Patents
Patents for C07D 401 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom (107,979)
07/2005
07/06/2005EP1549316A1 INHIBITORS OF TFG&bgr;
07/06/2005EP1373256B1 Ccr5 antagonists useful for treating aids
07/06/2005EP1212320B1 Phenylpiperazines as serotonin reuptake inhibitors
07/06/2005EP1140909B1 Novel inhibitors of farnesyl-protein transferase
07/06/2005EP1044001B1 Integrin receptor antagonists
07/06/2005EP0776327B1 New multimerizing agents
07/06/2005CN1636154A Di-substituted iminoheterocyclic compounds
07/06/2005CN1636011A Succinoylamino lactams as inhibitors and as a beta protein production
07/06/2005CN1636001A 2-amino-4-bicyclyl amino-6h-1.3.5-triazines, method for the production and use thereof as herbicides and plant growth regulators
07/06/2005CN1636000A 5-substituted arylpyrimidines
07/06/2005CN1635891A Tetrahydroquinoline analogues as muscarinic agonists
07/06/2005CN1635890A Neuroprotective 2-pyridinamine compositions and related methods
07/06/2005CN1635885A Improvement of nitric oxide synthase activity by using substituted indole compound
07/06/2005CN1635877A Treatment of affective disorders by the combined action of a nicotinic receptor agonist and a monoaminergic substance
07/06/2005CN1634918A 2-pyridyl-1H-benzimidazole-4-amide derivatives
07/06/2005CN1634893A 4, 5-disubstituted-1, 8-naphthoyl imide compounds and use thereof
07/06/2005CN1209368C Novel acetamide derivative and use thereof
07/06/2005CN1209362C Tetrazolyl-phenyl acetamide glucokinase activators
07/06/2005CN1209361C Hydantoin-containing glucokinase activators
07/06/2005CN1209360C 16-halogen-epothilone derivatives, process for producing them and their pharmaceutical use
07/06/2005CN1209359C Novel dihydric indole compound, their preparation process and medicinal compositions containing them
07/06/2005CN1209358C Inhibitors of alpha L beta 2 mediated cell adhesion
07/06/2005CN1209351C N-(4-aryloxypiperidin-1-ylalkyl) cinnamic amides as CCR3 receptor antagonists
07/06/2005CN1209016C Fungicides
07/05/2005US6914160 Oxytocin inhibitors
07/05/2005US6914069 Pharmaceutically active compounds and methods of use
07/05/2005US6914066 1,2-annelated quinoline derivatives
07/05/2005US6914062 Pyrazinone derivatives
07/05/2005US6914058 1-(p-(thiomorpholino)phenyl)-1,2,3-triazole derivatives
07/05/2005CA2309485C New 4-arylpiperidine derivatives for the treatment of pruritus
07/05/2005CA2160928C Compounds as pde iv and tnf inhibitors
06/2005
06/30/2005WO2005059107A2 Chemokine receptor binding compounds
06/30/2005WO2005059037A1 Reagent for detecting an analyte
06/30/2005WO2005058920A1 Regiospecific synthesis of nicotine derivatives
06/30/2005WO2005058885A2 Piperidine derivatives and their use as glycine transporter inhibitors
06/30/2005WO2005058884A2 Cyclopropane compounds and pharmaceutical use thereof
06/30/2005WO2005058883A1 2, 6 bisheteroaryl-4-aminopyrimidines as adenosine receptor antagonists
06/30/2005WO2005058882A1 Compounds having morpholinyl and piperidinyl groups for use as glyt1 and glyt2 inhibitors
06/30/2005WO2005058877A1 Novel chelating agents and highly luminescent and stable chelates and their use
06/30/2005WO2005058876A1 Pyrazine derivatives as effective compounds against infectious diseases
06/30/2005WO2005058874A1 5- or 6-substituted benzimidazole derivatives as inhibitors of respiratory syncytial virus replication
06/30/2005WO2005058873A1 Piperidine-amino-benzimidazole derivatives as inhibitors of respiratory syncytial virus replication
