Patents
Patents for C07D 401 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom (107,979)
08/2008
08/14/2008WO2008096746A1 Spiro compound and use thereof
08/14/2008WO2008096001A1 Hcv inhibiting macrocyclic phenylcarbamates
08/14/2008WO2008095928A1 Process for the preparation of a benzimidazole derivative
08/14/2008WO2008095852A1 Bronchorelaxing arylamides
08/14/2008WO2008095847A1 Bicyclic heterocycles, drugs containing said compounds, use thereof, and method for production thereof
08/14/2008WO2008095823A1 5 -amido- (ih- indol- 2 -yl) piperazin-1-yl-methanone derivatives as histamine h3 receptor ligands
08/14/2008WO2008095821A1 Indol-2-yl-piperazin-1-yl-methanone derivatives
08/14/2008WO2008095292A1 [1,2,3] triazolyl substituted quinolines and coumarins as inhibitors of leukotriene biosynthesis
08/14/2008WO2008079972A3 4-{4- [ ({3-tert-butyl-1- [3- (hydroxymethyl) phenyl] - 1h- pyrazol- 5 -yl } carbamoyl) -amin o] -3-chlorophenoxy} -n-methylpyridine-2-carboxamide as an inhibitor of the vegfr kinase for the treatment of cancer
08/14/2008WO2008076805A3 Arylpropionamide, arylacrylamide, arylpropynamide, or arylmethylurea analogs as factor xia inhibitors
08/14/2008WO2008076805A2 Arylpropionamide, arylacrylamide, arylpropynamide, or arylmethylurea analogs as factor xia inhibitors
08/14/2008WO2008067390A9 Metabolites of 5-fluoro-8-{4-[4-(6-methoxyquinolin-8-yl)piperazin-1-yl]piperidin-1-yl} quinoline and methods of preparation and uses thereof
08/14/2008WO2008038136A3 Substituted heterocyclylcarbonylamino-acetic-acid-derivatives as inhibitors of bacterial heptose synthesis, methods for their preparation and biological applications of said inhibitors
08/14/2008WO2008010984A3 Acridine activation of p53 and uses thereof
08/14/2008WO2008005670A3 One-pot condensation reduction methods for preparing substituted allylic alcohols
08/14/2008US20080194828 Method of Preparing Esomeprazole and Salts Thereof
08/14/2008US20080194826 4-aminopiperidines react with 2-furancarboxylic acid or 2-furoyl chloride; opiod antagonist
08/14/2008US20080194819 Avoids a laborious isolation and purification of intermediates and the final product; industrial scale; starting by reacting 2-methyl-5-nitroaniline with cyanamide and 3-acetylpyridine with N,N-dimethylformamide dimethyl acetal
08/14/2008US20080194643 Using pyrrolidonedicarboxamide compound; therapy for thrombosis, cardiovascular disorders; myocardoim infraction; restenosis; atherosclerosis; anticancer agents; sepsis; antidiabetic agents
08/14/2008US20080194640 Optically Active Tetrahydronaphthalene Derivative
08/14/2008US20080194629 3-Mono-and 3,5-Disubstituted Piperidine Derivatives as Renin Inhibitors
08/14/2008US20080194625 Tetrahydroquinoline derivatives as cannabinoid receptor modulators
08/14/2008US20080194605 Antitumor agents; kinase inhibitors; angiogenesis inhibitors; arteriosclerosis ; antiinflammatory agents
08/14/2008US20080194597 Platelet adp receptor inhibitors
08/14/2008US20080194595 Quinazolinone Derivatives Useful as Vanilloid Antagonists
08/14/2008US20080194588 Modulation of pathogcnicity
08/14/2008US20080194587 phosphodiesterase inhibitor; drug for respiratory system disorders
08/14/2008US20080194586 Controlling non-insulin dependent diabetes; hypoglycemic agents; antilipemic agents; hypercholesterolemia; obesity
