Patents for C07D 261 - Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings (11,459) |
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12/06/2005 | US6972295 Central nervous system disorders; psychological disorders; antiinflammatory agents; multiple sclerosis |
12/06/2005 | US6972290 Piperazine derivatives and their use as anti-inflammatory agents |
12/01/2005 | WO2005113519A1 Compounds and compositions as ppar modulators |
12/01/2005 | WO2005112945A2 Synthesis of tetracyclines and analogues thereof |
12/01/2005 | WO2005060456A3 Method for treating adamts-5-associate disease |
12/01/2005 | US20050267206 Thyroid receptor antagonists for the treatment of cardiac and metabolic disorders |
12/01/2005 | US20050267190 Solid-state form of celecoxib having enhanced bioavailability |
12/01/2005 | US20050267182 Urea derivatives as FLT-3 modulators |
12/01/2005 | US20050267175 Anticancer agents for, lungs, leukemia and ovarian cancer or prostate glands |
12/01/2005 | CA2767912A1 Synthesis of tetracyclines and analogues thereof |
12/01/2005 | CA2564429A1 Compounds and compositions as ppar modulators |
11/30/2005 | EP1600442A1 Heteroarylcarbamoylbenzene derivative |
11/30/2005 | EP1124827B1 3-(substituted phenyl)-5-(substituted heterocyclyl)-1,2,4-triazole compounds |
11/30/2005 | EP1091943B1 Non-peptidyl inhibitors of vla-4 dependent cell binding useful in treating inflammatory, autoimmune, and respiratory diseases |
11/30/2005 | CN1703395A Aryl and heteroaryl compounds and methods to modulate coagulation |
11/29/2005 | US6969713 Piperidine and piperazine acetamide derivatives |
11/29/2005 | US6969710 Compounds |
11/24/2005 | WO2005110971A1 Heteroaryl substituted cyclohexyl-1,4-diamine derivatives |
11/24/2005 | WO2005092011A3 Mitotic kinesin inhibitors |
11/24/2005 | US20050261503 Heteroaromatic glucokinase activators |
11/24/2005 | US20050261315 tyrosine kinase inhibitors such as N-(3-tert-butylisoxazol-5-yl)-2-(4-(benzyloxy)phenyl)acetamide, used for treating and preventing conditions and diseases, such as cancer, hematologic malignancies, cardiovascular disease, inflammation or multiple sclerosis |
11/24/2005 | US20050261291 1-Cyclopropylmethyl-4-[2-(3,3,5,5-tetramethylcyclohexyl)phenyl]piperazine or a salt or hydrate; exhibit excellent cell adhesion inhibitory action or cell infiltration inhibitory action; for treating inflammatory diseases and autoimmune diseases such as inflammatory bowel diseases and rheumatoid arthritis |
11/24/2005 | US20050261276 Novel sulphones for inhibition of gamma secretase |
11/24/2005 | US20050261273 Substituted urea and carbamate, phenacyl-2-hydroxy-3-diaminoalkane, and benzamide-2-hydroxy-3-diaminoalkane aspartyl-protease inhibitors |
11/24/2005 | CA2566212A1 Heteroaryl-substituted cyclohexyl-1,4-diamine derivatives |
11/23/2005 | EP1597243A1 Heterocyclic compounds useful as nurr-1 activators |
11/23/2005 | EP1372645B1 Reconstitutable parenteral composition containing a cox-2 inhibitor |
11/23/2005 | CN1228332C Chemical synthesis method of 3-(2-chlorophenyl)-5-methyl-4-isoxazole formyl chloride |
11/23/2005 | CN1228327C Carboxylic acid derivatives and drugs containing the same |
11/17/2005 | WO2005108347A2 Substituted enaminones, their derivatives and uses thereof |
11/17/2005 | WO2005107762A2 Certain chemical entities, compositions, and methods |
