Patents
Patents for C07D 261 - Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings (11,459)
09/2009
09/03/2009US20090220662 Isosorbide derivatives and their use as flavor modifiers, tastants, and taste enhancers
09/03/2009US20090220454 Use of the histone deacetylase inhibitor N-hydroxy-4-[2-(3-dimethylaminobenzofuran-2-ylcarbonylamino)ethoxy]benzamide (aka CRA-24781, PCI-24781) for treating myelogenous leukemia (MML) or acute myelogenous leukemia (AML), optionally in combination therapy
09/02/2009EP2094675A1 A salt of 3-benzyl-2-methyl-2,3,3a,4,5,6,7,7a-octahydrobenzo[d]isoxazol-4-one
09/02/2009EP2094674A1 A salt of 3-benzyl-2-methyl-2,3,3a,4,5,6,7,7a-octahydrobenzo[d]isoxazol-4-one
09/02/2009EP2094673A1 Compounds and methods for inhibiting the interaction of bcl proteins with binding partners
09/02/2009EP2094645A1 2-hydroxy-1,3-diaminopropane derivatives
09/01/2009US7582668 to treat cellular proliferative diseases, hyperplasias, solid tumor, cardiac hypertrophy, immune disorders and inflammation; modulators of one or more mitotic kinesins; N-(2-(2-dimethylamino-acetylamino)-1-{4-[8-(1-hydroxy-ethyl)-imidazo[1,2-a]pyridin-2-yl]-benzyl}-ethyl)-3-chloro-4-isopropoxy-benzamide
08/2009
08/27/2009WO2009105509A1 Amine and ether compounds which modulate the cb2 receptor
08/27/2009US20090216013 e.g.1,1-Dicyclohexyl-3-[5-(pyridin-2-ylsulfanyl)-thiazol-2-yl]-urea; useful for the management, treatment, control, or adjunct treatment of diseases, where increasing glucokinase activity is beneficial, in particular, type 2 diabetes
08/27/2009US20090215795 Cyclic amidine derivatives
08/27/2009US20090215768 Isoxazole derivatives and pharmaceutical compositions comprising the same
08/27/2009US20090215624 Alkoxyalkyl Spirocyclic Tetramic Acids and Tetronic Acids
08/27/2009CA2716515A1 Amine and ether compounds which modulate the cb2 receptor
08/26/2009CN101516839A Compounds which modulate the cb2 receptor
08/25/2009US7579465 For treatment of picornavirus infections in mammals
08/25/2009US7579313 Transglutaminase inhibitors and methods of use thereof
08/20/2009WO2009101082A1 Substituted sulfonic acid amide compounds
08/19/2009CN100528849C Process for the preparation of 1,2-dichloroethane free crystals of zonisamide and high pure crystals of zonisamide
08/19/2009CN100528154C Malonyl-COA decarboxylase inhibitors useful as metabolic modulators
08/18/2009US7576108 Substituted arylcyclopropylacetamides as glucokinase activators
08/13/2009WO2009003719A3 Indane-amine derivatives, their preparation and use as medicaments
08/12/2009EP2086948A2 Inhibitors of phosphodiesterase type-iv
08/12/2009CN101506148A Inhibitors for GLYT-1
08/06/2009US20090197928 Novel Receptor Antagonists and Their Methods of Use
08/05/2009EP2083816A2 Heterocyclic amide compounds useful as kinase inhibitors
08/05/2009EP2029559B1 Aryl-4-ethynyl-isoxazole derivatives
08/05/2009EP1888541B1 Benzo(d)isoxazol-3-yl-amine compounds and their use as vanilloid receptor ligands
08/05/2009EP1249233B9 Npyy5 antagonists
08/05/2009CN101500986A Di-aromatic substituted amides as inhibitors for GLYT1
08/05/2009CN100522952C Insecticidal phthalamide derivatives
08/05/2009CN100522174C Crystalline isoxazole derivative and medical preparation thereof
08/04/2009US7569727 Pesticidally active ketone and oxime derivatives
