Patents
Patents for C07D 401 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom (107,979)
07/2005
07/12/2005US6916957 Antiinflammatory agents; antihistamines; antiallergens
07/12/2005US6916927 Pyrazolopyrimidinones which inhibit type 5 cyclic guanosine 3′,5′-monophosphate phosphodiesterase (cGMP-PDE5) for the treatment of sexual dysfunction
07/12/2005US6916856 Thermosetting resin compositions containing maleimide and/or vinyl compounds
07/12/2005US6916841 Inhibitors of phospholipase enzymes
07/12/2005US6916830 Substituted tetrahydroisoquinolines as C5a receptor modulators
07/12/2005US6916820 Neurotrophic substituted pyrimidines
07/12/2005US6916819 Benzimidazole and pyridylimidazole derivatives
07/12/2005US6916817 Inhibitors of metalloproteinases
07/12/2005US6916814 Methods of treating cytokine mediated diseases
07/12/2005US6916813 (1-phenyl-2-heteoaryl)ethyl-guanidine compounds as inhibitors of mitochondrial F1F0 ATP hydrolase
07/12/2005US6916812 Dietetic agents
07/12/2005US6916810 αν integrin receptor antagonists
07/12/2005US6916809 Heterocyclic acridone inhibitors of IMPDH enzyme
07/12/2005US6916804 Pyrimidine A2b selective antagonist compounds, their synthesis and use
07/12/2005US6916798 Inhibitors of glycogen synthase kinase-3 (GSK-3), a serine/threonine protein kinase; for treatment and prevention of diabetes and Alzheimer's disease
07/12/2005US6916345 6-alkoxy-2,3-diaminopyridine couplers for dyeing keratin fibres
07/12/2005CA2341739C Quinolin-2-one derivatives useful as anticancer agents
07/12/2005CA2105867C Novel imidazole derivatives, their preparation and therapeutic applications
07/07/2005WO2005061519A1 Kinase inhibitors
07/07/2005WO2005061489A1 Heterocyclic derivatives as gpcr receptor agonists
07/07/2005WO2005061487A1 Hiv protease inhibiting compounds
07/07/2005WO2005061486A1 Crystalline form of 2-{4-‘3-(4-chloro-2-fluorophenyl)-4-pyrimidin-4-yl-1h-pyrazol-5-yl!piperidin-1-yl}-2-oxoethanol
07/07/2005WO2005061485A1 Process for making substituted pyrazoles
07/07/2005WO2005061484A1 1,2,3,4-tetrahydroisoquinoline derivatives, preparations thereof and uses thereof
07/07/2005WO2005061483A2 Modulators of peripheral 5-ht receptors
07/07/2005WO2005061477A1 Biaryl sulfonamides as mmp inhibitors
07/07/2005WO2005061467A2 Piperazine derivatives as bradykinin antagonists
07/07/2005WO2005061466A1 Novel phenylalanine derivative
07/07/2005WO2005061463A1 Pyrazole derivatives as protein kinase modulators
07/07/2005WO2005061458A2 Phosphodiesterase 4 inhibitors, including n-substituted diarylamine analogs
07/07/2005WO2005061457A1 Organic compounds
07/07/2005WO2005061455A1 2-(1h-indolylsulfanyl)-benzyl amine derivatives as ssri
07/07/2005WO2005061450A2 Hiv protease inhibiting sulfonamides
07/07/2005WO2005061442A1 Opioid receptor antagonists
07/07/2005WO2005060970A1 Pyrimidines with tie2 (tek) activity
07/07/2005WO2005060969A1 Pyrimidines with tie2 (tek) activity
07/07/2005WO2005060963A1 Benzenesulfonylamino-pyridin-2-yl derivatives and related compounds as inhibitors of 11-beta-hydroxysteroid dehydrogenase type 1 (11-beta-hsd-1) for the treatment of diabetes and obesity
07/07/2005WO2005060959A1 Pyrazole derivatives and use thereof as orexin receptor antagonists
07/07/2005WO2005060947A2 Agonist and antagonist ligands of the nociceptin receptor
