Patents for C07D 261 - Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings (11,459) |
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06/26/2008 | US20080152950 Anthracene derivative and organic electroluminescent device using the same |
06/26/2008 | DE102006060598A1 New tetrahydrobenzoisoxazole compounds are mitotic motor protein Eg5 modulators useful to treat and prevent cancer, and to treat e.g. monocyte leukemia, glioblastoma, colon carcinoma, myelotic leukemia and lymphatic leukemia |
06/25/2008 | EP1935892A1 Glycyrrhetinic acid-30-amide derivatives and the uses thereof |
06/25/2008 | EP1935888A1 Method for sulfonating 1,2-benzisoxazole-3-acetic acid |
06/25/2008 | EP1935887A1 Heterocyclic substituted carbonyl derivatives and their use as dopamine D3 receptor ligands |
06/25/2008 | EP1935886A1 Heterocyclyl-substituted-ethylamino-phenyl derivatives, their preparation and use as medicaments |
06/25/2008 | CN101208314A Benzisoxazole piperazine compounds and methods of use thereof |
06/25/2008 | CN101208082A Niacin receptor agonists, compositions containing such compounds and methods of treatment |
06/24/2008 | US7390908 Such as 2-[3,5-Di(2-chlorobenzyloxy)benzoyl)amino]-thiazole; for treatment of diabetes |
06/24/2008 | US7390833 osteoarthritis; compounds inhibit Aggrecanase Activity of a disintegrin and metalloprotease with thrombosondin type I motifs; biaryl sulfonamid derivatives; N-({4'-[2-4-methylisoquinolin-3-yl)ethyl]-1,1 '-biphenyl-4-yl}sulfonyl)-D-valine |
06/19/2008 | US20080146627 Thiazole, oxazole, imidazole, isoxazole and isoxazoline derivatives, e.g., butyl 2-(4-[1,1'-biphenyl]-4-yl-1H-imidazol-2-yl)ethylcarbamate inhibit lipidic peroxidation and monoamine oxidase and modulate sodium channels and are used for treating neurodegenerative disorders or pain. |
06/19/2008 | US20080146624 Amidines as modulators of indoleamine 2,3-dioxygenase |
06/19/2008 | US20080146620 Dibenzylamine Compounds and Pharmaceutical Use Thereof |
06/19/2008 | US20080145356 Administering glutenase to Celiac or dermatitis herpetiformis patient reduces levels of toxic gluten oligopeptides |
06/18/2008 | EP1932836A1 Isoxazoline-substituted benzamide compound and harmful organism-controlling agent |
06/18/2008 | EP1931205A2 Transglutaminase inhibitors and methods of use thereof |
06/18/2008 | CN101203498A Heterocyclic anti-viral compounds comprising metabolizable moieties and their uses |
06/18/2008 | CN101200456A Bromine difluoro methyl substituted isoxazole derivatives |
06/12/2008 | WO2007118323A8 Isoxazole derivatives as calcium channel blockers |
06/12/2008 | WO2007110237A3 Amide derivatives and their application for the treatment of g protein related diseases |
06/12/2008 | US20080139599 e.g. 4-[6-(5-methyl-2-phenyloxazol-4-ylmethoxy)-1-oxoindan-5-yl]benzoic acid; antidiabetic and antilipemic agent, obesity; atherosclerosis; coupling benzene derivatives folowed by hydration and alkylation |
06/12/2008 | US20080139547 N-Hydroxyalkynylbenzamide (or hydroxamate) derivatives; anticarcinogenic and antiproliferative agents |
06/12/2008 | US20080139390 Isoxazoline Derivatives and Their Use as Herbicides |
06/10/2008 | US7385063 Method for preparing imidazole derivatives |
06/10/2008 | US7384929 N-aryl azaspiroalkene and azaspiroalkane compounds and methods of preparation and use thereof |
06/10/2008 | CA2393995C Novel benzene sulfonamide derivatives, their preparation and pharmaceutical compositions containing them |
06/05/2008 | WO2008066131A1 Novel phenyl-isoxazol-3-ol derivative |
06/05/2008 | US20080132706 Compounds as PDE IV and TNF Inhibitors |
06/05/2008 | US20080132480 Biphenyloxyacetic Acid Derivatives for the Treatment of Respiratory Disease |
06/05/2008 | CA2668713A1 Novel phenyl-isoxazol-3-ol derivative |
06/04/2008 | EP1343775B1 Piperazine derivatives |
06/04/2008 | EP1204643B1 Fungicidal heterocyclic aromatic amides and their compositions, methods of use and preparation |
06/04/2008 | EP1193250B1 Phenyl sulfamate derivatives |