11/17/2005 | CA2565695A1 Certain chemical entities and compositions for use in the treatment of a cellular proliferative disease or disorder |
11/16/2005 | EP1594846A1 Bis(hetero)aryl carboxamide derivatives for use as pgi2 antagonists |
11/16/2005 | EP1594508A2 Novel bicyclic compounds and compositions |
11/16/2005 | EP1594505A2 Phenylglycine derivatives useful as serine protease inhibitors |
11/16/2005 | CN1227244C Herbicidal benzoyl derivatives |
11/16/2005 | CN1227012C Pharmaceutical compositions for topical delivery of cyclooxygenase-2 enzyme inhibitors |
11/15/2005 | US6965036 Intermediates for guanidine mimics as factor Xa inhibitors |
11/15/2005 | US6964983 Compounds that modulate PPAR activity and methods for their preparation |
11/15/2005 | US6964978 Dissolving with crystal growth inihibitos; drying |
11/15/2005 | US6964975 Isoxazole and thiazole compounds and use thereof as medicine |
11/10/2005 | WO2005105770A2 Arylphenylamino-, arylphenylamide-, and arylphenylether-sulfide derivatives |
11/10/2005 | WO2005105764A1 Butanoic acid derivatives, processes for the preparation thereof, pharmaceutical compositions comprising them, and therapeutic applications threreof |
11/10/2005 | WO2005105744A1 Histamine-3 receptor antagonists |
11/10/2005 | WO2005105733A1 Ortho substituted aryl or heteroaryl amide compounds |
11/10/2005 | WO2005082871A3 Guanidine compounds, and use thereof as binding partners for 5-ht5 receptors |
11/10/2005 | US20050250826 Compounds, compositions, processes of making, and methods of use related to inhibiting macrophage migration inhibitory factor |
11/10/2005 | US20050250822 Substituted benzanilide compound and noxious organism controlling agent |
11/10/2005 | US20050250818 Ortho substituted aryl or heteroaryl amide compounds |
11/10/2005 | US20050250816 Positive allosteric modulators of the nicotinic acetylcholine receptor |
11/10/2005 | CA2565184A1 Butanoic acid derivatives, processes for the preparation thereof, pharmaceutical compositions comprising them, and therapeutic applications threreof |
11/10/2005 | CA2564258A1 Histamine-3 receptor antagonists |
11/10/2005 | CA2562176A1 Arylphenylamino-, arylphenylamide-, and arylphenylether-sulfide derivatives |
11/09/2005 | EP1593677A2 Benzylidene-thiazolidinediones and analogues and their use in the treatment of diabetes |
11/09/2005 | EP1593671A1 DPP-IV inhibitors |
11/09/2005 | EP1501787B1 N-biphenylmethyl aminocycloalkanecarboxamide derivatives with a substiituent on the methyl useful as bradykinin antagonists |
11/09/2005 | EP1216223B1 Novel dicarboxylic acid derivatives with pharmaceutical properties |
11/09/2005 | EP1095016B1 Sulfur substituted sulfonylaminocarboxylic acid n-arylamides, their preparation, their use and pharmaceutical preparations comprising them |
11/09/2005 | EP0979226B1 Isoxazole derivatives |
11/08/2005 | US6962935 Anticoagulants; thrombosis therapy; cardiovascular disorders |
11/08/2005 | CA2155104C Heterocyclic-substituted alkyl amide acat inhibitors |
11/03/2005 | WO2005102980A1 Novel compounds, the preparation and the use thereof for a regiospesific synthesis of perfluor(alkyl) group heterocycles |
11/03/2005 | WO2004099165A3 Heterocyclic compounds and hydro isomers thereof |
11/03/2005 | US20050245747 e.g. 2-[2-(5-chloro-benzo[b]thiophen-2-yl)-phenylmethanesulfinyl]-acetamide; autoimmune disorders, antidepressant; narcolepsy, Parkinson's, Alzheimer's disease; attention deficit hyperactivity disorder; sleep disorder, fatigue |
