Patents
Patents for C07D 277 - Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings (33,621)
07/2003
07/31/2003WO2003002596A3 Use of dipeptidyl peptidase iv inhibitors as therapeutics for neurological disorders
07/31/2003WO2002051410A3 Phenylthiazole and thiazoline derivatives and their use as antiparasitics
07/31/2003WO2002020500A3 Materials and methods to potentiate cancer treatment
07/31/2003US20030144542 Use of propargyl glycine amino propargyl diol compounds for treatment of renal failure
07/31/2003US20030144526 Calcium receptor-active compounds
07/31/2003US20030144523 Epothilone derivatives, method for producing same and their pharmaceutical use
07/31/2003US20030144521 Hydrogenation of a corresponding nonracemic 1-(4-benzoxy phenyl)-2-(4-hydroxy-4- phenyl-piperidin-1-yl)-1-propanone using a catalyst system comprising ruthenium, a nonracemic diphosphine ligand, a bidentate amine ligand selected from
07/31/2003US20030144331 p53 inhibitors and therapeutic use of the same
07/31/2003US20030144329 N-substituted heterocycles for the treatment of hypercholesteremia, dyslipidemia and other metabolic disorders; cancer, and other diseases
07/31/2003US20030144323 Phenylalkynes
07/31/2003US20030144288 Sulfur compounds such as 4-fluoro-N-(4-methoxy-7-(tetrahydro-pyran-4-yl)-benzothiazol-2-yl) -benzamide, used as preferential adenosine receptor ligands for the prophylaxis of neurodegenerative disorders
07/31/2003US20030143633 Factors participating in degranulation of mast cells, dnas encoding the same, method of screening of these factors and the inhibitors
07/31/2003CA2474322A1 4(hetero-) aryl substituted (thia-/oxa-/pyra) zoles for inhibition of tie-2
07/31/2003CA2471989A1 2-aminothiazole allosteric enhancers of a1 adenosine receptors
07/31/2003CA2471389A1 Process for the preparation of nonracemic syn-1-(4-hydroxy-phenyl)-2-(4-hydroxy-4-phenyl-piperidin-1yl)-1-propanol compounds
07/30/2003EP1331224A1 Thiazole or oxazole derivatives
07/30/2003EP1331221A1 5-amidino-2-hydroxybenzenesulfonamide derivatives, pharmaceutical compositions containing the same and intermediates for their preparation
07/30/2003EP1330446A1 Process for the manufacture of thiazole derivatives with pesticidal activity
07/30/2003EP1052989B1 Use of 2-amino-6- trifluoromehthoxy- benzothiazole for preventing or treating cerebellum dysfunction
07/30/2003EP0991428B1 Delta1,2 bicyclo 4,4,0] functional dyes for contrast enhancement in optical imaging
07/30/2003EP0958296B1 Heterocyclic compounds process for their preparation and pharmaceutical compositions containing them and their use in the treatment of diabetes and related diseases
07/30/2003CN1433415A N-[5-[[[5-alkyl-2-oxazlyl]methyl]thio]-2-thiazolyl] carboxamide inhibitors of cyclin dependent kinases
07/30/2003CN1433414A Benzazole derivatives and their use as JNK modulators
07/30/2003CN1433408A Aminothiazole inhibitors of cyslin dependent kinases
07/30/2003CN1433297A Topical compositions comprising protected functional thiols
07/30/2003CN1116288C Urea derivatives as inhibitors of inosine-5'-phospho-dehydrogenase
07/29/2003US6600058 Vitamin D derivatives with carbo- or heterocyclic substituents at C-25, a process for their production, intermediate products and their use for producing medicaments
07/29/2003US6600035 6-(substituted methylene) penems and intermediates
07/29/2003US6599943 Preventive treatment, related to the radical generating nature of the xanthine dehydrogenase/xanthine oxidase
07/29/2003US6599932 Highly selective in killing tumor cells but not normal cells
07/29/2003US6599923 Insulin sensitivity enhancer in combination with other antidiabetics differing from the enhancer in the mechanism of action
07/29/2003US6599910 Substituted triazole compounds
07/29/2003US6599904 Sulphonamide derivatives, process for their preparation, and their use as medicaments
07/29/2003US6599903 Derivatives of 2-(iminomethyl)amino-phenyl, their preparation, their use as medicaments and the pharmaceutical compositions containing them
07/24/2003WO2003060078A2 Heterocyclic modulators of nuclear receptors
07/24/2003WO2003059900A1 Coumarin derivatives, process for their production and use thereof
07/24/2003WO2003059896A1 Method for producing halogenated 2-(3-butenylsulfanyl)-1,3-thiazoles
07/24/2003WO2003059895A1 Halogenobenzyl aminopropionic acid derivatives
07/24/2003WO2003059886A1 Acyl sulfonamide derivative
07/24/2003WO2003059873A1 Potassium channel modulators
07/24/2003WO2003059871A1 N-alkylsulfonyl-substituted amide derivatives
07/24/2003WO2003059864A2 Pheny(alkyl)carboxylic acid derivatives and dionic phenylalkylheterocyclic derivatives and their use as medicines with serum glucose and/or serum lipid lowering activity
07/24/2003WO2003059265A2 Compositions and methods for treating heart failure
07/24/2003WO2003059064A1 Insecticides containing hydrazone derivatives as the active ingredient and novel hydrazone derivatives
07/24/2003US20030139473 Novel compounds, their preparation and use
07/24/2003US20030139453 Difluorobutyric acid metalloprotease inhibitors