07/07/2005WO2005060749A1 Substituted arylpyrazoles as parasiticidal agents
07/07/2005WO2005060665A2 3-cycloalkylaminopyrrolidine derivatives as modulators of chemokine receptors
07/07/2005WO2005060571A2 Antiprotozoal imidazopyridine compounds
07/07/2005WO2005049593A3 N-acylsulfonamide apoptosis promoters
07/07/2005WO2005047258A3 Methods and compositions for selectin inhibition
07/07/2005WO2005042521A3 Piperidinyl-and piperazinyl-sulfonylmethyl hydroxamic acids and their use as protease inhibitors
07/07/2005WO2005042498A3 4-amino (aza) quinoline derivatives as capsaicin receptor agonists
07/07/2005WO2005037779A3 Novel dipeptidyl peptidase iv inhibitors used for functionally influencing different cells and treating immunological, inflammatory, neuronal, and other diseases
07/07/2005WO2005035495A3 Fibrinogen receptor antagonists and their use
07/07/2005WO2004058704A3 Quinazolinones as potassium channel modulators
07/07/2005US20050148777 (2R)-6-chloro-7-isobutyl-2-(trifluoromethyl)-2H-chromene-3-carboxylic acid; cyclooxygenase-2 mediated disorders
07/07/2005US20050148651 Processes for preparing 3-substituted 1-(chloromethyl)-1,2-dihydro-3h-[ring fused indol-5-yl-(amine- derived)] compounds and analogues thereof, and to products obtained therefrom
07/07/2005US20050148649 Substituted arylpyrazoles
07/07/2005US20050148646 Dicationic triaryl analogs as anti-protozoan agents
07/07/2005US20050148638 Increasing contractile force in cardiac muscle fiber by administering a N-[(3-yloxy)-phenyl]-arylamide derivatives; modulating at the cardiac sarcomere (cardiac beta myosin) for congestive heart failure
07/07/2005US20050148637 Neurotrophic low molecular weight ketones and tioester compounds for treatment of nervous system disorders and neurodegenerative conditions
07/07/2005US20050148636 Useful aroyl pyrrole heteroaryl methanones and methanols
07/07/2005US20050148635 3-imino-2-indolones for the treatment of depression and/or anxiety
07/07/2005US20050148634 1-N-Aminobenzimidazole derivatives
07/07/2005US20050148631 Modulation of steroid enzymes in mammals as antidiabetic agents, for treatment of obesity, vision defects, lowering fats in blood, for treatment of osteoporosis, tuberculosis or atherosclerosis in mammals
07/07/2005US20050148623 HIV protease inhibiting compounds
07/07/2005US20050148621 Acetylcholinesterase dual inhibitors
07/07/2005US20050148613 Carbonylamino-derivatives as novel inhibitors of histone deacetylase
07/07/2005US20050148608 Chymase enzyme inhibitors for drugs in vascular systems using sulfonylurea derivatives
07/07/2005US20050148601 Neurokinin-3 receptor modulators: diaryl imidazole derivatives
07/07/2005US20050148581 Quinolines; 1-(6-bromo-2-methoxy-quinolin-3-yl)-4-dimethylamino-2-naphthalen-1-yl-1-phenyl-butan-2-ol; Mycobacterium tuberculosis, M. bovis, M. avium and M. marinum; reduces the total length of treatment and the frequency of drug administration; multi-drug and antibiotic resistance
07/07/2005US20050148580 Non-opioid analgesics for chronic and acute pain; 1-[1-(p-phenylbenzyl)-4-piperidinyl]-2,1,3-benzothiadiazol-2,2-dione; modulation of the opioid and ORL I receptors; agonist or antagonist activity at the CNS mu, delta and kappa receptors greater than morphine
07/07/2005US20050148573 Benzimidazolone compounds having 5-HT4 receptor agonistic activity