06/03/2008 | US7381687 3-heteroaryl substituted 5-methyloxymethyl isoxazolines used as herbicides |
05/29/2008 | WO2008062044A1 2-hydroxy-1,3-diaminopropane derivatives |
05/29/2008 | US20080125470 N-(3-chloro-4-fluorophenyl)-N'-hydroxy-5-(2-(methylamino)-1,3-thiazol-4-yl)isoxazole-3-carboximidamide; cancer, viral infections, depression, a neurodegenerative disorder, trauma, age-related cataracts, organ transplant rejection, or an autoimmune disease |
05/29/2008 | CA2669839A1 2-hydroxy-1,3-diaminopropane derivatives |
05/28/2008 | EP1924569A2 Preparation of tetrahydro-1,8-dioxa-4a-aza-naphthalenes and their use in coating applications |
05/28/2008 | EP1924554A1 Sulphonamide derivatives |
05/27/2008 | US7378448 Diphenylether amide derivatives as opioid receptor antagonists |
05/27/2008 | US7378409 Substituted cycloalkylamine derivatives as modulators of chemokine receptor activity |
05/22/2008 | WO2008060569A1 Compounds and methods for inhibiting the interaction of bcl proteins with binding partners |
05/22/2008 | WO2008059023A1 New haloalkylsulfone substituted compounds useful for treating obesity and diabetes |
05/22/2008 | WO2008020007A3 Process for the preparation of 5-hydroxyisoxazolidines, 5-isoxazolidinones, b-amino acids, b-amino aldehydes and derivatives thereof |
05/22/2008 | CA2669860A1 New haloalkylsulfone substituted compounds useful for treating obesity and diabetes |
05/22/2008 | CA2669596A1 Compounds and methods for inhibiting the interaction of bcl proteins with binding partners |
05/21/2008 | EP1922311A2 Acyclic ikur inhibitors |
05/21/2008 | EP1482924B1 Cathepsin cysteine protease inhibitors |
05/21/2008 | EP1395551B1 Hydroxy alkyl amine derivatives as beta-secretase inhibitors and their use for the treatment of alzheimer's disease and similar diseases |
05/21/2008 | EP1362027B1 Acylated 6,7,8,9-tetrahydro-5h-benzocycloheptenyl amines and their use as pharmaceutical |
05/21/2008 | CN101184739A Polycyclic oxadiazoles or isoxazoles and their use as S1P receptor ligands |
05/21/2008 | CN100389110C Process of preparing aromatic ring substituted ixooxazoline compound |
05/20/2008 | US7375233 Process for the preparation of zonisamide and the intermediates thereof |
05/20/2008 | US7375134 N1-(1-cyanocyclopropyl)-4-fluoro-N2-{(1S)-2,2,2-trifluoro-1-[4'-(methylsulfonyl)-1,1'-biphenyl-4-yl]ethyl}-L-leucinamide; osteoporosis and other bone loss disorders |
05/15/2008 | WO2008057775A2 Heterocyclic amide compounds useful as kinase inhibitors |
05/15/2008 | WO2008057280A1 Multi-cyclic compounds and methods of use |
05/15/2008 | US20080114167 Compounds and Methods for Inhibiting the Interaction of BCL Proteins with Binding Partners |
05/15/2008 | US20080114044 Isoxazole compounds as Peroxisome Proliferator-Activated Receptor (PPAR) delta modulators; (5-{4-[2-(2,4-Dichloro-phenoxy)-ethyl-carbamoyl]-5-phenyl-isoxazol-3-yl}-phenyl)-acetic acid; diabetes, cardiovascular disorders, dyslipidemias, irritable bowel disease, cancer, skin disorders, eye disorders |
05/15/2008 | US20080113997 Compounds, compositions, processes of making, and methods of use related to inhibiting macrophage migration inhibitory factor |
05/15/2008 | CA2672956A1 Calcium receptor modulating agents |
05/14/2008 | EP1919882A2 Isoxazole combretastatin derivatives for the treatment of proliferative disorders |
05/14/2008 | EP1485365B1 Sulfonyl-derivatives as novel inhibitors of histone deacetylase |
05/13/2008 | US7371871 imidazole derivatives; Alzheimer's Disease, Down syndrome and Huntington's Disease; hypotensive agents, sleeping and eating disorders, anxiolytic agents, antidepressants, antiepileptic agents, drug abuse withdrawl |
05/13/2008 | US7371755 Antiviral agents |
05/13/2008 | CA2235298C Isoxazole derivatives |
05/08/2008 | WO2008053326A1 A salt of 3-benzyl-2-methyl-2,3,3a,4,5,6,7,7a-octahydrobenzo[d]isoxazol-4-one |
05/08/2008 | WO2008053325A1 A salt of 3-benzyl-2-methyl-2,3,3a,4,5,6,7,7a-octahydrobenzo[d]isoxazol-4-one |
05/08/2008 | US20080108679 Isoxazolic Derivative to Relieve Neuropathic Pain |