07/24/2003US20030139449 Anxiolytic agents; psychological disorders; cognition activators
07/24/2003US20030139405 6-Membered heterocyclic compounds useful for selective inhibition of the coagulation cascade
07/24/2003US20030139404 N-monoacylated derivatives of o-phenylenediamines, their analogs and their use as pharmaceutical agents
07/24/2003US20030139390 Compounds for the modulation of PPARgamma activity
07/24/2003US20030139379 Autoimmune disease, osteoporosis, rheumatic diseases, skin disorders
07/24/2003CA2473207A1 Halogenobenzylaminopropionic acid derivatives
07/24/2003CA2472419A1 Coumarin derivatives, process for their production and use thereof
07/24/2003CA2472209A1 Pheny(alkyl)carboxylic acid derivatives and dionic phenylalkylheterocyclic derivatives and their use as medicines with serum glucose and/or serum lipid lowering activity
07/23/2003EP1328271A2 Method for the treatment of neurological and neuropsychological disorders
07/23/2003EP1328270A2 Method for the treatment of neurological and neuropsychological disorders
07/23/2003EP1328265A2 Novel uses for thyroid hormones or thyroid hormone-like agonist compounds for treating dermis conditions
07/23/2003EP0929528B1 Aralkyl and aralkylidene heterocyclic lactams and imides
07/23/2003EP0808163B1 Use of thiazolium compounds for preventing and reversing the formation of advanced glycosylation endproducts
07/23/2003EP0695183B1 Use of thiazolidinediones for the treatment of atherosclerosis and eating disorders
07/23/2003CN1432004A Alkynyl phenyl heteroaromatic glucokinase activators
07/23/2003CN1431941A 挤压模 Extrusion die
07/22/2003US6596875 Method for synthesizing epothilones and epothilone analogs
07/22/2003US6596863 Matrix metalloproteinase inhibitor is useful as an anticancer agent, angiogenesis inhibitor, a tumor cell infiltration inhibitor or a tumor metastasis inhibitor; inflammatory diseases, osteoarthritis, rheumatoid arthritis
07/22/2003US6596754 Preventives/remedies for multiple organ failure
07/22/2003US6596746 Cyclic protein tyrosine kinase inhibitors
07/22/2003US6596744 Method for treating fibrotic diseases or other indications IIC
07/22/2003US6596741 Compounds of formula I exhibit activity as serotonin, norepinephrine, and dopamine reuptake inhibitors and can be used in the treatment of central nervous system and other disorders.
07/22/2003US6596718 7-Morpholin-4yl-benzothiazole amide derivatives
07/22/2003US6596716 2-propane-sulphonamide derivatives
07/22/2003US6596693 Dipeptide apoptosis inhibitors and the thereof
07/17/2003WO2003057681A1 Process for producing 2-cyanoimino-1,3-thiazolidine
07/17/2003WO2003057680A1 Process for producing 2-cyanoimino-1,3-thiazolidine
07/17/2003WO2003057666A2 Inhibitors of dipeptidyl peptidase iv
07/17/2003WO2003057200A2 Compositions comprising inhibitors of dpp-iv and nep enzymes for the treatment of diabetes
07/17/2003WO2003057169A2 4-dedimethylamino tetracycline compounds
07/17/2003WO2003057144A2 Change inhibitors of dipeptidyl peptidase iv
07/17/2003WO2003056922A1 Substituted thiazolyl sulfonyl urea compounds
07/17/2003US20030135066 Renin inhibitors for the treatment of hypertension and glaucoma.
07/17/2003US20030134885 Biaromatic ligand activators of PPARgamma receptors
07/17/2003US20030134883 Use in the treatment of cancer and other diseases characterized by undesired cellular hyperproliferation.
07/17/2003US20030134874 Multicyclic compounds which inhibit leukocyte adhesion mediated by VLA-4
07/17/2003US20030134859 Substituted 2-chloro-5-nitrobenzamides; treating retrograde osteoporosis and diabetes mellitus
07/17/2003US20030134857 Synergistic insecticide mixtures
07/17/2003US20030134855 P-acylaminomethyl-N-(4-methoxy-7-morpholin-4-yl-benzothiazol-2 -yl)-benzamides; treatment of diseases related to the adenosine receptor, such as Alzheimer's disease, depression, drug addiction, Parkinson's and ADHD
07/17/2003US20030134848 Substituted 1-aza-2-imino-heterocycles and their use as nicotinic acetylcholin receptors activators
07/17/2003US20030134802 Novel effectors of dipepetidyl peptidase IV
07/17/2003US20030134237 Methine dyes, manufacturing methods thereof, and silver halide photoraphic materials contaning same dyes
07/17/2003CA2471204A1 Inhibitors of dipeptidyl peptidase iv
07/16/2003EP1327887A2 Use of thiazolium compounds for preventing and reversing the formation of advanced glycosylation end products
07/16/2003EP1326861A1 Alpha-aryl ethanolamines and their use as beta-3 adrenergic receptor agonists
07/16/2003EP1326852A1 Aromatic and heterocyclic thiazolyl thiourea compounds and use
07/16/2003EP1326850A1 A process for the preparation of bis-benzazolyl compounds
07/16/2003EP1326835A1 Benzamide compounds as apo b secretion inhibitors
07/16/2003EP1326828A1 Beta-amino acid derivatives as integrin receptor antagonists
07/16/2003EP1326824A1 Pharmaceutical compounds
07/16/2003CN1430615A Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1
07/16/2003CN1430614A Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1
07/16/2003CN1430613A Method for producing 2-chloro-5-chloromethyl-1,3-thiazole
07/16/2003CN1430612A Hete rocyclic derivatives