08/04/2009US7569601 Such as (2E)-3-{4-[1-ethyl-2,2-bis(4-hydroxyphenyl)ethenyl]phenyl}-2-propenoic acid; for selective estrogen receptor modulation; menopausal or postmenopausal disorders, vasomotor symptoms, urogenital or vulvar vaginal atrophy, atrophic vaginitis, female sexual dysfunction, breast cancer, osteoporosis
07/2009
07/29/2009EP2081905A2 Sulfonyl compounds which modulate the cb2 receptor
07/29/2009CN101492416A Compounds effecting glucokinase
07/28/2009US7566803 Vitamin D receptor modulators
07/28/2009US7566715 Substituted sulfonamide compounds useful for the prophylaxis and treatment of conditions relating to obesity, type II diabetes and/or disorders of the central nervous system
07/23/2009US20090186905 Anaplastic lymphoma kinase modulators and methods of use
07/22/2009EP2080752A1 Pesticidally active ketone and oxime derivatives
07/22/2009EP2006286A9 Isoxazole derivative and isothiazole derivative having inhibitory activity on 11 beta -hydroxysteroid dehydrogenase type i
07/22/2009EP1391456B1 2-iminoimidazole derivatives
07/22/2009CN101490021A Insecticidal compounds
07/16/2009US20090181970 Functionalized diarylisoxazoles inhibitors of ciclooxygenase
07/14/2009US7560589 Cycloalkylidene compounds as modulators of estrogen receptor
07/14/2009US7560561 Such as terfenadine carboxylic acid metabolite and carebastine using a 4-(4-halo-1-oxobutyl)-alpha,alpha-dimethyl-alpha-substituted toluene intermediate
07/09/2009WO2008154642A3 Antibacterial agents
07/09/2009US20090176782 Inhibitors of tace
07/08/2009EP2076133A2 Synthesis of enone intermediate
07/08/2009CN101479238A Amine derivative having npyy5 receptor antagonist activity
07/08/2009CN100509790C Aryl- and heteroarylcarbonylpiperazines and their use for the treatment of benign and malignant oncoses
07/08/2009CN100509759C Novel alpha-oxygenated or alpha-thiolated carboxylic acid penethylamide derivatives
07/07/2009US7557133 Such as (3S)-5-[(2,6-dichlorobenzoyl)oxy]-3-({[5-methyl-3-phenyl-4,5-dihydro-5-isoxazolyl]carbonyl}amino)-4-oxopentanoic acid for preventing inflammation and apoptosis; crystallization
07/07/2009CA2438324C Acylated 6,7,8,9-tetrahydro-5h-benzocycloheptenyl amines and their use as pharmaceutical
07/02/2009WO2009081892A1 Novel catechol derivative, pharmaceutical composition containing the same, and use of those
07/02/2009US20090170911 Novel azole compound
07/02/2009US20090170824 Diarylsulfones as 5-HT2A Antagonists
07/01/2009EP2074084A1 Compounds which modulate the cb2 receptor
07/01/2009EP1756043B1 Ortho substituted aryl or heteroaryl amide compounds
07/01/2009EP1423362B1 New mandelic acid derivative and its use as thrombin inhibitor
07/01/2009CN100506788C Arylalkylcarbamate derivatives production and use thereof in therapy
06/2009
06/30/2009US7553972 Benzamide inhibitors of the P2X7 receptor
06/30/2009US7553966 Glucocorticoid mimetics, methods of making them, pharmaceutical compositions, and uses thereof
06/30/2009CA2406088C Novel phenyl-propargylether derivatives
06/25/2009WO2009077197A1 Insecticidal compounds
06/25/2009WO2009025983A4 Method for preparing 5-haloalkyl-4,5-dihydroisoxazole derivatives
06/25/2009US20090163549 Pharmaceutical Composition Comprising an Amide Derivative
06/25/2009CA2707612A1 Insecticidal compounds
06/24/2009CN100503576C Substituted azole compounds, preparation and application thereof
06/23/2009US7550489 N-[3-(4-chlorophenyl)-2-(3-cyanophenyl)-1-methylpropyl]-2-(5-trifluoromethyl-2-pyridyloxy)-2-methylpropanamide and phentermine, metformin, or bupropion; obesity; antipsychotic agents; synergistic; cannabinoid receptor antagonists