08/14/2008US20080194584 Nitrogen Heteroaromatic Compounds Which Bind To The Active Site Of Protein Kinase Enzymes
08/14/2008US20080194583 Tubulin Inhibitors
08/14/2008US20080194581 Pyrrole derivatives, intermediates therefor, preparation and therapeutic use thereof
08/14/2008US20080194578 Quinazoline based egfr inhibitors containing a zinc binding moiety
08/14/2008US20080194574 Pyrazine Derivatives As Effective Compounds Against Infectious Diseases
08/14/2008US20080194565 5-Phenyl-Pentanoic Acid Derivatives as Matrix Metalloproteinase Inhibitors for the Treatment of Asthma and Other Diseases
08/14/2008US20080194562 Pyrazole Derivatives For The Inhibition Of Cdk's And Gsk's
08/14/2008US20080194558 Quinazoline analogs as receptor Tyrosine Kinase inhibitors
08/14/2008US20080194549 Organic Compounds
08/14/2008US20080194520 Sulfonyl Amino Cyclic Derivatives and Use Thereof
08/14/2008US20080193924 Reacting astemizole with potassium channel moderators; complexing; calibration; kits
08/14/2008US20080193700 Metal Chelates and Their Use in Optical Recording Media Having High Storage Capacity
08/14/2008CA2677995A1 Acylguanidine derivative
08/14/2008CA2677481A1 Triazole compounds that modulate hsp90 activity
08/14/2008CA2677336A1 Bicyclic heterocycles, pharmaceutical compositions containing these compounds, the use thereof and processes for the preparation thereof
08/14/2008CA2677263A1 Compounds and compositions as modulators of gpr119 activity
08/14/2008CA2677015A1 Hcv inhibiting macrocyclic phenylcarbamates
08/14/2008CA2676498A1 [1,2,3] triazolyl substituted quinolines and coumarins as inhibitors of leukotriene biosynthesis
08/14/2008CA2676268A1 5 -amido- (ih- indol- 2 -yl) piperazin-1-yl-methanone derivatives as histamine h3 receptor ligands
08/14/2008CA2676265A1 Indol-2-yl-piperazin-1-yl-methanone derivatives
08/14/2008CA2675624A1 Process for the preparation of a benzimidazole derivative
08/14/2008CA2675558A1 Pi 3-kinase inhibitors and methods of their use
08/14/2008CA2675261A1 4-[(4-methyl-1-piperazinyl)methyl]-n-[4-methyl-3-[[4-(3-pyridyl)-2-pyrimidinyl]amino]phenyl]benzamide camsylate and method for preparing thereof
08/13/2008EP1956020A2 1-[2-(heterocyclyl-aminomethyl)-piperidin-1-YL]-1-(2-methyl-5-phenyl-heterocyclyl)-methanone derivatives and related compounds as orexin-1 antagonists for the treatment of obesity
08/13/2008EP1956018A1 Method of preparing a derivative of benzimidazole
08/13/2008EP1956017A1 Substituted 2-(2,6-dioxopiperidin-3-yl)-phthalimides and method of reducing TNF alpha levels
08/13/2008EP1956010A1 Bicyclical heterocycles, medicines containing these compounds, their application and method for their production
08/13/2008EP1956008A1 Organic compound, charge-transporting material, composition for charge-transporting material and organic electroluminescent device
08/13/2008EP1956004A1 Quinoline derivatives and their use as 5-HT6 ligands
08/13/2008EP1955697A1 2-aminobenzamide derivative
08/13/2008EP1954696A2 2-phenoxy-n-(1,3,4-thiadizol-2-yl)pyridin-3-amine derivatives and related compounds as p2y1 receptor inhibitors for the treatment of thromboembolic disorders
08/13/2008EP1954691A2 Amorphous and crystalline forms of pantoprazole magnesium salt
08/13/2008EP1954690A1 Benzamide compounds useful as histone deacetylase inhibitors
08/13/2008EP1954689A1 N-substituted-1h-quinoline-2, 4-diones, preparation method thereof, and pharmaceutical composition containing the same