06/30/2005WO2005058872A1 Crystalline forms of (+)- and (-)-erythro-mefloquine hydrochloride
06/30/2005WO2005058871A1 Morpholinyl containing benzimidazoles as inhibitors of respiratory syncytial virus replication
06/30/2005WO2005058870A1 Amino-benzimidazoles derivatives as inhibitors of respiratory syncytial virus replication
06/30/2005WO2005058869A1 Aminobenzimidazoles and benzimidazoles as inhibitors of respiratory syncytial virus replication
06/30/2005WO2005058868A1 N-(4-carbamimidoyl-benzyl) -2-alkoxy-2-heterocyclyl acetamides as inhibitors of the formation of coagulation factors xa, ixa and thrombin induced by factor viia
06/30/2005WO2005058857A1 Tetronic and tetramic acids as inhibitors of beta-secrease
06/30/2005WO2005058843A1 Substituted 6-cyclohexylalkyl substituted 2-quinolinones and 2-quinoxalinones as poly(adp-ribose) polymerase inhibitors
06/30/2005WO2005058841A2 Hiv protease inhibiting compounds
06/30/2005WO2005058837A1 Benzazepine derivatives as histamine h3 antagonists
06/30/2005WO2005058836A1 Insecticidal spiroindane derivatives
06/30/2005WO2005058834A2 Quinolines useful in treating cardiovascular disease
06/30/2005WO2005058833A1 2-pyridinylethylcarboxamide derivatives and their use as fungicides
06/30/2005WO2005058832A1 Diacylhydrazine derivatives
06/30/2005WO2005058830A1 Novel herbicides
06/30/2005WO2005058824A2 N-aryl piperidine substituted biphenylcarboxamides as inhibitors of apolipoprote in b
06/30/2005WO2005058822A1 Substituted amino-cycloalkanes
06/30/2005WO2005058821A1 Inhibitors of hepatitis c virus ns3/ns4a serine protease
06/30/2005WO2005058817A1 Prolinylarylacetamides
06/30/2005WO2005058311A1 Heterocyclic aspartyl protease inhibitors
06/30/2005WO2005058037A1 Picolinylpyrazoles as herbicides
06/30/2005WO2005058035A1 Use of (3-(1-(3-phenyl-propenyl)-piperidin-4-yl)-2,3-dihydro-indol-1-yl)-(pyridin-4-yl)-methanone derivatives and related compounds as insecticides
06/30/2005WO2005035504A3 5-h -benzo [d] naphth [2, 1-b] azepine derivative as selective d1/d5 receptor antagonists for the treatment of obesity and cns disorders
06/30/2005WO2005032493A8 Amide compounds as ion channel ligands and uses thereof
06/30/2005WO2005032484A3 Alkoxy substituted imidazoquinolines
06/30/2005WO2005020899A3 Substituted cycloalkyamine derivatives as modulators of chemokine receptor activity
06/30/2005WO2004089890A3 Process and intermediates for preparing benzazepines
06/30/2005WO2004055006A8 Novel compounds having selective inhibiting effect at gsk3
06/30/2005WO2004055005A8 Novel compounds having selective inhibiting effect at gsk3
06/30/2005WO2002058698A8 Malonyl-coa decarboxylase inhibitors useful as metabolic modulators
06/30/2005US20050143578 Compounds and methods
06/30/2005US20050143539 Polymerizable composition with free radicals and by controlling polymerization
06/30/2005US20050143456 Carboxamide-substituted phenylurea derivatives, process for their preparation and their use as medicaments
06/30/2005US20050143447 Mixing at least one nonaqueous, pharmaceutically acceptable solvent and a taxane compound
06/30/2005US20050143440 Excellent hypoglycemic agents for treating hyperglycemia, dyslipidemia, hypercholesterolemia, noninsulin-dependent type II diabetes, obesity, glucose intolerance, cardiovascular diabetic complications; reduced side effects due to absence of serotonin reuptake inhibition; imidazoline receptor pathologies
06/30/2005US20050143439 1-Aryl-2-N-, S- or O-substituted benzimidazole derivatives, their use for the production of pharmaceutical agents as well as pharmaceutical preparations that contain these derivatives