06/18/2009WO2009075080A1 Fluoroalkylsulfide derivative and pest control agent
06/18/2009US20090156643 Substituted isoxazoline compound and pesticide
06/17/2009EP2069020A2 Benzo[d]isoxazole derivatives as c-kit tyrosine kinase inhibitors for the treatment of disorders associated with the over production of histamine
06/17/2009EP1611088B1 Hydroxamates as therapeutic agents
06/17/2009CN101456846A Novel method for synthesizing acetyl-sulfisoxazole
06/16/2009CA2447640C Substituted anilide derivative, intermediate thereof, agricultural and horticultural chemical and its usage
06/11/2009WO2009051718A3 Calcium receptor modulating agents
06/11/2009US20090149459 P38 inhibitors and methods of use thereof
06/11/2009US20090149445 Tricyclic steroid hormone nuclear receptor modulators
06/11/2009US20090149425 Malononitrile compound as pesticides
06/11/2009US20090149415 Compounds for modulating the glycolysis enzyme complex and/or the transaminase complex
06/10/2009EP2066620A1 Di-aromatic substituted amides as inhibitors for glyt1
06/10/2009CN101454298A Novel crystal of 3-[5-[4-(cyclopentyloxy)-2- hydroxybenzoyl]-2-[(3-hydroxy-1,2-benzisoxazol-6- yl)methoxy]phenyl]propionic acid
06/10/2009CN101454297A Aryl-4-ethynyl-isoxazole derivatives
06/09/2009US7544704 Aryl-4-ethynyl-isoxazole derivatives
06/09/2009US7544701 Central nervous system disorders; psychological disorders
06/04/2009WO2009069643A1 Solid dispersion comprising 3-[5-[4-(cyclopentyloxy)- 2-hydroxybenzoyl]-2-[(3-hydroxy-1,2-benzisoxazol-6- yl)methoxy]phenyl]propionic acid or salt thereof, or composition comprising the solid dispersion
06/04/2009WO2009068557A1 Novel phenyl-acetamide and phenyl-propionamide derivatives useful as potassium channel modulators
06/04/2009WO2009068509A1 Novel benzamide derivatives useful as potassium channel modulators
06/04/2009US20090143435 GABA enhancers in the treatment of diseases relating to reduced neurosteroid activity
06/04/2009US20090143422 P38 inhibitors and methods of use thereof
06/04/2009US20090143365 Derivatives of alkylpiperazine- and alkylhomopiperazine-carboxylates, preparation method thereof and use of same as fatty acid amido hydrolase enzyme inhibitors
06/04/2009US20090143358 Inhibitors of ion channels
06/04/2009CA2707133A1 Chiral 3-(benzylsulfinyl)-5,5-dimethyl-4,5-dihydroisoxazole derivatives and 5,5-dimethyl-3-[(1h-pyrazol-4-ylmethyl)sulfinyl]-4,5-dihydroisoxazole derivatives, method for the production thereof, and use of same as herbicides and plant growth regulators
06/03/2009EP2065373A1 Chiral 3-(benzylsulfinyl)-5,5-dimethyl-4,5-dihydroisoxazole and 5,5-dimethyl-3-[(1H-pyrazol-4-ylmethyl) sulfinyl]-4,5-dihydroisoxazole derivatives, methods for their preparation and their use as herbicides and plant growth regulators
06/03/2009EP2064207A2 N-hydroxyamidinoheterocycles as modulators of indoleamine 2,3-dioxygenase
06/03/2009EP2064194A2 N-hydroxyamidinoheterocycles as modulators of indoleamine 2,3-dioxygenase
06/03/2009EP2064193A1 Heterocyclic gpr40 modulators
06/03/2009EP2064192A2 Compounds and methods for inhibiting the interaction of bcl proteins with binding partners
06/03/2009EP1140079B1 Assays for ligands for nuclear receptors
06/03/2009CN100494177C Bi-amido heterocyclic derivative with antitumour activity and its preparation method and use
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