08/13/2008EP1954683A1 2-(phenyl or heterocyclic)-1h-phenantrho(9,10-d)imidazoles as mpges-1 inhibitors
08/13/2008EP1954682A1 Novel 2-amino-imidazole-4-one compounds and their use in the manufacture of a medicament to be used in the treatment of cognitive impairment, alzheimer s disease, neurodegeneration and dementia
08/13/2008EP1954673A1 Hydroxy-substituted diphenylazetidinones for the treatment of hyperlipidaemia
08/13/2008EP1954277A2 Aminopyrimidines useful as kinase inhibitors
08/13/2008EP1954128A2 Diphenylmethane derivatives as inhibitors of leukotriene biosynthesis
08/13/2008EP1753763B1 Indazole and indolone derivatives and their use as pharmaceuticals
08/13/2008EP1664023B1 Sustituted isoquinoline derivatives and methods of use
08/13/2008EP1541558B1 Heterocyclic compounds having hiv integrase inhibitory activity
08/13/2008EP1501803B1 Tetrahydropyranyl cyclopentyl tetrahydroisoquinoline modulators of chemokine receptor activity
08/13/2008EP1467979B1 Fused heterocyclic compounds and analogs thereof modulators of nuclear hormone receptor function
08/13/2008EP1453501B1 N- aryl-n'-arylcycloalkyl-urea derivatives as mch antagonists for the treatment of obesity
08/13/2008EP1452528B1 Xanthine oxidase inhibitors
08/13/2008EP1427379B1 Use of potent, selective and non toxic c-kit inhibitors for treating interstitial cystitis
08/13/2008EP1322309B1 High affinity small molecule c5a receptor modulators
08/13/2008EP1020445B1 Fused pyridine derivatives
08/13/2008EP0996448B1 Treatment and prevention of adhesions
08/13/2008CN101243075A Novel 2,3-dihydroindole compounds
08/13/2008CN101243074A Heterocyclic compounds
08/13/2008CN101243073A Piperazine-piperidine antagonists and agonists of the 5-HT1A receptor
08/13/2008CN101243072A Piperidine derivatives useful as histamine H3 antagonists
08/13/2008CN101243071A Novel 2,4-dianilinopyrimidine derivatives, the preparation thereof, their use as medicaments, pharmaceutical compositions and, in particular, as ikk inhibitors
08/13/2008CN101243070A Trombin inhibiting 2,4-dioxo-3,4-dihydropyrimidine derivatives
08/13/2008CN101243069A Thrombin inhibiting 2-oxo-1,2,5,6-tetrahydropyridine derivatives
08/13/2008CN101243068A Compounds for the treatment of multi-drug resistant bacterial infections
08/13/2008CN101243067A Novel anthranilamides for controlling invertebrate pests
08/13/2008CN101243066A Delta and epsilon crystal forms of imatinib mesylate
08/13/2008CN101243065A Intermediates useful in the synthesis of alkylquinoline and alkylquinazoline kinase modulators and related methods of synthesis
08/13/2008CN101243055A Dihydropyrimidone multimers and their use as human neutrophil elastase inhibitors
08/13/2008CN101242844A Aminopyrimidines as kinase modulators
08/13/2008CN101242843A Aminopyrimidines as kinase modulators
08/13/2008CN101242834A Inhibitors of AKT activity
08/13/2008CN101239973A Substituted aminoquinazolinone (thione) derivative or salts thereof, intermediate compound therefor, pest-controlling agent and using method thereof
08/13/2008CN101239972A Heterocyclic n-aryl carboxamides as cytokine inhibitors
08/13/2008CN101239971A Biphenyl derivatives
08/13/2008CN101239970A Biphenyl derivatives
08/13/2008CN101239969A Biphenyl derivatives
08/13/2008CN101239968A Biphenyl derivatives
08/13/2008CN101239953A Antidepressant arylpiperazine derivatives of heterocycle-fused benzodioxans