07/07/2005US20050148572 2-(2,4-difluorophenyl)-2-[(3R,6R)-3-(2,3-dihydro-1H-inden-2-yl)-6-isobutyl-2,5-dioxopiperazin-1-yl]-N,N-dimethylethanamide; to suppress uterine contractions; cyclization of leucine analogs
07/07/2005US20050148034 Using reduced microvessel outgrowth of pluripotent stem cells as diagnostic indicator angoigenseis inhibition; antitumor agents
07/07/2005US20050147633 Insecticidal amides with nitrogen-containing benzo-Fused bicyclic ring systems
07/07/2005US20050147568 nanostructured acid addition salt of 1-[N2-[3,5-dibromo-N-[[4-(3,4-dihydro-2(1H)-oxoquinazolin-3-yl)-1-piperidinyl]carbonyl]-D-tyrosyl]-L-lysyl]-4-(4-pyridinyl)-piperazine, used for the treatment of headaches
07/07/2005DE10358539A1 Carbonsäureamidderivate Carboxamide
07/07/2005CA2792483A1 Hiv protease inhibiting sulfonamides
07/07/2005CA2550843A1 Novel phenylalanine derivatives
07/07/2005CA2550643A1 1,2,3,4-tetrahydroisoquinoline derivatives, preparations thereof and uses thereof
07/07/2005CA2550283A1 Crystalline form of 2-{4-[3-(4-chloro-2-fluorophenyl)-4-pyrimidin-4-yl-1h-pyrazol-5-yl]piperidin-1-yl}-2-oxoethanol
07/07/2005CA2549955A1 Heterocyclic derivatives as gpcr receptor agonists
07/07/2005CA2549651A1 Benzenesulfonylamino-pyridin-2-yl derivatives and related compounds as inhibitors of 11-beta-hydroxysteroid dehydrogenase type 1 (11-beta-hsd-1) for the treatment of diabetes and obesity
07/07/2005CA2549389A1 Hiv protease inhibiting sulfonamides
07/07/2005CA2549009A1 Opioid receptor antagonists
07/07/2005CA2548824A1 Phosphodiesterase 4 inhibitors, including n-substituted diarylamine analogs
07/07/2005CA2548518A1 Biaryl sulfonamides as mmp inhibitors
07/07/2005CA2548374A1 Pyrazole derivatives as protein kinase modulators
07/07/2005CA2529314A1 Piperazine derivatives and methods of use
07/06/2005EP1550668A1 Pyrazole derivative, medicinal composition containing the same, medicinal use thereof and intermediate in producing the same
07/06/2005EP1550660A1 Isoquinoline derivatives having kinasae inhibitory activity and drugs containing the same
07/06/2005EP1550657A1 Amine compounds and use thereof
07/06/2005EP1549646A2 Piperidine derivatives
07/06/2005EP1549645A1 4,6-diaminosubstituted-2-[oxy or aminoxy]-[1,3,5]triazines as protein tyrosine kinase inhibitors
07/06/2005EP1549643A2 Method for preparing fused oxazinones from ortho-amino aromatic carboxylic acid and a carboxylic acid in the presence of a sulfonyl chloride and pyridine
07/06/2005EP1549638A1 Indole-3-carboxamides as glucokinase (gk) activators
07/06/2005EP1549636A1 Imidazol-1-ylmethyl pyridazine derivatives
07/06/2005EP1549635A1 3,4-disubstituted pyrroles and their for use in treating inflammatory diseases
07/06/2005EP1549634A1 Novel substituted indoles
07/06/2005EP1549622A1 Sulfonylbenzodiazepinone acetamides as bradykinin antagonists
07/06/2005EP1549621A1 Fluorinated phenyl-naphthalenyl-urea compounds as inhibitors of cytokines involved in inflammatory processes
07/06/2005EP1549620A1 Indazolecarboxamide derivatives, preparation and use thereof as cdk1, cdk2 and cdk4 inhibitors
07/06/2005EP1549619A1 6-amino-1h-indazole and 4-aminobenzofuran compounds as phosphodiesterase 4 inhibitors
07/06/2005EP1549614A2 Vasculostatic agents and methods of use thereof
07/06/2005EP1549600A1 Ketones