11/03/2005 | US20050245592 2-Iminopyrrolidine derivatives |
11/03/2005 | US20050245543 Histamine-3 receptor antagonists |
11/02/2005 | EP1590321A2 Aryl alkyl carbamate derivatives production and use thereof in therapy |
11/02/2005 | EP1085016B1 Heterocycle-bearing thio phenol compounds, intermediates for the preparation of the same and processes for the preparation of both |
11/02/2005 | CN1691944A Oxadiazoles as modulators of metabotropic glutamate receptor-5 |
11/02/2005 | CN1690050A Aryl-substituted iso-oxazoline compounds used as bactericide |
11/01/2005 | US6960688 Use of compounds for the elevation of pyruvate dehydrogenase activity |
11/01/2005 | US6960614 Oxygenated esters of 4-lodo phenylamino benzhydroxamic acids |
11/01/2005 | US6960607 Naphthyl benzoxazoles and benzisoxazoles as estrogenic agents |
11/01/2005 | CA2177586C 4-benzoylisoxazoles and their use as herbicides |
10/27/2005 | WO2005100308A1 Thio-substituted biaryl-methanesulfinyl derivatives |
10/27/2005 | WO2005100298A1 Cetp inhibitors |
10/27/2005 | WO2005034848A3 Inhibitors of cathepsin s |
10/27/2005 | WO2005021515B1 Inhibitors of phosphodiesterase type-iv |
10/27/2005 | WO2004089366A8 Bicyclic compounds as nr2b receptor antagonists |
10/27/2005 | US20050240023 Cathepsin cysteine protease inhibitors |
10/27/2005 | US20050239899 Beta-secretase inhibitors |
10/27/2005 | US20050239769 Therapeutic compounds for treating dyslipidemic conditions |
10/27/2005 | US20050239751 e.g. tert-Butyl 6-(2-(3-(2,6-Dichlorophenyl)isoxazol-5-yl)pyridin-4-ylamino)-2-methyl-4-oxohexan-3-ylcarbamate; Hepatitis C virus (HCV) infections |
10/27/2005 | CA2562082A1 Cetp inhibitors for the treatment and prevention of atherosclerosis |
10/26/2005 | EP1589007A2 5-membered heterocycle derivatives, production thereof and their use as medicaments |
10/26/2005 | CN1688545A Phosphodiesterase 4 inhibitors, including n-substituted phenylamine and diphenylamine analogs |
10/26/2005 | CN1688527A Fused benzene derivative and use |
10/26/2005 | CN1688315A Use of selective COX-2 inhibitors for the treatment of urinary incontinence |
10/25/2005 | US6958356 Guanidine mimics factor Xa inhibitors |
10/25/2005 | US6958355 Materials and methods for the treatment of diabetes, hyperlipidemia, hypercholesterolemia, and atherosclerosis |
10/25/2005 | US6958331 sulfonyl amine derivatives such as {2-(2,2-diphenyl-ethylamino)-5-[4-(4-isopropyl-piperazine-1-carbonyl)-piperidine-1-sulfonyl]-phenyl}-morpholin-4-yl-methanone; pain, inflammation, septic shock |
10/20/2005 | WO2005097765A1 Anaplastic lymphoma kinase modulators and methods of use |
10/20/2005 | WO2005097760A1 Heterocyclic anti-viral compounds comprising metabolizable moieties and their uses |
10/20/2005 | WO2005097751A2 Non-imidazole heterocyclic compounds as histamine h3-receptor ligands |
10/20/2005 | WO2005066143A3 Benzo[d]isoxazol-3-ol daao inhibitors |
10/20/2005 | WO2005058845A3 Novel glucagon antagonists/inverse agonists |
10/20/2005 | WO2005055715A3 Insecticidal n-(heteroarylalkyl) alkanediamine derivatives |
10/20/2005 | WO2005051931A3 Phosphodiesterase inhibitors |
10/20/2005 | US20050234111 D-homo-17-chlor-16(17)-ene steroids |
10/20/2005 | US20050234106 1-aryl-1-heteroarylaminoalkylene-substituted, e.g., 1-[fluorophenylcyclohexylmethyl]isoquinolin-1-ylamine; antiarrhythmia agents; cardiovascular disorders |