05/08/2008 | US20080108668 compounds with biological activity against all sorts of plant diseases and insects at very low dosage, to control plant diseases like cucumber downy mildew, cucumber grey mold, cucumber powdery mildew, tomato early blight, tomato late blight, phytophthora blight of pepper, grape downy mildew and etc |
05/08/2008 | US20080108601 anticancer agents; catalytic hydrogenation |
05/08/2008 | US20080108595 Inhibitors of cathepsin s |
05/08/2008 | CA2667515A1 A salt of 3-benzyl-2-methyl-2,3,3a,4,5,6,7,7a-octahydrobenzo[d]isoxazol-4-one |
05/08/2008 | CA2667513A1 A salt of 3-benzyl-2-methyl-2,3,3a,4,5,6,7,7a-octahydrobenzo[d]isoxazol-4-one |
05/07/2008 | EP1916896A2 Non-steroidal antiandrogens |
05/07/2008 | EP1436272B1 Biphenylcarboxylic amide derivatives as p38 kinase inhibitors |
05/07/2008 | CN101172983A Substituted phenylacetic acids |
05/06/2008 | US7368578 superior in an adipose tissue weight decreasing action and a retinoid-related receptor function regulating action; to treat obesity, diabetes mellitus, hyperlipidemia, impaired glucose tolerance, hypertension; fewer side effects; 4-{[2-(2-furyl)-1,3-oxazol-4-yl]methoxy}-3-methoxybenzaldehyde |
05/06/2008 | US7368572 Anticancer agents |
05/06/2008 | US7368473 Paclitaxel enhancer compounds |
05/06/2008 | US7368224 Photopolymerizable composition |
05/06/2008 | CA2430601C Piperazine derivatives |
05/06/2008 | CA2377803C Phenyl sulfamate derivatives |
05/02/2008 | WO2008050167A1 New phenylsulfamoyl benzamide derivatives as bradykinin antagonists |
04/30/2008 | CN100384418C Isoxazolopyridinones and use thereof in the treatment of parkinson's disease |
04/29/2008 | US7365088 Indazole-derivatives as factor Xa inhibitors |
04/29/2008 | US7365068 Hepatitis C virus infections; -(3-cyclopropyl-4-(pentyloxy)phenyl)-3-nicotinoylthiourea;methyl 2-oxo-2-(5-((3-(4-(pentyloxy)-3-(trifluoromethyl)phenyl)thioureido)carbonyl)pyridin-2-ylamino)acetate |
04/29/2008 | CA2394037C New derivatives of benzene sulfonamide, their preparation process and pharmaceutical compositions that contain them |
04/29/2008 | CA2363875C Method crystallising n-(4-trifluoromethylphenyl)-5-methyl-isoxazole-4-carboxamide |
04/29/2008 | CA2336474C C-terminal modified oxamyl dipeptides as inhibitors of the ice/ced-3 family of cysteine proteases |
04/24/2008 | WO2008011080A3 Benzo(d) isoxazole derivatives as c-kit tyrosine kinase inhibitors for the treatment of disorders associated with the over production of histamine |
04/24/2008 | US20080096943 Urea derivatives, for example, 1-(3,5-dimethyl-isoxazole-4-yl)-3-[4-[(4-fluorobenzyl)methylamino]-butyl]-urea; use in treating inflammatory or allergic condition such as an inflammatory or obstructive airways disease |
04/24/2008 | US20080096936 Sulfur substituted sulfonylaminocarboxylic acid N-arylamides, their preparation, their use and pharmaceutical preparations comprising them |
04/24/2008 | US20080096873 New compounds |
04/22/2008 | US7361679 Integrin VLA-4 ( alpha 4 beta 1) and/or integrin LPAM-1 ( alpha 4 beta 7) antagonists, cell adhesion inhibitor; bioavailability, oral administration;treating inflammatory diseases; e.g. 3-[2-(2,6-dichlorobenzoylamino)pyrid-5-yl]-2-{3-[(2,2-dimethylpropionyl)isobutylamino]-4-methoxyphenyl}propionic acid |
04/17/2008 | WO2008044767A1 Aromatic amine derivative and use thereof |
04/17/2008 | WO2008043263A1 Isoxazole derivatives and methods of treating diseases |
04/17/2008 | WO2008024337A3 Compounds and methods for inhibiting the interaction of bcl proteins with binding partners |
04/17/2008 | WO2008005528A3 Compositions and methods for the modulation of detrusor activity |
04/17/2008 | US20080090860 Side effect reduction; 2-carboxy-4-(2-propoxy-3,5-di-tert-butylphenyl)-benzo[b]thiophene for example; syndrome X, non-insulin dependent diabetes mellitus, cancer, photoaging, acne, psoriasis, obesity, cardiovascular disease, atherosclerosis, uterine leiomyomata, inflamatory or neurodegenerative disease |
04/17/2008 | US20080090840 Heterocyclic GPR40 Modulators |