06/30/2005US20050143438 N3 alkylated benzimidazole derivatives as MEk inhibitors
06/30/2005US20050143436 N-acylamino with fused nitrogen heterocyclic ring compound; capase enzyme inhibitors; antiinflammatory agents; oral bioavailability; autoimmune diseases, destructive bone disorders, proliferative disorders, infectious diseases, degenerative diseases, and necrotic diseases
06/30/2005US20050143426 Osteoporosis, bone disorders, or diseases associated with excessive secretion of PTH, such as hyperparathyroidism; reduce or inhibit parathyroid hormone (PTH) secretion
06/30/2005US20050143423 Antiulcer; antisecretory; solubility, bioavailability; slow hydrolysis; full inhibition of acid secretion in oral therapy by prolonged presence in body; 1-(carboxythiophenesulfonyl)- 2-(substituted pyridylmethylsulfinyl) benzimidazoles; also with LANSOPRAZOLE, OMEPRAZOLE, PANTOPRAZOLE, or RABEPRAZOLE
06/30/2005US20050143422 N-({4'-[(1-benzofuran-2-ylcarbonyl)amino]-1,1'-biphenyl-4-yl}sulfonyl)glycine; metalloproteinase inhibitors; arthritis, macular degeneration, graft versus host disease, cancer, osteoarthritis
06/30/2005US20050143419 Guanidine and amidine derivatives as factor Xa inhibitors
06/30/2005US20050143418 Pesticidal heterocycles
06/30/2005US20050143407 Process for porducing quinolonecarboxylic acid derivative
06/30/2005US20050143405 Dipeptidyl peptidase inhibitors that lower plasma glucose; treatment and prophylaxis of diabetes, non-insulin dependent diabetes; 2-amino-3aminomethyl-4-phenylpyridines
06/30/2005US20050143403 Substituted pyrimidinones and pyrimidinthiones
06/30/2005US20050143390 piperidines or piperazines 1-linked to a 1-(1-carbonylpiperidin-4-yl)piperidinyl- group through an optionally substituted methyl group; treating Human Immuno-deficiency Virus, solid organ transplant rejection, arthritis, rheumatoid arthritis, and multiple sclerosis
06/30/2005US20050143387 Preserving cosmetic, household or technical products, use in paper treatment liquors, printing thickeners, printing thickeners of starch or cellulose derivatives and paints
06/30/2005US20050143375 Imidazole derivatives
06/30/2005US20050143372 Compounds, pharmaceutical compositions and methods of use therefor
06/30/2005US20050143318 ((1R)-2-indol-3-yl-1-{N-[1-(2-oxo-1-phenyl-2-pyrrolidinylethyl)imidazol-4-yl]carbamoyl)ethyl)-2-[(tert-butoxy)carbonylamino]-2-methylpropanamide; combinded with bone-antiresorptive agent selected from selective estrogen receptor modulators, bisphosphonates, calcitonin, and PTH; carrieres, excipients
06/30/2005US20050143316 Hepatitis C virus inhibitors
06/30/2005US20050142614 Methods for ligand discovery
06/30/2005DE10354584A1 Kationische Diaminopyrazole, ein Verfahren zu deren Herstellung und diese Verbindungen enthaltende Färbemittel Cationic diaminopyrazoles, a process for their preparation and compositions containing these compounds colorant
06/30/2005CA2551944A1 2, 6 bisheteroaryl-4-aminopyrimidines as adenosine receptor antagonists
06/30/2005CA2550074A1 Novel chelating agents and highly luminescent and stable chelates and their use
06/30/2005CA2550012A1 Urea derivative, process for producing the same and use
06/30/2005CA2549825A1 N-(4-carbamimidoyl-benzyl) -2-alkoxy-2-heterocyclyl acetamides as inhibitors of the formation of coagulation factors xa, ixa and thrombin induced by factor viia
06/30/2005CA2549741A1 Reagent for detecting an analyte