 | EP1537086A2 Novel phenanthridines |
06/08/2005 | EP1537085A1 Oxytocin inhibitors |
06/08/2005 | EP1537084A1 Substituted 2-alkylamine nicotinic amide derivatives and use there of |
06/08/2005 | EP1537081A1 Dihydropyridine derivatives for use as human neutrophil elastase inhibitors |
06/08/2005 | EP1537078A1 Indoles having anti-diabetic activity |
06/08/2005 | EP1537075A2 Diarylurea derivatives and their use as chloride channel blockers |
06/08/2005 | EP1537074A1 Cathepsin cysteine protease inhibitors |
06/08/2005 | EP1536799A1 Novel 2-amino-4-oxoquinazolones as lxr nuclear receptor binding compounds with partial agonistic properties |
06/08/2005 | EP1536797A1 1-amido-4-phenyl-4-benzyloxymethyl-piperidine derivatives and related comounds as neurokinin-1 (nk-1) antagonsists for the treatment of emesis, depression, anxiety and cough |
06/08/2005 | EP1536796A1 N-aryl piperidine substituted biphenylcarboxamides as inhibitors of apolipoprotein b secretion |
06/08/2005 | EP1536784A1 Hetero biaryl derivatives as matrix metalloproteinase inhibitors |
06/08/2005 | EP1536684A2 Method for the prevention and/or treatment of atherosclerosis |
06/08/2005 | EP1458706A4 Diaryl 1,2,4-triazole derivatives as a highly selective cyclooxygenase-2 inhibitor |
06/08/2005 | EP1370528B1 Mch antagonists and their use in the treatment of obesity |
06/08/2005 | EP1337526B1 Substituted imidazoles useful in the treatment of inflammatory diseases |
06/08/2005 | EP1294710B1 Indole derivatives useful for the treatment of cns disorders |
06/08/2005 | EP1263301A4 Method and system for assay and removal of harmful toxins during processing of tobacco products |
06/08/2005 | EP1252133B1 Pharmaceutical compounds |
06/08/2005 | EP1089735B1 4-benzyl piperidine alkylsulfoxide heterocycles and their use as subtype-selective nmda receptor antagonists |
06/08/2005 | EP1019045B1 Antithrombotic agents |
06/08/2005 | CN1625555A Quinazoline compounds |
06/08/2005 | CN1625410A 2, 4, 6-triamino-1, 3, 5-triazine derivative |
06/08/2005 | CN1625400A 2, 4-pyrimidinediamine compounds and their uses |
06/08/2005 | CN1623984A Fused-ring compounds and use thereof as drugs |
06/08/2005 | CN1623537A Biaryl sulfonamides and its using method |
06/08/2005 | CN1205205C Sodium-hydrogen exchanger type 1 inhibitor crystals |
06/08/2005 | CN1205202C N-carbanilides used as pesticides |
06/08/2005 | CN1205188C 4,5-dihydro-1h-pyrazole derivatives having CB1-antagonistic activity |
06/08/2005 | CN1205185C Nitrogenous cyclic compounds and pharmaceutical compositions containing the same |
06/08/2005 | CN1205183C New amidino derivatives and their use as thrombin inhibitors |
06/07/2005 | US6903218 Substituted or unsubstituted aryl-1-hydroxyethylaminocarbonylalkyl-chroman-sulfonamide compounds are useful in the treatment of beta-3 receptor mediated conditions |
06/07/2005 | US6903217 Heterocyclylalkylpiperidine derivatives, their preparation and compositions containing them |
06/07/2005 | US6903216 Antiarrhythmic agents for the treatment and prophylaxis of atrial arrhythmias, atrial fibrillation (AF) or atrial flutter; potassium channel modulators, beta-blocker |
06/07/2005 | US6903215 Glucocorticoid mimetics, methods of making them, pharmaceutical compositions, and uses thereof |
06/07/2005 | US6903213 HIV inhibiting pyrimidine derivatives |
06/07/2005 | US6903131 Administering to a patient an antiangiogenesis or anticancer agent (N,N-disubstituted-3,4-diamino-2,4-dione-pyrroline derivatives for the treatment of chemokine-mediated diseases such as acute and chronic inflammatory disorders and cancer |
06/07/2005 | US6903126 1-Aryl-2-N-, S- or O-substituted benzimidazole derivatives, their use for the production of pharmaceutical agents as well as pharmaceutical preparations that contain these derivatives |
06/07/2005 | US6903123 Antitussive agents, anxiolytic agents, analgesics for treating cough, anxiety and pain |